@book{CTT100793624, author = {布施新一郎}, title = {マイクロフローアミド化法を基盤とする高効率ペプチド合成法の開発}, publisher = {一般社団法人触媒学会}, year = 2019, } @book{CTT100786726, author = {布施新一郎}, title = {第III部実用編 第18章 実践光化学}, publisher = {化学同人}, year = 2018, } @book{CTT100759913, author = {布施新一郎}, title = {マイクロフロー法によるペプチド合成}, publisher = {株式会社シーエムシー出版}, year = 2018, } @book{CTT100774005, author = {布施新一郎}, title = {フローマイクロリアクターによるペプチド合成}, publisher = {技術情報協会}, year = 2017, } @book{CTT100673959, author = {布施新一郎 and 高橋孝志}, title = {フロー・マイクロ合成 基礎から実際の合成・製造まで}, publisher = {化学同人}, year = 2014, } @book{CTT100658212, author = {布施新一郎 and 高橋孝志}, title = {3 ケミカルバイオロジーのための化合物群合成}, publisher = {丸善出版}, year = 2013, } @book{CTT100635511, author = {Shinichiro Fuse and Kazuhiro Machida and Takashi Takahashi}, title = {Efficient Synthesis of Natural Products Aided by Automated Synthesizers and Microreactors}, publisher = {Wiley-VCH}, year = 2012, } @book{CTT100592777, author = {高橋孝志 and 布施新一郎}, title = {ラボオートメーション技術を活用したタキソールおよび9員環エンジイン化合物の合成}, publisher = {シーエムシー出版}, year = 2009, } @book{CTT100561145, author = {布施新一郎 and 土井隆行 and 高橋孝志}, title = {タキソール}, publisher = {アイピーシー}, year = 2007, } @article{CTT100881362, author = {H. Kitamura and Y. Otake and N. Sugisawa and H. Sugisawa and T. Ida and H. Nakamura and S. Fuse and Hiroyuki Nakamura}, title = {Sequential Selective Introduction of Alcohols against Phosphorus Trichloride in a Continuous-Flow Reactor and Consideration of a Mechanism for Reduced Overreaction via the Addition of Imidazole}, journal = {Chemistry}, year = 2022, } @article{CTT100858990, author = {N. Sugisawa and H. Sugisawa and Y. Otake and R. V. Krems and H. Nakamura and S. Fuse}, title = {Rapid and Mild One-Flow Synthetic Approach to Unsymmetrical Sulfamides Guided by Bayesian Optimization}, journal = {Chemistry Methods}, year = 2021, } @article{CTT100833090, author = {Shinichiro. Fuse and Wataru Moriya and Shinichi Sato and Hiroyuki Nakamura}, title = {Investigation into the influence of an acrylic acid acceptor in organic D-π-A sensitizers against phototoxicity}, journal = {Bioorg. Med. Chem.}, year = 2020, } @article{CTT100833099, author = {Jun. Kawamura and Hiroshi. Kitamura and Yuma. Otake and Shinichiro. Fuse and Hiroyuki. Nakamura}, title = {Size-Controllable and Scalable Production of Liposomes Using a V-Shape Mixer Micro-Flow Reactor}, journal = {Org. Process Res. Dev.}, year = 2020, } @article{CTT100852985, author = {盛田 大輝 and 布施 新一郎 and 中村 浩之}, title = {Novel Photochemical Conversion of Isoxazoles to 5-Hydroxyimidazolines: Possible Protein Labeling at Lysine Residues}, journal = {Org. Lett}, year = 2020, } @article{CTT100843293, author = {Y. Otake and Y. Shibata and Y. Hayashi and S. Kawauchi and H. Nakamura and S. Fuse}, title = {N-Methylated Peptide Synthesis through Acyl N-Methylimidazolium Cation Generation Accelerated by a Brønsted Acid}, journal = {Angew. Chem. Int. Ed.}, year = 2020, } @article{CTT100810170, author = {S. Fuse and K. Suzuki and T. Kuchimaru and T. Kadonosono and H. Ueda and S. Sato and S. Kizaka-Kondoh and H. Nakamura}, title = {Design, synthesis, and evaluation of indeno[2,1-c]pyrazolones for use as inhibitors against hypoxia-inducible factor (HIF)-1 transcriptional activity}, journal = {Bioorg. Med. Chem}, year = 2019, } @article{CTT100809276, author = {S. Fuse and K. Masuda and Y. Otake and H. Nakamura}, title = {Peptide chain elongation using unprotected amino acids in a micro-flow reactor}, journal = {Chem. Eur. J}, year = 2019, } @article{CTT100793622, author = {T. Nakamura and Y. Ishikura and N. Arakawa and M. Hori and M. Sato and M. Endo and H. Masui and S. Fuse and T. Takahashi and Y. Murata and R. Murdey and A. Wakamiya}, title = {Donor–acceptor polymers containing thiazole-fused benzothiadiazole acceptor units for organic solar cells}, journal = {RSC Advances}, year = 2019, } @article{CTT100786555, author = {布施新一郎}, title = {マイクロフロー法によるペプチド合成}, journal = {月刊ファインケミカル}, year = 2019, } @article{CTT100809286, author = {N. Sugisawa and Y. Otake and H. Nakamura and S. Fuse}, title = {Single-step, rapid, and mild synthesis of β-amino acid N-carboxy anhydrides using micro-flow technologies}, journal = {Chem. Asian J.}, year = 2019, } @article{CTT100809182, author = {福原 信太郎 and S. Yugandar and 布施 新一郎 and 中村 浩之}, title = {Synthesis of 3-Hydroxy-4-substituted-picolinonitriles from 4-Propargylaminoisoxazoles via Stepwise and One-pot Isoxazolopyridine Formation/N-O Bond Cleavage Sequence}, journal = {ACS. Omega.