"Y. Asawa,S. Hatsuzawa,A. Yoshimori,K. Yamada,A. Katoh,H. Kouji,H. Nakamura","Comprehensive Exploration of Chemical Space Using Trisubstituted Carboranes",,"Sci. Rep.",,"  11","  24101",,2021,Dec.
"Kohei Umedera,Taiki Morita,Hiroyuki Nakamura","Synthesis of sp3-carbon rich azatricyclododecene framework via gold-catalized Conia-ene reaction","Pacifichem",,,,,,2021,Dec.
"Masato Tsuda,Taiki Morita,Shintaro Fukuhara,Hiroyuki Nakamura","Cationic Gold(I)-Catalyzed Propargyl Aza-Claisen Rearrangement: Synthesis of 5-Allenyl-4-aminoisoxazoles","Pacifichem",,,,,,2021,Dec.
"Taiki Morita,Shinichiro Fuse,Hiroyuki Nakamura","Photochemical conversion of isoxazoles to 5-hydroxyimidazolines","Pacifichem",,,,,,2021,Dec.
"Hiroyuki Nakamura,Yijin Wen,Kazuki Miura,Michihiko Tsushima,Hideya Yuasa","Target protein knockdown using photocatalysts: Application to photodynamic therapy","Pacifichem",,,,,,2021,Dec.
"Hiroyuki Nakamura,Michihiko Tsushima,Shinichi Sato,Kazuki Miura","Development of photocatalytic-proximity protein labeling for profiling protein-protein interaction in intracellular microenvironments","Pacifichem",,,,,,2021,Dec.
"Haruna Shiono,Akira Takakado,Hiroyuki Nakamura,Koichi Iwata","Evaluation of viscosity of lipid bilayer nanodiscs","Pacifichem",,,,,,2021,Dec.
"Natsumi Okada,Masayuki Iwamoto,Akira Takado,Hiroyuki Nakamura,Shigetoshi Oiki,Koichi Iwata","The effect of local anesthetics on lipid bilayer membranes evaluated by picosecond time-resolved fluorescence spectroscopy","Pacifichem",,,,,,2021,Dec.
"Hiroyuki Nakamura","Development of PBC-IP as a Novel Boron Agent: Unexpectedly High BNCT Effect on Rat Brain Tumor","The 3rd Taiwan-Japan Neutron Capture Therapy Academic Communication of Elite (3rd TJNCTACE)",,,,,,2021,Dec.
"Yasunobu Asawa,Saki Hatsuzawa,Atsushi Yoshimori,Kentaro Yamada,Akira Katoh,Hiroyuki Kouji,Hiroyuki Nakamura","Comprehensive exploration of three-dimensional chemical space by trisubstituted carboranes for discovery of bioactive molecule","The 13th AFMC International Medicinal Chemistry Symposium (AIMECS-2021)",,,,,,2021,Nov.
"Hiroki Murakami,Taiki Morita,Hiroyuki Nakamura","パラジウム触媒を用いた1,2-アザボリン類のN-H/B-H二官能基化法の開発","第119回有機合成シンポジウム",,,,,,2021,Nov.
"Yasunobu Asawa,Kei Nishida,Kazuki Kawai,Kiyotaka Domae,Hyun Seung Ban,Akihiro Kitazaki,Hiroya Asami,Jun-Ya Kohno,Satoshi Okada,Hiraku Tokuma,Daisuke Sakano,Shoen Kume,Masaru Tanaka,Hiroyuki Nakamura","Carborane as an Alternative Efficient Hydrophobic Tag for Protein Degradation",,"Bioconjugate Chemistry",,,,,2021,Nov.
"H. Kashiwagi,S. Kawabata,K. Yoshimura,Y. Fukuo,T. Kanemitsu,K. Takeuchi,R. Hiramatsu,K. Nishimura,K. Kawai,T. Takata,H. Tanaka,T. Watanabe,M. Suzuki,S. Miyatake,H. Nakamura,M. Wanibuchi","Boron neutron capture therapy using dodecaborated albumin conjugates with maleimide is effective in a rat glioma model",,"Investigational new drugs",,,,,2021,Nov.
