"S. Ogawa,Y. Asawa,M. Iiyama,A. Yoshimori,H. Nakamura,M. Oda","Regulation of binding between CD28 cytoplasmic region and SH2 domains of Grb2 and PI3K by carborane compounds for T-cell activation",,"BIOORG. MED. CHEM. LETT.",,"Vol. 78",," 129049",2022,Dec. "Hiroyuki Nakamura,Yasunobu Asawa","Comprehensive Exploration of Chemical Space Using Trisubstituted Carboranes","The 9th European Conference on Boron Chemistry",,,,,,2022,July "浅輪泰允","低分子医薬品の標的分子拡充を志向したカルボランの創薬研究",,,,,,,2022,Mar. "浅輪泰允","低分子医薬品の標的分子拡充を志向したカルボランの創薬研究",,,,,,,2022,Mar. "浅輪泰允","低分子医薬品の標的分子拡充を志向したカルボランの創薬研究",,,,,,,2022,Mar. "T. Morita,H. Murakami,Y. Asawa,H. Nakamura","Enantioselective Synthesis of Oxazaborolidines by Palladium-Catalyzed N−H/B−H Double Activation of 1,2-Azaborines",,"Angew. Chem. Int. Ed.",,"Vol. 61","Issue 7",,2022,Feb. "Y. Asawa,S. Hatsuzawa,A. Yoshimori,K. Yamada,A. Katoh,H. Kouji,H. Nakamura","Comprehensive Exploration of Chemical Space Using Trisubstituted Carboranes",,"Sci. Rep.",," 11"," 24101",,2021,Dec. "Yasunobu Asawa,Kei Nishida,Kazuki Kawai,Kiyotaka Domae,Hyun Seung Ban,Akihiro Kitazaki,Hiroya Asami,Jun-Ya Kohno,Satoshi Okada,Hiraku Tokuma,Daisuke Sakano,Shoen Kume,Masaru Tanaka,Hiroyuki Nakamura","Carborane as an Alternative Efficient Hydrophobic Tag for Protein Degradation",,"Bioconjugate Chemistry",,,,,2021,Nov. "Yasunobu Asawa,Saki Hatsuzawa,Atsushi Yoshimori,Kentaro Yamada,Akira Katoh,Hiroyuki Kouji,Hiroyuki Nakamura","Comprehensive exploration of three-dimensional chemical space by trisubstituted carboranes for discovery of bioactive molecule","The 13th AFMC International Medicinal Chemistry Symposium (AIMECS-2021)",,,,,,2021,Nov. "浅輪 泰允,中村 浩之","カルボランを基盤とした立体的分子による3次元ケミカルスペースの探索と新規PPI制御分子の創成","バイオインタラクション研究会",,,,,,2021,Nov. "浅輪泰允,中村浩之","疎水性ホウ素クラスターによる新規タンパク質分解誘導剤の開発とその機構解明","第25回がん分子標的治療学会学術大会",,,,,,2021,May "Y. Asawa,A. V. Arsent’eva,S. A. Anufriev,A. A. Anisimov,K. Yu. Suponitsky,O. A. Filippov,H. Nakamura,I. B. Sivaev","Synthesis of Bis(Carboranyl)amides 1,1’-μ-(CH2NH(O)C(CH2)n- 1,2-C2B10H11)2 (n = 0, 1) and Attempt of Synthesis of Gadolinium Bis(Dicarbollide",,"Molecules",,"Vol. 26","No. 5","pp. 1321",2021,Mar. "村上弘樹,盛田大輝,浅輪泰允,中村浩之","パラジウム触媒を用いた1,2-アザボリン類のN-H/B-H二官能基化法の開発","日本化学会第101春季年会(オンライン)",,,,,,2021,Mar. "浅輪泰允,吉森篤史,山田健太郎,小路弘行,中村浩之","カルボランを基盤とした立体的分子による3次元ケミカルスペースの探索とそのPPI制御機能評価","日本薬学会第141年会(オンライン)",,,,,,2021,Mar. "初澤早貴,浅輪泰允,吉森篤史,山田健太郎,小路弘行,真崎康博,中村浩之","PPI阻害剤を志向した三置換メタカルボランライブラリー化合物の合成とその生物活性評価","日本薬学会第141年会(オンライン)",,,,,,2021,Mar. "R. Yudi Utomo,Y. Asawa,S. Okada,A. Yoshimori,J. Bajorath,H. Nakamura","Development of curcumin-based amyloid β aggregation inhibitors for Alzheimer's disease using the SAR matrix-approach","The International Center for Chemical and Biological Sciences (ICCBS-2021)","Bioorg. Med. Chem.",," 46,"," 116357",,2021,Feb. "Takahiro Shimizu,NorihitoTakahashi,Vincent J.Huber,Yasunobu Asawa,Hiroki Ueda,Atsushi Yoshimori,Yukiko Muramatsu,Hiroyuki Seimiya,Hiroyuki Kouji,Hiroyuki Nakamura,Hiroki