"H. Kitamura,Y. Otake,N. Sugisawa,H. Sugisawa,T. Ida,H. Nakamura,S. Fuse,Hiroyuki Nakamura","Sequential Selective Introduction of Alcohols against Phosphorus Trichloride in a Continuous-Flow Reactor and Consideration of a Mechanism for Reduced Overreaction via the Addition of Imidazole",,"Chemistry",," 28"," 37"," e202200932",2022,July "北村宙士,小竹佑磨,杉澤直斗,杉澤宏樹,井田朋智,中村浩之,布施新一郎","非対称リン酸トリエステルのマイクロフロー合成および反応機構解明","創薬懇話会2022",,,,,,2022,June "北村宙士,小竹佑磨,杉澤直斗,杉澤宏樹,井田朋智,中村浩之,布施新一郎","非対称リン酸トリエステルのマイクロフロー合成および反応機構解明","第120回有機合成シンポジウム",,,,,,2022,June "社本乙華,小室敬史,杉澤直斗,中村浩之,布施新一郎","マイクロフローリアクター内での環状ペプチド合成法の開発","日本化学会第102春季年会",,,,,,2022,Mar. "Taiki Morita,Shinichiro Fuse,Hiroyuki Nakamura","Photochemical conversion of isoxazoles to 5-hydroxyimidazolines","Pacifichem",,,,,,2021,Dec. "北村宙士,小竹佑磨,杉澤直斗,杉澤宏樹,井田朋智,中村浩之,布施新一郎","マイクロフローリアクターを用いる非対称リン酸トリエステルの高速合成","第11回CSJ化学フェスタ2021",,,,,,2021,Oct. "N. Sugisawa,H. Sugisawa,Y. Otake,R. V. Krems,H. Nakamura,S. Fuse","Rapid and Mild One-Flow Synthetic Approach to Unsymmetrical Sulfamides Guided by Bayesian Optimization",,"Chemistry Methods",,,,,2021,July "小室敬史,小竹佑磨,中村浩之,布施新一郎","マイクロフローリアクター内でのトリホスゲンを用いた迅速なラクタム合成法の開発","日本化学会第101春季年会(オンライン)",,,,,,2021,Mar. "北村宙士,小竹佑磨,中村浩之,布施新一郎","マイクロフローリアクターを用いる非対称リン酸トリエステルの高速合成","日本化学会第101春季年会(オンライン)",,,,,,2021,Mar. "杉澤直斗,中村浩之,布施新一郎","マイクロフローリアクター内での瞬間両基質活性化を駆使したβ-アミノ酸誘導体の合成","日本化学会第101春季年会(オンライン)",,,,,,2021,Mar. "杉澤直斗,小竹佑磨,中村浩之,布施新一郎","マイクロフローリアクター内でのpH瞬間転換と両基質同時活性化を駆使したβ-アミノ酸-N-カルボン酸無水物の合成と誘導体化","第117回有機合成シンポジウム(オンライン)",,,,,,2020,Oct. "Shinichiro. Fuse,Wataru Moriya,Shinichi Sato,Hiroyuki Nakamura","Investigation into the influence of an acrylic acid acceptor in organic D-π-A sensitizers against phototoxicity",,"Bioorg. Med. Chem.",,"Vol. 28","No. 13","pp. 115558",2020,July "Jun. Kawamura,Hiroshi. Kitamura,Yuma. Otake,Shinichiro. Fuse,Hiroyuki. Nakamura","Size-Controllable and Scalable Production of Liposomes Using a V-Shape Mixer Micro-Flow Reactor",,"Org. Process Res. Dev.",,"Vol. 24","No. 10","pp. 2122-2127",2020,June "盛田 大輝,布施 新一郎,中村 浩之","Novel Photochemical Conversion of Isoxazoles to 5-Hydroxyimidazolines: Possible Protein Labeling at Lysine Residues",,"Org. Lett",,,,,2020,Apr. "Y. Otake,Y. Shibata,Y. Hayashi,S. Kawauchi,H. Nakamura,S. Fuse","N-Methylated Peptide Synthesis through Acyl N-Methylimidazolium Cation Generation Accelerated by a Br?nsted Acid",,"Angew. Chem. Int. Ed.",,"Vol. 59","No. 31","pp. 12925-12930",2020,Apr. "森谷渉,布施新一郎,中村浩之","光線力学療法を志向したDπA光増感剤の構造光毒性相関の解明","日本化学会第100春季年会",,,,,,2020,Mar. "杉澤直斗,小竹佑磨,中村浩之,布施新一郎","β-アミノ酸-N-カルボン酸無水物の迅速かつ温和なワンフロー合成","日本化学会第100春季年会",,,,,,2020,Mar. "S. Fuse,K. Suzuki,T. Kuchimaru,T. Kadonosono,H. Ueda,S. Sato,S. Kizaka-Kondoh,H. Nakamura","Design, synthesis, and evaluation of indeno[2,1-c]pyrazolones for use as inhibitors against hypoxia-inducible factor (HIF)-1 transcriptional activity",,"Bioorg. Med. Chem",,,,,2019,Nov. "森谷渉,布施新一郎,中村浩之","光線力学療法を指向したDπA光増感剤の合成と作用機序の解明","PhotoDynamic Medicine PDM 2019",,,,,,2019,Sept. "布施新一郎","奥深いアミド化の世界へのご招待ーマイクロフロー合成法を道具としてー","第18回化学系若手研究者セミナー",,,,,,2019,Sept. "小竹佑磨,柴田裕介,林慶浩,川内進,中村浩之,布施新一郎","アシルイミダゾリウムカチオン中間体を利用するマイクロフローN?メチル化ペプチド合成法の開発とPterulamide I-IVの全合成","第61回天然有機化合物討論会",,,,,,2019,Sept. "S. Fuse,K. Masuda,Y. Otake,H. Nakamura","Peptide chain elongation using unprotected amino acids in a micro-flow reactor",,"Chem. Eur. J",,,,,2019,Aug. "布施新一郎,小竹佑磨,柴田裕介,林慶浩,川内進,中村浩之","N?メチル化ペプチドの超高効率マイクロフロー合成法の開発","第9回物質・デバイス領域共同研究拠点活動報告会 平成30年度ダイナミック・アライアンス成果報告会",,,,,,2019,July "Shinichiro Fuse","Investigation of amide bond formation based on micro-flow technologies","2nd SMARC Symposium: New Stream of Chemical Biology",,,,,,2019,July "布施新一郎","Nーメチル化ペプチドの超高効率マイクロフロー合成法の開発","2019 旭硝子財団 助成研究発表会",,,,,,2019,July "杉澤直斗,小竹佑磨,中村浩之,布施新一郎","マイクロフロー合成法による瞬間混合を駆使したβ?アミノ酸?N?カルボキシ無水物の合成とその応用","第115回有機合成シンポジウム",,,,,,2019,June "柴田裕介,林慶浩,小竹佑磨,中村浩之,布施新一郎,川内進","イミダゾール誘導体を触媒とするN-メチルアミド化反応機構の理論的解明","日本コンピューター化学会 2019年春季年会",,,,,,2019,June "Yuma Otake,Hiroyuki Nakamura,Shinichiro Fuse","Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor","11th Workshop on Organic Chemistry for Junior Chemists (WOCJC-11)",,,,,,2019,June "小竹佑磨,柴田裕介,林慶浩,川内進,中村浩之,布施新一郎","アシルイミダゾリウムカチオン中間体を利用するマイクロフローNーメチル化ペプチド合成法の開発","第77回有機合成化学協会関東支部シンポジウム",,,,,,2019,May "布施新一郎","マイクロフロー法を駆使するN?