"佐藤伸一,中村公亮,中村浩之","酵素Horseradish Peroxidaseを利用したタンパク質化学修飾","ファイブスターアソシエーション・ダイナミックアライアンスG3分科会",,,,,,2016,Dec. "中村浩之","生体高分子を用いたホウ素デリバリーシステムの構築","ファイブスターアソシエーション・ダイナミックアライアンスG3分科会",,,,,,2016,Dec. "G. Dorm?n,H. Nakamura,A. Pulsipher,G. D. Prestwich","The Life of Pi Star: Exploring the Exciting and Forbidden Worlds of the Benzophenone Photophore",,"Chem. Rev.",,"Vol. 116","No. 24","Page 15284?15398",2016,Dec. "石井秀一,布施新一郎,佐藤伸一,中野洋文,中村浩之","天然物タンシノンIIAを基盤とした新規HIF-1α阻害剤の開発","第5回「次世代がん治療推進専門家養成プランシンポジウム」",,,,,,2016,Dec. "中村浩之","世界をリードする次世代低侵襲がん治療:中性子捕捉療法","第2回神奈川県ヘルスケア・ニューフロンティア講座「次世代医療に向けた医理工学融合研究とその産業応用」",,,,,,2016,Dec. "Y. Mifune,H. Nakamura,S. Fuse","A Rapid and Clean Synthetic Approach to Cyclic Peptides via Micro-flow Peptide Chain Elongation and Photochemical Cyclization: Synthesis of a Cyclic RGD Peptide",,"Organic & Biomolecular Chemistry",,"Vol. 14","No. 47","page 11244-11249",2016,Nov. "Hiroyuki Nakamura,Kikuchi,Daisuke Kanoh,Shinichi Sato,Yoshinori Sakurai,Minoru Suzuki","Maleimide-Functionalized closo-Dodecaborate Albumin Conjugate: Unique Ligation at Cysteine and Lysine Residues Enables Efficient Boron Delivery to Tumor for Neutron Capture Therapy","3rd International Conference on Biomaterials Science in Tokyo (ICBS2016)",,,,,,2016,Nov. "中村浩之","リポソーム包埋型およびアルブミン結合型ホウ素キャリアー","大阪医科大学附属病院がんセンター先端医療開発部門 シンポジウム",,,,,,2016,Nov. "小竹佑磨,中村浩之,布施新一郎","マイクロフロー合成法を駆使するN-メチル化ペプチドの合成法開発","第6回CSJ化学フェスタ2016",,,,,,2016,Nov. "石井秀一,布施新一郎,佐藤伸一,中野洋文,中村浩之","天然物タンシノンIIAを基盤とした新規HIF-1α阻害剤の開発研究","第14回がんとハイポキシア研究会",,,,,,2016,Nov. "石井秀一,布施新一郎,中村浩之","多環性オルトキノン化合物の短段階合成を志向したPd触媒による脱水素型環化反応の開発","第6回CSJ化学フェスタ2016",,,,,,2016,Nov. "S. Fuse,T. Ohuchi,Y. Asawa,S. Sato,H. Nakamura","Development of 1-Aryl-3-furanyl/Thienyl-imidazopyridine Templates for Inhibitors against Hypoxia Inducible Factor (HIF)-1 Transcriptional Activity",,"Bioorganic and Medicinal Chemistry Letters",,"Vol. 26","No. 24","page 5887-5890",2016,Nov. "S. Fuse,Y. Mifune,H. Nakamura,H. Tanaka","Total Synthesis of Feglymycin based on a Linear/Convergent Hybrid Approach using Micro-flow Amide Bond Formation","The 10th International Symposium on Integrated Synthesis (ISONIS-10)",,,,,,2016,Nov. "Shinichiro Fuse,Yuto Mifune,Hiroyuki Nakamura,Hiroshi Tanaka","Total synthesis of feglymycin based on a linear/convergent hybrid approach using micro-flow amide bond formation",,"Nature Communications",,,"No. 13491",,2016,Nov. "Hiroyuki Nakamura","Enhanced Permeability and Retention (EPR) Effect-Based Efficient Boron Delivery Systems for BNCT","17th International Congress on Neutron Capture