}, year = 2018, } @article{CTT100786973, author = {S. Fuse and M. Takizawa and S. Sato and S. Okazaki and H. Nakamura}, title = {Elucidating the mode of action for thiophene-based organic D-π-A sensitizers for use in photodynamic therapy}, journal = {Bioorganic & Medicinal Chemistry}, year = 2018, } @article{CTT100758249, author = {M. Inai and N. Honda and H. Hazama and S. Akter and S. Fuse and H. Nakamura and T. Nishikawa and Y. Kaneda and K. Awazu}, title = {Photodynamic therapy with cell membrane-targeting drug delivery and direct cytotoxicity using hemagglutinating virus of Japan envelope incorporating lipidated protoporphyrin IX}, journal = {Photodiag. Photodyn. Ther.}, year = 2018, } @article{CTT100822219, author = {Y. Otake and H. Nakamura and S. Fuse}, title = {Rapid and mild synthesis of amino acid N-carboxy anhydrides using basic-to-acidic flash switching in a micro-flow reactor}, journal = {Angewandte Chemie}, year = 2018, } @article{CTT100771183, author = {Y. Otake and H. Nakamura and S. Fuse}, title = {Rapid and mild synthesis of amino acid N-carboxy anhydrides using basic-to-acidic flash switching in a micro-flow reactor}, journal = {Angewandte Chemie International Edition}, year = 2018, } @article{CTT100770717, author = {S. Fuse and K. Matsumura and M. Takizawa and S. Sato and H. Nakamura}, title = {The design, synthesis, and evaluation of organic dithienopyrrole-based D-π-A dyes for use as sensitizers in photodynamic therapy}, journal = {Bioorganic and Medicinal Chemistry Letters}, year = 2018, } @article{CTT100766630, author = {Xi Zeng and Yosuke Mizuno and Kentaro Nakamura and Shinichiro Fuse and Hiroyuki Nakamura}, title = {Compact test set for sensitivity evaluation of photoacoustic contrast agent}, journal = {Acoustical Science and Technology}, year = 2018, } @article{CTT100828134, author = {Taiki Morita and Somaraju Yugandar and Shinichiro Fuse and Nakamura}, title = {Recent progresses in the synthesis of functionalized isoxazoles}, journal = {Tetrahedron Letters}, year = 2018, } @article{CTT100828135, author = {T. Morita and S. Fukuhara and S. Fuse and H. Nakamura}, title = {Gold(I)-Catalyzed Intramolecular SEAr Reaction: Efficient Synthesis of Isoxazole-Containing Fused Heterocycles}, journal = {Organic Letters}, year = 2018, } @article{CTT100760774, author = {Shinichiro Fuse and Megumi Inaba and Shinichi Sato and Manjusha Joshi and Hiroyuki Nakamura}, title = {Synthesis of Pyrazolofuropyrazine via One-Pot SNAr Reaction and Intramolecular Direct C–H Arylation}, journal = {Synthesis}, year = 2018, } @article{CTT100759663, author = {H. Masui and M. M. Maitani and S. Fuse and A. Yamamura and Y. Ogomi and S. Hayase and T. Kaiho and H. Tanaka and Y. Wada and T. Takahashi}, title = {D–π–A dyes containing novel hydantoin anchoring groups for dye-sensitized solar cells}, journal = {Asian Journal of Organic Chemistry}, year = 2018, } @article{CTT100757543, author = {布施新一郎 and 田中浩士 and 高橋孝志 and 土井隆行}, title = {マンノペプチマイシンアグリコンの合成と立体配置訂正}, journal = {有機合成化学協会誌}, year = 2017, } @article{CTT100751759, author = {布施新一郎}, title = {チオフェン含有有機Donor-p-Acceptor色素の系統的合成と構造-機能相関解明}, journal = {有機合成化学協会誌}, year = 2017, } @article{CTT100752996, author = {S. Fuse and M. Takizawa and K. Matsumura and S. Sato and S. Okazaki and H. Nakamura}, title = {Thiophene-based, Organic D-π-A dyes as Potent Sensitizers for Photodynamic Therapy}, journal = {}, year = 2017, } @article{CTT100828137, author = {S. Fuse and T. Morita and H. Nakamura}, title = {Step-by-Step Multifunctionalization of Isoxazoles based on SEAr Reactions and C-H Direct Arylations.}, journal = {Synthesis}, year = 2017, } @article{CTT100735480, author = {H. Masui and S. Yosugi and S. Fuse and T. Takahashi}, title = {Solution-phase automated synthesis of α-amino aldehyde as a versatile intermediate.}, journal = {Beilstein Journal of Organic Chemistry}, year = 2017, } @article{CTT100734825, author = {S. Fuse and K. Matsumura and K. Johmoto and H. Uekusa and H. Tanaka and T. Hirose and T. Sunazuka and S. Ōmura and T. Takahashi}, title = {The Design, Synthesis, and Evaluation of 1,5,7-Trisubstituted-3-pyridyl-xanthones for Use as Insecticides Starting from Pyripyropene A}, journal = {Chemistry A European Journal}, year = 2016, } @article{CTT100734669, author = {S. Fuse and T. Ohuchi and Y. Asawa and S. Sato and H. Nakamura}, title = {Development of 1-Aryl-3-furanyl/Thienyl-imidazopyridine Templates for Inhibitors against Hypoxia Inducible Factor (HIF)-1 Transcriptional Activity}, journal = {Bioorganic and Medicinal Chemistry Letters}, year = 2016, } @article{CTT100734541, author = {Y. Mifune and H. Nakamura and S. Fuse}, title = {A Rapid and Clean Synthetic Approach to Cyclic Peptides via Micro-flow Peptide Chain Elongation and Photochemical Cyclization: Synthesis of a Cyclic RGD Peptide}, journal = {Organic & Biomolecular Chemistry}, year = 2016, } @article{CTT100734523, author = {Shinichiro Fuse and Yuto Mifune and Hiroyuki Nakamura and Hiroshi Tanaka}, title = {Total synthesis of feglymycin based on a linear/convergent hybrid approach using micro-flow amide bond formation}, journal = {Nature Communications}, year = 2016, } @article{CTT100828139, author = {T. Morita and S. Fuse and H. Nakamura}, title = {Generation of 4-Isoxazolyl Anion Species: Facile Access to 4-Substituted Isoxazoles}, journal = {Angewandte Chemie International Edition}, year = 2016, } @article{CTT100828138, author = {T. Morita and S. Fuse and H. Nakamura}, title = {Generation of 4-Isoxazolyl Anion Species: Facile Access to 4-Substituted Isoxazoles}, journal = {Angewandte Chemie International Edition}, year = 2016, } @article{CTT100713406, author = {N. Shiraishi and Motofumi Kumazoe and S. Fuse and Hirofumi Tachibana and H. Tanaka}, title = {The Synthesis of trans-Flavan-3-ol Gallates by Regioselective Oxidative Etherification and Their Biological Evaluation}, journal = {Chemistry a European Journal}, year = 2016, } @article{CTT100712302, author = {H. Hamagami and M. Kumazoe and Y. Yamaguchi and S. Fuse and H. Tachibana and H. Tanaka}, title = {6-Azido-6-deoxy-L-idose as a hetero-bifunctional spacer for the synthesis of azido-containing chemical probes}, journal = {Chemistry a European Journal}, year = 2016, } @article{CTT100711514, author = {Ryota Suzuki and Shinichiro Fuse and Hiroshi Tanaka}, title = {Synthesis of Asymmetrically Terminal Bifunctionlized Alkanes by Sequential Suzuki-Miyaura Coupling using B-Thexyl Boracyclanes}, journal = {Eur J Org Chem}, year = 2016, } @article{CTT100709322, author = {Taku Aoyagi and Shuichi Ohira and Shinichiro Fuse and Jun Uzawa and Yoshiki Yamaguchi and Hiroshi Tanaka}, title = {The α-Glycosidation of partially Unprotected N-Acetyl and N-Glycolyl Sialyl Donors in the Absence of a Nitrile Solvent Effect.}, journal = {Chem. Eur. J.}, year = 2016, } @article{CTT100700992, author = {Shunsuke Irie and Shinichiro Fuse and Masato M. Maitani and Yuji Wada and Yuhei Ogomi and Shuzi Hayase and Tatsuo Kaiho and Hisashi Masui and Hiroshi Tanaka and Takashi Takahashi}, title = {Synthesis of D-A’-π-A Dyes via One-Pot Three-Component Suzuki-Miyaura Coupling and an Evaluation of the Photovoltaic Properties for Use in DSSCs}, journal = {Chemistry a European Journal}, year = 2016, } @article{CTT100801748, author = {Irie, S. and Shinichiro Fuse and Maitani, M.M. and Yuji Wada and Ogomi, Y. and Hayase, S. and Kaiho, T. and Masui, H. and Tanaka, H. and Takahashi, T.}, title = {Rapid Synthesis of D-A'-π-A Dyes through a One-Pot Three-Component Suzuki-Miyaura Coupling and an Evaluation of their Photovoltaic Properties for Use in Dye-Sensitized Solar Cells}, journal = {Chemistry - A European Journal}, year = 2016, } @article{CTT100700898, author = {Shinichiro Fuse and Ryota Takahashi and Masato M. Maitani and Yuji Wada and Tatsuo Kaiho and Hiroshi Tanaka and Takashi Takahashi}, title = {Synthesis and Evaluation of Thiophene-based Organic Dyes Containing a Rigid and Non-Planar Donor with Secondary Electron Donors for Use in Dye-Sensitized Solar Cells}, journal = {European Journal of Organic Chemistry}, year = 2015, } @article{CTT100724218, author = {Shinichiro Fuse and T. Morita and Johmoto Kohei and H. Uekusa and H. Tanaka}, title = {Directing/Protecting-Group-Free Synthesis of Tetraaryl-Substituted Pyrazoles through Four Direct Arylations on an Unsubstituted Pyrazole Scaffold}, journal = {Chem.-Eur. J.}, year = 2015, } @article{CTT100698164, author = {Shinichiro Fuse and Yuma Otake and Yuto Mifune and Hiroshi Tanaka}, title = {A Facile Preparation of a-Aryl Carboxylic Acid via One-Flow Arndt–Eistert Synthesis}, journal = {Australian Journal of Chemistry}, year = 2015, } @article{CTT100695009, author = {布施新一郎}, title = {サイト選択的マイクロフロー反応を駆使する天然物合成}, journal = {化学と工業}, year = 2015, } @article{CTT100696668, author = {増井悠 and 布施新一郎 and 高橋孝志}, title = {ワンポット多成分連結反応を基盤とした機能性分子のコンビナトリアル合成}, journal = {Organometallic News}, year = 2015, } @article{CTT100696829, author = {Shinichiro Fuse and Taiki Morita and Kohei Johmoto and Hidehiro Uekusa and Hiroshi Tanaka}, title = {Directing/Protecting-Group-Free Synthesis of Tetraaryl-Substituted Pyrazoles through Four Direct Arylations on an Unsubstituted Pyrazole Scaffold}, journal = {Chemistry A Europian Journal}, year = 2015, } @article{CTT100724222, author = {T. Morita and D. Kobayashi and K. Matsumura and Johmoto Kohei and H. Uekusa and Shinichiro Fuse and T. Takahashi}, title = {Sequential SNAr Reaction/Suzuki-Miyaura Coupling/C-H Direct Arylations Approach for the Rapid Synthesis of Tetraaryl-Substituted Pyrazoles}, journal = {Chem.