メチル化ペプチドの高効率合成","反応集積化が導く中分子戦略 高次生物機能分子の創製 第8回公開成果報告会",,,,,,2019,May "増田耕志郎,小竹佑磨,中村浩之,布施新一郎","無保護アミノ酸連結を基盤とするマイクロフローペプチド鎖伸長法の開発","第77回有機合成化学協会関東支部シンポジウム",,,,,,2019,May "Shinichiro Fuse","Innovation of Peptide Synthesisbased on Micro-Flow Technology","Let's leap! Challenges in Organic Chemistry",,,,,,2019,Apr. "布施新一郎","高速マイクロフローアミド結合形成法の開発とペプチド合成の革新","原薬の連続生産に関する研究開発と規制動向に関するシンポジウム",,,,,,2019,Apr. "布施新一郎","マイクロフローアミド化法を基盤とする高効率ペプチド合成法の開発",,"触媒技術の動向と展望2019","一般社団法人触媒学会",,,"page 124-134",2019,Apr. "Yuma Otake,Hiroyuki Nakamura,Shinichiro Fuse","An efficient synthesis of N-methylated peptides using micro-flow technology","日本化学会第99春季年会",,,,,,2019,Mar. "Shinichiro Fuse,Yuma Otake,Hiroyuki Nakamura","Development of Amide Bond Formation of N-Methyl Amino Acids Using Micro-Flow Technology","日本化学会第99春季年会",,,,,,2019,Mar. "T. Nakamura,Y. Ishikura,N. Arakawa,M. Hori,M. Sato,M. Endo,H. Masui,S. Fuse,T. Takahashi,Y. Murata,R. Murdey,A. Wakamiya","Donor?acceptor polymers containing thiazole-fused benzothiadiazole acceptor units for organic solar cells",,"RSC Advances",,,"No. 9","page 7107-7114",2019,Mar. "福原信太郎,Somaraju Yugandar,布施新一郎,中村浩之","イソキサゾロピリジン形成と窒素ー酸素結合開裂を経由するプロパルギルイソオキサゾールからの3ーヒドロキシー4ー置換ピコリノニトリルの一気合成","日本化学会第99春季年会",,,,,,2019,Mar. "増田 耕志郎,小竹 佑磨,中村 浩之,布施 新一郎","マイクロフロー法を駆使する無保護アミノ酸を用いたペプチド鎖伸長法の開発","日本化学会第99春季年会",,,,,,2019,Mar. "Taiki Morita,Shinichiro Fuse,Hiroyuki Nakamura","Photochemical conversion of isoxazoles to 5-hydroxyimidazolines and its application for protein labeling","日本化学会第99春季年会",,,,,,2019,Mar. "布施新一郎","高速混合技術を基盤とする効率的有機合成手法の開発","平成30年度一般社団法人先端膜工学研究推進機構活動報告会及び 春季講演会",,,,,,2019,Mar. "Shinichiro Fuse","Highly Efficient Amide Bond Formation using Micro-Flow Technology","Flow Chemistry Europe 2019",,,,,,2019,Feb. "布施新一郎","マイクロフロー法によるペプチド合成",,"月刊ファインケミカル",,"Vol. 48","No. 1","page 13-21",2019,Jan. "布施新一郎","マイクロフロー技術を駆使する高収率・省スペースかつ低コストの革新的ペプチド合成法の開発","日本医療研究開発機構(AMED)平成30年度 創薬基盤推進研究事業 公開シンポジウム",,,,,,2019,Jan. "N. Sugisawa,Y. Otake,H. Nakamura,S. Fuse","Single-step, rapid, and mild synthesis of β-amino acid N-carboxy anhydrides using micro-flow technologies",,"Chem. Asian J.",,,,,2019, "Shinichiro Fuse","Highly Efficient Amide Bond Formation Using Micro-flow Technology","10th Singapore International Chemistry Conference (SICC-10)",,,,,,2018,Dec. "S. Fuse,M. Takizawa,S. Sato,S. Okazaki,H. Nakamura","Elucidating the mode of action for thiophene-based organic D-π-A sensitizers for use in photodynamic therapy",,"Bioorganic & Medicinal Chemistry",,"Vol. 27","No. 2","page 315-321",2018,Dec. "布施新一郎","第III部実用編 第18章 実践光化学",,"光化学フロンティア 未来材料を生む有機光化学の基礎","化学同人",,,"page 388-399",2018,Dec. "福原 信太郎,S. Yugandar,布施 新一郎,中村 浩之","Synthesis of 3-Hydroxy-4-substituted-picolinonitriles from 4-Propargylaminoisoxazoles via Stepwise and One-pot Isoxazolopyridine Formation/N-O Bond Cleavage Sequence",,"ACS. Omega.",,"Vol. 3","No. 13","Page 16472?16476",2018,Dec. "M. Inai,N. Honda,H. Hazama,S. Akter,S. Fuse,H. Nakamura,T. Nishikawa,Y. Kaneda,K. Awazu","Photodynamic therapy with cell membrane-targeting drug delivery and direct cytotoxicity using hemagglutinating virus of Japan envelope incorporating lipidated protoporphyrin IX",,"Photodiag. Photodyn. Ther.",,"Vol. 20",,"page 238-245",2018,Nov. "Shinichiro Fuse,Yuma Otake,Hiroyuki Nakamura","Rapid and mild synthesis of amino acid N-carboxy anhydrides using basic-to-acidic flash switching in a micro-flow reactor","The 4th International Symposium on Middle Molecular Strategy (ISMMS-4)",,,,,,2018,Nov. "布施新一郎,小竹佑磨,中村浩之","マイクロフローリアクター内での瞬間pH転換に基づくNーカルボキシ無水物の高効率合成","2018年度 人・環境と物質をつなぐイノベーション創出ダイナミックアライアンス 生命機能 物質・デバイスシステムG3分科会",,,,,,2018,Nov. "伊東篤志,小川潤一,村山広大,花瀬勇貴,石垣美歌,布施新一郎,中村浩之,宮崎俊一,佐藤英俊,尾崎幸洋","近赤外分光法によるペプチド化学合成反応インラインモニタリング技術の開発","第34回近赤外フォーラム",,,,,,2018,Nov. "布施新一郎","マイクロフローアミド結合形成法を駆動力とするペプチド合成の革新","第四回魚住触媒研究会",,,,,,2018,Nov. "布施新一郎","マイクロフロー内での瞬間pH転換に基づくN?カルボキシ無水物の高効率合成","Tokyo Tech Research Festival",,,,,,2018,Nov. "布施新一郎,滝沢美織,佐藤伸一,岡崎茂俊,中村浩之","光線力学療法用有機DπA増感剤の作用機序の解明","第28回日本光線力学学会学術講演会",,,,,,2018,Nov. "大石 司,布施新一郎,Xi Zeng,中村健太郎,中村浩之","光音響イメージングを指向した新規DπAアゾ色素の合成と機能評価","第8回CSJ化学フェスタ",,,,,,2018,Oct. "Shinichiro Fuse,Yuma Otake,Hiroyuki Nakamura","Peptide Synthesis Utilizing Micro‐flow Technology",,"Chemistry - An Asian Journal",,"Vol. 13","No. 24","page 3818-3832",2018,Oct. "布施新一郎","フローマイクロリアクターによるペプチド合成","ペプチド医薬品の合成・製造技術とスケールアップ ?原薬の化学合成/マイクロ波による製造/マイクロフロー合成?",,,,,,2018,Oct. "盛田大輝,佐藤伸一,布施新一郎,中村浩之","イソオキサゾールの光分解を利用したイミダゾリンの合成とタンパク質ラベル化への応用","日本化学会第8回CSJ化学フェスタ",,,,,,2018,Oct. "布施新一郎,小竹佑磨,中村浩之","マイクロフローリアクター内での瞬間pH転換に基づくN-カルボキシ無水物の高効率合成","第35回有機合成化学セミナー",,,,,,2018,Sept. "布施新一郎","高速マイクロフローアミド結合形成法の開発とペプチド合成の革新","新学術領域「中分子戦略」「分子夾雑化学」ジョイントシンポジウム 第21回生命化学研究会",,,,,,2018,Sept. "盛田大輝,福原信太郎,布施新一郎,中村浩之","イソオキサゾールの直接修飾法の開発と新規縮環系への展開","第48回複素環化学討論会",,,,,,2018,Sept. "盛田大輝,福原信太郎,布施新一郎,中村浩之","金(I)触媒による分子内環化反応を用いた縮環イソオキサゾールの合成法開発","第65回有機金属化学討論会",,,,,,2018,Sept. "Y. Otake,H. Nakamura,S. Fuse","Rapid and mild synthesis of amino acid N-carboxy anhydrides using basic-to-acidic flash switching in a micro-flow reactor",,"Angewandte Chemie",,"Vol. 130","No. 35","page 11559-11563",2018,Aug. "布施新一郎","高速マイクロフローアミド結合形成法の開発とペプチド合成の革新","日本プロセス化学会2018サマーシンポジウム",,,,,,2018,July "S. Fuse,K. Matsumura,M. Takizawa,S. Sato,H. Nakamura","The design, synthesis, and evaluation of organic dithienopyrrole-based D-π-A dyes for use as sensitizers in photodynamic therapy",,"Bioorganic and Medicinal Chemistry Letters",,"Vol. 28","No. 18","page 3099-3104",2018,July "Atsushi Ito,Yuki Hanase,Koudai Murayama,Jun-ichi Ogawa,Shinichiro Fuse,Mika Ishigaki,Shun-ichi Miyazaki,Yukihiro Ozaki","The quantitative and non-destructive monitoring method of the amount of amide bonds in a peptide chemosynthetic model by NIR spectroscopy","International Conference on Advancing Molecular Spectroscopy",,,,,,2018,July "Y. Otake,H. Nakamura,S. Fuse","Rapid and mild synthesis of amino acid N-carboxy anhydrides using basic-to-acidic flash switching in a micro-flow reactor",,"Angewandte Chemie International Edition",,"Vol. 57","No. 35","page 11389-11393",2018,July "布施新一郎","マイクロフローリアクターを用いる高速・高効率アシル化反応","平成30年度 前期(春季)有機合成化学講習会",,,,,,2018,June "布施新一郎","マイクロフローアミド結合形成法を駆動力とするペプチド合成の革新","第15回フッ素相模セミナー",,,,,,2018,June "布施新一郎,小竹佑磨,中村浩之","マイクロフローリアクター内での瞬間pH転換に基づくN?