"Y. Honda,Haruna Haraguchi,T. Tsuda,Rui Ko,K. Muguruma,H. Guo,T. Nomoto,Y. Miura,N. Nishiyama","Metal-phenolic network-based polymeric nanocarriers facilitating antibody cytoplasmic delivery and anti-tumor effects to orthotopic breast tumors",,"J. Control. Release",,,," in press",2025,Apr. "飯田啓介,松井 誠,六車 共平,本田雄士,三浦 裕,西山 伸宏","一型糖尿病の治療を目指した抗体フラグメント-高分子結合型医薬品の創製","日本薬学会第145年会",,,,,,2025,Mar. "柳田浩毅,小林基晃,Chintrakulchai Wanphiwat,高田 郁人,尾木 公一,道西 准也,大嶽 知之,六車 共平,本田 雄士,武元 宏泰,三浦 裕,西山 伸宏","PEGジレンマを解決する新規脂質ナノ粒子の開発とがん治療への展開","日本薬学会第145年会",,,,,,2025,Mar. "千野利純,松尾 拓海,本田 雄士,刑部 祐里子,Guo Haochen,六車 共平,三浦裕,西山 伸宏","CRISPR/Cas9-sgRNA RNP搭載三元系複合体による臓器選択的in vivoゲノム編集","日本薬学会第145年会",,,,,,2025,Mar. "Nozomi Matsudaira,Yuto Honda,Kyohei Muguruma,Haochen Guo,Yutaka Miura,Nobuhiro Nishiyama","Self-Assembly Ternary Complex Comprising Cyclic RGD-installed Polymer and Tannic Acid for Selective and Effective Protein Delivery to Tumor","第34回日本MRS年次大会",,,,,,2024,Dec. "千野利純,松尾拓海,本田雄士,刑部 祐里子,Guo Haochen,六車共平,三浦裕,西山伸宏","Cas9 RNP三元系複合体の高分子側鎖アミン構造調整によるゲノム編集制御","日本バイオマテリアル学会シンポジウム2024",,,,,,2024,Oct. "津田雄流,本田雄士,リチャードソンJ.ジョセフ,六車共平,Guo Haochen,三浦裕,西山伸宏","金属イオン‐ポリフェノール錯体を基盤としたPEG被覆技術の構築及び物性評価","日本バイオマテリアル学会シンポジウム2024",,,,,,2024,Oct. "松平 望,本田 雄士,六車 共平,GUO Haochen,三浦 裕,西山 伸宏","環状RGDペプチド導入高分子とタンニン酸からなる腫瘍細胞標的型三元系複合体の開発","日本バイオマテリアル学会シンポジウム2024",,,,,,2024,Oct. "金子彩海,本田雄士,松平望,Guo Haochen,喜納宏昭,六車共平,三浦裕,西山伸宏","肝実質細胞を標的可能にするGalNAc搭載アデノ随伴ウイルス三元系複合体の開発","日本バイオマテリアル学会シンポジウム2024",,,,,,2024,Oct. "黄 若言,津田 雄流,本田 雄士,Haochen Guo,六車 共平,三浦 裕,西山伸宏","CRISPR-Cas9/sgRNA RNPのゲノム編集効率を向上させる高分子ナノキャリアの開発","日本バイオマテリアル学会シンポジウム2024",,,,,,2024,Oct. "津田雄流,本田雄士,リチャードソンJ.ジョセフ,六車共平,三浦裕,西山伸宏","金属イオン‐ポリフェノール錯体を基盤としたPEG被覆中空マイクロカプセルの 構築及び物性評価","第73回高分子討論会",,,,,,2024,Sept. "Imai Kyosuke,Kyohei Muguruma,Ambara R. Pradipta,Katsunori Tanaka","In vivo synthetic anticancer approach by resourcing mouse blood albumin as a biocompatible artificial metalloenzyme",,"Angewandte Chemie International Edition",,,,,2024,July "Minagi Mukaiyama,Chihiro Uchiyama,Akane Fukuda,Yoshiki Nakazawa,Yuka Kuramochi,Yudai Shibata,Sho Konno,Kyohei Muguruma,Naohiro Matsugaki,Tomo Asari,Kazuyoshi Ogawa,Akihiro Taguchi,Kentaro Takayama,Atsuhiko Taniguchi,Yoko Nagumo,Toshiya Senda,Yoshio Hayashi,Takeo Usui","X-Ray Conformation and Structure?Activity Relationships of MA026, a Reversible Tight Junction Opener",,"Journal of Medicinal Chemistry",,,,,2023,July "Yudai Ode,Ambara R. Pradipta,Peni Ahmadi,Akihiro Ishiwata,Akiko Nakamura,Yasuko Egawa,Yuriko Kusakari,Kyohei Muguruma,Yang Wang,Xiaojie Yin,Nozomi Sato,Hiromitsu Haba,Katsunori Tanaka","Therapeutic efficacy of 211At-radiolabeled 2,6-diisopropylphenyl azide in mouse models of human lung cancer",,"Chemical Science",,,,,2023,June "Tsung-Che Chang,Igor Nasibullin,Kyohei Muguruma,Yuriko Kusakari,Taiji Shimoda,Katsunori Tanaka","Evaluation of acute toxicity of cancer-targeting albumin-based artificial metalloenzymes",,"Bioorganic & Medicinal Chemistry",,,,,2022,Nov. "Ahmadi P,Muguruma K,Chang TC,Tamura S,Tsubokura K,Egawa Y,Suzuki T,Dohmae N,Nakao Y,Tanaka K","In vivo metal-catalyzed SeCT therapy by a proapoptotic peptide.",,"Chemical science",,,,,2021,Sept. "Pradipta AR,Ahmadi P,Terashima K,Muguruma K,Fujii M,Ichino T,Maeda S,Tanaka K","Targeted 1,3-dipolar