"Y. Tsuji,N. Nonoguchi,D. Okuzaki,Y. Wada,D. Motooka,Y. Hirota,T. Toho,N. Yoshikawa,M. Furuse,S. Kawabata,S.-I. Miyatake,H. Nakamura,R. Yamamoto,S. Nakamura,T. Kuroiwa,M. Wanibuchi","Chronic pathophysiological changes in the normal brain parenchyma caused by radiotherapy accelerate glioma progression",,"Sci. Rep",,"  11","  22110",,2021,Nov.
"Hiroyuki Nakamura,Satoshi Okada,Jeff Delacruz","3D細胞培養系の構築と抗がん剤ライブラリースクリーニング","がんとハイポキシア研究会2021",,,,,,2021,Nov.
"H. Yanagie,M. Yanagawa,K. Mouri,Y. Morishita,A. Shinohara,N. Dewi,Y. Nonaka,Y. Furuya,R. Mizumachi,Y. Murata,H. Nakamura,M. Suzuki,Y. Sakurai,H. Tanaka,S. Masunaga,K. Ono,T. Sugihara,M. Nashimoto,H. Yamauchi,M. Ono,J. Nakajima,H. Terada,H. Takahashi","Suppression of Tumor Growth in a Rabbit Hepatic Cancer Model by Boron Neutron Capture Therapy With Liposomal Boron Delivery Systems",,"In Vivo",,"Vol. 35","no. 6","pp. 3125?3135",2021,Nov.
"浅輪泰允,中村浩之","カルボランを基盤とした立体的分子による3次元ケミカルスペースの探索と新規PPI制御分子の創成","バイオインタラクション研究会",,,,,,2021,Nov.
"Kai Nishimura,Taiki Morita,Satoshi Okada,Takumi Ogawara,Takushi Takata,Minoru Suzuki,Hiroyuki Nakamura","Development of an albumin-based boron delivery system for neutron capture therapy","The 13th AFMC International Medicinal Chemistry Symposium (AIMECS-2021)",,,,,,2021,Nov.
"Kohei Umedera,Taiki Morita,Atsushi Yoshimori,Kentaro Yamada,Akira Katoh,Hiroyuki Kouji,Hiroyuki Nakamura","Synthesis of Three-Dimensional Diazatricyclododecene Scaffold and Design of Peptidomimetics","The 13th AFMC International Medicinal Chemistry Symposium (AIMECS-2021)",,,,,,2021,Nov.
"Yuka Takashima,?安聡子,Satoshi Okada,Hiroyuki Nakamura","磁場による薬物徐放を志向したポリマーコーティング酸化鉄ナノ粒子の開発","第81回有機合成化学協会関東支部シンポジウム ?群馬・前橋シンポジウム?",,,,,,2021,Nov.
"Hiroshi Kitamura,Yuma Otake,Naoto Sugisawa,杉澤宏樹,井田朋智,Hiroyuki Nakamura,Shinichiro Fuse","マイクロフローリアクターを用いる非対称リン酸トリエステルの高速合成","第11回CSJ化学フェスタ2021",,,,,,2021,Oct.
"Kohei Umedera,Taiki Morita,吉森篤史,Kentaro Yamada,小路弘之,Hiroyuki Nakamura","三次元骨格ジアザトリシクロドデセンの開発とペプチド模倣分子への応用","第11回CSJ化学フェスタ2021",,,,,,2021,Oct.
"Satoshi OKADA,Satoko TAKAYASU,Akira SUMIYOSHI,Ichio AOKI,Hiroyuki NAKAMURA","MRI-based Glucose Assay Using Magnetic Nanoparticle Sensors",,"Anal. Sci.",,,,,2021,Oct.