カルボキシ無水物の高効率合成","第8回物質・デバイス領域共同研究拠点活動報告会 平成29年度 人・環境と物質をつなぐイノベーション創出 ダイナミック・アライアンス成果報告会",,,,,,2018,June "布施新一郎,小竹佑磨,中村浩之","マイクロフローリアクター内での瞬間pH転換に基づくN-カルボキシ無水物の高効率合成","新学術領域研究 反応集積化が導く中分子戦略 高次生物機能分子の創製",,,,,,2018,May "Xi Zeng,Yosuke Mizuno,Kentaro Nakamura,Shinichiro Fuse,Hiroyuki Nakamura","Compact test set for sensitivity evaluation of photoacoustic contrast agent",,"Acoustical Science and Technology",,"vol. 39","no. 3","pp. 259-262",2018,May "Yuma Otake,Hiroyuki Nakamura,Shinichiro Fuse","Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor","日本化学会第98春季年会",,,,,,2018,Mar. "K. C. S. Pradeepa,S. Fuse,H. Nakamura","AlCl3-meidated Dehydrogenative Cyclization of Diaryl-1,2-diones under Solvent-Free Conditions","International CLS Forum 2018",,,,,,2018,Mar. "盛田大輝,佐藤伸一,布施新一郎,中村浩之","イソオキサゾールの光分解反応を利用したタンパク質の新規ラベル化法の開発","日本化学会第98春季年会",,,,,,2018,Mar. "福原信太郎,盛田大輝,布施新一郎,中村浩之","カチオン性金(I)触媒を用いたイソオキサゾール5位選択的環化反応","日本化学会第98春季年会",,,,,,2018,Mar. "増井悠,Santida Decharin,布施新一郎,高橋孝志","α?ケトカルボン酸類縁体の簡便な合成法の開発とそのヘテロ環合成への応用","日本薬学会第138年会",,,,,,2018,Mar. "小竹佑磨,中村浩之,布施新一郎","マイクロフローリアクター内での瞬間pH転換に基づくN?カルボキシ無水物の高効率合成","日本化学会第98春季年会",,,,,,2018,Mar. "滝沢美織,布施新一郎,岡崎茂俊,中村浩之","光線力学療法用DπA色素の合成と作用機序解明","日本化学会第98春季年会",,,,,,2018,Mar. "大石司,布施新一郎,Xi Zeng,中村健太郎,中村浩之","光音響イメージングを志向した新規DπA色素の合成と機能評価","日本化学会第98春季年会",,,,,,2018,Mar. "植田大樹,佐藤伸一,布施新一郎,中村浩之","低酸素誘導因子(HIF-1)を標的としたα―ヘリックス模倣PPI阻害低分子の設計・合成・生物活性評価","日本化学会第98春季年会",,,,,,2018,Mar. "布施新一郎","マイクロフローアミド結合形成法を駆動力とするペプチド合成の革新","日本薬学会第138年会",,,,,,2018,Mar. "鈴木健介,布施新一郎,川村淳,佐藤伸一,中村浩之","低酸素誘導因子(HIF)阻害剤を志向した新規インデノピラゾロンの短段階合成と生物活性評価","日本化学会第98春季年会",,,,,,2018,Mar. "布施新一郎","マイクロフロー法によるペプチド合成",,"中分子創薬に資するペプチド・核酸・糖鎖の合成技術","株式会社シーエムシー出版",,,"page 49-58",2018,Feb. "Taiki Morita,Somaraju Yugandar,Shinichiro Fuse,Nakamura","Recent progresses in the synthesis of functionalized isoxazoles",,"Tetrahedron Letters",,"Vol. 59","No. 13","pp. 1159-1171",2018,Feb. "S. Fuse","Highly Efficient Amide Bond Formation using Micro-flow Technology","Tokyo Tech - KAIST Joint Workshop",,,,,,2018,Feb. "T. Morita,S. Fukuhara,S. Fuse,H. Nakamura","Gold(I)-Catalyzed Intramolecular SEAr Reaction: Efficient Synthesis of Isoxazole-Containing Fused Heterocycles",,"Organic Letters",,"Vol. 20","No. 2","page 433-436",2018,Jan. "Shinichiro Fuse,Megumi Inaba,Shinichi Sato,Manjusha Joshi,Hiroyuki Nakamura","Synthesis of Pyrazolofuropyrazine via One-Pot SNAr Reaction and Intramolecular Direct C?H Arylation",,"Synthesis",,"Vol. 50","No. 7","pp. 1493-1498",2018,Jan. "Shinichiro Fuse","Highly Efficient Amide Bond Formation Using Micro-flow Technology","The First International Conference on Automated Flow and Microreactor Synthesis (ICAMS-1)",,,,,,2018,Jan. "Yuma Otake,Hiroyuki Nakamura,Shinichiro Fuse","Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor","The First International Conference on Automated Flow and Microreactor Synthesis (ICAMS-1)",,,,,,2018,Jan. "布施新一郎","マイクロフローアミド化法を駆使するN-メチルアミノ酸の連結","反応集積化が導く中分子戦略高次生物機能分子の創製 第5回公開成果報告会",,,,,,2018,Jan. "H. Masui,M. M. Maitani,S. Fuse,A. Yamamura,Y. Ogomi,S. Hayase,T. Kaiho,H. Tanaka,Y. Wada,T. Takahashi","D?π?A dyes containing novel hydantoin anchoring groups for dye-sensitized solar cells",,"Asian Journal of Organic Chemistry",,"Vol. 7","No. 2","page 458-464",2018,Jan. "滝沢美織,布施新一郎,松村圭介,岡崎茂俊,中村浩之","光線力学療法用光増感剤の開発を志向したチオフェン含有DπA色素の合成と機能評価","第44回有機典型元素化学討論会",,,,,,2017,Dec. "布施新一郎","フローマイクロリアクターによるペプチド合成",,"ペプチド医薬品開発のためのスクリーニング・安定化・製剤化技術","技術情報協会",,,"page 162-173",2017,Dec. "布施新一郎","マイクロフローアミド結合形成法を駆動力とするペプチド合成の革新","「有機合成を基盤とした生物活性分子の創製」第1回講演会",,,,,,2017,Dec. "布施新一郎,田中浩士,高橋孝志,土井隆行","マンノペプチマイシンアグリコンの合成と立体配置訂正",,"有機合成化学協会誌",,"Vol. 75","No. 12","page 1274-1285",2017,Dec. "布施新一郎","マイクロフロー法を駆使するペプチドの高効率合成","人・環境と物質をつなぐイノベーション創出ダイナミックアライアンス 2017年度生命機能 物質・デバイス・システムプロジェクトグループ(G3)分科会",,,,,,2017,Nov. "J. Kawamura,Y. Otake,S. Fuse,H. Nakamura","Preparation of boron cluster encapsulating liposomes using microflow system","9th Young Researchers' BNCT Meeting",,,,,,2017,Nov. "布施新一郎","マイクロフロー法を駆使する天然物の高効率合成法の開発","大塚有機合成シンポジウム2017",,,,,,2017,Nov. "Shinichiro Fuse","Highly Efficienty Amide Bond Formation Using Micro-flow Technology","The 12th International Conference on Cutting-Edge