-Asian J.}, year = 2015, } @article{CTT100694955, author = {Taiki Morita and Daisuke Kobayashi and keisuke Matumura and Kohei Johmoto and Hidehiro Uekusa and Shinichiro Fuse and Takashi Takahashi}, title = {Sequential SNAr Reaction/Suzuki–Miyaura Coupling/C−H Direct Arylations Approach for the Rapid Synthesis of Tetraaryl-Substituted Pyrazoles}, journal = {Chemistry an Asian Journal}, year = 2015, } @article{CTT100724217, author = {Shinichiro Fuse and A. Ikebe and K. Oosumi and T. Karasawa and K. Matsumura and M. Izumikawa and Johmoto Kohei and H. Uekusa and K. Shin-Ya and T. Doi and T. Takahashi}, title = {Asymmetric Total Synthesis of ent-PyripyropeneA}, journal = {Chem.-Eur. J.}, year = 2015, } @article{CTT100693264, author = {Shinichiro Fuse and Hirotaka Sugiyama and Daisuke Kobayashi and Yusuke Iijima and Keisuke Matsumura and Hiroshi Tanaka and Takashi Takahashi}, title = {Regioselective, One-Pot, Three-Component Synthesis of 1,3,4- and 1,3,5-Triarylpyrazoles from 1- and 2-Aryl-1-alkenyl Sulfones}, journal = {European Journal of Organic Chemistry}, year = 2015, } @article{CTT100695285, author = {Hisashi Masui and Natsumi Ishizawa and Shinichiro Fuse and Takashi Takahashi}, title = {Palladium-catalyzed double carbonylation-based diversity-oriented synthesis of 3,4-dihydroisoquinoline-1-carboxamides}, journal = {Tetrahedron}, year = 2015, } @article{CTT100691828, author = {Shinichiro Fuse and Ayako Ikebe and Kazuya Oosumi and Tomoya Karasawa and Keisuke Matsumura and Miho Izumikawa and Kohei Johmoto and Hidehiro Uekusa and Kazuo Shin-ya and Takayuki Doi and Takashi Takahashi}, title = {Asymmetric Total Synthesis of ent-Pyripyropene A}, journal = {Chemistry A Europian Journal}, year = 2015, } @article{CTT100691829, author = {Keisuke Matsumura and Soichi Yoshizaki and Masato. M. Maitani and Yuji Wada and Yuhei Ogomi and Shuzi Hayase and Tatsuo Kaiho and Shinichiro Fuse and Hiroshi Tanaka and Takashi Takahashi}, title = {Rapid Synthesis of Thiophene-Based, Organic Dyes for DSSCs via a One-Pot, Four-Component Coupling Approach}, journal = {Chemistry A Europian Journal}, year = 2015, } @article{CTT100690756, author = {Shinichiro Fuse and Ryota Takahashi and Takashi Takahashi}, title = {Facile, One-Step Synthesis of 5-Substituted Thieno[3,4-c]pyrrole-4,6-dione by Palladium-Catalyzed Carbonylative Amidation}, journal = {European Journal of Organic Chemistry}, year = 2015, } @article{CTT100802240, author = {布施新一郎 and 高橋 孝志}, title = {マイクロフロー光反応·イミドイル化反応·アシル化反応を駆使する効率的な有機合成}, journal = {有機合成化学協会誌}, year = 2015, } @article{CTT100678333, author = {Shinichiro Fuse and Kentarou Nakamura and Yuto Mifune and Hironori Marubayashi and Ichiro Hijikuro and Shuichi Nojima and Hiroshi Tanaka and Takashi Takahashi}, title = {Rapid library synthesis of amphiphiles based on a dioxinone scaffold and identification of nonlamellar liquid crystals}, journal = {SYNLETT}, year = 2014, } @article{CTT100677373, author = {Shinichiro Fuse and Yuya Asai and Sakae Sugiyama and Keisuke Matsumura and Masato M. Maitani and Yuji Wada and Yuhei Ogomi and Shuzi Hayase and Tatsuo Kaiho and Takashi Takahashi}, title = {Synthesis of EDOT-containing organic dyes via one-pot, four component Suzuki Miyaura coupling and the evaluation of their photovoltaic properties}, journal = {Tetrahedron}, year = 2014, } @article{CTT100676025, author = {Shinichiro Fuse and Keisuke Matsumura and Atsushi Wakamiya and Hisashi Masui and Hiroshi Tanaka and Susumu Yoshikawa and Takashi Takahashi}, title = {Elucidation of the structure-property relationship of p-type organic semiconductors through rapid library construction via a one-pot, Suzuki-Miyaura coupling reaction}, journal = {ACS Combinatorial Science}, year = 2014, } @article{CTT100679417, author = {Yuto Mifune and Shinichiro Fuse and Hiroshi Tanaka}, title = {Synthesis of N-allyloxycarbonyl 3,5-dihydroxyphenylglycine via photochemical Wolff rearrangement/nucleophilic addition sequence in a micro-flow reactor}, journal = {Journal of Flow Chemistry}, year = 2014, } @article{CTT100675101, author = {Shinichiro Fuse and keisuke Matumura and Yuki Fujita and Hachiro Sugimoto and Takashi Takahashi}, title = {Development of dual targeting inhibitors against