@article{CTT100842475, author = {Naoto Sugisawa and Hiroyuki Nakamura and Sinichiro Fuse}, title = {Recent advances in the continuous-flow reactions using metal-free homogeneous catalysts}, journal = {Catalysts}, year = 2020, } @article{CTT100842474, author = {Somaraju Yugandar and Taiki Moritai and Hiroyuki Nakamura}, title = {Rhodium(III)-Catalyzed Direct C-H Functionalization of Isoxazoles with Alkynes, Alkenes and Sulfoxonium Ylides}, journal = {Org. Biomol. Chem}, year = 2020, } @article{CTT100833095, author = {Shinichi Sato and Hiroyuki Nakamura}, title = {Labeling of Peroxidase-Induced Oxidative Stress Hotspots by Hemin-Catalyzed Tyrosine Click}, journal = {Chem. Pharm. Bull.}, year = 2020, } @article{CTT100843378, author = {S. A. Anufriev and I. B. Sivaev and Hiroyuki Nakamura}, title = {Two possible ways to combine boron and gadolinium for Gd-guided BNCT. A concept}, journal = {Phosphorus, Sulfur and Silicon}, year = 2020, } @article{CTT100833117, author = {Yasunobu. Asawa and A. Yoshimori and J. Bajorath and Hiroyuki. Nakamura}, title = {Prediction of an MMP-1 Inhibitor Activity Cliff Using the SAR Matrix Approach and Its Experimental Validation}, journal = {Sci. Rep}, year = 2020, } @article{CTT100833118, author = {T. Masuzawa and S. Sato and T. Niwa and H. Taguchi and H. Nakamura and T. Oyoshi}, title = {G-Quadruplex-Proximity Protein Labeling Based on Peroxidase Activity}, journal = {Chem. Commun.}, year = 2020, } @article{CTT100833119, author = {Kazuki Kawai and Kai Nishimura and Satoshi Okada and Shinichi Sato and Minoru Suzuki and T. Takata and Hiroyuki Nakamura}, title = {Cyclic RGD-Functionalized closo-Dodecaborate Albumin Conjugates as Integrin Targeting Boron Carriers for Neutron Capture Therapy}, journal = {Mol. Pharm.}, year = 2020, } @article{CTT100833116, author = {Sei-ichi Tanuma and Takahiro Oyama and Atsushi Yoshimori and Kiyotaka Katsuragi and Yuri Shibasaki and Yasunobu Asawa and Hiroaki Yamazaki and Kosho Makino and Miwa Okazawa and Yoko Ogino and Yoshimi Sakamoto and Miyuki Nomura and Akira Sato and Hideaki Abe and Hiroyuki Nakamura and Hideyo Takahashi and Nobuhiro Tanuma and Fumiaki Uchiumi}, title = {Structural insights into the tunnel-shaped cavity of human nicotinamide phosphoribosyltransferase using a close structural set of azacyclohexane-motif inhibitors}, journal = {Molecules}, year = 2020, } @article{CTT100833115, author = {Fumiko Nakagawa and H. Kawashima and Taiki. Morita and Hiroyuki. Nakamura}, title = {Water-soluble closo-Docecaborate-conjugated Pteroyl Derivatives for Boron Neutron Capture Therapy: Evidence of Targeting to Folate Receptor-Mediated Cell Uptake}, journal = {Cells}, year = 2020, } @article{CTT100833090, author = {Shinichiro. Fuse and Wataru Moriya and Shinichi Sato and Hiroyuki Nakamura}, title = {Investigation into the influence of an acrylic acid acceptor in organic D-π-A sensitizers against phototoxicity}, journal = {Bioorg. Med. Chem.}, year = 2020, } @article{CTT100833099, author = {Jun. Kawamura and Hiroshi. Kitamura and Yuma. Otake and Shinichiro. Fuse and Hiroyuki. Nakamura}, title = {Size-Controllable and Scalable Production of Liposomes Using a V-Shape Mixer Micro-Flow Reactor}, journal = {Org. Process Res. Dev.