Organic Chemistry in Asia / The 3rd Advanced Research Network on Cutting-Edge Organic Chemistry in Asia",,,,,,2017,Nov. "福原信太郎,盛田大輝,布施新一郎,中村浩之","カチオン性金(I)触媒を用いたイソオキサゾールの芳香族求電子置換型分子内環化反応","第7回CSJ化学フェスタ2017",,,,,,2017,Oct. "布施新一郎,御舩悠人,小竹佑磨,高橋孝志,田中浩士,中村浩之","迅速かつ強力なカルボン酸の活性化を基盤とするマイクロフローペプチド合成法の開発","第35回メディシナルケミストリーシンポジウム",,,,,,2017,Oct. "布施新一郎,御舩悠人,小竹佑磨,高橋孝志,田中浩士,中村浩之","迅速かつ強力なカルボン酸の活性化を基盤とするマイクロフローペプチド合成法の開発","第35回メディシナルケミストリーシンポジウム",,,,,,2017,Oct. "布施新一郎","マイクロフローアミド化法を駆使するペプチドの高効率合成","化学とマイクロ・ナノシステム学会第36回研究会",,,,,,2017,Oct. "S. Fuse,M. Takizawa,K. Matsumura,S. Sato,S. Okazaki,H. Nakamura","Thiophene-based, Organic D-π-A dyes as Potent Sensitizers for Photodynamic Therapy",,,,,"No. 34","page 5170-5177",2017,Sept. "布施新一郎","超高速マイクロフローアミド化反応の開発とペプチド合成の革新","千葉大学大学院薬学研究院第11回化学系若手研究者講演会",,,,,,2017,Sept. "布施新一郎","ペプチドの低コスト生産を志向したマイクロフローアミド結合形成法の開発","第5回バイオ関連化学シンポジウム若手フォーラム",,,,,,2017,Sept. "布施新一郎","チオフェン含有有機Donor-p-Acceptor色素の系統的合成と構造?機能相関解明",,"有機合成化学協会誌",,"Vol. 75","No. 9","page 941-954",2017,Sept. "福原信太郎,盛田大輝,布施新一郎,中村浩之","カチオン性金(I)触媒を用いた4-(プロパルギルアミノ)イソオキサゾールの5位選択的環化反応の開発","第64回有機金属化学討論会",,,,,,2017,Sept. "布施新一郎,御舩悠人,高橋孝志,田中浩士,中村浩之","マイクロフローアミド結合形成法を駆使するフェグリマイシンの全合成","第59回天然有機化合物討論会",,,,,,2017,Sept. "布施新一郎","迅速かつ強力なカルボン酸の活性化を基盤とするマイクロフローペプチド合成法の開発","第34回有機合成化学セミナー",,,,,,2017,Sept. "布施新一郎","微小流路中での高速アミド化反応(秒単位)を駆使するペプチド合成","第49回若手ペプチド夏の勉強会",,,,,,2017,Aug. "Shinichiro Fuse,Yuma Otake,Hiroyuki Nakamura","Integrated Micro-Flow Synthesis Based on Photochemical Wolff Rearrangement",,"European Journal of Organic Chemistry","Wiley","Volume 2017"," Issue 44","pp. 6466-6473",2017,Aug. "布施新一郎","マイクロフロー法を駆使する最強のアミド化法開発を目指して","新学術領域研究「反応集積化が導く中分子戦略:高次生物機能分子の創製」 若手シンポジウム",,,,,,2017,Aug. "布施新一郎,松村圭介,滝沢美織,岡崎茂俊,中村浩之","ジチエノピロール含有DπA色素の迅速合成と機能評価","第27回日本光線力学学会学術講演会",,,,,,2017,July "布施新一郎","マイクロフローアミド化法を駆使するN?メチルアミノ酸の連結","新学術領域研究 反応集積化が導く中分子戦略高次生物機能分子の創製",,,,,,2017,July "布施新一郎","マイクロフローアミド化法を駆使するN?メチルアミノ酸の連結","新学術領域研究 反応集積化が導く中分子戦略高次生物機能分子の創製第4回成果報告会",,,,,,2017,July "洪瑛淳,稲井瑞穂,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","複製能欠損ウイルス粒子とプロトポルフィリンIX脂質を用いたPDTにおける腫瘍選択性向上のための治療条件の検討","第27回日本光線力学学会学術講演会",,,,,,2017,July "滝沢美織,松村圭介,布施新一郎,岡崎茂俊,中村浩之","光線力学療法用有機DπA色素の作用機序解明","第27回日本光線力学学会学術講演会",,,,,,2017,July "布施新一郎","マイクロフロー法を駆使するペプチドの高効率合成","平成28年度附置研アライアンス成果報告会",,,,,,2017,June "布施新一郎","マイクロフロー合成を駆使するアミド化法の開発とペプチド合成の革新","第49回触媒化学融合研究センター講演会",,,,,,2017,June "小竹佑磨,中村浩之,布施新一郎","マイクロフロー法を駆使するN-メチル化ペプチドの効率的合成","第111回有機合成シンポジウム",,,,,,2017,June "Shinichiro Fuse","Highly Efficient Amide Bond Formation Using Micro‐flow Technology","The International Symposium on Pure & Applied Chemistry (ISPAC) 2017",,,,,,2017,June "盛田大輝,布施新一郎,中村浩之","イソオキサゾリルアニオンを利用するイソオキサゾール合成法の開発","第73回有機合成化学協会関東支部シンポジウム",,,,,,2017,May "S. Fuse,T. Morita,H. Nakamura","Step-by-Step Multifunctionalization of Isoxazoles based on SEAr Reactions and C-H Direct Arylations.",,"Synthesis",,"Vol. 49","No. 11","page 2351-2360",2017,Apr. "石井 秀一,布施 新一郎,佐藤 伸一,中野 洋文,中村 浩之","多環性オルトキノン化合物の短段階合成法を指向したPd触媒による脱水素型環化反応の開発","日本化学会第97回年会",,,,,,2017,Mar. "布施 新一郎","マイクロフローペプチド合成法の開発 ?奥深いアミド化の世界?","東工大応用化学系 次世代を担う若手シンポジウム",,,,,,2017,Mar. "Shinichiro Fuse","An efficient amide bond formation through rapid and strong activation of carboxylic acids in a micro-flow reactor","7th CCS-CSJ Young Chemists Forum 2017 ?Frontier in Organic Synthesis toward Middle Molecular Strategy-",,,,,,2017,Mar. "布施 新一郎,御舩 悠人,中村 浩之","マイクロフローアミド化・光環化反応を駆使する高効率環状ペプチドの合成法の開発","日本化学会第97回年会",,,,,,2017,Mar. "小竹 佑磨,中村 浩之,布施 新一郎","マイクロフロー法を駆使するN?メチル化ペプチドの革新的合成","日本化学会第97回年会",,,,,,2017,Mar. "Keisuke Matsumura,Miori Takizawa,Shinichiro Fuse,Hiroyuki Nakamura","Synthesis and Evaluation of Organic DπA Dye Containing Dithienopyrrole as the Photosensitizer for Photodynamic Therapy","日本化学会第97回年会",,,,,,2017,Mar. "滝沢 美織,松村 圭介,布施 新一郎,中村 浩之","光線力学療法のための有機DπA型色素の作用機序解明","日本化学会第97回年会",,,,,,2017,Mar. "福原 信太郎,盛田 大輝,布施 新一郎,中村 浩之","カチオン性金(I)触媒を用いた4-(プロパルギルアミノ)イソオキサゾールの分子内ヒドロアリール化反応の開発","日本化学会第97回年会",,,,,,2017,Mar. "Taiki Morita,Shinichiro Fuse,Hiroyuki Nakamura","Generation of 4-Isoxazolyl Anion Species and Its Application for Synthesis of Multifunctionalized Isoxazoles","日本化学会第97回年会",,,,,,2017,Mar. "鈴木 健介,布施 新一郎,佐藤 伸一,中村 浩之","創薬を指向した新規インデノピラゾロンの短段階合成法の開発と生物活性評価","日本化学会第97回年会",,,,,,2017,Mar. "稲葉 恵,峯岸 秀充,布施 新一郎,佐藤 伸一,中村 浩之","HIF阻害剤の創出を指向したベンゾフロピラゾールおよびピラゾロフロピラジンの合成法開発と生物活性評価","日本化学会第97回年会",,,,,,2017,Mar. "布施 新一郎","マイクロフローアミド結合形成法を駆使するフェグリマイシンの全合成","反応集積化が導く中分子戦略高次生物機能分子の創製 第3回公開成果報告会",,,,,,2017,Jan. "H. Masui,S. Yosugi,S. Fuse,T. Takahashi","Solution-phase automated synthesis of α-amino aldehyde as a versatile intermediate.",,"Beilstein Journal of Organic Chemistry",,"Vol. 13",,"page 106-110",2017,Jan. "古山祐,稲井瑞穂,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","複製能欠損ウイルス粒子をキャリアとした新規光感受性物質による光線力学治療の作用機序の検討","レーザー学会学術講演会第37回年次大会",,,,,,2017,Jan. "石井秀一,布施新一郎,佐藤伸一,中野洋文,中村浩之","天然物タンシノンIIAを基盤とした新規HIF-1α阻害剤の開発","第5回「次世代がん治療推進専門家養成プランシンポジウム」",,,,,,2016,Dec. "布施新一郎","マイクロフローアミド結合形成法の開発?