aggregations of amyloid-β and tau protein}, journal = {European Journal of Medicinal Chemistry}, year = 2014, } @article{CTT100676024, author = {Shinichiro Fuse and Hirotsugu Koinuma and Atsushi Kimbara and Miho Izumikawa and Yuto Mifune and Haiyin He and Kazuo Shin-ya and Takashi Takahashi and Takayuki Doi}, title = {Total synthesis and stereochemistry revision of mannopeptimycin aglycone}, journal = {Journal of the American Chemical Society}, year = 2014, } @article{CTT100674719, author = {Shinichiro Fuse and Hayato Yoshida and Kazuya Oosumi and Takashi Takahashi}, title = {Rapid and structurally diverse synthesis of multi-substituted β-keto amide derivatives based on a dioxinone scaffold}, journal = {European Journal of Organic Chemistry}, year = 2014, } @article{CTT100675775, author = {Shinichiro Fuse and Yuto Mifune and Nobutake Tanabe and Takashi Takahashi}, title = {Micro-flow Technology: Another Solution for the Site-Selective Modification of Multi-functionalized Molecules}, journal = {Synlett}, year = 2014, } @article{CTT100675092, author = {Shinichiro Fuse and Sakae Sugiyama and Masato M. Maitani and Yuji Wada and Yuhei Ogomi and Shuzi Hayase and Ryuzi Katoh and Tatsuo Kaiho and Takashi Takahashi}, title = {Elucidating the structure-property relationship of donor-pi-acceptor dyes for DSSCs through rapid library synthesis via a one-pot procedure}, journal = {Chemistry A European Journal}, year = 2014, } @article{CTT100665960, author = {Shinichiro Fuse and Yuto Mifune and Takashi Takahashi}, title = {Efficient Amide Bond Formation through a Rapid and Strong Activation of Carboxylic Acids in a Microflow Reactor}, journal = {Angewandte Chemie International Edition}, year = 2013, } @article{CTT100662494, author = {Shinichiro Fuse and Nobutake Tanabe and Akio Tannna and Yohei Konishi and Takashi Takahashi}, title = {Micro-flow synthesis and structural analysis of sterically crowded, diimine ligands with five aryl rings}, journal = {Beilstein Journal of Organic Chemistry}, year = 2013, } @article{CTT100658211, author = {Shinichiro Fuse and Kennichi Inaba and Motoki Takagi and Masahiro Tanaka and Takatsugu Hirokawa and Kohei Johmoto and Hidehiro Uekusa and Kazuo Shin-ya and Takashi Takahashi and Takayuki Doi}, title = {Design and synthesis of 2-phenyl-1,4-dioxa-spiro[4.5]deca-6,9-dien-8-ones as potential anticancer agents starting from cytotoxic spiromamakone A}, journal = {European Journal of Medicinal Chemistry}, year = 2013, } @article{CTT100641417, author = {Hisashi Masui and Shinichiro Fuse and Takashi Takahashi}, title = {A one-pot, three-component coupling approach to the synthesis of α-iminocarboxamides}, journal = {Organic Letters}, year = 2012, } @article{CTT100644620, author = {Shinichiro Fuse and Hiroaki Tago and Masato M. Maitani and Yuji Wada and Takashi Takahashi}, title = {Sequential Coupling Approach to the Synthesis of Nickel(II) Complexes with N-aryl-2-amino Phenolates}, journal = {ACS Combinatorial Science}, year = 2012, } @article{CTT100638881, author = {Shinichiro Fuse and Hayato Yoshida and Takashi Takahashi}, title = {An Iterative Approach to the Synthesis of Thiophene-based Organic Dyes}, journal = {Tetrahedron Letters}, year = 2012, } @article{CTT100639419, author = {Shinichiro Fuse and Yuto Mifune and Nobutake Tanabe and Takashi Takahashi}, title = {Continuous-flow synthesis of activated vitamin D3 and its analogues}, journal = {Organic & Biomolecular Chemistry}, year = 2012, } @article{CTT100631601, author = {Shinichiro Fuse and Nobutake Tanabe and Takashi Takahashi}, title = {Continuous in-situ generation and reaction of phosgene in a microflow system}, journal = {Chemical Communications}, year = 2011, } @article{CTT100632681, author = {Shinichiro Fuse and Hisashi Masui and Akio Tannna and Fumihiko Shimizu and Takashi Takahashi}, title = {Combinatorial Synthesis and Evaluation of α-Iminocarboxamide-Nickel (II) Catalysts for the Copolymerization of Ethylene and a Polar Monomer}, journal = {ACS Combinatorial Science}, year = 2011, } @article{CTT100625626, author = {Keiichiro Motohashi and Kennichi Inaba and Shinichiro Fuse and Takayuki Doi and Miho Izumikawa and Shams Tabrez Khan Motoki Takagi and Takashi Takahashi and Kazuo Shin-ya}, title = {JBIR-56 and JBIR-57, 2(1H)-Pyrazinones from a Marine Sponge-Derived Streptomyces sp. SpD081030SC-03}, journal = {Journal of Natural Product}, year = 2011, } @article{CTT100620985, author = {Yukinori Ohshiro and Eiji Nakajima and Yuki Goto and Shinichiro Fuse and Takashi Takahashi and Takayuki Doi and Hiroaki Suga}, title = {Ribosomal Synthesis of Backbone-Macrocyclic Peptides Containing γ-Amino Acids}, journal = {ChemBioChem}, year = 2011, } @article{CTT100625632, author = {Sakae Sugiyama and Shinichiro Fuse and Takashi Takahashi}, title = {Three-Component Coupling Approach Toward the Synthesis of a Resorcylic Acid Lactone Framework}, journal = {Tetrahedron}, year = 2011, } @article{CTT100620583, author = {Shinichiro Fuse and Kumiko Okada and Yusuke Iijima and Asami Munakata and Kazuhiro Machida and Takashi Takahashi and Motoki Takagi and Kazuo Shin-ya and Takayuki Doi}, title = {Total synthesis of spiruchostatin B aided by an automated synthesizer}, journal = {Organic & Biomolecular Chemistry}, year = 2011, } @article{CTT100616120, author = {Shinichiro Fuse and Sakae Sugiyama and Takashi Takahashi}, title = {Rapid Assembly of Resorcylic Acid Lactone Frameworks through Sequential Palladium-Catalyzed Coupling Reactions}, journal = {Chemistry an Asian Journal}, year = 2010, } @article{CTT100615602, author = {Shinichiro Fuse and Nobutake Tanabe and Masahito Yoshida and Hayato Yoshida and Takayuki Doi and Takashi Takahashi}, title = {Continuous-Flow Synthesis of Vitamin D3}, journal = {Chemical Communications}, year = 2010, } @article{CTT100612746, author = {Motoki Takagi and Keiichiro Motohashi and Aya Nagai and Miho Izumikawa and Masahiro Tanaka and Shinichiro Fuse and Takayuki Doi and Keiichiro Iwase and Atsushi Kawaguchi and Kyosuke Nagata and Takashi Takahashi and Kazuo Shin-ya}, title = {Anti-influenza virus compound from Streptomyces sp. RI18}, journal = {Organic Letters}, year = 2010, } @article{CTT100610547, author = {Takayuki Serizawa and Shigeru Miyamoto and Shinichiro Fuse and Takayuki Doi and Takashi Takahashi}, title = {Construction of the ABC Ring System of Taxanes via Stereoselective One-Pot Three-Component Coupling and Intramolecular Alkylation of a Protected Cyanohydrin Ether}, journal = {Bulletin of the Chemical Society of Japan}, year = 2010, } @article{CTT100608413, author = {Shinichiro Fuse and Hirokazu Tsukamoto and Yanqiu Yuan and Tsung-Shing Andrew Wang and Yi Zhang and Megan Bolla and Suzanne Walker and Piotr Sliz and Daniel Kahne}, title = {Functional and Structural Analysis of a Key Region of the Cell Wall Inhibitor Moenomycin.}, journal = {ACS Chemical Biology}, year = 2010, } @article{CTT100603592, author = {Jun Takahashi and Ichiro Hijikuro and Takeshi Kihara and Modachur G. Murugesh and Shinichiro Fuse and Yoshinori Tsumura and Akinori Akaike and Tetsuhiro Niidome and Takashi Takahashi and Hachiro Sugimoto}, title = {Design, synthesis and evaluation of carbamate-modified (-)-N 1-phenetylnorphysostigmine derivatives as selective butyrylcholinesterase inhibitors}, journal = {Bioorganic and Medicinal Chemistry Letters}, year = 2010, } @article{CTT100603587, author = {Jun Takahashi and Ichiro Hijikuro and Takeshi Kihara and Modachur G. Murugesh and Shinichiro Fuse and Yoshinori Tsumura and Akinori Akaike and Tetsuhiro Niidome and Takashi Takahashi and Hachiro Sugimoto}, title = {Design, synthesis and evaluation and QSAR analysis of (-)-N 1-substituted norcymserine derivatives as selective butyrylcholinesterase inhibitors}, journal = {Bioorganic and Medicinal Chemistry Letters}, year = 2010, } @article{CTT100592776, author = {Kazuhiro Machida and Yoichiro Hirose and Shinichiro Fuse and Tohru Sugawara and Takashi Takahashi}, title = {Development and Application of a Solution-Phase Automated Synthesizer,}, journal = {Chemical & Pharmaceutical Bulletin}, year = 2010, } @article{CTT100592775, author = {Yoshikazu Tanaka and Shinichiro Fuse and Hiroshi Tanaka and Takayuki Doi and Takashi Takahashi}, title = {An Efficient Synthesis of a Cyclic Ether Key Intermediate for 9-Membered Masked}, journal = {Organic Process Research & Development}, year = 2009, } @article{CTT100590060, author = {Bohdan Ostash and Emma H. Doud and Cecilie Lin and Iryna Ostash and Deborah L. Perlstein and Shinichiro Fuse and Manuel Wolpert and Daniel Kahne and Suzanne Walker}, title = {Complete Characterization of the Seventeen Step Moenomycin Biosynthetic Pathway}, journal = {Biochemistry}, year = 2009, } @article{CTT100572423, author = {Takayuki Serizawa and Yoshitaka Numajiri and Shinichiro Fuse and Takayuki Doi and Takashi Takahashi}, title = {Stereoselective one-pot three-component coupling approach towards the synthesis of the AC ring system of taxanes}, journal = {Tetrahedron Letters}, year = 2009, } @article{CTT100561006, author = {Yanqiu Yuan and Shinichiro Fuse and Bohdan Ostash and Piotr Sliz and Daniel Kahne