}, year = 2020, } @article{CTT100833092, author = {Michihiko Tsushima and Shinichi Sato and Keita Nakane and Hiroyuki Nakamura}, title = {Target protein identification on the photocatalyst-functionalized magnetic affinity beads}, journal = {Current Protocol.}, year = 2020, } @article{CTT100833091, author = {Guangzhe Li, and Chengdong Wang and Yueqing Li, and Kun Shao and Guo Yu and Shisheng Wang, and Xiuhan Guo, and Weijie Zhao and H. Nakamura}, title = {Zinc (II)-Catalyzed Intramolecular Hydroarylation-Redox Cross-Dehydrogenative Coupling of N-Propargylamines with sp and sp3 Carbon Pronucleophiles: Facile Access to Multifunctionalized Tetrahydroquinolines}, journal = {Chem. Commun.}, year = 2020, } @article{CTT100833085, author = {S. Sato and K. Nakane and H. Nakamura}, title = {Laccase-Catalysed Tyrosine Click Reaction}, journal = {Org. Biomol. Chem}, year = 2020, } @article{CTT100826199, author = {Wanaporn Yimchuen and Tetsuya Kadonosono and Yumi Ota and Shinichi Sato and Maika Kitazawa and Tadashi Shiozawa and Takahiro Kuchimaru and Masumi Taki and Yuji Ito and Hiroyuki Nakamura and Shinae Kizaka-Kondoh}, title = {Strategic design to create HER2-targeting proteins with target-binding peptides immobilized on a fibronectin type III domain scaffold}, journal = {RSC Advances}, year = 2020, } @article{CTT100852985, author = {盛田 大輝 and 布施 新一郎 and 中村 浩之}, title = {Novel Photochemical Conversion of Isoxazoles to 5-Hydroxyimidazolines: Possible Protein Labeling at Lysine Residues}, journal = {Org. Lett}, year = 2020, } @article{CTT100843293, author = {Y. Otake and Y. Shibata and Y. Hayashi and S. Kawauchi and H. Nakamura and S. Fuse}, title = {N-Methylated Peptide Synthesis through Acyl N-Methylimidazolium Cation Generation Accelerated by a Brønsted Acid}, journal = {Angew. Chem. Int. Ed.}, year = 2020, } @article{CTT100826198, author = {Shinichi Sato and Masaki Matsumura and Tetsuya Kadonosono and Satoshi Abe and Takafumi Ueno and Hiroshi Ueda and Hiroyuki Nakamura}, title = {Site-selective protein chemical modification of exposed tyrosine residues using tyrosine click reaction}, journal = {Bioconjugate Chemistry}, year = 2020, } @article{CTT100822307, author = {中村浩之}, title = {ホウ素中性子捕捉療法:がん細胞内でα線を発生させる次世代放射線治療}, journal = {DDS学会誌}, year = 2020, } @article{CTT100822137, author = {Hiroyuki Nakamura}, title = {Carrier proteins-based boron delivery to tumor}, journal = {Applied Radiation and Isotopes}, year = 2020, } @article{CTT100822138, author = {Hiroyuki Nakamura}, title = {Suppression of HIF-1α accumulation by betulinic acid through proteasome activation in hypoxic cervical cancer}, journal = {Biochemical and Biophysical Research Communications}, year = 2020, } @article{CTT100822136, author = {Hiroyuki Nakamura}, title = {Boron Neutron Capture Therapy Study of 10B Enriched Nanostructured Boron Carbide Against Cervical Cancer and Glioblastoma Cell Line}, journal = {Journal of Cluster Science}, year = 2020, } @article{CTT100822311, author = {中村浩之}, title = {中性子捕捉療法のためホウ素薬剤研究開発の進展-ホウ素薬剤が今後適応疾患拡大の鍵を握る!