単純なようで奥深いアミド化の世界?","第11回プロセス化学ラウンジ",,,,,,2016,Dec. "S. Fuse,T. Ohuchi,Y. Asawa,S. Sato,H. Nakamura","Development of 1-Aryl-3-furanyl/Thienyl-imidazopyridine Templates for Inhibitors against Hypoxia Inducible Factor (HIF)-1 Transcriptional Activity",,"Bioorganic and Medicinal Chemistry Letters",,"Vol. 26","No. 24","page 5887-5890",2016,Nov. "S. Fuse,Y. Mifune,H. Nakamura,H. Tanaka","Total Synthesis of Feglymycin based on a Linear/Convergent Hybrid Approach using Micro-flow Amide Bond Formation","The 10th International Symposium on Integrated Synthesis (ISONIS-10)",,,,,,2016,Nov. "小竹佑磨,中村浩之,布施新一郎","マイクロフロー合成法を駆使するN-メチル化ペプチドの合成法開発","第6回CSJ化学フェスタ2016",,,,,,2016,Nov. "布施新一郎","わずか5秒以内でアミノ酸を連結する超高速マイクロフローペプチド合成法の開発","第6回CSJ化学フェスタ2016",,,,,,2016,Nov. "石井秀一,布施新一郎,佐藤伸一,中野洋文,中村浩之","天然物タンシノンIIAを基盤とした新規HIF-1α阻害剤の開発研究","第14回がんとハイポキシア研究会",,,,,,2016,Nov. "S. Fuse,K. Matsumura,K. Johmoto,H. Uekusa,H. Tanaka,T. Hirose,T. Sunazuka,S. ?mura,T. Takahashi","The Design, Synthesis, and Evaluation of 1,5,7-Trisubstituted-3-pyridyl-xanthones for Use as Insecticides Starting from Pyripyropene A",,"Chemistry A European Journal",,"Vol. 22","No. 51","page 18450-18455",2016,Nov. "石井秀一,布施新一郎,中村浩之","多環性オルトキノン化合物の短段階合成を志向したPd触媒による脱水素型環化反応の開発","第6回CSJ化学フェスタ2016",,,,,,2016,Nov. "Y. Mifune,H. Nakamura,S. Fuse","A Rapid and Clean Synthetic Approach to Cyclic Peptides via Micro-flow Peptide Chain Elongation and Photochemical Cyclization: Synthesis of a Cyclic RGD Peptide",,"Organic & Biomolecular Chemistry",,"Vol. 14","No. 47","page 11244-11249",2016,Nov. "Shinichiro Fuse,Yuto Mifune,Hiroyuki Nakamura,Hiroshi Tanaka","Total synthesis of feglymycin based on a linear/convergent hybrid approach using micro-flow amide bond formation",,"Nature Communications",,,"No. 13491",,2016,Nov. "布施新一郎","強力かつ迅速なカルボン酸の活性化を基盤とするマイクロフローペプチド合成法の開発","2016年度第7回マイクロ化学プロセス分科会主催講演会",,,,,,2016,Nov. "稲井瑞穂,古山祐,洪暎淳,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","複製能欠損ウイルス粒子を用いた光感受性薬剤の細胞内局在と腫瘍選択性の検討","第37回日本レーザー医学会総会",,,,,,2016,Oct. "松村圭介,布施新一郎,池邊彩子,大角和也,柄澤智哉,田中浩士,廣瀬友靖,砂塚敏明,大村智,高橋孝志","ent-ピリピロペンAおよび構造簡略化ピリピロペン類縁体の合成と殺虫活性評価","第58回天然有機化合物討論会",,,,,,2016,Sept. "T. Morita,S. Fuse,H. Nakamura","Generation of 4-Isoxazolyl Anion Species: Facile Access to 4-Substituted Isoxazoles",,"Angewandte Chemie International Edition",,"Vol. 55","No. 43","page 13580-13584",2016,Sept. "T. Morita,S. Fuse,H. Nakamura","Generation of 4-Isoxazolyl Anion Species: Facile Access to 4-Substituted Isoxazoles",,"Angewandte Chemie International Edition",,"Vol. 55","No. 43","page 13580-13584",2016,Sept. "洪暎淳,稲井瑞穂,古山祐,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","抗がん剤耐性前立腺がん細胞への迅速な薬剤輸送に向けた複製能欠損ウイルス粒子への光感受性物質の封入",,"電気学会 光・量子デバイス研究会",,,,,2016,Sept. "盛田大輝,布施新一郎,中村浩之","4?イソオキサゾリルアニオンを利用したイソオキサゾール4位の官能基化","第63回有機金属化学討論会",,,,,,2016,Sept. "布施新一郎","フロー反応でしか実現できない高効率合成法開発を目指して","電磁波励起反応場第188委員会 平成28年度 第1回化学材料分科会",,,,,,2016,Sept. "Shinichiro Fuse","Elucidating the structure-property relationship of donor-π-acceptor dyes for DSSCs through rapid library synthesis","AEARU 6th Energy and Environmental Workshop",,,,,,2016,Aug. "H. Hamagami,M. Kumazoe,Y. Yamaguchi,S. Fuse,H. Tachibana,H. Tanaka","6-Azido-6-deoxy-L-idose as a hetero-bifunctional spacer for the synthesis of azido-containing chemical probes",,"Chemistry a European Journal",,"Vol. 22","No. 36","page 12884-12890",2016,Aug. "N. Shiraishi,Motofumi Kumazoe,S. Fuse,Hirofumi Tachibana,H. Tanaka","The Synthesis of trans-Flavan-3-ol Gallates by Regioselective Oxidative Etherification and Their Biological Evaluation",,"Chemistry a European Journal",,"Vol. 22","No. 37","page 13050-13053",2016,Aug. "Taiki Morita,Shinichiro Fuse,Hiroyuki Nakamura","Preparation of 4-isoxazolyl Grignard reagent and its application for divergent synthesis of 4-substituted isoxazoles","27th International Conference on Organometallic Chemistry (ICOMC 2016)",,,,,,2016,July "滝沢美織,布施新一郎,中村浩之","有機D-π-A色素の構造?PDT活性相関の解明","第26回日本光線力学学会学術講演会",,,,,,2016,June "布施新一郎,滝沢美織,中村浩之","新規PDT用有機色素の開発を志向したD?π?A色素の迅速合成と機能評価","第26回日本光線力学学会学術講演会",,,,,,2016,June "洪暎淳,稲井瑞穂,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","迅速な薬剤輸送に向けた複製能欠損センダイウイルス粒子への光感受性物質の封入条件の検討","第26回日本光線力学学会学術講演会",,,,,,2016,June "古山祐,稲井瑞穂,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","複製能欠損ウィルス粒子とプロトポルフィリンIV脂質を利用したPDT過程のタイムラプス撮影による作用機序の検討","第26回日本光線力学学会学術講演会",,,,,,2016,June "布施新一郎,滝沢美織,中村浩之","新規PDT用有機色素の開発を志向したD-π-A色素の迅速合成と機能評価","第26回日本光線力学学会学術講演会",,,,,,2016,June "布施新一郎,〇杉山寛崇,小林大輔,田中浩士","ワンポット[3+2]環化付加反応を基盤とした三置換ピラゾールの位置選択的合成法の開発","第109回有機合成シンポジウム",,,,,,2016,June "稲葉恵,峯岸秀充,佐藤伸一,布施新一郎,中村浩之","ベンゾフロピラゾール類縁体の設計、合成およびHIF-1阻害能評価","第109回有機合成シンポジウム",,,,,,2016,June "Ryota Suzuki,Shinichiro Fuse,Hiroshi Tanaka","Synthesis of Asymmetrically Terminal Bifunctionlized Alkanes by Sequential Suzuki-Miyaura Coupling using B-Thexyl Boracyclanes",,"Eur J Org