Therapy",,,,,,2016,Oct. "中村浩之","中性子捕捉療法用ホウ素高集積リポソームの開発","第6回DDS製剤臨床応用FG合宿討論会",,,,,,2016,Oct. "中村浩之","化学でがんの根治に挑む","都立新宿高校模擬講義",,,,,,2016,Oct. "S. Ishii,S. Kikuchi,S. Sato,H. Nakamura","Development of closo-Dodecaborate-Serum Albumin Conjugates via Ruthenium-Photocatalyzed Tyrosine Modification for Neutron Capture Therapy","17th International Congress on Neutron Capture Therapy",,,,,,2016,Oct. "稲井瑞穂,古山祐,洪暎淳,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","複製能欠損ウイルス粒子を用いた光感受性薬剤の細胞内局在と腫瘍選択性の検討","第37回日本レーザー医学会総会",,,,,,2016,Oct. "Hiroyuki Nakamura","Zinc(II)-Catalyzed Intramolecular Hydroarylation-Redox Cross-Dehydrogenative Coupling of Propargylic Amines","International Conference Nature Inspired Initiative in Chemical Trends 2016",,,,,,2016,Sept. "中村浩之","Boron compounds suitable for BNCT","1st NRW-Fukushima Joint Symposium on Advances in Medicine",,,,,,2016,Sept. "洪暎淳,稲井瑞穂,古山祐,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","抗がん剤耐性前立腺がん細胞への迅速な薬剤輸送に向けた複製能欠損ウイルス粒子への光感受性物質の封入",,"電気学会 光・量子デバイス研究会",,,,,2016,Sept. "T. Morita,S. Fuse,H. Nakamura","Generation of 4-Isoxazolyl Anion Species: Facile Access to 4-Substituted Isoxazoles",,"Angewandte Chemie International Edition",,"Vol. 55","No. 43","page 13580-13584",2016,Sept. "佐藤伸一,中村公亮,中村浩之","生体内ヘムの鉄酸化状態変化を利用したタンパク質ラベリング","第89回日本生化学会大会",,,,,,2016,Sept. "大西宏明,大塚弘毅,松島早月,渡邊卓,中村浩之,広川貴次","蛋白質立体構造解析と分子動力学に基づくEGFR分子標的薬の効果予測","第63回日本臨床検査医学会学術大会",,,,,,2016,Sept. "T. Morita,S. Fuse,H. Nakamura","Generation of 4-Isoxazolyl Anion Species: Facile Access to 4-Substituted Isoxazoles",,"Angewandte Chemie International Edition",,"Vol. 55","No. 43","page 13580-13584",2016,Sept. "佐藤伸一,中村公亮,中村浩之","Horseradish Peroxidaseを触媒として利用したタンパク質チロシン残基ラベル化反応","第10回バイオ関連化学シンポジウム",,,,,,2016,Sept. "Hiroyuki Nakamura,Kikuchi,Daisuke Kanoh,Shinichi Sato,Yoshinori Sakurai,Minoru Suzuki","Maleimide-Functionalized closo-Dodecaborate Albumin Conjugates: Unique Ligation at Cysteine and Lysine Residues Enables Efficient Boron Delivery to Tumor for Neutron Capture Therapy","7th European Conference on Boron Chemistry",,,,,,2016,Sept. "盛田大輝,布施新一郎,中村浩之","4?イソオキサゾリルアニオンを利用したイソオキサゾール4位の官能基化","第63回有機金属化学討論会",,,,,,2016,Sept. "Syifa Asatyas,林智広,望月誠仁,佐藤伸一,中村浩之","顕微ラマン分光イメージング法による単一細胞中のホウ素化合物の濃度分布の可視化","第13回日本中性子捕捉療法学会学術大会","第13回日本中性子捕捉療法学会学術大会",,,,,2016,Aug. "石井里武,菊地俊介,佐藤伸一,中村浩之","新規ホウ素キャリアを指向したホウ素修飾アルブミンの開発―チロシン残基修飾法の利用","第13回日本中性子捕捉療法学会学術大会",,,,,,2016,Aug. "中村浩之","化学でがんを克服できるか?","東京工業大学オープンキャンパス模擬授業",,,,,,2016,Aug. "佐藤伸一,菊地俊介,石井里武,中村浩之","新規ホウ素キャリアを指向したホウ素修飾アルブミンの開発―ホウ素クラスター共役マレイミドの利用―",,"第13回日本中性子捕捉療法学会学術大会",,,,,2016,Aug. "Taiki Morita,Shinichiro Fuse,Hiroyuki Nakamura","Preparation of 4-isoxazolyl Grignard