}, journal = {日本原子力学会誌}, year = 2020, } @article{CTT100822140, author = {Naoto Sugisawa and Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {Single‐Step, Rapid, and Mild Synthesis of β‐Amino Acid N ‐Carboxy Anhydrides Using Micro‐Flow Technology}, journal = {Chemistry – An Asian Journal}, year = 2020, } @article{CTT100809277, author = {A. Kumar; M. Kaur; P. Singh; K. Singh; U. S. Gaharwar; R. Meena; M. Kumar; K. Nakagawa; S. Wu; M. Suzuki; H. Nakamura and Hiroyuki Nakamura}, title = {Boron Nitride (10BN) a prospective material for treatment of cancer by Boron Neutron Capture Therapy (BNCT)}, journal = {Materials Letters}, year = 2020, } @article{CTT100822141, author = {Shinichiro Fuse and Tsukasa Oishi and Keisuke Matsumura and Yoshihiro Hayashi and Susumu Kawauchi and Hiroyuki Nakamura}, title = {Design, synthesis, and evaluation of azo D–π-A dyes as photothermal agents}, journal = {Organic & Biomolecular Chemistry}, year = 2020, } @article{CTT100822142, author = {Naoto Sugisawa and Hiroyuki Nakamura and Shinichiro Fuse}, title = {Micro-flow synthesis of β-amino acid derivatives via a rapid dual activation approach}, journal = {Chemical Communications}, year = 2020, } @article{CTT100822144, author = {Hiroyuki Nakamura}, title = {Suppression of HIF-1α accumulation by betulinic acid through proteasome activation in hypoxic cervical cancer}, journal = {Biochemical and Biophysical Research Communications}, year = 2020, } @inproceedings{CTT100844790, author = {Hiroyuki Nakamura}, title = {Development of Protein Chemical Labeling: From Target Identification to Cancer Therapy}, booktitle = {}, year = 2020, } @inproceedings{CTT100844789, author = {Hiroyuki Nakamura}, title = {Albumin-Dodecaborate Conjugates as Efficient Boron Carriers for Neutron Capture Therapy}, booktitle = {}, year = 2020, } @inproceedings{CTT100836673, author = {Hiroyuki Nakamura}, title = {Development of Boron Agents for BNCT}, booktitle = {}, year = 2020, } @inproceedings{CTT100836670, author = {津田 正仁 and 盛田 大輝 and 福原 信太郎 and 中村 浩之}, title = {金(I)触媒を用いたプロパルギルアザClaisen転位反応による5-アレニルイソオキサゾールの合成}, booktitle = {}, year = 2020, } @inproceedings{CTT100844788, author = {Hiroyuki Nakamura and Kazuki Kawai and Kai Nishimura and Satoshi Okada and Takushi Takata and Minoru Suzuki}, title = {Albumin-Based Boron Delivery for Active Targeting to Tumor}, booktitle = {}, year = 2020, } @inproceedings{CTT100844787, author = {中村 浩之}, title = {がんの低侵襲治療法(中性子捕捉療法):承認までの軌跡と今後の展望}, booktitle = {}, year = 2020, } @inproceedings{CTT100836672, author = {杉澤直斗 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフローリアクター内でのpH瞬間転換と両基質同時活性化を駆使したβ-アミノ酸-N-カルボン酸無水物の合成と誘導体化}, booktitle = {}, year = 2020, } @inproceedings{CTT100836671, author = {岡田夏実 and 高門輝 and 岩本真幸 and 老木成稔 and 中村浩之 and 岩田耕一}, title = {ピコ秒時間分解けい光分光法を用いて評価した局所麻酔薬の脂質二重膜への影響}, booktitle = {}, year = 2020, } @inproceedings{CTT100836669, author = {YU Guo and ZHANG Xuhai and LI Guangzhe and Hiroyuki Nakamura}, title = {Synthesis of 2-Phosphonotetrahydroquinoline with Site-Selective C-H Bond Functionalization