"Hiroyuki Nakamura","Boron Delivery System for Neutron Capture Therapy","Asia Pacific Consortium of Gene and Cell Therapy 2019",,,,,,2019,Dec. "Hiroyuki Nakamura","Site-selective Protein Chemical Modification Using Tyrosine Click Reaction","The 20th General Assembly of the Federation of Asian Chemical Societies and The 18th Asian Chemical Congress",,,,,,2019,Dec. "佐藤伸一,中根啓太,對馬理彦,中村浩之","ナノメートルスケールの局所反応場を利用したタンパク質ラベル化反応による抗体の部位特異的修飾","第78回有機合成化学協会関東支部シンポジウム",,,,,,2019,Nov. "Shinichiro Fuse,Koshiro Masuda,Yuma Otake,Hiroyuki Nakamura","Peptide‐Chain Elongation Using Unprotected Amino Acids in a Micro‐Flow Reactor",,"Chemistry ? A European Journal",,,,,2019,Nov. "Shinichi Sato,Michihiko Tsushima,Keita Nakane,Hiroyuki Nakamura","Site-selective antibody chemical modification using photocatalyst-proximity labeling reaction","The 2nd edition of the International Symposium of CEFMS-NCTU, RCAS-AS (Taiwan) and 5-star Alliance (Japan)",,,,,,2019,Nov. "S. Fuse,K. Suzuki,T. Kuchimaru,T. Kadonosono,H. Ueda,S. Sato,S. Kizaka-Kondoh,H. Nakamura","Design, synthesis, and evaluation of indeno[2,1-c]pyrazolones for use as inhibitors against hypoxia-inducible factor (HIF)-1 transcriptional activity",,"Bioorg. Med. Chem",,,,,2019,Nov. "對馬理彦,中根啓太,佐藤伸一,中村浩之","標的タンパク質の部位選択的ラベル化を志向した光触媒担持ビーズ上での近接ラベル化法の開発","第9回CSJ化学フェスタ2019",,,,,,2019,Oct. "Takuya Asai,Hanqin Liu,Yasuyuki Ozeki,Shinichi Sato,Tomohiro Hayashi,Hiroyuki Nakamura","Imaging of Cellular Uptake of Boron Cluster Compound by Stimulated Raman Scattering Microscopy",,"Applied Physics Express",,,,,2019,Oct. "Hiroyuki Nakamura","Current Status and Future prospects for boron agents in BNCT","1st Russia BNCT Conference ? School of Young Scientists",,,,,,2019,Oct. "増田耕志郎,小竹佑磨,中村浩之","マイクロフロー法を駆使する無保護アミノ酸直接連結によるペプチド鎖伸長法の開発","第9回CSJ化学フェスタ2019",,,,,,2019,Oct. "Hiroyuki Nakamura","Albumin-Based Boron Delivery to Tumor on BNCT","The 3rd A3 Foresight Symposium on Organic/Inorganic Nanohybrid Platforms for Precision Tumor Imaging and Therapy",,,,,,2019,Oct. "Michihiko Tsushima,Shinichi Sato,Tatsuya Niwa,HIDEKI TAGUCHI,Hiroyuki Nakamura","Catalyst-proximity protein chemical labelling on affinity beads targeting endogenous lectins.",,"Chemical communications (Cambridge, England)",,"Vol. 55","No. 88","Page 13275-13278",2019,Oct. "J.-H. Choy,H. Nakamura,S. Eom,G. Choi","2-Dimensional Nanomaterials with Imaging and Diagnostic Functions for Nanomedicine",,"Bull. Chem. Soc. Jpn",,,"No. 93","pp. 1-12",2019,Oct. "S. Sato,H. Nakamura","Protein Chemical Labeling Using Biomimetic Radical Chemistry",,"Molecules",,"Vol. 24","No. 21"," 3890",2019,Oct. "塩野晴菜,林春菜,高門輝,?