"東礎代子,佐藤伸一,Hiroyuki Nakamura","HIF-1αの分解に関わるHsp60のシャペロン活性を阻害するカルボラン化合物の開発","第10回がんとハイポキシア研究会",,,,,,2012,Dec. "松川卓也 峯岸秀充 中村浩之,松川卓也,峯岸秀充,Hiroyuki Nakamura","ジアリールカルボラン骨格を有するHIF-1阻害剤の開発","第10回がんとハイポキシア研究会",,,,,,2012,Dec. "Hiroyuki Nakamura","closo-Dodecaborate-conjugated cholesterols: Synthesis and click imaging of their liposomes in cells,","Trilaterla Meeting of BNCT in Taipei",,,,,,2012,Dec. "Hayato Koganei,Manabu Ueno,Shoji Tachikawa,Lisa Tasaki,Hyun Seung Ban,Minoru Suzuki,Kouichi Shiraishi,Kumi Kawano,Masayuki Yokoyama,Yoshie Maitani,Koji Ono,Hiroyuki Nakamura","Development of High Boron Content Liposomes and Their Promising Antitumor Effect for Neutron Capture Therapy of Cancers",,"Bioconjugate Chemistry",,"Vol. 24",,"pp. 124-132",2012,Dec. "Hiroyuki Nakamura,Yuka Yasui,Minako Maruyama,Hidemitsu Minegishi,Hyun Seung Ban,Shinichi Sato","Development of hypoxia-inducible factor (HIF)-1ホア inhibitors: Effect of ortho-carborane substituents on HIF transcriptional activity under hypoxia",,"Bioorganic & Medicinal Chemistry Letters",,"Vol. 23",,"pp. 806-810",2012,Dec. "Hiroyuki Nakamura","Boron-Based Drug Design: Discovery of HIF-1α Degradation Induced by Inhibition of HSP60 under Hypoxia","Korea University, Seminar, 依頼講演",,,,,,2012,Dec. "峯岸秀充,安井友香,丸山美菜子,潘鉉承,佐藤伸一,Hiroyuki Nakamura","カルボラン骨格を基軸としたHIF-1阻害剤の開発","第10回がんとハイポキシア研究会",,,,,,2012,Dec. "Tsuyuka Sugiishi,Hiroyuki Nakamura","CH vs CC Bond Activation of Propargylic Amines in the Presence of Pd, Cu or Zn Catalysts","12th International Kyoto Congress of Organich Chemistry (IKCOC-12)",,,,,,2012,Nov. "H. Minegishi,S. Fukashiro,H. S. Ban,H. Nakamura","Discovery of Indenopyrazoles as HIF-1α Inhibitors","12th International Kyoto Congress of Organich Chemistry (IKCOC-12)",,,,,,2012,Nov. "Hiroyuki Nakamura","Neutron Capture Therapy ?Principles and Applications",,,"Springer",,,,2012,Nov. "東礎代子,安井友香,峯岸秀充,佐藤伸一,Hiroyuki Nakamura","カルボラン含有低酸素誘導因子HIF-1α阻害剤の開発","第30回メディシナルケミストリーシンポジウム",,,,,,2012,Nov. "佐藤伸一,安井友香,丸山美菜子,峯岸秀充,潘鉉承,Hiroyuki Nakamura","カルボラン骨格を基盤とした新規Hsp60阻害剤の開発","第30回メディシナルケミストリーシンポジウム",,,,,,2012,Nov. "T. Matsukawa,L. Tazaki,H. S. Ban,H. Nakamura","Diphenylcarboranes as a new class of hypoxia inducible factor inhibitors","12th International Kyoto Congress of Organich Chemistry (IKCOC-12)",,,,,,2012,Nov. "Hiroyuki Nakamura","Boron-Based Drug Design: From Chemical Biology to Neutron Capture Therapy","the Institute of Medical Biology (IMB) Poland Academy of Science, Seminar",,,,,,2012,Oct. "Hiroyuki Nakamura","Development of inhibitors targeting hypoxia cell signaling","2th COLLOQUE FRANCO-ROUMAIN DE CHIMIE MEDICINALE",,,,,,2012,Oct. "Hiroyuki Nakamura","Discovery of HIF-1a Degradation Induced by