"Satoshi Okada,Vivian Hsieh,Satoko Takayasu,Akira Sumiyoshi,Ichio Aoki,Alan Jasanoff,Hiroyuki Nakamura","Development of neurotransmitter-responsive magnetic nanoprobes","The 5th A3 Foresight Symposium on Organic/Inorganic Nanohybrid Platforms for Precision Tumor Imaging and Therapy",,,,,,2021,Oct.
"Ayana Uehara,Taiki Morita,佐々木雄彦,Hiroyuki Nakamura","リゾホスファチジルイノシトール（４，５）ビスリン酸の合成研究","第11回CSJ化学フェスタ2021",,,,,,2021,Oct.
"Kai Nishimura,Taiki Morita,Satoshi Okada,Takumi Ogawara,Takushi Takata,Minoru Suzuki,Hiroyuki Nakamura","Development of an albumin-based boron delivery system for neutron capture therapy","The 19th International Congress on Neutron Capture Therapy (ICNCT 19)",,,,,,2021,Sept.
"T. Morita,S. Yugandar,H. Nakamura","Novel Direct Functionalization and Photochemical Reaction of Isoxazoles","XI International Conference on Chemistry  for Young Scientists (Mendeleev 2021)",,,,,,2021,Sept.
"M. Tsuda,T. Morita,S. Fukuhara,H. Nakamura","Gold(I)-Catalyzed Intramolecular Electrophilic Aromatic Substitution of Isoxazoles","XI International Conference on Chemistry  for Young Scientists (Mendeleev 2021)",,,,,,2021,Sept.
"H. Nakamura,M. Tsushima,M. Matsumura,S. Sato","Boron Neutron Capture Therapy: A New Modality of Radiation Therapy","XI International Conference on Chemistry  for Young Scientists (Mendeleev 2021)",,,,,,2021,Sept.
"Satoshi Okada,Vivian Hsieh,?安 聡子,住吉 晃,Alan Jasanoff,Ichio Aoki,Hiroyuki Nakamura","磁場照射で脳機能を観察・操作する磁性ナノツールの開発","2021年第82回応用物理学会秋季学術講演会",,,,,,2021,Sept.
"Hiroyuki Nakamura","チロシン残基特異的ラベル化技術の開発","同仁化学研究所セミナー",,,,,,2021,Sept.
"Shinichi Sato,Masaki Matsumura,Hiroshi Ueda,Hiroyuki Nakamura","Preparation of an antigen-responsive fluorogenic immunosensor by tyrosine chemical modification of the antibody complementarity determining region",,"Chemical Communications","RSC",,,,2021,Aug.
"N. Sugisawa,H. Sugisawa,Y. Otake,R. V. Krems,H. Nakamura,S. Fuse","Rapid and Mild One-Flow Synthetic Approach to Unsymmetrical Sulfamides Guided by Bayesian Optimization",,"Chemistry Methods",,,,,2021,July
"Hiroyuki Nakamura,Kai Nishimura,Taiki Morita,Satoshi Okada,磯山翔,玉城尚美,旦慎吾","低分子ホウ素薬剤PBC-IPの細胞選択性評価","第17回日本中性子捕捉療法学会",,,,,,2021,July