屋智久,中村浩之,岩田耕一","脂質二重膜ナノディスクの粘度評価の試み","分子科学討論会",,,,,,2019,Sept. "津田正仁,盛田大輝,福原信太郎,中村浩之","カチオン性金(I)触媒を用いたアザープロパルギルClaisen転位反応による5-アレニルイソオキサゾールの合成","第66回有機金属化学討論会",,,,,,2019,Sept. "中村浩之","ISNCTにおけるchemistry技術部会の方向性","第16回日本中性子捕捉療法学会学術大会",,,,,,2019,Sept. "佐藤伸一,松村雅喜,上田宏,中村浩之","チロシン残基修飾による抗体の部位選択的修飾と蛍光免疫センサー分子作成法への応用","第13回バイオ関連化学シンポジウム",,,,,,2019,Sept. "平松亮,川端信司,中村浩之,Vicente MGH,田中浩基,櫻井良憲,小野公二,黒岩敏彦,鰐淵昌彦","新規ホウ素化ポルフィリン・クロリンのconvection enhanced deliveryを用いたPDTおよびBNCTの有用性","PhotoDynamic Medicine PDM 2019",,,,,,2019,Sept. "岡田夏実,岩本真幸,林春菜,高門輝,老木成稔,中村浩之,岩田耕一","脂質二重膜に対する膜標的薬物の効果のピコ秒時間分解けい光分光法による検出","分子科学討論会",,,,,,2019,Sept. "呉尚沢,中川史子,中村浩之","中性子捕捉療法のための水溶性ホウ素クラスター含有葉酸誘導体の開発","日本薬学会関東支部大会",,,,,,2019,Sept. "中根啓太,對馬理彦,佐藤伸一,中村浩之","Ru光触媒担持アフィニティービーズを駆使した抗体のFc領域選択的化学修飾の開発","第13回バイオ関連化学シンポジウム",,,,,,2019,Sept. "森谷渉,布施新一郎,中村浩之","光線力学療法を指向したDπA光増感剤の合成と作用機序の解明","PhotoDynamic Medicine PDM 2019",,,,,,2019,Sept. "Shinichi Sato,Michihiko Tsushima,Keita Nakane,Hiroyuki Nakamura","Photocatalyst-Proximity-Dependent Protein Chemical Modification","he 14th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-14)",,,,,,2019,Sept. "Hiroyuki Nakamura,Kazuki Kawai,Takushi Takata,Minoru Suzuki","Development of Cyclic RGD-functionalized Maleimide-closo-dodecaborate Albumin Conjugate (cRGD-MID-AC) as a Tumor Targeting Boron Carrier","yBNCT10",,,,,,2019,Sept. "中村浩之","ホウ素を基軸としたがん治療戦略","九州大学先導物質化学研究所特別講演会",,,,,,2019,Sept. "Hiroyuki Nakamura","Tyrosine-Specific Protein Chemical Labeling","ICPAC Yangon 2019",,,,,,2019,Aug. "M. Mochizuki,S. Asatyas,S. Sato,F. Nakagawa,T. Hayashi,H. Nakamura","Distribution and Concentration of Small Molecules in Single Cells Visualized by νB-H Raman Microscopy",,"RSC Advance",,"Vol. 9",,"Page 23973?23978",2019,Aug. "S. Fuse,K. Masuda,Y. Otake,H. Nakamura","Peptide chain elongation using unprotected amino acids in a micro-flow reactor",,"Chem. Eur. J",,,,,2019,Aug. "M. Mochizuki,S. Sato,S. Asatyas,Z. J. Lesnikowski,T. Hayashi,H. Nakamura","Raman cell imaging with boron cluster molecules conjugated with biomolecules",,"Rsc Adv",,"Vol. 9","No. 41","pp. 23973-23978",2019,Aug. "布施新一郎,小竹佑磨,柴田裕介,林慶浩,川内進,中村浩之","N?