"Hiroyuki Nakamura","Design of Boron Cluster Lipids for Liposomal Boron Delivery System on NeutronCapture Therapy of Cancers","2006 International Conference on Bio and Pharmaceutical Scienceand Technology",,,,,,2006,Dec. "H. Nakamura,Y. Miyajima,Y. Kuwata,S. Masunaga,K. Ono,K. Maruyama,Hiroyuki Nakamura","Boron Nano Capsule: Tumor Targeting Boron Delivery System for Neutron CaptureTherapy","NANOBIO-TOKYO2006",,,,,,2006,Dec. "Hiroyuki Nakamura","病院併設型加速器中性子捕捉がん治療実用化に向けたホウ素デリバリーシステム","第12回創剤フォーラム若手シンポジウム",,,,,,2006,Dec. "堀越良爾,潘鉉承,Hiroyuki Nakamura","4-アニリノキナゾリン環上のホウ酸基置換部位によるEGFR及びVEGFRチロシンキナーゼ阻害活性の制御","第25回メディシナルケミストリーシンポジウム",,,,,,2006,Nov. "H. Nakamura,T. Usui,R. Horikoshi,H. Kuroda,H. S. Ban","Design of Organoboronic Acids for Targeting to Tumoral Vasculature System","10thInternational Kyoto Conference on New Aspects of Organic Chemistry",,,,,,2006,Nov. "Hiroyuki Nakamura,Shinya Onagi,Makoto Ishikura,Tsuyuka Sugiishi,TakayaKamakura","Synthesis of Allenes via Palladium-Catalyzed Hydride Transfer Reaction ofPropargylic Amines","10thInternational Kyoto Conference on New Aspects of Organic Chemistry",,,,,,2006,Nov. "Masaharu Uno,Yusuke Sasaki,Tomohiro Yoshikawa,Toru Asano,Hyun Seung Ban,HiroyukiNakamura","Synthesis and Biological Evaluation of Benzamides and Benzamidines as SelectiveInhibitors of VEGFR Tyrosine Kinases","10thInternational Kyoto Conference on New Aspects of Organic Chemistry",,,,,,2006,Nov. "Taikou Usui,Hyun Seung Ban,MInako Maruyama,Junpei Kawada,Takatsugu Hirokawa,Hiroyuki Nakamura,Taikou Usui,Hyun Seung Ban,MInako Maruyama,Junpei Kawada,Takatsugu Hirokawa,Hiroyuki Nakamura","Structure Based Drug Design and Synthesis of Indenopyrazoles as EpidermalGrowth Factor Receptor Tyrosine Kinase Inhibitors by in silico Libraly Screening","Structure Based Drug Design and Synthesis of Indenopyrazoles as EpidermalGrowth Factor Receptor Tyrosine Kinase Inhibitors by in silico Libraly Screening",,,,,,2006,Nov. "Hiroyuki Nakamura,Jong-Dae Lee,○Manabu Ueno,Yusuke Miyajiama,Hyun SeungBan","Synthesis and Liposome Formation of Boron Ion Cluster Lipid: New Boron DeliverySystem for Neutron Capture Therapy","10thInternational Kyoto Conference on New Aspects of Organic Chemistry",,,,,,2006,Nov. "Hiroyuki Nakamura,臼井大晃,堀越良爾,鍋山航,潘鉉承","4?アニリノキナゾリン骨格へのホウ酸基導入によるEGFR およびVEGFRチロシンキナーゼ阻害活性制御","第28回生体膜と薬物の相互作用シンポジウム",,,,,,2006,Nov. "Hiroyuki Nakamura","チロシンキナーゼ分子標的とホウ素薬剤の分子設計","静岡県立大学、依頼講演",,,,,,2006,Nov. "Hiroyuki Nakamura,宮島祐介,桑田康弘,増永慎一郎,小野公二,丸 山一雄","Transferrin-Conjugated Boron Cluster Liposome: Synthesis and IntracellularTargeting to Solid Tumors for Boron Neutron Capture Therapy","12th International Congress onneutron Capture Therapy、Plenary Session",,,,,,2006,Sept. "李宗大,Hiroyuki Nakamura","Synthesis and Liposome Formation of B12H11S-Substituted Lipids for BoronNeutron Capture Therapy","12th International Congress onneutron Capture Therapy、Plenary Session",,,,,,2006,Sept. "A. Matsumura,Y. Mori,Y. Kaneda,K. Hashimoto,H. Nakamura,T. Yamamoto,K.Nakai","A New NEDO Research Project towards Hospital Based Accelerator BNCT UsingAdvanced DDS System","12th International Congress onneutron Capture Therapy、Plenary Session",,,,,,2006,Sept. "Hiroyuki Nakamura,石倉誠,杉石露佳","Synthesis of 1,3-Disubstituted Allenes from Propargylic Amines via Palladium-CatalyzedHydride-Transfer Reaction","第53回有機金属化学討論会",,,,,,2006,Sept. "李宗大,Hiroyuki Nakamura","Synthesis and Liposome Formation of B-10 Enriched B12H11S-Substituted Lipidsfor Boron Neutron Capture Therapy","22th International Symposium on the Organic Chemistryof Sulfur (ISOCS-22)",,,,,,2006,Aug. "Hiroyuki Nakamura,臼井大晃,堀越良爾,潘鉉承,上原至雅,渋谷正史","Synthesis of Boron Containing Quinazolines: Unprecedented Control of Inhibitionstoward EGFR and VEGFR2 Protein Tyrosine Kinases by a Boronic Acid Substituent","Boron