"H. Minegishi,M. Maruyama,Y. Yasui,K. Shimizu,H. Ban,H. Nakamura","Discovery of carboranes as 20S proteasome activators","2010環太平洋国際化学会議",,,,,,2010,Dec. "S. Tachikawa,H. Nakamura","Development of closo-dodecaborates for liposomal boron delivery of neutron capture therapy","2010環太平洋国際化学会議",,,,,,2010,Dec. "A. Takeuchi,A. Shoji,H. Ban,T. Yamori,H. Nakamura","Discovery of carborane-conjugated triazines as topoisomerase inhibitors","2010環太平洋国際化学会議",,,,,,2010,Dec. "H. Ban,K. Shimizu,H. Minegishi,H. Nakamura","Action mechanism of HIF-1α inhibitor GN26361: Identification of target protein with multifunctional molecular probe","2010環太平洋国際化学会議",,,,,,2010,Dec. "H. Nakamura,M. E. El-Zaria,H. Ban,A. R. Genady","Synthesis of triazolyl methyl-substituted thio-, amino-, and oxy-undecahydrododecaborates for potential application to boron neutron capture therapy","2010環太平洋国際化学会議",,,,,,2010,Dec. "H. Nakamura,M. Ueno,N. Ueda,R. Inomata,H. Ban","Development of boron lipid liposomes for neutron capture therapy","2010環太平洋国際化学会議",,,,,,2010,Dec. "H. Nakamura,M. Ueno,N. Ueda,R. Inomata,H. Ban","Development of boron lipid liposomes for neutron capture therapy","2010環太平洋国際化学会議",,,,,,2010,Dec. "Y. Koma,M. Uno,H. Ban,H. Nakamura","Structure-activity relationship of 1-[4-(N-benzylamino)phenyl]-3-phenylurea derivatives as HIF-1α inhibitors","2010環太平洋国際化学会議",,,,,,2010,Dec. "中村 浩之","低酸素誘導因子シグナルを標的とした創薬研究の現状","日本放射線腫瘍学会第23回学術大会",,,,,,2010,Nov. "三好達郎,Mohamed E. El-Zaria,潘鉉承,中村浩之","カルボラニルトリアジン誘導体の選択的トポイソメラーゼ阻害活性","第29回メディシナルケミストリーシンポジウム",,,,,,2010,Nov. "峯岸秀充,潘鉉承,丸山美菜子,安井友香,清水一希,中村浩之,中村浩之","カルボラン含有低分子20S プロテアソーム活性化剤の開発","第29回メディシナルケミストリーシンポジウム",,,,,,2010,Nov. "竹内彩乃,東海林篤,潘鉉承,矢守隆夫,中村浩之","ホウ素含有コレステロールの開発:クリック反応によるイメージングとリポソーム化","第29回メディシナルケミストリーシンポジウム",,,,,,2010,Nov. "F. Yoshida,K. Nakai,T. Isobe,R. Inomata,A. Zaboronok,Y. Yamamoto,M. Shirakawa,T. Yamamoto,A. Matsumura,H. Nakamura","Biodistribution of BSH-encapsulated boron liposome in mouse glioma","14th International Congress Neutron Capture Therapy, Buenos Aires",,,,,,2010,Oct. "H. Nakamura,N. Ueda,H. S. Ban,K. Maruyama,M. E. El-Zaria","Boron Lipid Liposomes: EPR Effect and Fluorescence Imaging","14th International Congress Neutron Capture Therapy, Buenos Aires",,,,,,2010,Oct. "R. Inomata,M. E. El-Zaria,H. S. Ban,H. Nakamura","Development of Boron-Containing Protoporphyrin IX Derivatives for Boron Neutron Capture Therapy and Photodynamic Therapy","14th International Congress Neutron Capture Therapy, Buenos Aires",,,,,,2010,Oct. "R. Inomata,M. E. El-Zaria,H. S. Ban,H. Nakamura","Development of Boron-Containing Protoporphyrin IX Derivatives for Boron Neutron Capture Therapy and Photodynamic Therapy","14th International Congress Neutron Capture Therapy, Buenos Aires",,,,,,2010,Oct. "東海林篤,竹内彩乃,潘鉉承,Kang Sang Ook,矢守隆夫,中村浩之","カルボラン含有トリアジン誘導体のトポイソメラーゼ阻害活性","第40回複素環化学討論会",,,,,,2010,Oct. "中村 浩之","ホウ素の力でがんに挑む","学習院大学生命科学シンポジウム『生命の秘密を解く鍵をもとめて』(第8回) 