メチル化ペプチドの超高効率マイクロフロー合成法の開発","第9回物質・デバイス領域共同研究拠点活動報告会 平成30年度ダイナミック・アライアンス成果報告会",,,,,,2019,July "Hiroyuki Nakamura","Protein Engineering Using Chemical Labeling Technology","Emerging Trends in Chemistry 2019",,,,,,2019,July "金光拓也,平松亮,福村匡央,川端信司,鈴木実,増永慎一郎,中川史子,宮武伸一,黒岩敏彦,小野公二,中村浩之","F98ラットグリオーマモデルに対する葉酸受容体標的新規ホウ素化合物を用いたホウ素中性子捕捉療法","第9回物質・デバイス領域共同研究拠点活動報告会・平成30年度ダイナミック・アライアンス成果報告会",,,,,,2019,July "川井一輝,佐藤伸一,中村浩之","中性子捕捉療法のためのcyclicRGDペプチドを用いた腫瘍選択的なホウ素送達法の開発","第35回DDS学会学術集会",,,,,,2019,July "Y. Asawa,K. Katsuragi,A. Sato,A. Yoshimori,S. Tanuma,H. Nakamura","Structure-based drug design of novel carborane-containing nicotinamide phosphoribosyltransferase inhibitors",,"Bioorg. Med. Chem.",,"Vol. 27","No. 13","Page 2832-2844",2019,July "中村浩之,川井一輝,高田卓志,鈴木実","cRGDペプチドを利用したアルブミンーホウ素キャリアの腫瘍ターゲティング","第25回癌治療増感研究会",,,,,,2019,June "Yuma Otake,Hiroyuki Nakamura,Shinichiro Fuse","Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor","11th Workshop on Organic Chemistry for Junior Chemists (WOCJC-11)",,,,,,2019,June "Yasunobu Asawa,Kiyotaka Katsuragi,Akira Sato,Atsushi Yoshimori,Sei-ichi Tanuma,Hiroyuki Nakamura","Structure-based Drug Design of Novel Carborane-containing NAMPT Inhibitors","11th Workshop on Organic Chemistry for Junior Chemists (WOCJC-11)",,,,,,2019,June "S. Yugandar,H. Nakamura","Rhodium(III)-catalyzed oxidative [4+2] annulation of isoxazolyl-4-carboxylic acids with alkynes: Oxidants control the tormation of pyra-noisoxazolones and isoquinolines",,"Chem. Commun",,"Vol. 55",,"Page 8382-8385",2019,June "Wanaporn Yimchuen,Tetsuya Kadonosono,Shinichi Sato,Takahiro Nomoto,Kyra See,Hiroyuki Nakamura,Nobuhiro Nishiyama,Shinae Kizaka-Kondoh","Development of photoimmunotherapy probe using a small antibody mimetic with structurally constrained anti-HER2 CDR peptides","11th International Peptide Symposium",,,,,,2019,June "Hiroyuki Nakamura,Shinichi Sato,Michihiko Tsushima,Keita Nakane","Protein Engineering Using Tyrosine-Specific Chemical Labeling Technology","11th Workshop on Organic Chemistry for Junior Chemists(WOCJC-11)",,,,,,2019,June "佐藤伸一,松村雅喜,中村浩之","抗体の部位選択的チロシン残基修飾に基づく蛍光免疫センサー分子の作成技術","日本ケミカルバイオロジー学会第14回年会",,,,,,2019,June "中村浩之","反応有機化学から生命分子夾雑科学へ","第30回記念 万有仙台シンポジウム",,,,,,2019,June "對馬理彦,佐藤伸一,中村浩之","アフィニティービーズ上での触媒近接標識のためのラベル化剤開発","日本ケミカルバイオロジー学会第14回年会",,,,,,2019,June "中根啓太,對馬理彦,佐藤伸一,中村浩之","Ru光触媒担持アフィニティービーズを用いた抗体のFc領域選択的修飾法の開発","日本ケミカルバイオロジー学会第14回年会",,,,,,2019,June "柴田裕介,林慶浩,小竹佑磨,中村浩之,布施新一郎,川内進","イミダゾール誘導体を触媒とするN-メチルアミド化反応機構の理論的解明","日本コンピューター化学会 2019年春季年会",,,,,,2019,June "對馬理彦,佐藤伸一,中村浩之","Ru光触媒近傍で起こる一電子移動反応を利用した標的タンパク質のケミカルラベリング","第115回有機合成シンポジウム",,,,,,2019,June "杉澤直斗,小竹佑磨,中村浩之,布施新一郎","マイクロフロー合成法による瞬間混合を駆使したβ?アミノ酸?N?