Chem",,"Vol. 21",,"pp. 3471-3481",2016,May "松村圭介,吉崎聡一,米谷真人,和田雄二,尾込裕平,早瀬修二,海宝龍夫,布施新一郎,田中浩士,中村浩之,高橋孝志","化学選択的ワンポット連結反応を駆使した色素増感太陽電池用DπA色素の効率的合成法の開発とその機能評価","第71回有機合成化学協会関東支部シンポジウム",,,,,,2016,May "御舩悠人,田中浩士,中村浩之,布施新一郎","マイクロフローアミド結合形成法を基盤とするフェグリマイシンの全合成","日本化学会第96春季年会",,,,,,2016,Mar. "布施新一郎,池邊彩子,大角和也,柄澤智哉,松村圭介,泉川美穂,上本紘平,植草秀裕,新家一男,土井隆行,高橋孝志","塩化チタノセン触媒によるタンデムラジカル環化反応を駆使するピリピロペンAの不斉全合成","日本化学会第96春季年会",,,,,,2016,Mar. "唐崎貴史,佐瀬祥平,布施新一郎,田中浩士,後藤敬","「クレードルドセレノシステイン」を活用した抗酸化酵素反応過程のモデル研究","日本化学会第96春季年会",,,,,,2016,Mar. "稲葉 恵,峯岸 秀充,布施 新一郎,中村 浩之","ベンゾフロピラゾール骨格をもつ 新規HIF-1阻害剤の開発研究","日本薬学会 第136年会",,,,,,2016,Mar. "Taku Aoyagi,Shuichi Ohira,Shinichiro Fuse,Jun Uzawa,Yoshiki Yamaguchi,Hiroshi Tanaka","The α-Glycosidation of partially Unprotected N-Acetyl and N-Glycolyl Sialyl Donors in the Absence of a Nitrile Solvent Effect.",,"Chem. Eur. J.",,"Vol. 22",,"pp. 6968-6973",2016,Mar. "中村浩之,佐藤伸一,立川将士,布施新一郎,間久直,粟津邦男,金田安史","光感受性ポルフィリン脂質の開発とナノ粒子化による光線力学的治療効果","第4回次世代がん治療推進専門家養成プランシンポジウム",,,,,,2016,Jan. "Shunsuke Irie,Shinichiro Fuse,Masato M. Maitani,Yuji Wada,Yuhei Ogomi,Shuzi Hayase,Tatsuo Kaiho,Hisashi Masui,Hiroshi Tanaka,Takashi Takahashi","Synthesis of D-A’-π-A Dyes via One-Pot Three-Component Suzuki-Miyaura Coupling and an Evaluation of the Photovoltaic Properties for Use in DSSCs",,"Chemistry a European Journal",,"Vol. 22","No. 7","page 2185-2538",2016,Jan. "Irie, S.,Shinichiro Fuse,Maitani, M.M.,Yuji Wada,Ogomi, Y.,Hayase, S.,Kaiho, T.,Masui, H.,Tanaka, H.,Takahashi, T.","Rapid Synthesis of D-A'-π-A Dyes through a One-Pot Three-Component Suzuki-Miyaura Coupling and an Evaluation of their Photovoltaic Properties for Use in Dye-Sensitized Solar Cells",,"Chemistry - A European Journal",,"Vol. 22","No. 7","pp. 2507-2514",2016, "Hiroki Hamagami,Yukinori Hatasa,Yoshiki Yamaguchi,Shinichiro Fuse,Takahiro Shibata,Hirofumi Tachibana,Koji Uchida,Hiroshi Tanaka","Synthesis of Sugar-Modified EGCGs by Direct C-Glycosylation and Its Application to a Chemical Biology","The International Chemical Congress of Pacific Basin Societies 2015 (Pacifichem 2015)",,,,,,2015,Dec. "Shinichiro Fuse,Ryota Takahashi,Masato M. Maitani,Yuji Wada,Tatsuo Kaiho,Hiroshi Tanaka,Takashi Takahashi","Synthesis and Evaluation of Thiophene-based Organic Dyes Containing a Rigid and Non-Planar Donor with Secondary Electron Donors for Use in Dye-Sensitized Solar Cells",,"European Journal of Organic Chemistry",,,"No. 3","page 508-517",2015,Dec. "Nana Shiraishi,Motofumi Kumazoe,Shinichiro Fuse,Hirofumi Tachibana,Hiroshi Tanaka","Synthesis of Optically Active 3-O-Acylated Catechin Analogs by Oxidative Cyclization","The International Chemical Congress of Pacific Basin Societies 2015 (Pacifichem 2015)",,,,,,2015,Dec. "Taku Aoyagi,Syuichi Ohira,Shinichiro Fuse,Hiroshi Tanaka","Partially Unprotected N-Acetyl Sialyl Donors Undergoing α-Sialylation without the Nitrile Effect","The International Chemical Congress of Pacific Basin Societies 2015 (Pacifichem 2015)",,,,,,2015,Dec. "Taiki Morita,Shinichiro Fuse,Keisuke Matsumura,Hirotaka Sugiyama,Daisuke Kobayashi,Hiroshi Tanaka,Hiroyuki Nakamura,Takashi Takahashi","Rapid synthesis of tri/tetraaryl-substituted pyrazoles via [3+2] cycloadditon and C-H direct arylation approaches","The International Chemical Congress of Pacific Basin Societies 2015 (Pacifichem 2015)",,,,,,2015,Dec. "Ryota Suzuki,Kou Sato,Shinichiro Fuse,Hiroshi Tanaka","One-pot Sequential Palladium-Catalyzed Cross-Coupling Reaction of Cyclic Boron Compounds","The International Chemical Congress of Pacific Basin Societies 2015 (Pacifichem 2015)",,,,,,2015,Dec. "布施新一郎","生物活性天然物のマイクロフロー合成:「マイクロフロー法ならでは」の手法論開発を目指して","マイクロ化学生産研究コンソーシアム講演会および成果報告会",,,,,,2015,Dec. "Shinichiro Fuse,Yuto Mifune,Nobutake Tanabe,Hiroyuki Nakamura,Takashi Takahashi","Utilization of microflow technology for the site-selective modification of multifunctionalized molecules","The International Chemical Congress of Pacific Basin Societies 2015 (Pacifichem 2015)",,,,,,2015,Dec. "布施新一郎,小竹佑磨,御舩悠人,中村浩之,田中浩士","マイクロフローリアクター内での四連続反応によるαアリールカルボニル化合物合成法の開発","第70回記念有機合成化学協会関東支部シンポジウム?新潟(長岡)シンポジウム?",,,,,,2015,Nov. "盛田大輝,田中浩士,中村浩之,布施新一郎","4連続の直接アリール化による4置換ピラゾールの合成とその発光特性","第108回有機合成シンポジウム",,,,,,2015,Nov. "Shinichiro Fuse,T. Morita,Johmoto Kohei,H. Uekusa,H. Tanaka","Directing/Protecting-Group-Free Synthesis of Tetraaryl-Substituted Pyrazoles through Four Direct Arylations on an Unsubstituted Pyrazole Scaffold",,"Chem.