in the Americas X (BORAM X)",,,,,,2006,Aug. "Hiroyuki Nakamura,臼井大晃,堀越良爾,潘鉉承,上原至雅,渋谷正史","EGFRチロシンキナーゼ阻害剤を指向したホウ酸キナゾリン誘導体の合成と生物活性","第10回がん分子標的治療研究会総会",,,,,,2006,June "Hiroyuki Nakamura,宮島祐介,桑田康弘,増永慎一郎,小野公二,丸山一 雄","Synthesis of Transferrin-loaded nido-Carborane Liposome. Intracellular Targetingto Solid Tumors for Boron Neutron Capture Therapy","10th Liposome Research Days Conference",,,,,,2006,May "Hiroyuki Nakamura","Transferrin-Loaded nido-Carborane Liposome: Synthesis and IntracellularTargeting to Solid Tumors for Boron Neutron Capture Therapy","Particles 2006",,,,,,2006,May "小名木信耶,Hiroyuki Nakamura","EGFRチロシンキナーゼ阻害を指向したアレニルキナゾリン誘導体の合成および生物活性評価","日本化学会第86回春季年会",,,,,,2006,Mar. "堀越良爾,上原至雅,Hiroyuki Nakamura","EGFRチロシンキナーゼ阻害剤を指向したホウ素含有アニリノキナゾリン誘導体の合成および生物活性評価","日本化学会第86回春季年会",,,,,,2006,Mar. "佐々木悠介,上原至雅,Hiroyuki Nakamura","EGFR及びVEGFRチロシンキナーゼ阻害剤を指向したベンズアミジン誘導体の合成と生物活性評価","日本化学会第86回春季年会",,,,,,2006,Mar. "田代智史,蒲倉貴耶,Hiroyuki Nakamura","パラジウム触媒を用いた温和な条件下におけるプロパルギルアミンからのエン-アレン化合物の合成","日本化学会第86回春季年会",,,,,,2006,Mar. "Hiroyuki Nakamura","計算を活用した創薬アプローチの現状と今後の課題 ―有機合成化学者の立場から―","みずほ情報総研 「計算を活用した創薬の現状」セミナー",,,,,,2006,Mar. "H. Nakamura,T. Usui,R. Horikoshi,W. Nabeyama,H. S. Ban","Selective Inhibition of EGFR and VEGER Tyrosine Kinases Controlled by a Boronic Acid Substituent on 4-Anilinoquinazolines",,"Yakugaku Zasshi",,,"No. 126"," 164-165",2006, "A. Matsumura,Y. Mori,Y. Kaneda,K. Hashimoto,K. Nakai,T. Yamamoto,H. Nakamura,K. Akamatsu,T. Asano,S. Lee,Y. Sakurai,H. Kumada,K. Yamamoto,Y. Shibata,T. Shibata,T. Nakahara,M. Mutoh,H. Sakae,Y. Satoh,H. Sakurabata,S. Muraki,T. Nagayama","A New NEDO Reseach Project Toward Hospital Based Accelerator BNCT using Advanced DDS system",,"Advances in Neutron Capture Therapy",,,,"pp. 74-76",2006, "H. Nakamura,Y. Miyajima,Y. Kuwata,S. Masunaga,K. Ono,K. Maruyama","Transferrin-Loaded nido-Carborane Liposomes: Synthesis and Intracellular Targeting to Solid Tumors for Boron Neutron Capture Therapy",,"Advances in Neutron Capture Therapy",,,,"pp. 195-198",2006, "J.-D. Lee,H. Nakamura","Synthesis and Liposome Formation of B-10 Enriched B12H11S-Substituted Lipid for Boron Delivery System on BNCT",,"Advances in Neutron Capture Therapy",,,,"pp. 238-241",2006, "H Nakamura,S Onagi","Synthesis and biological evaluation of allenic quinazolines using palladium-catalyzed hydride-transfer reaction",,"Tetrahedron Letters",,"Vol. 47",,"pp. 2539-2542",2006, "H Nakamura,T Kamakura,S Onagi","1,2-Bis(diphenylphosphino)carborane as a dual mode ligand for both the sonogashira coupling and hydride-transfer steps in palladium-catalyzed one-pot synthesis of allenes from aryl iodides",,"Organic Letters",,"Vol. 8",,"pp. 2095-2098",2006, "Hiroyuki Nakamura,Yusuke Sasaki,Masaharu Uno,Tomohiro Yoshikawa,Toru Asano,Hyun Seung Ban,Hidesuke Fukazawa,Masabumi Shibuya,Yoshimasa Uehara","Synthesis and biological evaluation of benzamides and benzamidines as selective inhibitors of VEGFR tyrosine kinases",,"Bioorganic & Medicinal Chemistry Letters",,"Vol. 16",,"pp. 5127-5131",2006, "Hiroyuki Nakamura,Hirokazu Kuroda,Hiroyuki Saito,Ryo Suzuki,Takao Yamori,Kazuo Maruyama,Tatsuya Haga","Synthesis and biological evaluation of boronic acid containing cis-stilbenes as apoptotic tubulin polymerzation inhibitors",,"Chemmedchem",,"Vol. 1",,"pp. 729-740",2006, "Yusuke Miyajima,Hiroyuki Nakamura,Yasuhiro Kuwata,Jong-Dae Lee,Shinichiro Masunaga,Koji Ono,Kazuo Maruyama","Transferrin-loaded nido-carborane liposomes: Tumor-targeting boron delivery system for neutron capture therapy",,"Bioconjugate Chemistry",,"Vol. 17",,"pp. 1314-1320",2006, "CH Lee,JM Oh,JD Lee,H Nakamura,J Ko,SO Kang","Synthesis of THIQ derivatives as potential boron neutron capture therapy agents: N-functionalized o-carboranylmethyl benzopiperidines",,"Synlett",,,,"pp. 275-278",2006,