"Kai Nishimura,Taiki Morita,Satoshi Okada,Takumi Ogawara,柏木秀基,福尾祐介,松本孔貴,高田卓志,Minoru Suzuki,中井啓,川端信司,Hiroyuki Nakamura","中性子捕捉療法のためのアルブミンをプラットホームとした低分子ホウ素薬剤PBC-IPの開発","第17回日本中性子捕捉療法学会",,,,,,2021,July
"Hiroyuki Nakamura","中性子捕捉療法：承認までの軌跡と今後の展望","第17回フッ素相模セミナー",,,,,,2021,July
"Keita Nakane,Tatsuya Niwa,Michihiko Tsushima,HIDEKI TAGUCHI,友重秀介,Hiroyuki Nakamura,石川稔,Shinichi Sato","一重項酸素を活用したヒスチジン残基近接標識法の開発","日本ケミカルバイオロジー学会第１５回年会",,,,,,2021,June
"Kazuki Miura,Michihiko Tsushima,Shinichi Sato,Tatsuya Niwa,HIDEKI TAGUCHI,Hiroyuki Nakamura","細胞内タンパク質間相互作用解析のための光触媒近接タンパク質標識法の開発","日本ケミカルバイオロジー学会第１５回年会（オンライン）",,,,,,2021,June
"Kohei Umedera,Hiroyuki Nakamura","含窒素三環性骨格を基盤としたHIF転写活性阻害剤の開発","第25回がん分子標的治療学会学術大会",,,,,,2021,May
"M. Tsuda,T. Morita,H. Nakamura","Suzuki-Miyaura Cross-coupling of 3,4-disubstituted 5-bromoisoxazoles: An efficient access to trisubstituted isoxazoles",,"Tetrahedron Lett",,,,,2021,May
"Hiroki Ueda,Peter Wipf,Hiroyuki Nakamura","ケミカルスペースの開拓を志向した三次元骨格の新規構築反応開発","有機合成化学協会 第79回関東支部シンポジウム（オンライン",,,,,,2021,May
"Yasunobu Asawa,Hiroyuki Nakamura","疎水性ホウ素クラスターによる新規タンパク質分解誘導剤の開発とその機構解明","第25回がん分子標的治療学会学術大会",,,,,,2021,May
"SUSUMU KAJIWARA,Tenagy,Shuji Tsuchida,Ayana Uehara,陳馨?,Hiroyuki Nakamura","抗マラセチア薬開発に資する脂肪酸取込阻害","第95回日本感染症学会学術講演会",,,,,,2021,May
"Masato Tsuda,Taiki Morita,Hiroyuki Nakamura","金(I)触媒およびパラジウム触媒を用いたイソオキサゾール5位修飾反応の開発","有機合成化学協会 第79回関東支部シンポジウム",,,,,,2021,May
"Paviter Singh,Manjot Kaur,Kulwinder Singh,Gurpreet Kaur,Ramovatar Meena,Manpreet Kaur,Bikramjeet Singh,Anup Thakur,Jeewan Sharma,Ajay Singh,Manjeet Kumar,Ju-Hyung Yun,Fumiko Nakagawa,Minoru Suzuki,Hiroyuki Nakamura,Akshay Kumar","Fluorescent Boron Carbide Quantum dots synthesized with a low-temperature solvothermal approach for boron neutron capture therapy",,"Physica E: Low-Dimensional Systems and Nanostructures.",,"  132, 114766",,,2021,Apr.
"H. S. Ban,H. Nakamura","Design of Carborane-Based Hypoxia-Inducible Factor Inhibitors",,"Boron-Based Compounds: Potential and Emerging Applications in Medicine",,,,,2021,Apr.
"Hiroyuki Nakamura","細胞内タンパク質?タンパク質相互作用解析を可能とする光ラベル化技術の開発","新学術領域研究「分子夾雑の生命化学」第5回班会議",,,,,,2021,Apr.
"K. Nakane,S. Sato,T. Niwa,M. Tsushima,S. Tomoshige,H. Taguchi,M. Ishikawa,H. Nakamura","Proximity Histidine Labeling by Umpolung Strategy Using Singlet Oxygen",,"J. Am. Chem. Soc.",,"  143, 20, 7726?7731",,,2021,Apr.