-Eur. J.",,"Vol. 21","No. 41","pp. 14370-14375",2015,Oct. "Shinichiro Fuse","An efficient amide bond formation through the rapid and strong activation of carboxylic acids in a micro-flow reactor","International Conference on Nascent Developments in Chemical Sciences 2015 (NDCS-2015): Opportunities for Academia-Industry Collaboration",,,,,,2015,Oct. "盛田大輝,田中浩士,中村浩之,布施新一郎","連続的C?H結合直接アリール化による4置換ピラゾールの合成","第62回有機金属化学討論会",,,,,,2015,Sept. "御舩悠人,布施新一郎,田中浩士,中村浩之,高橋孝志","カルボン酸の迅速かつ強力な活性化を基盤とするマイクロフローペプチド合成法の開発とフェグリマイシンの合成研究","第32回有機合成化学セミナー",,,,,,2015,Sept. "増井悠,布施新一郎,高橋孝志","ワンポット多成分連結反応を基盤とした機能性分子のコンビナトリアル合成",,"Organometallic News",,,"No. 3","page 100-104",2015,Aug. "布施新一郎","サイト選択的マイクロフロー反応を駆使する天然物合成",,"化学と工業",,"Vol. 68","No. 8","page 733-734",2015,Aug. "Shinichiro Fuse,Taiki Morita,Kohei Johmoto,Hidehiro Uekusa,Hiroshi Tanaka","Directing/Protecting-Group-Free Synthesis of Tetraaryl-Substituted Pyrazoles through Four Direct Arylations on an Unsubstituted Pyrazole Scaffold",,"Chemistry A Europian Journal",,"Vol. 21","No. 41","page 14370-14375",2015,Aug. "Shinichiro Fuse,Yuma Otake,Yuto Mifune,Hiroshi Tanaka","A Facile Preparation of a-Aryl Carboxylic Acid via One-Flow Arndt?Eistert Synthesis",,"Australian Journal of Chemistry",,"Vol. 68","No. 11","page 1657-1661",2015,Aug. "T. Morita,D. Kobayashi,K. Matsumura,Johmoto Kohei,H. Uekusa,Shinichiro Fuse,T. Takahashi","Sequential SNAr Reaction/Suzuki-Miyaura Coupling/C-H Direct Arylations Approach for the Rapid Synthesis of Tetraaryl-Substituted Pyrazoles",,"Chem.-Asian J.",,"Vol. 10","No. 8","pp. 1626-1630",2015,Aug. "Taiki Morita,Daisuke Kobayashi,keisuke Matumura,Kohei Johmoto,Hidehiro Uekusa,Shinichiro Fuse,Takashi Takahashi","Sequential SNAr Reaction/Suzuki?Miyaura Coupling/C−H Direct Arylations Approach for the Rapid Synthesis of Tetraaryl-Substituted Pyrazoles",,"Chemistry an Asian Journal",,"Vol. 10","No. 8","page 1626-1630",2015,June "Hisashi Masui,Natsumi Ishizawa,Shinichiro Fuse,Takashi Takahashi","Palladium-catalyzed double carbonylation-based diversity-oriented synthesis of 3,4-dihydroisoquinoline-1-carboxamides",,"Tetrahedron",,"Vol. 71","No. 37","page 6354-6360",2015,June "布施新一郎","サイト選択的反応を駆使する多官能基性生物活性分子の合成","平成27年度 環境調和材料・デバイスプロジェクトグループ(G4)分科会",,,,,,2015,June "Shinichiro Fuse,Hirotaka Sugiyama,Daisuke Kobayashi,Yusuke Iijima,Keisuke Matsumura,Hiroshi Tanaka,Takashi Takahashi","Regioselective, One-Pot, Three-Component Synthesis of 1,3,4- and 1,3,5-Triarylpyrazoles from 1- and 2-Aryl-1-alkenyl Sulfones",,"European Journal of Organic Chemistry",,,"No. 21","page 4756?4764",2015,June "Shinichiro Fuse,A. Ikebe,K. Oosumi,T. Karasawa,K. Matsumura,M. Izumikawa,Johmoto Kohei,H. Uekusa,K. Shin-Ya,T. Doi,T. Takahashi","Asymmetric Total Synthesis of ent-PyripyropeneA",,"Chem.-Eur. J.",,"Vol. 21","No. 26","pp. 9454-9460",2015,June "Keisuke Matsumura,Soichi Yoshizaki,Masato. M. Maitani,Yuji Wada,Yuhei Ogomi,Shuzi Hayase,Tatsuo Kaiho,Shinichiro Fuse,Hiroshi Tanaka,Takashi Takahashi","Rapid Synthesis of Thiophene-Based, Organic Dyes for DSSCs via a One-Pot, Four-Component Coupling Approach",,"Chemistry A Europian Journal",,"Vol. 21","No. 27","page 9742-9747",2015,May "Shinichiro Fuse,Ayako Ikebe,Kazuya Oosumi,Tomoya Karasawa,Keisuke Matsumura,Miho Izumikawa,Kohei Johmoto,Hidehiro Uekusa,Kazuo Shin-ya,Takayuki Doi,Takashi Takahashi","Asymmetric Total Synthesis of ent-Pyripyropene A",,"Chemistry A Europian Journal",,"Vol. 21","No. 26","page 9454-9460",2015,May "Shinichiro Fuse,Ryota Takahashi,Takashi Takahashi","Facile, One-Step Synthesis of 5-Substituted Thieno[3,4-c]pyrrole-4,6-dione by Palladium-Catalyzed Carbonylative Amidation",,"European Journal of Organic Chemistry",,"Vol. 2015","No. 16","page 3430-3434",2015,Apr. "青?拓,大平脩一,布施新一 郎,田中浩士","遊離水酸基を有するN-アセチルシアル酸供与体を用いたα選択的シアリル化反応","日本化学会第95春季年会",,,,,,2015,Mar. "布施新一郎","マイクロフロー合成法を駆使する高 選択的反応を基軸とした天然物合成","日本化学会第95春季年会",,,,,,2015,Mar. "増井悠,布施新一郎,米谷真 人,和田雄二,尾込裕平,早瀬修二,高橋孝志","新規アンカー基含有色素の合成とその機能評価","日本化学会第95春季年会",,,,,,2015,Mar. "御舩悠人,布施新一郎,田中浩 士","マイクロフロー合成法を駆使したペプチド系天然物フェグリマイシンの合成研究","日本化学会第95春季年会",,,,,,2015,Mar. "布施新一郎","マイクロフローリアクター内での四連続反応によるαアリールカルボニル化合物合成法の開発","日本化学会第95春季年会",,,,,,2015,Mar. "布施新一郎,盛田大輝,田 中浩士","4 連続のN-H およびC-H 結合直接アリール化を駆使した4置換ピラゾールの合成研究","日本化学会第95春季年会",,,,,,2015,Mar. "布施新一郎,吉崎聡一,田中浩士","C-H結合直接アリール化を駆使するD-π-A色素合成法の開発","日本化学会第95春季年会",,,,,,2015,Mar. "入江俊介,布施新一郎,米谷真人,和田雄二,尾込裕平,早瀬修 二,海宝龍夫,増井悠,田中浩士,高橋孝志","DA’πA型近赤外光吸収色素の設計・合成およびその機能評価","日本化学会第95春季年会",,,,,,2015,Mar. "松村圭介,布施新一郎,藤田有紀,杉本八郎,高橋孝志","4成分ワンポット連結反応を駆使した機能性色素の合成とアミ ロイドβおよびタウタンパクの凝集阻害活性評価","日本化学会第95春季年会",,,,,,2015,Mar. "布施新一郎,杉山寛崇,小林大輔,田中浩士","ワンポット[3+2]環化付加反応を基盤とした三置換ピラゾールの位置選択的合成法の開発","日本化学会第95春季年会",,,,,,2015,Mar. "白石奈々,布施新一郎,田中浩士","酸化的環化反応を用いた光学活性3-O-アシル化カテキン類縁体の合成研究","日本化学会第95春季年会",,,,,,2015,Mar. "布施新一郎,高橋 孝志","マイクロフロー光反応?イミドイル化反応?