cycloaddition with acrolein for cancer prodrug activation.",,"Chemical science",,,,,2021,Apr. "Muguruma K,Osawa R,Fukuda A,Ishikawa N,Fujita K,Taguchi A,Takayama K,Taniguchi A,Ito Y,Hayashi Y","Development of a High-Affinity Antibody-Binding Peptide for Site-Specific Modification.",,"ChemMedChem",,,,,2021,Mar. "Sasaki K,Muguruma K,Osawa R,Fukuda A,Taniguchi A,Kishimura A,Hayashi Y,Mori T,Katayama Y","Synthesis and biological evaluation of a monocyclic Fc-binding antibody-recruiting molecule for cancer immunotherapy.",,"RSC medicinal chemistry",,,,,2021,Jan. "Muguruma K,Pradipta AR,Ode Y,Terashima K,Michiba H,Fujii M,Tanaka K","Disease-associated acrolein: A possible diagnostic and therapeutic substrate for in vivo synthetic chemistry.",,"Bioorganic & medicinal chemistry",,,,,2020,Oct. "Muguruma K,Fujita K,Fukuda A,Kishimoto S,Sakamoto S,Arima R,Ito M,Kawasaki M,Nakano S,Ito S,Shimizu K,Taguchi A,Takayama K,Taniguchi A,Hayashi Y","Kinetics-Based Structural Requirements of Human Immunoglobulin G Binding Peptides.",,"ACS omega",,,,,2019,Aug. "Muguruma K,Ito M,Fukuda A,Kishimoto S,Taguchi A,Takayama K,Taniguchi A,Ito Y,Hayashi Y","Synthesis and structure-activity relationship studies of IgG-binding peptides focused on the C-terminal histidine residue.",,"MedChemComm",,,,,2019,Aug. "Muguruma K,Shirasaka T,Akiyama D,Fukumoto K,Taguchi A,Takayama K,Taniguchi A,Hayashi Y","An Efficient Method for the Conjugation of Hydrophilic and Hydrophobic Components by Solid-Phase-Assisted Disulfide Ligation.",,"Angewandte Chemie (International ed. in English)",,,,,2018,Jan. "Takayama K,Rentier C,Asari T,Nakamura A,Saga Y,Shimada T,Nirasawa K,Sasaki E,Muguruma K,Taguchi A,Taniguchi A,Negishi Y,Hayashi Y","Development of Potent Myostatin Inhibitory Peptides through Hydrophobic Residue-Directed Structural Modification.",,"ACS medicinal chemistry letters",,,,,2017,June "Taguchi A,Kobayashi K,Kotani A,Muguruma K,Kobayashi M,Fukumoto K,Takayama K,Hakamata H,Hayashi Y","3-Nitro-2-pyridinesulfenates as Efficient Solution- and Solid-Phase Disulfide Bond Forming Agents.",,"Chemistry (Weinheim an der Bergstrasse, Germany)",,,,,2017,May "Yakushiji F,Muguruma K,Hayashi Y,Shirasaka T,Kawamata R,Tanaka H,Yoshiwaka Y,Taguchi A,Takayama K,Hayashi Y","Click strategy using disodium salts of amino acids improves the water solubility of plinabulin and KPU-300.",,"Bioorganic & medicinal chemistry",,,,,2017,May "Muguruma K,Yakushiji F,Kawamata R,Akiyama D,Arima R,Shirasaka T,Kikkawa Y,Taguchi A,Takayama K,Fukuhara T,Watabe T,Ito Y,Hayashi Y","Novel Hybrid Compound of a Plinabulin Prodrug with an IgG Binding Peptide for Generating a Tumor Selective Noncovalent-Type Antibody-Drug Conjugate.",,"Bioconjugate chemistry",,,,,2016,July "Hayashi Y,Takeno H,Chinen T,Muguruma K,Okuyama K,Taguchi A,Takayama K,Yakushiji F,Miura M,Usui T,Hayashi Y","Development of a new benzophenone-diketopiperazine-type potent antimicrotubule agent possessing a 2-pyridine structure.",,"ACS medicinal chemistry letters",,,,,2014,July "Yakushiji F,Tanaka H,Muguruma K,Iwahashi T,Yamazaki Y,Hayashi Y","Water-soluble prodrug of antimicrotubule agent plinabulin: effective strategy with click chemistry.",,"Chemistry (Weinheim an der Bergstrasse, Germany)",,,,,2011,Sept.