"Hiroki Ueda,Peter WIPF,Hiroyuki Nakamura","ケミカルスペースの開拓を志向した三次元骨格の新規構築反応開発とタンパク質間相互作用（Protein-proteinInteraction, PPI）阻害活性評価","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"Masato Tsuda,Taiki Morita,Shintaro Fukuhara,Hiroyuki Nakamura","プロパルギルアザClaisen転位反応による5-アレニルイソオキサゾールの合成とイソオキサゾロアザボリン環構築への展開","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"Taiki Morita,Somaraju Yugandar,Hiroyuki Nakamura","ロジウム（III）触媒を用いた脱炭酸を伴うイソオキサゾールのC-H官能基化反応の開発","日本化学会第101春季年会",,,,,,2021,Mar.
"初澤早貴,Yasunobu Asawa,吉森篤史,Kentaro Yamada,小路弘行,真崎康博,Hiroyuki Nakamura","PPI阻害剤を志向した三置換メタカルボランライブラリー化合物の合成とその生物活性評価","日本薬学会第141年会（オンライン）",,,,,,2021,Mar.
"Kai Nishimura,Kazuki Kawai,Satoshi Okada,Shinichi Sato,Minori Suzuki,高田卓志,Hiroyuki Nakamura","中性子捕捉療法のための、インテグリンをターゲットとしたホウ素キャリア、環状RGDペプチド結合型ホウ素化アルブミンの開発","日本薬学会第141年会（オンライン）",,,,,,2021,Mar.
"Kohei Umedera,Taiki Morita,吉森篤史,Kentaro Yamada,小路弘行,Hiroyuki Nakamura","含窒素三環性骨格を足場とするペプチド模倣分子の開発","日本薬学会第141年会（オンライン）",,,,,,2021,Mar.
"Y. Asawa,A. V. Arsent’eva,S. A. Anufriev,A. A. Anisimov,K. Yu. Suponitsky,O. A. Filippov,H. Nakamura,I. B. Sivaev","Synthesis of Bis(Carboranyl)amides 1,1’-μ-(CH2NH(O)C(CH2)n- 1,2-C2B10H11)2 (n = 0, 1) and Attempt of Synthesis of Gadolinium Bis(Dicarbollide",,"Molecules",,"Vol. 26","No. 5","pp. 1321",2021,Mar.
"Yasunobu Asawa,吉森篤史,Kentaro Yamada,小路弘行,Hiroyuki Nakamura","カルボランを基盤とした立体的分子による3次元ケミカルスペースの探索とそのPPI制御機能評価","日本薬学会第141年会（オンライン）",,,,,,2021,Mar.
"Ayana Uehara,Taiki Morita,佐々木雄彦,Hiroyuki Nakamura","リゾホスファチジルイノシトール（4,5）ビスリン酸の合成研究","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"Keiji Komuro,Yuma Otake,Hiroyuki Nakamura,Shinichiro Fuse","マイクロフローリアクター内でのトリホスゲンを用いた迅速なラクタム合成法の開発","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"Michihiko Tsushima,Shinichi Sato,Hiroyuki Nakamura","細胞内微小空間で起こるタンパク質間相互作用の解析を可能にする光触媒近接タンパク質ラベル化法の開発","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"Aaron Li Hsin Chang,Michihiko Tsushima,Hiroyuki Nakamura","Photocatalytic proximity labelling of ligand-binding proteins utilizing single-electron transfer mediate radical reaction","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"Hiroki Murakami,Taiki Morita,Yasunobu Asawa,Hiroyuki Nakamura","パラジウム触媒を用いた1,2-アザボリン類のN-H/B-H二官能基化法の開発","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"Hiroshi Kitamura,Yuma Otake,Hiroyuki Nakamura,Shinichiro Fuse","マイクロフローリアクターを用いる非対称リン酸トリエステルの高速合成","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"Naoto Sugisawa,Hiroyuki Nakamura,Shinichiro Fuse","マイクロフローリアクター内での瞬間両基質活性化を駆使したβ-アミノ酸誘導体の合成","日本化学会第101春季年会（オンライン）",,,,,,2021,Mar.