Inhibition of HSP60 under Hypoxia","1st International Symposium on Chemical Biology of Natural Products:Target ID and Regulation of Bioactivity",,,,,,2012,Oct. "小金井逸人,上野学,立川将士,鈴木実,小野公二,Hiroyuki Nakamura","高ホウ素化リポソームの開発と中性子照射による抗腫瘍効果","第21回DDSカンファランス",,,,,,2012,Sept. "F. Yoshida,K. Nakei,T. Yamamoto,M. Shirakawa,H. Nakamura,Alexander Zaboronok,Akira Matsumura","Pretreatment with buthionine sulfoximine enhanced uptake and retention of BSH for BNCT","15th International congress on Neutron Capture Therapy",,,,,,2012,Sept. "H. Nakamura,T. Miyoshi,S. Tachikawa,H. Koganei,S. Kojima,M. Suzuki,K. Ono","closo-Dodecaborate-conjugated cholesterols:Synthesis and click imaging of their liposomesin cells","15th International congress on Neutron Capture Therapy",,,,,,2012,Sept. "S. Tachikawa,T. Miyoshi,H. Koganei,D. Kanoh,H. Ban,M. Suzuki,M. Kirrihara,K. Ono,H. Nakamura","Development of liposomal boron agents for neutron capture therapy","15th International congress on Neutron Capture Therapy",,,,,,2012,Sept. "Ayano Takeuchi,Makihito Hori,Shinichi Sato,Hyun Seung Ban,Takahiro Kuchimaru,Shinae Kizaka-Kondoh,Takao Yamori,Hiroyuki Nakamura","Synthesis and biological activity of furanylindazoles as inhibitors of hypoxia inducible factor (HIF)-1 transcriptional activity",,"MedChemComm",,"Vol. 3",,"pp. 1455-1461",2012,Sept. "Agnieszka B. Olejniczak,S. Tachikawa,H. Nakamura,Z. J. Lesnikowski","Cholesterol-boron cluster conjugates:Synthesis via dioxane ring opening of the oxonium derivative of the boron cluster and preliminary physicochemical and biological evaluation Magdalena Bialek-Pietras","4th Congress of the European Association for Chemical and Molecular Sciences Prague",,,,,,2012,Aug. "Makoto Sakai,Naohiro Fujimoto,Katsunori Ishii,Hiroyuki Nakamura,Yasufumi Kaneda,Kunio Awazu","In vitro investigation of efficient photodynamic therapy using a nonviral vector; hemagglutinating virus of Japan envelope",,"Journal of Biomedical Optics",,"Vol. 17",,,2012,July "Hiroyuki Nakamura,三好達郎,立川将士,小金井逸人,鈴木実,小野公二","中性子捕捉療法のためのホウ素コレステロールの開発-リポソーム化と細胞内イメージング","日本DDS学会学術集会",,,,,,2012,July "Masaharu Uno,Yosuke Koma,Hyun Seung Ban,Hiroyuki Nakamura","Discovery of 1-[4-(N-benzylamino)phenyl]-3-phenylurea derivatives as non-peptidic selective SUMO-sentrin specific protease (SENP)1 inhibitors",,"Bioorganic & Medicinal Chemistry Letters",,"Vol. 22",,"pp. 5169-5173",2012,July "峯岸 秀充,矢守 隆夫,Hiroyuki Nakamura","インデノピラゾール化合物の細胞増殖抑制効果に関する研究","第16回日本がん分子標的治療学会学術集会",,,,,,2012,June "Hiroyuki Nakamura","Boron-Based Drug Design:From Chemical Biology to Neutron Capture Therapy","Paris Tech Seminar",,,,,,2012,June "佐藤伸一,竹内彩乃,堀牧人,潘鉉承,口丸高弘,近藤科江,矢守隆夫,Hiroyuki