依頼講演",,,,,,2010,Oct. "杉石露佳,中村浩之","1価の銅触媒存在下におけるプロパルギルアミン類のアルキン置換反応","第57回有機金属化学討論会",,,,,,2010,Sept. "上野学,潘鉉承,中村浩之","リポソームを用いる中性子捕捉治療",,"Drug Delivery System",,"Vol. 25","No. 5","pp. 474-482",2010,Sept. "M. E. El- Zaria,A. R. Genady,中村浩之","New Strategy for Synthesis of Mercaptoundecahydrododecaborate Derivatives via Click Chemistry: Possible Boron Carriers and Visualization in Cells for Neutron Capture Therapy","第7回日本中性子捕捉療法学会学術集会",,,,,,2010,Aug. "猪俣竜,上野学,立川将士,三好達郎,Mohamed E. El-Zaria,潘鉉承,小田雄介,鈴木亮,丸山一雄,中村浩之","トランスフェリン修飾ホウ素リポソームによるBNCT効果","第7回日本中性子捕捉療法学会学術集会",,,,,,2010,Aug. "潘鉉承,清水一希,峯岸秀充,中村浩之","カルボラン含有小分子化合物GN26361による低酸素誘導因子(HIF)阻害と作用機序","第7回日本中性子捕捉療法学会学術集会",,,,,,2010,Aug. "中村 浩之","がんの低酸素環境応答に着目した創薬アプローチ","日本化学会第4回関東支部大会 依頼講演",,,,,,2010,Aug. "潘鉉承,清水一希,峯岸秀充,中村浩之","低酸素誘導因子(HIF) 阻害剤GN26361 の作用機序の解明","第14回日本がん分子標的治療学会学術集会",,,,,,2010,July "中村浩之,宇野正治,潘鉉承","脱SUMO 化酵素SENP-1 阻害剤の発見","第14回日本がん分子標的治療学会学術集会",,,,,,2010,July "峯岸秀充,清水一希,潘鉉承,中村浩之","カルボラン含有低分子20S プロテアソーム活性化剤の開発","第14回日本がん分子標的治療学会学術集会",,,,,,2010,July "東海林篤,潘鉉承,矢守隆夫,中村浩之","カルボラン含有トリアジン類のトポイソメラーゼ阻害活性","第14回日本がん分子標的治療学会学術集会",,,,,,2010,July "Hiroyuki Nakamura","Boron-Containing Phenoxyacetanilide DHypoxia-Inducible Factor (HIF)-1α Inhibitors","Boron in the Americas XII",,,,,,2010,June "Hiroyuki Nakamura","Liposomal Boron Delivery System for Neutron Capture Therapy of Cancers","第49回日本生体医工学会大会",,,,,,2010,June "峯岸秀充,潘鉉承,丸山美菜子,安井友香,清水一希,中村浩之","カルボラン含有低分子20Sプロテアソーム活性化剤の開発","第59回有機合成化学協会関東支部シンポジウム",,,,,,2010,May "竹内彩乃,東海林篤,潘鉉承,矢守隆夫,中村浩之","カルボラン含有トリアジン類のトポイソメラーゼ阻害活性","日本ケミカルバイオロジー学会 第5回年会",,,,,,2010,May "中村浩之,宇野正治,潘鉉承","脱SUMO化酵素SENP-1阻害剤の発見と低酸素誘導因子抑制作用","日本ケミカルバイオロジー学会 第5回年会",,,,,,2010,May "M. E. El-Zaria,A. R. Genady,潘鉉承,中村浩之","イオン性ホウ素クラスターのクリック型環化反応の開発と細胞内イメージング","日本ケミカルバイオロジー学会 第5回年会",,,,,,2010,May "中村浩之","中性子捕捉治療のためのナノカプセル型ホウ素薬剤送達システム(BDS)の開発",,"Pharm. Tech. Japan (invited)",,,"No. 26","pp. 1005-1012",2010,May "高麗洋佑,宇野正治,潘鉉承,中村浩之","低酸素誘導因子(HIF)-1α阻害剤の開発","第59回有機合成化学協会関東支部シンポジウム",,,,,,2010,May "潘鉉承,宇野正治,中村浩之","VEGFR阻害剤によるHIF活性化抑制とその作用機序","日本薬学会第130回年会",,,,,,2010,Mar. "田中優子,臼井大晃,潘鉉承,浅井章良,中村浩之","インデノピラゾール骨格を有する新規HIF-1α 阻害剤の開発","日本薬学会第130回年会",,,,,,2010,Mar. "清水一希,中村浩之","アリルトリフルオロボレートを用いた触媒的ビス-π- アリルパラジウム反応","日本薬学会第130回年会",,,,,,2010,Mar. "峯岸秀充,丸山美菜子,安井友香,清水一希,潘鉉承,中村浩之","カルボラン含有低分子プロテアソーム活性化剤の開発","日本薬学会第130回年会",,,,,,2010,Mar. "宇野正治,潘鉉承,中村浩之","新規SUMO 特異的プロテアーゼ(SENP)阻害剤の開発","日本薬学会第130回年会",,,,,,2010,Mar. "高麗洋佑,潘鉉承,近藤科江,平岡眞寛,中村浩之","HIF-1α 抑制剤GN6767誘導体の創薬研究 宇野正治","日本薬学会第130回年会",,,,,,2010,Mar. "中村 浩之","ホウ素の中性子捕捉反応を利用した低侵襲細胞選択的放射線療法","日本薬学会第130回年会シンポジウム「異分野技術の融合による次世代の医療基盤技術の構築に向けて」、オーガナイザー",,,,,,2010,Mar. "上田記子,潘鉉承,中村浩之","蛍光標識ホウ素ナノカプセルの開発と細胞内イメージング","日本薬学会第130回年会",,,,,,2010,Mar. "Hyun Seung Ban,Hidemitsu Minegishi,Kazuki Shimizu,Minako Maruyama,Yuka Yasui,Hiroyuki Nakamura","Discovery of Carboranes as Inducers of 20S Proteasome Activity",,"Chemmedchem",,"Vol. 5",,"pp. 1236-1241",2010, "Manabu Ueno,Hyun Seung Ban,Kei Nakai,Ryu Inomata,Yasufumi Kaneda,Akira Matsumura,Hiroyuki Nakamura","Dodecaborate lipid liposomes