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石川智久 2006年 研究業績一覧 (16件 / 185件)
論文
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Shirasaka Y,
Onishi Y,
Sakurai A,
Nakagawa H,
Ishikawa T,
Yamashita S.
Evaluation of Human P-Glycoprotein (MDR1/ABCB1) ATPase Activity Assay Method by Comparing with in Vitro Transport Measurements: Michaelis-Menten Kinetic Analysis to Estimate the Affinity of P-Glycoprotein to Drugs.,
Biol. Pharm. Bull.,
Vol. 29,
No. 12,
pp. 2465-2471,
2006.
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Tamura A,
Wakabayashi K,
Onishi Y,
Nakagawa H,
Tsuji M,
Matsuda Y,
Ishikawa T.
Genetic polymorphisms of human ABC transporter ABCG2: Development of the standard method for functional validation of SNPs by using the Flp recombinase system.,
J. Exp. Ther. Oncol.,
Vol. 6,
No. 1,
pp. 1-11,
2006.
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Tamura A,
Watanabe M,
Saito H,
Nakagawa H,
Kamachi T,
Okura I,
Ishikawa T.
Functional validation of the genetic polymorphisms of human ATP-binding cassette (ABC) transporter ABCG2: identification of alleles that are defective in porphyrin transport.,
Mol. Pharmacol.,
Vol. 70,
No. 1,
pp. 287-296,
2006.
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Hirano H,
Kurata A,
Onishi Y,
Sakurai A,
Saito H,
Nakagawa H,
Nagakura M,
Tarui S,
Kanamori Y,
Kitajima M,
Ishikawa T.
High-Speed Screening and QSAR Analysis of Human ATP-Binding Cassette Transporter ABCB11 (Bile Salt Export Pump) To Predict Drug-Induced Intrahepatic Cholestasis.,
Mol. Pharm.,
Vol. 3,
No. 3,
pp. 252-265,
2006.
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Wakabayashi K,
Tamura A,
Saito H,
Onishi Y,
Ishikawa T.
Human ABC transporter ABCG2 in xenobiotic protection and redox biology.,
Drug Metab. Rev.,
Vol. 38,
No. 3,
pp. 371-391,
2006.
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Yoshiura K,
Kinoshita A,
Ishida T,
Ninokata A,
Ishikawa T,
Kaname T,
Bannai M,
Tokunaga K,
Sonoda S,
Komaki R,
Ihara M,
Saenko VA,
Alipov GK,
Sekine I,
Komatsu K,
Takahashi H,
Nakashima M,
Sosonkina N,
Mapendano CK,
Ghadami M,
Nomura M,
Liang DS,
Miwa N.
A SNP in the ABCC11 gene is the determinant of human earwax type.,
Nat. Genet.,
Vol. 38,
No. 3,
pp. 324-330,
2006.
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Wakabayashi K,
Nakagawa H,
Adachi T,
Kii I,
Kobatake E,
Kudo A,
Ishikawa T.
Identification of cysteine residues critically involved in homodimer formation and protein expression of human ATP-binding cassette transporter ABCG2: a new approach using the flp recombinase system.,
J. Exp. Ther. Oncol.,
Vol. 5,
No. 3,
pp. 205-222,
2006.
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Ishikawa T,
Ikegami Y,
Sano K,
Nakagawa H,
Sawada S.
Transport mechanism-based drug molecular design: novel camptothecin analogues to circumvent ABCG2-associated drug resistance of human tumor cells.,
Curr. Pharm. Des.,
Vol. 12,
No. 3,
pp. 313-325,
2006.
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Nakagawa H,
Saito H,
Ikegami Y,
Aida-Hyugaji S,
Sawada S,
Ishikawa T.
Molecular modeling of new camptothecin analogues to circumvent ABCG2-mediated drug resistance in cancer.,
Cancer Lett.,
Vol. 234,
No. 1,
pp. 81-89,
2006.
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Nakata K,
Tanaka Y,
Nakano T,
Adachi T,
Tanaka H,
Kaminuma T,
Ishikawa T.
Nuclear receptor-mediated xenobiotic procession loops in phase I, II, and III drug metabolizing systems.,
Drug Metab. Pharmacokinet.,
Vol. 21,
pp. 437-457,
2006.
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Saito H,
Hirano H,
Nakagawa H,
Fukami T,
Oosumi K,
Murakami K,
Kimura H,
Kouchi T,
Konomi M,
Tao E,
Tsujikawa N,
Tarui S,
Nagakura M,
Osumi M,
Ishikawa T.
A new strategy of high-speed screening and quantitative structure-activity relationship analysis to evaluate human ATP-binding cassette transporter ABCG2-drug interactions.,
J. Pharmacol. Exp. Ther.,
Vol. 317,
No. 3,
pp. 1114-1124,
2006.
著書
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石川智久.
CMCテクニカルライブラリー DNAチップの開発II・第4章 薬物トランスポーターに基づく創薬分子デザイン -21世紀ゲノム創薬にむけた産学連携の提案-,
シーエムシー出版,
pp. 148-157,
Dec. 2006.
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Susan P.C. Cole,
Ian F. Tannock 【訳=石川智久】.
がんのベーシックサイエンス・第18章 薬剤耐性,
メディカル・サイエンス・インターナショナル,
pp. 419-444,
Nov. 2006.
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石川智久,
櫻井亜季,
田村藍,
大西裕子,
宝田裕,
橋本幸蔵,
川瀬三雄.
『バイオ解析・診断技術のテーラーメイド医療への応用』・第2章 薬物トランスポーターの遺伝子多型:機能バリデーション法の国際標準化とSNP診断システムの開発,
シーエムシー出版,
pp. 219-231,
Oct. 2006.
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蔵田敦夫,
櫻井亜季,
大西裕子,
平野弘之,
石川智久.
毒性質問箱<医薬品副作用予測の最前線> 安全性評価研究会編集企画委員会編・ 薬物性胆汁鬱滞の予測:胆汁酸トランスポーター(ABCB11/BSEP/sPGP)の高速スクリーニングと定量的幸蔵活性相関(QSAR)解析,
サイエンティスト社,
pp. 15-24,
June 2006.
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