through Intramolecular Hydroarylation-Redox CDC Reaction}, booktitle = {}, year = 2020, } @inproceedings{CTT100836668, author = {小室 敬史 and 小竹 佑磨 and 中村 浩之 and 布施 新一郎}, title = {マイクロフローリアクター内でのトリホスゲンを用いた環状ペプチド合成法の開発}, booktitle = {}, year = 2020, } @inproceedings{CTT100836667, author = {浅輪 泰允 and 吉森 篤史 and BAJORATH J?rgen and 中村 浩之}, title = {SAR空間の可視化によるActivity cliffの予測とその実験的検証}, booktitle = {}, year = 2020, } @inproceedings{CTT100836666, author = {對馬理彦 and Yijin Wen and 津賀雄輝 and 金森功吏 and 湯浅英哉 and 中村浩之}, title = {リガンド連結型有機光触媒を用いた標的タンパク質の酸化的不活性化と抗腫瘍活性}, booktitle = {}, year = 2020, } @inproceedings{CTT100836663, author = {岡田夏実 and 岩本真幸 and 高門輝 and 中村浩之 and 老木成稔 and 岩田耕一}, title = {ピコ秒時間分解けい光分光法で評価した脂質二重膜の粘度に対する局所麻酔薬の影響―脂質分子の極性基による違い}, booktitle = {}, year = 2020, } @inproceedings{CTT100836662, author = {塩野晴菜 and 高門輝 and 髙屋智久 and 中村浩之 and 岩田耕一}, title = {時間分解けい光分光法による脂質二重膜ナノディスクの粘度評価}, booktitle = {}, year = 2020, } @inproceedings{CTT100836661, author = {Hiroyuki Nakamura and Kawai Kazuki and Shinichi Sato and Minoru Suzuki and }, title = {Albumin-Based Boron Delivery to Tumor by Active Targeting via αvβ3 Integrin}, booktitle = {}, year = 2020, } @inproceedings{CTT100836660, author = {佐藤伸一 and 増澤樹 and 大吉崇文 and 丹羽達也 and 田口英樹 and 中村浩之}, title = {ペルオキシダーゼ活性の変化と近接標識を利用したグアニン四重鎖結合タンパク質の選択的化学修飾}, booktitle = {}, year = 2020, } @inproceedings{CTT100836665, author = {對馬理彦 and 佐藤伸一 and 中村浩之}, title = {タンパク質-タンパク質相互作用の解析を志向した細胞内触媒近接ラベル化の開発}, booktitle = {}, year = 2020, } @inproceedings{CTT100836664, author = {Rohmad Yudi Utomo and Yasunobu Asawa and Atsushi Yoshimori and Hiroyuki Nakamura}, title = {Novel Curcumin Derivatives Generated from SAR Matrix Possess as Amyloid β Inhibitors for Alzheimer?s Disease}, booktitle = {}, year = 2020, } @inproceedings{CTT100844786, author = {中村 浩之}, title = {BNCT 用ホウ素薬剤:現在の状況と将来の展望、}, booktitle = {}, year = 2020, } @inproceedings{CTT100844785, author = {中村 浩之}, title = {細胞内タンパク質-タンパク質相互作用解析を可能とする光ラベル化技術の開発}, booktitle = {}, year = 2020, } @inproceedings{CTT100844783, author = {Hiroyuki Nakamura and Eva Hey-Hawkins}, title = {Boron Compounds}, booktitle = {}, year = 2020, } @inproceedings{CTT100844784, author = {Hiroyuki Nakamura}, title = {Boron Delivery Agents for BNCT: Current Status and Future Prospects}, booktitle = {}, year = 2020, } @inproceedings{CTT100823567, author = {浅輪泰允 and 吉森篤史 and 山田健太郎 and 邵玉潔 and 李廣晢 and 加藤明良 and 小路弘行 and 中村浩之}, title = {タンパク質の2次構造を模倣した新規カルボランPPI制御分子の設計・合成とその機能評価}, booktitle = {}, year = 2020, } @inproceedings{CTT100823566, author = {増澤樹 and 佐藤伸一 and 中村浩之 and 大吉崇文}, title = {ヘミンによって活性化したルミノール誘導体によるグアニン四重鎖結合タンパク質の選択的修飾}, booktitle = {}, year = 2020, } @inproceedings{CTT100823565, author = {Takahiro Shimizu and Huber Vincent and Atsushi Yoshimori and Hiroki Ueda and Hiroyuki Nakamura and Hiroyuki Koji and Hiroki Oguri}, title = {Design, synthesis and biological evaluation of α-helix mimetics composed of skeletally diverse macrocyclic mid-sized scaffolds,}, booktitle = {}, year = 2020, } @inproceedings{CTT100823564, author = {YU Guo and Xuhai Zhang and 李 廣哲 and 中村 浩之}, title = {Synthesis of tetrahydroquinoline