"R. Yudi Utomo,Y. Asawa,S. Okada,A. Yoshimori,J. Bajorath,H. Nakamura","Development of curcumin-based amyloid β aggregation inhibitors for Alzheimer's disease using the SAR matrix-approach","The International Center for Chemical and Biological Sciences (ICCBS-2021)","Bioorg. Med. Chem.",,"  46,","  116357",,2021,Feb.
"Hiroyuki Nakamura","BNCTの薬剤と中性子の反応",,"月刊インナービジョン特集号",,"Vol. 36","No. 2","pp. 40-42",2021,Feb.
"中村 浩之","中性子捕捉療法：承認までの奇跡と今後の展望","岡山大学次世代研究G講演会（ナノ・ハ?イオ融合によるエネルキ?ー集積・高度利用研究拠点形成）招待講演（オンライン）",,,,,,2021,Feb.
"Hiroyuki Nakamura","Boron Neutron Capture Therapy: A New Modality of Radiation Therapy","The International Center for Chemical and Biological Sciences (ICCBS-2021), Keynote Lecture (online, Tokyo)",,,,,,2021,Feb.
"H. S. Ban,Y. Uto,H. Nakamura","Hypoxia-inducible factor (HIF) inhibitors: a patent survey (2016-2020)",,"Expert Opin. Ther. Pat.",,,,,2021,Jan.
"Hiroshi Kitamura,Yuma Otake,Jun Kawamura,布施 新一郎,Hiroyuki Nakamura","入手容易なマイクロミキサーを用いたリポソーム調製法の開発",,"製剤機械技術学会誌",,"Vol. 29","No. 4","  407-413",2021,Jan.
"M. Tsuda,S. Fukuhara,Taiki Morita,H. Nakamura","Synthesis of 4-Amino-5-allenylisoxazoles via Gold(I)-Catalyzed Propar-gyl Aza-Claisen Rearrangement: Application to an Isoxazoloazaborine Ring System",,"Org. Biomol. Chem",,,"No. 19","pp. 1358-1364",2021,Jan.
"K. Umedera,T. Morita,A. Yoshimori,K. Yamada,A. Katoh,H. Koji,H. Nakamura","Synthesis of Three-Dimensional (3D) (Di)azatricyclododecene Scaffold and its Application to Peptidomimetics",,"Chem. Eur. J",,,,,2021,Jan.
"S. Fuse,K. Komuro,Y. Otake,H. Masui,H. Nakamura","Rapid and Mild Lactamization Using Highly Electrophilic Triphosgene in a Micro-Flow Reactor",,"Chem. Eur. J",,"Vol. 2021","No. 27","pp. 1-9",2021,Jan.
"Hiroyuki Nakamura","Boron Neutron Capture Therapy: A New Modality of Radiation Therapy","Dalian University of Technology Online Exchange Conference, Invited Lecture (online, China)",,,,,,2021,Jan.
"Takahiro Shimizu,NorihitoTakahashi,Vincent J.Huber,Yasunobu Asawa,Hiroki Ueda,Atsushi Yoshimori,Yukiko Muramatsu,Hiroyuki Seimiya,Hiroyuki Kouji,Hiroyuki Nakamura,Hiroki Oguri","Design and synthesis of 14 and 15-membered macrocyclic scaffolds exhibiting inhibitory activities of hypoxia-inducible factor 1α",,"Bioorg. Med. Chem.",,,"No. 30","pp. 115949",2021,Jan.
"G. Li,Y. Shao,Y. Pan,Y. Li,Y. Wang,L. Wan],K. Shao,S. Wang,H. Dong,X. W,X. Guo,W. Zhao,H. Nakamura","Total synthesis and biological evaluation of 7-Hydroxyneolamellarin A as hypoxia-inducible factor-1α inhibitor for cancer therapy",,"BIOORG. MED. CHEM. LETT.",,"  50","  128338",,2021,