アシル化反応を駆使する効率的な有機合成",,"有機合成化学協会誌","The Society of Synthetic Organic Chemistry, Japan","Vol. 73","No. 5","pp. 442-451",2015, "Shinichiro Fuse","Utilization of micro-flow technology for the site-selective modification of multi-functionalized molecules","8th Singapore International Chemistry Conference 2014",,,,,,2014,Dec. "Hirotsugu Koinuma,Shinichiro Fuse,Atsushi Kimbara,Miho Izumikawa,Yuto Mifune,Haiyin He,Kazuo Shin-ya,Takashi Takahashi,Takayuki Doi","Total synthesis and stereochemistry revision of mannopeptimycin aglycone","8th Singapore International Chemistry Conference 2014",,,,,,2014,Dec. "布施新一郎,入江俊介,杉山 栄,米谷真人,和田雄二,尾込裕平,早瀬修二,海宝龍夫,高橋孝志","ワンポットパラジウムカップリング反応によるD-π-A色素ライブラリーの迅速合成と構造-機能相関解明","第四回CSJ化学フェスタ2014",,,,,,2014,Oct. "Shinichiro Fuse,Kentarou Nakamura,Yuto Mifune,Hironori Marubayashi,Ichiro Hijikuro,Shuichi Nojima,Hiroshi Tanaka,Takashi Takahashi","Rapid library synthesis of amphiphiles based on a dioxinone scaffold and identification of nonlamellar liquid crystals",,"SYNLETT",,"Vol. 25","No. 19","page 2806-2813",2014,Oct. "鈴木涼太,布施新一郎,田中浩士","環状ホウ素化合物の合成とその連続的クロスカップリング反応への応用","第106回有機合成シンポジウム",,,,,,2014,Oct. "鈴木涼太,布施新一郎,田中浩士","環状ホウ素化合物の合成とその連続的クロスカップリング反応への応用","第106回有機合成シンポジウム",,,,,,2014,Oct. "布施新一郎,盛田大輝,田中浩士","C-H結合直接アリール化を駆使した4置換ピラゾールの合成研究","第四回CSJ化学フェスタ2014",,,,,,2014,Oct. "Shinichiro Fuse,Yuya Asai,Sakae Sugiyama,Keisuke Matsumura,Masato M. Maitani,Yuji Wada,Yuhei Ogomi,Shuzi Hayase,Tatsuo Kaiho,Takashi Takahashi","Synthesis of EDOT-containing organic dyes via one-pot, four component Suzuki Miyaura coupling and the evaluation of their photovoltaic properties",,"Tetrahedron",,"Vol. 70","No. 45","page 8690-8695",2014,Sept. "濱上大基,布施新一郎,田中浩士","C - グリコシルポリフェノール類の合成を指向した水中 C - グリコシル化反応の開発研究","第 33 回 日本糖質学会年会",,,,,,2014,Aug. "布施新一郎","フローでおこなうペプチドの超高速合成","新学術領域研究「反応集積化の合成化学 革新的手法の開拓と有機物質創成への展開」研究成果とりまとめシンポジウム",,,,,,2014,Aug. "青柳拓,大平脩一,布施新一郎,田中浩士","4 位遊離水酸基を有する N - アセチルシアル酸供与体を用いる α 選択的シアリル化反応","第 33 回 日本糖質学会年会",,,,,,2014,Aug. "Shinichiro Fuse,Keisuke Matsumura,Atsushi Wakamiya,Hisashi Masui,Hiroshi Tanaka,Susumu Yoshikawa,Takashi Takahashi","Elucidation of the structure-property relationship of p-type organic semiconductors through rapid library construction via a one-pot, Suzuki-Miyaura coupling reaction",,"ACS Combinatorial Science",,"Vol. 16","No. 9","page 494-499",2014,Aug. "布施新一郎,高橋孝志","フロー・マイクロ合成 基礎から実際の合成・製造まで",,,"化学同人",,,"page 203-215",2014,July "Shinichiro Fuse,Hirotsugu Koinuma,Atsushi Kimbara,Miho Izumikawa,Yuto Mifune,Haiyin He,Kazuo Shin-ya,Takashi Takahashi,Takayuki Doi","Total synthesis and stereochemistry revision of mannopeptimycin aglycone",,"Journal of the American Chemical Society",,"Vol. 136","No. 34","page 12011-12017",2014,July "布施新一郎,高橋孝志","マイクロフローリアクターを駆使したペプチドの迅速合成",,"現代化学","東京化学同人",,"No. 520","page 24-28",2014,July "Shinichiro Fuse,keisuke Matumura,Yuki Fujita,Hachiro Sugimoto,Takashi Takahashi","Development of dual targeting inhibitors against aggregations of amyloid-β and tau protein",,"European Journal of Medicinal Chemistry",,"Vol. 85",,"page 228-234",2014,July "Yuto Mifune,Shinichiro Fuse,Hiroshi Tanaka","Synthesis of N-allyloxycarbonyl 3,5-dihydroxyphenylglycine via photochemical Wolff rearrangement/nucleophilic addition sequence in a micro-flow reactor",,"Journal of Flow Chemistry",,"Vol. 4","No. 4","page 172-178",2014,July "Shinichiro Fuse,Sakae Sugiyama,Masato M. Maitani,Yuji Wada,Yuhei Ogomi,Shuzi Hayase,Ryuzi Katoh,Tatsuo Kaiho,Takashi Takahashi","Elucidating the structure-property relationship of donor-pi-acceptor dyes for DSSCs through rapid library synthesis via a one-pot procedure",,"Chemistry A European Journal",,"Vol. 20","No. 34","page 10685-10694",2014,June "Shinichiro Fuse,Yuto Mifune,Nobutake Tanabe,Takashi Takahashi","Micro-flow Technology: Another Solution for the Site-Selective Modification of Multi-functionalized Molecules",,"Synlett",,"Vol. 25","No. 15","page 2087-2092",2014,June "Shinichiro Fuse,Hayato Yoshida,Kazuya Oosumi,Takashi Takahashi","Rapid and structurally diverse synthesis of multi-substituted β-keto amide derivatives based on a dioxinone scaffold",,"European Journal of Organic Chemistry",,"Vol. 2014","No. 22","page 4854-4860",2014,June "松村圭介,布施新一郎,増井悠,若宮淳志,吉川暹,高橋孝志,田中浩士","有機薄膜太陽電池用p 型有機半導体を指向したオリゴヘテロ芳香環化合物の効率的合成法の開発とその機能評価","第67回有機合成化学協会関東支部シンポジウム(横浜シンポジウム)",,,,,,2014,May "布施 新一郎,高橋 良多,増井 悠,若宮 淳志,吉川 暹,高橋 孝志,田中 浩士","多様な側鎖構造の有機薄膜太陽電池用高分子p型半導体創出を指向したモノマーの迅速合成法の開発","日本化学会第94春季年会",,,,,,2014,Mar. "増井悠,高橋良太,布施新一郎,若宮淳志,吉川暹,高橋孝志","高分子有機半導体のライブラリー合成とその評価","日本化学会第94春季年会",,,,,,2014,Mar. "布施 新一郎,デーシャリン サンティダー,増井 悠,高橋 孝志,田中 浩士","α-シアノ酢酸エステルを基盤とするアザビシクロ化合物の効率合成法の開発","日本化学会第94春季年会",,,,,,2014,Mar. "布施 新一郎,中村 研太郎,御舩 悠人,中村 沙季,高橋 孝志,田中 浩士","ジオキシノンを分子集積プラットフォームとして活用する非ラメラ液晶ライブラリーの構築と評価","日本化学会第94春季年会",,,,,,2014,Mar. "鈴木 涼太,布施 新一郎,田中 浩士","環状ボラン化合物に対する 連続的鈴木・宮浦クロスカップリング 反応の開発","日本化学会第94春季年会",,,,,,2014,Mar. "米谷 真人,尾込 裕平,布 施 新一郎,野上 顕吾,望月 大,鈴木 榮一,早瀬 修二,加藤 隆二,高橋 孝 志,和田 雄二","アナターゼ型酸化チタン表面の D-pi-A 系有機色素吸着形態による色素増感太陽電池の電子移動特性への影響","日本化学会第94春季年会",,,,,,2014,Mar. "布施 新一郎,盛田 大輝,小林 大輔,松村 圭介,高橋 孝志,田中 浩士","C-H 結合直接アリール化を駆使した アリール4 置換ピラゾールの合成","日本化学会第94春季年会",,,,,,2014,Mar. "布施 新一郎,松村 圭介,増井 悠,若宮 淳志,吉川 暹,高橋 孝志,田中 浩士","有機薄膜太陽電池用p 型有機半導体を指向したオリゴヘテロ芳香環化合物の効率的合成法の開発とその機能評価","日本化学会第94春季年会",,,,,,2014,Mar. "MIFUNE Yuto,Shinichiro,TANAKA Hiroshi,TAKAHASHI Takashi","Efficient Amide Bond Formation through a Rapid and Strong Activation of Carboxylic Acid, and its Application for a Synthesis of Feglymycin","日本化学会第94春季年会",,,,,,2014,Mar.