カルボキシ無水物の合成とその応用","第115回有機合成シンポジウム",,,,,,2019,June "Somaraju Yugandar,Hiroyuki Nakamura","Rhodium(III)-Catalyzed Carboxylate-Directed C-H Functionalizations of Isoxazoles with Alkynes","第77回有機合成化学協会関東支部シンポジウム",,,,,,2019,May "佐藤伸一,對馬理彦,中村浩之","タンパク質ケミカルラベリングにおける一電子移動反応の活用 Utilization of Single Electron Transfer Reaction in Protein",,"有機合成化学協会誌",,"Vol. 77","No. 5","Page 463-471",2019,May "中根啓太,對馬理彦,佐藤伸一,中村浩之","Ru光触媒担持アフィニティービーズを用いた抗体の部位選択的修飾法の開発","第77回有機合成化学協会関東支部シンポジウム",,,,,,2019,May "小竹佑磨,柴田裕介,林慶浩,川内進,中村浩之,布施新一郎","アシルイミダゾリウムカチオン中間体を利用するマイクロフローNーメチル化ペプチド合成法の開発","第77回有機合成化学協会関東支部シンポジウム",,,,,,2019,May "増田耕志郎,小竹佑磨,中村浩之,布施新一郎","無保護アミノ酸連結を基盤とするマイクロフローペプチド鎖伸長法の開発","第77回有機合成化学協会関東支部シンポジウム",,,,,,2019,May "浅輪泰允,吉森篤史,中村浩之","SBDDによる新規カルボラン含有NAMPT阻害剤の開発","第77回有機合成化学協会関東支部シンポジウム",,,,,,2019,May "中村浩之","タンパク質夾雑空間解析を可能とする光触媒ー近接標識法の開発","分子夾雑の生命科学 第3回領域会議",,,,,,2019,May "S. Ishii,S. Sato,H. Asami,T. Hasegawa,J. Kohno,H. Nakamura","Design of S-S Bond Containing Maleimide-conjugated closo-Dodecaborate (SSMID): Identification of Unique Modification Sites on Albumin and Investigation of Intracellular Uptake",,"Org. Biomol. Chem",,"Vol. 17","No. 22",,2019,Apr. "Hiroyuki Nakamura","Isoxazole-Based Transformations via Direct C-H Activations","The Fifth International Scientific Conference "Advances in Synthesis and Complexing"",,,,,,2019,Apr. "Hiroyuki Nakamura","Protein Engineering Using Chemical Labeling Technology","ICMDA&ICCFE 2019",,,,,,2019,Apr. "浅輪泰允,中村浩之","ジカルボラン骨格を有する新規NAMPT阻害剤の理論的設計と合成、生物活性評価","日本化学会第99春季年会",,,,,,2019,Mar. "Hiroyuki Nakamura","In vivo tumor-targeting using small boron molecules: Limitation and possible solutions","Kyoto/Osaka-Taiwan BNCT International Conference",,,,,,2019,Mar. "Yuma Otake,Hiroyuki Nakamura,Shinichiro Fuse","An efficient synthesis of N-methylated peptides using micro-flow technology","日本化学会第99春季年会",,,,,,2019,Mar. "佐藤伸一,對馬理彦,中村浩之","アフィニティービーズ表面での局所的タンパク質ケミカルラベリング法の開発","日本薬学会第139年会",,,,,,2019,Mar. "Michihiko Tsushima,Shinichi Sato,Hiroyuki Nakamura","Proximity-dependent labeling on ruthenium photocatalyst-functionalized affinity beads","日本化学会第99春季年会",,,,,,2019,Mar. "中根啓太,對馬理彦,佐藤伸一,中村浩之","Ru光触媒担持アフィニティービーズを用いた抗体の部位選択的修飾法の開発","日本化学会第99春季年会",,,,,,2019,Mar. "川井一輝,佐藤伸一,中村浩之","中性子捕捉療法を志向した腫瘍アクティブターゲティングのための cyclic RGD ペプチド結合ホウ素化アルブミンの開発","日本化学会第99春季年会",,,,,,2019,Mar. "佐藤伸一,松村雅喜,中村浩之","チロシン残基ラベル化反応による抗体の相補性決定領域選択的修飾","日本化学会第99春季年会",,,,,,2019,Mar. "中村浩之","加速器中性子源を用いた中性子捕捉療法の現状と今後の展望",,"BIO Clinica",,"Vol. 34","No. 4","Page 431-434",2019,Mar. "Shinichiro Fuse,Yuma Otake,Hiroyuki Nakamura","Development