Oguri","Design and synthesis of 14 and 15-membered macrocyclic scaffolds exhibiting inhibitory activities of hypoxia-inducible factor 1α",,"Bioorg. Med. Chem.",,,"No. 30","pp. 115949",2021,Jan. "浅輪 泰允,吉森 篤史,BAJORATH J?rgen,中村 浩之","SAR空間の可視化によるActivity cliffの予測とその実験的検証","第10回CSJ化学フェスタ2020(オンライン)",,,,,,2020,Oct. "Rohmad Yudi Utomo,Yasunobu Asawa,Atsushi Yoshimori,Hiroyuki Nakamura","Novel Curcumin Derivatives Generated from SAR Matrix Possess as Amyloid β Inhibitors for Alzheimer?s Disease","第64回日本薬学会関東支部大会(オンライン)",,,,,,2020,Sept. "Yasunobu. Asawa,A. Yoshimori,J. Bajorath,Hiroyuki. Nakamura","Prediction of an MMP-1 Inhibitor Activity Cliff Using the SAR Matrix Approach and Its Experimental Validation",,"Sci. Rep",,,"No. 10","pp. 14710",2020,Sept. "Sei-ichi Tanuma,Takahiro Oyama,Atsushi Yoshimori,Kiyotaka Katsuragi,Yuri Shibasaki,Yasunobu Asawa,Hiroaki Yamazaki,Kosho Makino,Miwa Okazawa,Yoko Ogino,Yoshimi Sakamoto,Miyuki Nomura,Akira Sato,Hideaki Abe,Hiroyuki Nakamura,Hideyo Takahashi,Nobuhiro Tanuma,Fumiaki Uchiumi","Structural insights into the tunnel-shaped cavity of human nicotinamide phosphoribosyltransferase using a close structural set of azacyclohexane-motif inhibitors",,"Molecules",,"Vol. 25","No. 16","pp. 3633",2020,Aug. "Rohmad Yudi Utomo,Yasunobu Asawa,Shinichi Sato,Atsushi Yoshimori,Hiroyuki Nakamura","Novel Curcumin Derivatives Generated from SAR Matrix Possess as Amyloid β Inhibitors","日本薬学会第140年会",,,,,,2020,Mar. "浅輪泰允,吉森篤史,山田健太郎,邵玉潔,李廣晢,加藤明良,小路弘行,中村浩之","タンパク質の2次構造を模倣した新規カルボランPPI制御分子の設計・合成とその機能評価","日本薬学会第140年会",,,,,,2020,Mar. "Y. Asawa,K. Katsuragi,A. Sato,A. Yoshimori,S. Tanuma,H. Nakamura","Structure-based drug design of novel carborane-containing nicotinamide phosphoribosyltransferase inhibitors",,"Bioorg. Med. Chem.",,"Vol. 27","No. 13","Page 2832-2844",2019,July "Yasunobu Asawa,Kiyotaka Katsuragi,Akira Sato,Atsushi Yoshimori,Sei-ichi Tanuma,Hiroyuki Nakamura","Structure-based Drug Design of Novel Carborane-containing NAMPT Inhibitors","11th Workshop on Organic Chemistry for Junior Chemists (WOCJC-11)",,,,,,2019,June "浅輪泰允,吉森篤史,中村浩之","SBDDによる新規カルボラン含有NAMPT阻害剤の開発","第77回有機合成化学協会関東支部シンポジウム",,,,,,2019,May "浅輪泰允,中村浩之","ジカルボラン骨格を有する新規NAMPT阻害剤の理論的設計と合成、生物活性評価","日本化学会第99春季年会",,,,,,2019,Mar. "浅輪泰允,葛城粛貴,佐藤聡,吉森篤史,田沼靖一,中村浩之","疎水性ファーマコフォアとしてカルボランを導入した新規NAMPT阻害剤の開発","第36回メディシナルケミストリーシンポジウム",,,,,,2018,Nov. "浅輪泰允,葛城粛貴,佐藤聡,吉森篤史,田沼靖一,中村浩之","疎水性ファーマコフォアとしてカルボランを導入した新規NAMPT阻害剤の開発","日本化学会秋季事業 第8回CSJ化学フェスタ2018",,,,,,2018,Oct. "浅輪泰允,葛城粛貴,佐藤聡,吉森篤史,田沼靖一,中村浩之","疎水性ファーマコフォアとしてカルボランを導入した新規NAMPT阻害剤の開発","日本化学会第98春季年会",,,,,,2018,Mar. "浅輪泰允,葛城粛貴,佐藤聡,吉森篤史,田沼靖一,中村浩之","疎水性ファーマコフォアとしてカルボランを導入した新規Nampt阻害剤の開発","第35回メディシナルケミストリーシンポジウム",,,,,,2017,Oct. "S. Fuse,T. Ohuchi,Y. Asawa,S. Sato,H. Nakamura","Development of 1-Aryl-3-furanyl/Thienyl-imidazopyridine Templates for Inhibitors against Hypoxia Inducible Factor (HIF)-1 Transcriptional Activity",,"Bioorganic and Medicinal Chemistry Letters",,"Vol. 26","No. 24","page 5887-5890",2016,Nov.