with site-selective C-H bond functionalization through IH-Redox CDC reaction}, booktitle = {}, year = 2020, } @inproceedings{CTT100823563, author = {津田正仁 and 盛田大輝 and 福原信太郎 and 中村浩之}, title = {金(I)触媒を用いたアザプロパルギルClaisen転位反応による5-アレニルイソオキサゾールの合成}, booktitle = {}, year = 2020, } @inproceedings{CTT100823562, author = {杉澤直斗 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {β-アミノ酸-N-カルボン酸無水物の迅速かつ温和なワンフロー合成}, booktitle = {}, year = 2020, } @inproceedings{CTT100823561, author = {梅寺倖平 and 盛田大輝 and 中村浩之}, title = {飽和炭素に富むアザトリシクロドデセン骨格の合成}, booktitle = {}, year = 2020, } @inproceedings{CTT100823560, author = {森谷渉 and 布施新一郎 and 中村浩之}, title = {光線力学療法を志向したDπA光増感剤の構造光毒性相関の解明}, booktitle = {}, year = 2020, } @inproceedings{CTT100823559, author = {中根啓太 and 佐藤伸一 and 對馬理彦 and 丹羽達也 and 田口英樹 and 中村浩之}, title = {アフィニティー担体上でのチロシン残基修飾による抗体の部位選択的修飾}, booktitle = {}, year = 2020, } @inproceedings{CTT100823558, author = {佐藤伸一 and 中村浩之}, title = {チロシン残基ラベル化における触媒的手法と電気化学的手法の比較}, booktitle = {}, year = 2020, } @inproceedings{CTT100823557, author = {Takahiro Shimizu and Huber Vincent and Atsushi Yoshimori and Hiroki Ueda and Hiroyuki Nakamura and Hiroyuki Koji and Hiroki Oguri}, title = {Design, synthesis and biological evaluation of α-helix mimetics composed of skeletally diverse macrocyclic mid-sized scaffolds}, booktitle = {}, year = 2020, } @inproceedings{CTT100823568, author = {Rohmad Yudi Utomo and Yasunobu Asawa and Shinichi Sato and Atsushi Yoshimori and Hiroyuki Nakamura}, title = {Novel Curcumin Derivatives Generated from SAR Matrix Possess as Amyloid β Inhibitors}, booktitle = {}, year = 2020, } @misc{CTT100882394, author = {中村浩之 and 梅寺倖平 and 盛田大輝 and 小路 弘行 and 吉森 篤史}, title = {新規含窒素三環性骨格化合物およびその使用}, howpublished = {公開特許}, year = 2022, month = {}, note = {特願2020-204328(2020/12/09), 特開2022-091476(2022/06/21)} } @misc{CTT100868492, author = {布施新一郎 and 増田耕志郎 and 小竹佑磨 and 中村浩之}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2021-501811(2020/02/03), 再表2020/175023(2021/12/16)} } @misc{CTT100826091, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {フローリアクターを用いるN-カルボキシ無水物の合成方法}, howpublished = {登録特許}, year = 2023, month = {}, note = {特願2019-094952(2019/05/21), 特開2020-011948(2020/01/23), 特許第7362055号(2023/10/06)} } @misc{CTT100835044, author = {中村浩之 and 佐藤伸一 and 深瀬 浩一}, title = {電気化学的手法を用いたハロゲン化物の製造方法}, howpublished = {登録特許}, year = 2022, month = {}, note = {特願2018-239130(2018/12/21), 特開2020-100865(2020/07/02), 特許第7166531号(2022/10/28)} } @misc{CTT100826082, author = {佐藤伸一 and 中村浩之}, title = {電気化学的手法による修飾タンパク質の製造方法}, howpublished = {公開特許}, year = 2020, month = {}, note = {特願2018-124834(2018/06/29), 特開2020-002095(2020/01/09)} } @misc{CTT100785207, author = {佐藤伸一 and 中村浩之 and 中野 洋文}, title = {チロシンホスファターゼ及びチロシンキナーゼ活性の測定方法}, howpublished = {登録特許}, year = 2020, month = {}, note = {特願2017-544450(2016/09/26), 特開(再表)2017/061288(2018/09/06), 特許第6770750号(2020/09/30)} } @misc{CTT100808478, author = {中村浩之}, title = {ホウ素含有化合物とタンパク質とのコンジュゲートを含む医薬組成物}, howpublished = {登録特許}, year = 2020, month = {}, note = {特願2017-534171(2016/07/26), 再表2017/026276(2018/05/24), 特許第6788278号(2020/11/04)} }