"S. Ogawa,Y. Asawa,M. Iiyama,A. Yoshimori,H. Nakamura,M. Oda","Regulation of binding between CD28 cytoplasmic region and SH2 domains of Grb2 and PI3K by carborane compounds for T-cell activation",,"BIOORG. MED. CHEM. LETT.",,"Vol. 78",," 129049",2022,Dec. "Hiroyuki Nakamura","Chemical Manipulation of Target Proteins Using Ruthenium bis(Bipyridine) Complexes","The 27th International SPACC Symposium",,,,,,2022,Dec. "Kohei Umedera,Atsushi Yoshimori,Hengwei Chen,Hiroyuki Kouji,Hiroyuki Nakamura,Jurgen Bajorath","DeepCubist: Molecular Generator for Designing Peptidomimetics based on Complex three-dimensional scaffolds",,"Journal of Computer-Aided Molecular Design",,"Vol. 37","No. 2","pp. 107-115",2022,Dec. "Hiroyuki Nakamura","BNCTの適応拡大を目指したホウ素薬剤開発","日本量子医科学会第2回学術大会",,,,,,2022,Dec. "Hiroyuki Nakamura","Design of MMP-1 Inhibitors via SAR Transfer and Experimental Validation",,,,,,,2022,Dec. "K. Umedera,T. Morita,H. Nakamura","Asymmetric construction of densely functionalized three-dimensional aza-tetracyclic scaffolds for drug discovery",,"Chem. Commun",,,,,2022,Nov. "Hiroyuki Nakamura","Development of Intracellular Photocatalytic Proximity Protein Labeling (iPPL) for Profiling Protein?Protein Interactions","International Congress of Pure and Applied Chemistry (ICPACK)2022",,,,,,2022,Nov. "Kazuki Miura,Yijin Wen,Michihiko Tsushima,Hiroyuki Nakamura","Photodynamic therapy by glucose transporter 1?selective light inactivation",,"ACS Omega",," 7"," 38"," 34685?34692",2022,Sept. "H. Nakamura,T. Morita,H. Murakami","Development of 1,2-Azaborine-fused Heterocycles and Their Novel Functionalization","The VIth International Conference",,,,,,2022,Sept. "Hiroyuki Nakamura","光触媒を用いた生細胞内標的タンパク質近接場標識法(iPPL 法)の開発","バイオインタラクション研究会第18回ワークショップ",,,,,,2022,Sept. "Hiroyuki Nakamura","ホウ素クラスターの創薬化学","第66回日本薬学会関東支部大会",,,,,,2022,Sept. "K. Nishimura,S. Harrison,K. Kawai,T. Morita,K. Miura,S. Okada,H. Nakamura","Iodophenyl-conjugated closo-dodecaborate as a promising small boron molecule that binds to serum albumin and accumulates in tumor",,"BIOORG. MED. CHEM. LETT.",,"Vol. 72",," 128869",2022,Sept. "Hiroyuki Nakamura","ホウ素の拓く創薬ワールド",,"細胞「特集 低分子モダリティの進化―元素・光・分子機能に注目して」",," 54"," 9",,2022,Aug. "Taiki Morita,Hiroki Murakami,Hiroyuki Nakamura","Asymmetric Synthesis of Oxazaborolidines via Palladium-Catalyzed N-H/B-H Double Functionalization of 1,2-Azaborines","The 9th European Conference on Boron Chemistry",,,,,,2022,July "Hiroyuki Nakamura,Yasunobu Asawa","Comprehensive Exploration of Chemical Space Using Trisubstituted Carboranes","The 9th European Conference on Boron Chemistry",,,,,,2022,July "H. Kitamura,Y. Otake,N. Sugisawa,H. Sugisawa,T. Ida,H. Nakamura,S. Fuse,Hiroyuki Nakamura","Sequential Selective Introduction of Alcohols against Phosphorus Trichloride in a Continuous-Flow