as new vehicles for boron delivery system of neutron capture therapy",,"Bioorganic & Medicinal Chemistry",,"Vol. 18",,"pp. 3059-3065",2010, "Tsuyuka Sugiishi,Akifumi Kimura,Hiroyuki Nakamura","Copper(I)-Catalyzed Substitution Reactions of Propargylic Amines: Importance of C(sp)-C(sp(3)) Bond Cleavage in Generation of Iminium Intermediates",,"Journal of the American Chemical Society",,"Vol. 132",,"pp. 5332-+",2010, "Kazuki Shimizu,Minako Maruyama,Yuka Yasui,Hidemitsu Minegishi,Hyun Seung Ban,Hiroyuki Nakamura","Boron-containing phenoxyacetanilide derivatives as hypoxia-inducible factor (HIF)-1 alpha inhibitors",,"Bioorganic & Medicinal Chemistry Letters",,"Vol. 20",,"pp. 1453-1456",2010, "Hiroyuki Nakamura,Ryoji Horikoshi,Taikou Usui,Hyun Seung Ban","Selective inhibition of EGFR and VEGFR2 tyrosine kinases controlled by a boronic acid substituent on 4-anilinoquinazolines",,"Medchemcomm",,"Vol. 1",,"pp. 282-286",2010, "Kenji Ishihara,Shuhei Okuyama,Shun Kumano,Koji Iida,Hiroshi Hamana,Michio Murakoshi,Toshimitsu Kobayashi,Shinichi Usami,Katsuhisa Ikeda,Yoichi Haga,Kohei Tsumoto,Hiroyuki Nakamura,Noriyasu Hirasawa,Hiroshi Wada","Salicylate restores transport function and anion exchanger activity of missense pendrin mutations",,"Hearing Research",,"Vol. 270",,"pp. 110-118",2010, "Afaf R. Genady,Hiroyuki Nakamura","Undecahydro-closo-dodecaborates as good leaving groups in organic synthesis: generation of substituted styrenes via elimination of arylethyl dodecaborates",,"Organic & Biomolecular Chemistry",,"Vol. 8",,"pp. 4427-4435",2010, "Mohamed E. El-Zaria,Afaf R. Genady,Hiroyuki Nakamura","Synthesis of triazolyl methyl-substituted amino- and oxy-undecahydrododecaborates for potential application in boron neutron capture therapy",,"New Journal of Chemistry",,"Vol. 34",,"pp. 1612-1622",2010, "Mohamed E. El-Zaria,Hyun Seung Ban,Hiroyuki Nakamura","Boron-Containing Protoporphyrin IX Derivatives and Their Modification for Boron Neutron Capture Therapy: Synthesis, Characterization, and Comparative In Vitro Toxicity Evaluation",,"Chemistry-a European Journal",,"Vol. 16",,"pp. 1543-1552",2010, "Hyun Seung Ban,Masaharu Uno,Hiroyuki Nakamura","Suppression of hypoxia-induced HIF-1 alpha accumulation by VEGFR inhibitors: Different profiles of AAL993 versus SU5416 and KRN633",,"Cancer Letters",,"Vol. 296",,"pp. 17-26",2010, "Hyun Seung Ban,Yuko Tanaka,Wataru Nabeyama,Masako Hatori,Hiroyuki Nakamura","Enhancement of EGFR tyrosine kinase inhibition by C-C multiple bonds-containing anilinoquinazolines",,"Bioorganic & Medicinal Chemistry",,"Vol. 18",,"pp. 870-879",2010, "中村 浩之","ホウ素の中性子捕捉反応を利用した低侵襲細胞選択的放射線療法",,"Yakugaku Zasshi",,,"No. 130","pp. 1687-1694",2010, "Hyun Seung Ban,Kazuki Shimizu,Hidemitsu Minegishi,Hiroyuki Nakamura","Identification of HSP60 as a Primary Target of o-Carboranylphenoxyacetanilide, an HIF-1 alpha Inhibitor",,"Journal of the American Chemical Society",,"Vol. 132",,"pp. 11870-11871",2010,