reagent and its application for divergent synthesis of 4-substituted isoxazoles","27th International Conference on Organometallic Chemistry (ICOMC 2016)",,,,,,2016,July "S. Sato,K. Morita,H. Nakamura","Protein modification using ligand-directed Ru(bpy)3 photocatalysts,","27th International Conference on Organometallic Chemistry (ICOMC 2016)",,,,,,2016,July "中村浩之,佐藤伸一","タンパク質化学修飾法のパラダイムシフト","新学術領域「天然物ケミカルバイオロジー?分子標的と活性制御?」研究成果報告シンポジウム",,,,,,2016,July "Shunsuke Kikuchi,Daisuke Kanoh,Shinichi Sato,Yoshinori Sakurai,Minoru Suzuki,Hiroyuki Nakamura","Maleimide-Functionalized closo-Dodecaborate Albumin Conjugates (MID-AC): The Unique Ligation at both Cysteine and Lysine Residues Enabling to Efficient Boron Delivery to Tumor for Neutron Capture Therapy",,"J. CONTROL. RELEASE",,"Vol. 237","No. 10","pp. 160-167",2016,July "Shunsuke Kikuchi,Daisuke Kanoh,Shinichi Sato,Yoshinori Sakurai,Minoru Suzuki,Hiroyuki Nakamura","Maleimide-functionalized closo-dodecaborate albumin conjugates (MID-AC): Unique ligation at cysteine and lysine residues enables efficient boron delivery to tumor for neutron capture therapy",,"Journal of Controlled Release",,"Vol. 237",,"pp. 160-167",2016,July "滝沢美織,布施新一郎,中村浩之","有機D-π-A色素の構造?PDT活性相関の解明","第26回日本光線力学学会学術講演会",,,,,,2016,June "稲葉恵,峯岸秀充,佐藤伸一,布施新一郎,中村浩之","ベンゾフロピラゾール類縁体の設計、合成およびHIF-1阻害能評価","第109回有機合成シンポジウム",,,,,,2016,June "羽田野兼資,佐藤伸一,中村浩之","Ru(bpy)3触媒によるチロシン残基修飾法の分子機構の解明研究","第109回有機合成シンポジウム",,,,,,2016,June "佐藤 伸一,中村 公亮,中村 浩之","Horseradish Peroxidaseを触媒としたチロシン残基選択的なタンパク質ラベル化反応","日本ケミカルバイロジー学会第11回年会",,,,,,2016,June "中村浩之,立川将士,平松亮,川端信司,黒岩敏彦","ホウ素クラスター含有水溶性プロトポルフィリン誘導体の合成とPDT効果","第26回日本光線力学学会学術講演会",,,,,,2016,June "對馬 理彦,佐藤 伸一,中村 浩之","ビーズ固相表面における一電子酸化的なタンパク質修飾法の開発","日本ケミカルバイロジー学会第11回年会",,,,,,2016,June "布施新一郎,滝沢美織,中村浩之","新規PDT用有機色素の開発を志向したD?π?A色素の迅速合成と機能評価","第26回日本光線力学学会学術講演会",,,,,,2016,June "洪暎淳,稲井瑞穂,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","迅速な薬剤輸送に向けた複製能欠損センダイウイルス粒子への光感受性物質の封入条件の検討","第26回日本光線力学学会学術講演会",,,,,,2016,June "古山祐,稲井瑞穂,本多典広,間久直,布施新一郎,中村浩之,金田安史,粟津邦男","複製能欠損ウィルス粒子とプロトポルフィリンIV脂質を利用したPDT過程のタイムラプス撮影による作用機序の検討","第26回日本光線力学学会学術講演会",,,,,,2016,June "布施新一郎,滝沢美織,中村浩之","新規PDT用有機色素の開発を志向したD-π-A色素の迅速合成と機能評価","第26回日本光線力学学会学術講演会",,,,,,2016,June "中村浩之","Development of Boron Delivery Nano Vehicles for Neutron Capture Therapy of Cancers","The Chinese University of Hong Kong, Seminar",,,,,,2016,May "佐藤 伸一,中村 公亮,中村 浩之","活性化ヘム検出に立脚した活性酸素誘導性細胞死の評価系開発","新学術領域「ダイイングコード」平成28年班会議",,,,,,2016,May "稲葉 恵,峯岸 秀充,佐藤 伸一,中村 浩之","ベンゾフロピラゾール類縁体の設計、合成およびHIF-1阻害能評価","第20回日本がん分子標的治療学会学術集会",,,,,,2016,May "松村圭介,吉崎聡一,米谷真人,和田雄二,尾込裕平,早瀬修二,海宝龍夫,布施新一郎,田中浩士,中村浩之,高橋孝志","化学選択的ワンポット連結反応を駆使した色素増感太陽電池用DπA色素の効率的合成法の開発とその機能評価","第71回有機合成化学協会関東支部シンポジウム",,,,,,2016,May "中村浩之","Identification and Modification of Target Protein using Small Molecules with Light","The Chinese University of Hong Kong, Seminar",,,,,,2016,May "Guangzhe Li,Hiroyuki Nakamura","Synthesis of 2-Indolyltetrahydroquinolines by Zinc (II)-Catalyzed Intramolecular Hydroarylation-Redox Cross-Dehydrogenative Coupling of N-Propargylanilines with Indoles",,"Angewandte Chemie International Edition",,"Vol. 55","No. 23","pp. 6758-6761",2016,Apr. "御舩悠人,田中浩士,中村浩之,布施新一郎","マイクロフローアミド結合形成法を基盤とするフェグリマイシンの全合成","日本化学会第96春季年会",,,,,,2016,Mar. "Hiroyuki Nakamura","Development of Efficient Boron Delivery Nano Carriers for Neutron Capture Therapy","IAEA-Southern Tohoku Hospital Group Joint Workshop on BNCT",,,,,,2016,Mar. "中村浩之","外部エネルギーと局所増感型ナノデバイスによる低侵襲がん治療","LSC研究発表会",,,,,,2016,Mar. "佐藤 伸一,中村 公亮,中野 洋文,中村 浩之","チロシン残基選択的化学修飾法を用いたチロシンホスファターゼ活性スクリーニング法の開発","日本化学会第96回年会",,,,,,2016,Mar. "羽田野 兼資,佐藤 伸一,中村 浩之","光触媒を用いたTyr残基修飾反応における一電子移動範囲の解明","日本化学会第96回年会",,,,,,2016,Mar. "稲葉 恵,峯岸 秀充,布施 新一郎,中村 浩之","ベンゾフロピラゾール骨格をもつ 新規HIF-1阻害剤の開発研究","日本薬学会 第136年会",,,,,,2016,Mar. "佐藤 伸一,中村 公亮,中村 浩之,","ルミノール誘導体を用いたチロシン残基選択的な化学修飾法開発","日本化学会第96回年会",,,,,,2016,Mar. "北村 捷,京極 信輔,Manjusha Joshi,中村 浩之,岩田 耕一","ピコ秒時間分解けい光分光法で観測された単一成分脂質二重膜における不均一構造","日本化学会第96回年会",,,,,,2016,Mar. "Masao Sasai,Hiroyuki Nakamura,Nagao Sougawa,Yoshinori Sakurai,Minoru Suzuki,Chun Man Lee","Novel Hyaluronan Formulation Enhances the Efficacy of Boron Neutron Capture Therapy for Murine Mesothelioma",,"Anticancer research",,"Vol. 36","No. 3","pp. 907-911",2016,Feb. "Hyun Seung Ban,Yoshikazu Uto,Misun Won,Hiroyuki Nakamura","Hypoxia-inducible factor (HIF) inhibitors: a patent survey (2011-2015)",,"Expert opinion on therapeutic patents",,"Vol. 26","No. 3","pp. 309-322",2016,Feb. "Hiroyuki Nakamura,M Yamauchi,N Honda,H Hazama,S Tachikawa,K Awazu","Effective Photodynamic Therapy in Drug-Resistant Prostate Cancer Cells Utilizing a Non-Viral Antitumor Vector",,"Laser Therapy",,"Vol. 25","No. 1",,2016,Jan. "中村浩之","ホウ素を使ってがんに挑む 〜ホウ素創薬の最前線〜","第8回「国際的キャリア展望に向けた生命化学研究者による講演会」",,,,,,2016,Jan. "佐藤伸一,中村公亮,中村浩之","ヘムを触媒とする酸化的チロシン修飾法開発とその応用","新学術領域「酸素生物学」&「ダイイングコード」合同若手会議",,,,,,2016,Jan. "中村浩之,佐藤伸一,立川将士,布施新一郎,間久直,粟津邦男,金田安史","光感受性ポルフィリン脂質の開発とナノ粒子化による光線力学的治療効果","第4回次世代がん治療推進専門家養成プランシンポジウム",,,,,,2016,Jan. "田中健,中村浩之,岩本武明,斎藤雅一,柴田高範,長澤和夫,西林仁昭","ウェイド「有機化学」問題の解き方",,,"丸善",,,,2016,Jan. "S. Sato,H. Nakamura","Heme-Catalyzed Tyrosine Click Reaction","The 8th Takeda Science Foundation Symposium on PharmaSciences",,,,,,2016,Jan. "中村浩之","外部エネルギーと局所増感型ナノデバイスによる低侵襲がん治療","LSC研究発表会",,,,,,2016,