Reactor and Consideration of a Mechanism for Reduced Overreaction via the Addition of Imidazole",,"Chemistry",," 28"," 37"," e202200932",2022,July "A. M.Hughes,J. A. Goldfinger,M. A. Palmieri,P. Ramos,I. S. Santa Cruz,L. De Leo,M. A. Garabalino,S. I. Thorp,P. Curotto,E. C.C. Pozzi,K. Kawai,S. Sato,M. E. Itoiz,V.A. Trivillin,J. S. Guidobono,H. Nakamura,A. E. Schwint","Boron neutron capture therapy (BNCT) mediated by maleimide-functionalized closo-dodecaborate albumin conjugates (MID:BSA) for oral cancer: Biodistribution studies and in vivo BNCT in the hamster cheek pouch oral cancer model",,"Life (Basel)",," 12"," 7"," 1082",2022,July "Hiroyuki Nakamura","光反応を利用したタンパク質の化学修飾","第27回ケムステVシンポ『有機光反応の化学 』(オンライン)",,,,,,2022,July "Hiroshi Kitamura,Yuma Otake,Naoto Sugisawa,杉澤宏樹,井田朋智,Hiroyuki Nakamura,Shinichiro Fuse","非対称リン酸トリエステルのマイクロフロー合成および反応機構解明","創薬懇話会2022",,,,,,2022,June "Hiroshi Kitamura,Yuma Otake,Naoto Sugisawa,杉澤宏樹,井田朋智,Hiroyuki Nakamura,Shinichiro Fuse","非対称リン酸トリエステルのマイクロフロー合成および反応機構解明","第120回有機合成シンポジウム",,,,,,2022,June "A. R Jalilian,A. Shahi,I. P. Swainson,H. Nakamura,M. Venkatesh,J. A. Osso Jr","Potential theranostic BNCT agents as multimodal radiopharmaceuticals",,"Cancer Biotherapy and Radiopharmaceuticals",,"Vol. 37"," 5",,2022,June "Hiroyuki Nakamura,Kai Nishimura,Taiki Morita,Satoshi Okada,Kazuki Miura,柏木秀基,福尾祐介,松本孔貴,Minoru Suzuki,中井啓,川端信司","中性子捕捉療法のための血清アルフ?ミンを利用したホウ素キャリアの開発","第27 回癌治療増感研究会",,,,,,2022,Apr. "Hiroyuki Nakamura","Boron Delivery using Serum Albumin","NCI Workshop on Neutron Capture Therapy for Cancer",,,,,,2022,Apr. "Taiki Morita,Hiroyuki Nakamura","ピペラジン酸およびN-ヒドロキシアミノ酸の直接縮合を基盤としたDentigerumycin Aの合成研究","日本化学会第102春季年会",,,,,,2022,Mar. "Kazuki Miura,Yijin Wen,Michihiko Tsushima,Hiroyuki Nakamura","細胞透過型有機光触媒による標的タンパク質選択的不活性化と抗腫瘍活性プローブへの応用","日本薬学会142春季年会",,,,,,2022,Mar. "Rohmad.Yudi Utomo,Atsushi Sugie,Satoshi Okada,Kazuki Miura,Hiroyuki Nakamura","Curcumin誘導体のアミロイドβ繊維の解離を介した解毒作用とショウジョウバエのアルツハイマー病モデルにおける検証","日本薬学会142春季年会",,,,,,2022,Mar. "Kai Nishimura,Taiki Morita,Satoshi Okada,Kazuki Miura,柏木秀基,福尾祐介,松本孔貴,高田卓志,Minoru Suzuki,中井啓,川端信司,Hiroyuki Nakamura","中性子捕捉療法のための、アルブミンリガンドを基軸としたホウ素キャリアの開発","日本薬学会142春季年会",,,,,,2022,Mar. "社本乙華,Keiji Komuro,Naoto Sugisawa,Hiroyuki Nakamura,Shinichiro Fuse","マイクロフローリアクター内での環状ペプチド合成法の開発","日本化学会第102春季年会",,,,,,2022,Mar. "Ayana Uehara,Taiki Morita,佐々木雄彦,Hiroyuki Nakamura","リゾホスファチジルイノシトール(4,5)ビスリン酸の合成研究","日本化学会第102春季年会",,,,,,2022,Mar. "Hiroyuki Nakamura,Rohmad.Yudi Utomo,Satoshi Okada,住吉晃,Ichio Aoki","アミロイドβ繊維化を検出・阻害するMRIプローブの開発","日本化学会第102春季年会",,,,,,2022,Mar. "Hiroki Murakami,Taiki Morita,Hiroyuki Nakamura","パラジウム触媒を用いた1,2-アザボリン類の不斉N-H/B-H二官能基化法の開発","日本化学会第102春季年会",,,,,,2022,Mar. "Masato Tsuda,Taiki Morita,Hiroyuki Nakamura","金(I)触媒によるプロパルギルアザClaisen転位反応を用いたイソオキサゾロアザボリンの合成と亜鉛カルベノイドによるN−O結合へのメチレン挿入反応の開発","日本化学会第102春季年会",,,,,,2022,Mar. "Hiroyuki