Nakamura","HIF-1α転写阻害剤YC-1の誘導展開と作用機構解析","新学術領域研究「天然物ケミカルバイオロジー:分子標的と活性制御」第 1回若手研究者ワークショップ",,,,,,2012,June "Hiroyuki Nakamura","Carboranylphenoxyacetanilides as HIF-1 Inhibitors:Photoaffinity Probe Design for Identification of Heat Shock Protein 60, a Primary Target","A celebration of Organic Chemistry",,,,,,2012,June "Hiroyuki Nakamura","Dodecaborate Lipid Liposomes as New Vehicles for Boron Delivery System of Neutron Capture Therapy","The 13th Boron In The Americas Conference",,,,,,2012,June "Hiroyuki Nakamura","ホウ素脂質リポソームの開発と中性子捕捉治療効果","第16回日本がん分子標的治療学会学術集会",,,,,,2012,June "Hiroyuki Nakamura","ホウ素でがんに挑む","第69回学習院大学理学部技術交流会",,,,,,2012,May "堀牧人,潘鉉承,Hiroyuki Nakamura","低酸素誘導因子(HIF)? 1α 阻害剤YC ? 1誘導体の合成","日本薬学会第131年会",,,,,,2012,Mar. "深代真司,峯岸秀充,潘鉉承,Hiroyuki Nakamura","インデノピラゾール骨格を基軸としたHIF-1阻害剤の開発","第132回日本薬学会年会",,,,,,2012,Mar. "小金井逸人,立川将士,三好達郎,鈴木実,小野公二,Hiroyuki Nakamura","ホウ素脂質リポソームの 中性子照射における抗腫瘍効果","第132回日本薬学会年会",,,,,,2012,Mar. "Hayato Koganei,Shoji Tachikawa,Minoru Suzuki,Koji Ono,Hiroyuki Nakamura","Antitumor Activity of Boron Lipid Liposomes with Neutron Irradiation","SIMS2012",,,,,,2012,Mar. "Hiroyuki Nakamura","ホウ素リポソームの高集積化を目指して","平成23年度京都大学原子炉実験所専門研究会",,,,,,2012,Feb. "Hiroyuki Nakamura","がんの低酸素応答を標的とした創薬研究の現状","筑波大学医学医療系 セミナー 依頼講演",,,,,,2012,Feb. "Hiroyuki Nakamura","がんの低酸素環境応答と分子標的","第2回Cancer Cell Informaticsによる創薬研究会",,,,,,2012,Feb. "Tsuyuka Sugiishi,Hiroyuki Nakamura","Zinc(II)-Catalyzed Redox Cross-Dehydrogenative Coupling of Propargylic Amines and Terminal Alkynes for Synthesis of N-Tethered 1,6-Enynes",,"Journal of the American Chemical Society",,"Vol. 134",,"pp. 2504-2507",2012,Jan. "Hyun Seung Ban,Kazuki Shimizu,Hidemitsu Minegishi,Hiroyuki Nakamura","Identification of heat shock protein 60 as the regulator of the hypoxia-inducible factor subunit HIF-1 alpha",,"Pure and Applied Chemistry",,"Vol. 84",,"pp. 2325-2337",2012, "Yongeun Kim,Hiroyuki Nakamura","Copper(I)-Catalysed Deacetylenative Cross-Coupling Reaction of Terminal Alkynes with Propargylic Amines via C(sp)-C(sp(3)) Bond Cleavage",,"Synlett",,,,"pp. 1686-1690",2012, "Hiroyuki Nakamura,Hirokazu Kuroda,Hidemitsu Minegishi","Synthesis and biological evaluation of boronic acid-containing phenstatin analogues",,"Arkivoc",,,,"pp. 79-87",2012, "N. Ueda,H. Koganei,M. Ueno,S. Tachikawa,M. Suzuki,K. Ono,H. Nakamura","Development of fluorescence-labeled boron lipid: liposome formation and in vitro and in vivo imaging",,"Progress in Drug Delivery System XXI",,,,"pp. 68-73",2012, "Takeuchi A,Hori M Hyun,Ban S,Kuchimaru T,Kizaka-Kondoh S,Yamori T,Hiroyuki Nakamura","Synthesis and biological evaluation of furylindazoles as hypoxia inducible factor (HIF)-1α inhibitors.",,"Med Chem Commun",,"Vol. 3",,"p. 1455",2012,