of Amide Bond Formation of N-Methyl Amino Acids Using Micro-Flow Technology","日本化学会第99春季年会",,,,,,2019,Mar. "S. Sato,M. Yoshida,K. Hatano,M. Matsumura,H.Nakamura","N’-Acyl-N-methylphenylenediamine as a Novel Proximity Labeling Agent for Signal Amplification in Immunohistochemisty",,"Bioorg. Med. Chem.,",,"Vol. 27","No. 6","Page 1110-1118",2019,Mar. "akahiro Shimizu,Huber Vincent,Atsushi Yoshimori,Hiroki Ueda,Hiroyuki Nakamura,Hiroyuki Koji,Hiroki Oguri","Design, synthesis and biological evaluation of α-helix mimetics composed of skeletally diverse macrocyclic mid-sized scaffolds","The Fourth A3 Young Scientist Meeting,",,,,,,2019,Mar. "小林勇気,佐藤 伸一,丹羽 達也,田口英樹,中村浩之,田中寛","Analysis of initiation of organelle DNA replication in red alga Cyanidioschyzon merolae紅藻Cyanidioschyzon merolaeにおけるオルガネラDNA複製開始機構の解析","第61回日本植物生理学会年会",,,,,,2019,Mar. "浅井卓也,劉寒沁,小関泰之,林智広,佐藤伸一,中村浩之","ホウ素クラスター化合物の生細胞への取り込みの誘導ラマンイメーシ?ンク?","第66回応用物理学会春期学術講演会","第66回応用物理学会春期学術講演会",,,,,2019,Mar. "Taiki Morita,Shinichiro Fuse,Hiroyuki Nakamura","Photochemical conversion of isoxazoles to 5-hydroxyimidazolines and its application for protein labeling","日本化学会第99春季年会",,,,,,2019,Mar. "福原信太郎,Somaraju Yugandar,布施新一郎,中村浩之","イソキサゾロピリジン形成と窒素ー酸素結合開裂を経由するプロパルギルイソオキサゾールからの3ーヒドロキシー4ー置換ピコリノニトリルの一気合成","日本化学会第99春季年会",,,,,,2019,Mar. "増田 耕志郎,小竹 佑磨,中村 浩之,布施 新一郎","マイクロフロー法を駆使する無保護アミノ酸を用いたペプチド鎖伸長法の開発","日本化学会第99春季年会",,,,,,2019,Mar. "〇Yugandar Somaraju,Hiroyuki Nakamura","Rhodium(III)-Catalyzed Oxidative Coupling of Isoxazolyl-4-carboxylic acids with Alkynes: Oxidants Control the Formation of Pyranoisoxazolones and Isoquinolines","日本化学会第99春季年会",,,,,,2019,Mar. "Hiroyuki Nakamura","Boron Neutron Capture Therapy: Current Status and Future Aspect,","Conference on Chemistry and Chemical Process (ICCCP 2019)",,,,,,2019,Feb. "N. Sugisawa,Y. Otake,H. Nakamura,S. Fuse","Single-step, rapid, and mild synthesis of β-amino acid N-carboxy anhydrides using micro-flow technologies",,"Chem. Asian J.",,,,,2019, "Somaraju Yugandar,Hiroyuki Nakamura","Rhodium(iii)-catalysed carboxylate-directed C?H functionalizations of isoxazoles with alkynes",,"Chemical Communications",,"Vol. 55","No. 58","pp. 8382-8385",2019, "Shinichi Sato,Michihiko Tsushima,Keita Nakane,Hiroyuki Nakamura","SITE-SELECTIVE ANTIBODY MODIFICATION USING RADICAL-MEDIATED TYROSINE CLICK REACTION","第56回ペプチド討論会",,,,,,2019, "Hiroyuki Nakamura","Rhodium(iii)-catalysed carboxylate-directed C?H functionalizations of isoxazoles with alkynes",,"Chemical Communications",,,,,2019,