Nakamura","中性子捕捉療法:承認までの軌跡と今後の展望","第19回同位体科学研究会",,,,,,2022,Mar. "Hiroyuki Nakamura","Development of Intracellular Photocatalytic Proximity Protein Labeling (iPPL)","9th International Conference on Chemical and Biological Sciences (ICCBS 2022)",,,,,,2022,Mar. "S. Koyama,H. Sato,H. Sugai,M. Murakoshi,T. Kobayashi,S. Usami,K. Ikeda,Y. Haga,K. Tsumoto,H. Nakamura,N. Hirasawa,Kenji ISHIHARA,H. Wada","Effects of Salicylate Derivatives on Changes in Localization of H723R Pendrin Mutant Expressed in HEK293 Cells",,"Auris Nasus Larynx",,,,,2022,Mar. "T. Morita,H. Murakami,Y. Asawa,H. Nakamura","Enantioselective Synthesis of Oxazaborolidines by Palladium-Catalyzed N−H/B−H Double Activation of 1,2-Azaborines",,"Angew. Chem. Int. Ed.",,"Vol. 61","Issue 7",,2022,Feb. "R. Y. Utomo,S. Okada,A. Sumiyoshi,I. Aoki,H. Nakamura","Development of an MRI contrast agent for both detection and inhibition of the amyloid-β fibrillation process",,"RSC Adv.",,,,,2022,Feb. "Tae-Hee Han,M. K. Park,H. Nakamura,H. S. Ban","Capsaicin inhibits HIF-1α accumulation through suppression of mitochondrial respiration in lung cancer cells",,"Biomedicine & Pharmacotherapy",,"Volume 146"," 112500",,2022,Feb. "Hiroyuki Nakamura","BODIPY Catalyzes Proximity‐Dependent Histidine Labellin",,,,,,,2022,Feb. "M. Tsushima,S. Sato,K. Miura,T. Niwa,HIDEKI TAGUCHI,H. Nakamura","Intracellular photocatalytic-proximity labeling for profiling protein?protein interactions in microenvironments",,"Chem. Commun.",," 58"," 1926-1929",,2022,Jan. "H. Ueda,P.Wipf,H. Nakamura","Synthesis of sp3-rich chiral bicyclo[3.3.1]nonanes for chemical space expansion and study of biological activities",,"Bioorganic & Medicinal Chemistry",,"Volume 54"," 116561",,2022,Jan. "G. Li,G. Yu,C. Wang,T. Morita,X. Zhang,H. Nakamura","Copper(I)-catalysed intramolecular hydroarylation-redox cross-dehydrogenative coupling of N-propargylanilines with phosphites",,"Org. biomol. chem.",,," 20"," 113-116",2022,Jan. "Hiroyuki Nakamura","タンパク質夾雑空間解析のための細胞内光触媒近接場標識法(iPPL法)の開発","新学術領域研究「分子夾雑の生命化学」第6回班会議",,,,,,2022,Jan. "Michihiko Tsushima,Kazuki Miura,Shinichi Sato,Hiroyuki Nakamura","Intrecellular photocatalytic proximity labeling for profiling protein-protein interactins in multimolecular crowding","The 2nd International Symposium on Chemistry for Multimolecular Vrouding Biosystems",,,,,,2022,Jan. "R. Y. Utomo,A. Sugie,S. Okada,K. Miura,H. Nakamura","Detoxification of amyloid β fibrils by curcumin derivatives and their verification in a Drosophila Alzheimer's model",,"Chem. Commun.",," 58"," 2576-2579",,2022,Jan. "M. Tsuda,T. Morita,H. Nakamura","Synthesis of isoxazoloazaborines via gold(i)-catalyzed propargyl aza-Claisen rearrangement/borylative cyclization cascade",,"Chem. Commun.",," 58"," 1942-1945",,2022,Jan.