and Suzanne Walker}, title = {Structural analysis of the contacts anchoring moenomycin to peptidoglycan glycosyltransferases and inplications for antibiotic design}, journal = {ACS Chemical Biology}, year = 2008, } @article{CTT100562747, author = {Takayuki Doi and Shinichiro Fuse and Shigeru Miyamoto and Kazuoki Nakai and Daisuke Sasuga and Takashi Takahashi}, title = {A formal total synthesis of taxol aided by an automated synthesizer}, journal = {Chemistry an Asian Journal}, year = 2006, } @article{CTT100561007, author = {Shinichiro Fuse and Malcoln Hanochi and Takashi Takahashi and Takayuki Doi}, title = {Ti(III) catalyzed radical cyclization of 6, 7-epoxygeranyl acetate}, journal = {Tetrahedron letters}, year = 2004, } @inproceedings{CTT100877627, author = {北村宙士 and 小竹佑磨 and 杉澤直斗 and 杉澤宏樹 and 井田朋智 and 中村浩之 and 布施新一郎}, title = {非対称リン酸トリエステルのマイクロフロー合成および反応機構解明}, booktitle = {}, year = 2022, } @inproceedings{CTT100877626, author = {北村宙士 and 小竹佑磨 and 杉澤直斗 and 杉澤宏樹 and 井田朋智 and 中村浩之 and 布施新一郎}, title = {非対称リン酸トリエステルのマイクロフロー合成および反応機構解明}, booktitle = {}, year = 2022, } @inproceedings{CTT100875467, author = {社本乙華 and 小室敬史 and 杉澤直斗 and 中村浩之 and 布施新一郎}, title = {マイクロフローリアクター内での環状ペプチド合成法の開発}, booktitle = {}, year = 2022, } @inproceedings{CTT100864823, author = {Taiki Morita and Shinichiro Fuse and Hiroyuki Nakamura}, title = {Photochemical conversion of isoxazoles to 5-hydroxyimidazolines}, booktitle = {}, year = 2021, } @inproceedings{CTT100864814, author = {北村宙士 and 小竹佑磨 and 杉澤直斗 and 杉澤宏樹 and 井田朋智 and 中村浩之 and 布施新一郎}, title = {マイクロフローリアクターを用いる非対称リン酸トリエステルの高速合成}, booktitle = {}, year = 2021, } @inproceedings{CTT100853232, author = {北村宙士 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフローリアクターを用いる非対称リン酸トリエステルの高速合成}, booktitle = {}, year = 2021, } @inproceedings{CTT100853231, author = {杉澤直斗 and 中村浩之 and 布施新一郎}, title = {マイクロフローリアクター内での瞬間両基質活性化を駆使したβ-アミノ酸誘導体の合成}, booktitle = {}, year = 2021, } @inproceedings{CTT100853236, author = {小室敬史 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフローリアクター内でのトリホスゲンを用いた迅速なラクタム合成法の開発}, booktitle = {}, year = 2021, } @inproceedings{CTT100836672, author = {杉澤直斗 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフローリアクター内でのpH瞬間転換と両基質同時活性化を駆使したβ-アミノ酸-N-カルボン酸無水物の合成と誘導体化}, booktitle = {}, year = 2020, } @inproceedings{CTT100823560, author = {森谷渉 and 布施新一郎 and 中村浩之}, title = {光線力学療法を志向したDπA光増感剤の構造光毒性相関の解明}, booktitle = {}, year = 2020, } @inproceedings{CTT100823562, author = {杉澤直斗 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {β-アミノ酸-N-カルボン酸無水物の迅速かつ温和なワンフロー合成}, booktitle = {}, year = 2020, } @inproceedings{CTT100804153, author = {小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之 and 布施新一郎}, title = {アシルイミダゾリウムカチオン中間体を利用するマイクロフローN-メチル化ペプチド合成法の開発とPterulamide I-IVの全合成}, booktitle = {}, year = 2019, } @inproceedings{CTT100806154, author = {森谷渉 and 布施新一郎 and 中村浩之}, title = {光線力学療法を指向したDπA光増感剤の合成と作用機序の解明}, booktitle = {}, year = 2019, } @inproceedings{CTT100804000, author = {布施新一郎}, title = {奥深いアミド化の世界へのご招待ーマイクロフロー合成法を道具としてー}, booktitle = {}, year = 2019, } @inproceedings{CTT100800122, author = {布施新一郎 and 小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之}, title = {N-メチル化ペプチドの超高効率マイクロフロー合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100802417, author = {布施新一郎}, title = {Nーメチル化ペプチドの超高効率マイクロフロー合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100800890, author = {Shinichiro Fuse}, title = {Investigation of amide bond formation based on micro-flow technologies}, booktitle = {}, year = 2019, } @inproceedings{CTT100798655, author = {杉澤直斗 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフロー合成法による瞬間混合を駆使したβ-アミノ酸-N-カルボキシ無水物の合成とその応用}, booktitle = {}, year = 2019, } @inproceedings{CTT100798810, author = {柴田裕介 and 林慶浩 and 小竹佑磨 and 中村浩之 and 布施新一郎 and 川内進}, title = {イミダゾール誘導体を触媒とするN-メチルアミド化反応機構の理論的解明}, booktitle = {}, year = 2019, } @inproceedings{CTT100822791, author = {Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor}, booktitle = {}, year = 2019, } @inproceedings{CTT100795963, author = {増田耕志郎 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {無保護アミノ酸連結を基盤とするマイクロフローペプチド鎖伸長法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100798357, author = {布施新一郎}, title = {マイクロフロー法を駆使するN-メチル化ペプチドの高効率合成}, booktitle = {}, year = 2019, } @inproceedings{CTT100795962, author = {小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之 and 布施新一郎}, title = {アシルイミダゾリウムカチオン中間体を利用するマイクロフローNーメチル化ペプチド合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100793957, author = {Shinichiro Fuse}, title = {Innovation of Peptide Synthesisbased on Micro-Flow Technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100793958, author = {布施新一郎}, title = {高速マイクロフローアミド結合形成法の開発とペプチド合成の革新}, booktitle = {}, year = 2019, } @inproceedings{CTT100792102, author = {Taiki Morita and Shinichiro Fuse and Hiroyuki Nakamura}, title = {Photochemical conversion of isoxazoles to 5-hydroxyimidazolines and its application for protein labeling}, booktitle = {}, year = 2019, } @inproceedings{CTT100792418, author = {布施新一郎}, title = {高速混合技術を基盤とする効率的有機合成手法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100792096, author = {増田 耕志郎 and 小竹 佑磨 and 中村 浩之 and 布施 新一郎}, title = {マイクロフロー法を駆使する無保護アミノ酸を用いたペプチド鎖伸長法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100792094, author = {Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {An efficient synthesis of N-methylated peptides using micro-flow technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100792085, author = {Shinichiro Fuse and Yuma Otake and Hiroyuki Nakamura}, title = {Development of Amide Bond Formation of N-Methyl Amino Acids Using Micro-Flow Technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100792099, author = {福原信太郎 and Somaraju Yugandar and 布施新一郎 and 中村浩之}, title = {イソキサゾロピリジン形成と窒素ー酸素結合開裂を経由するプロパルギルイソオキサゾールからの3ーヒドロキシー4ー置換ピコリノニトリルの一気合成}, booktitle = {}, year = 2019, } @inproceedings{CTT100789460, author = {Shinichiro Fuse}, title = {Highly Efficient Amide Bond Formation using Micro-Flow Technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100787105, author = {布施新一郎}, title = {マイクロフロー技術を駆使する高収率・省スペースかつ低コストの革新的ペプチド合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100783302, author = {Shinichiro Fuse}, title = {Highly Efficient Amide Bond Formation Using Micro-flow Technology}, booktitle = {}, year = 2018, } @inproceedings{CTT100779988, author = {Shinichiro Fuse and Yuma Otake and Hiroyuki Nakamura}, title = {Rapid and mild synthesis of amino acid N-carboxy anhydrides using basic-to-acidic flash switching in a micro-flow reactor}, booktitle = {}, year = 2018, } @inproceedings{CTT100778333, author = {伊東篤志 and 小川潤一 and 村山広大 and 花瀬勇貴 and 石垣美歌 and 布施新一郎 and 中村浩之 and 宮崎俊一 and 佐藤英俊 and 尾崎幸洋}, title = {近赤外分光法によるペプチド化学合成反応インラインモニタリング技術の開発}, booktitle = {}, year = 2018, } @inproceedings{CTT100774352, author = {布施新一郎 and 滝沢美織 and 佐藤伸一 and 岡崎茂俊 and 中村浩之}, title = {光線力学療法用有機DπA増感剤の作用機序の解明}, booktitle = {}, year = 2018, } @inproceedings{CTT100777555, author = {布施新一郎}, title = {マイクロフロー内での瞬間pH転換に基づくN-カルボキシ無水物の高効率合成}, booktitle = {}, year = 2018, } @inproceedings{CTT100778332, author = {布施新一郎}, title = {マイクロフローアミド結合形成法を駆動力とするペプチド合成の革新}, booktitle = {}, year = 2018, } @inproceedings{CTT100778684, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {マイクロフローリアクター内での瞬間pH転換に基づくNーカルボキシ無水物の高効率合成}, booktitle = {}, year = 2018, } @inproceedings{CTT100813234, author = {大石 司 and 布施新一郎 and Xi Zeng and 中村健太郎 and 中村浩之}, title = {光音響イメージングを指向した新規DπAアゾ色素の合成と機能評価}, booktitle = {}, year = 2018, } @inproceedings{CTT100813230, author = {盛田大輝 and 佐藤伸一 and 布施新一郎 and 中村浩之}, title = {イソオキサゾールの光分解を利用したイミダゾリンの合成とタンパク質ラベル化への応用}, booktitle = {}, year = 2018, } @inproceedings{CTT100773743, author = {布施新一郎}, title = {フローマイクロリアクターによるペプチド合成}, booktitle = {}, year = 2018, } @inproceedings{CTT100771191, author = {布施新一郎}, title = {高速マイクロフローアミド結合形成法の開発とペプチド合成の革新}, booktitle = {}, year = 2018, } @inproceedings{CTT100813229, author = {盛田大輝 and 福原信太郎 and 布施新一郎 and 中村浩之}, title = {金(I)触媒による分子内環化反応を用いた縮環イソオキサゾールの合成法開発}, booktitle = {}, year = 2018, } @inproceedings{CTT100771440, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {マイクロフローリアクター内での瞬間pH転換に基づくN-カルボキシ無水物の高効率合成}, booktitle = {}, year = 2018, } @inproceedings{CTT100771184, author = {盛田大輝 and 福原信太郎 and 布施新一郎 and 中村浩之}, title = {イソオキサゾールの直接修飾法の開発と新規縮環系への展開}, booktitle = {}, year = 2018, } @inproceedings{CTT100769173, author = {Atsushi Ito and Yuki Hanase and Koudai Murayama and Jun-ichi Ogawa and Shinichiro Fuse and Mika Ishigaki and Shun-ichi Miyazaki and Yukihiro Ozaki}, title = {The quantitative and non-destructive monitoring method of the amount of amide bonds in a peptide chemosynthetic model by NIR spectroscopy}, booktitle = {}, year = 2018, } @inproceedings{CTT100770112, author = {布施新一郎}, title = {高速マイクロフローアミド結合形成法の開発とペプチド合成の革新}, booktitle = {}, year = 2018, } @inproceedings{CTT100768805, author = {布施新一郎}, title = {マイクロフローリアクターを用いる高速・高効率アシル化反応}, booktitle = {}, year = 2018, } @inproceedings{CTT100768477, author = {布施新一郎}, title = {マイクロフローアミド結合形成法を駆動力とするペプチド合成の革新}, booktitle = {}, year = 2018, } @inproceedings{CTT100769407, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {マイクロフローリアクター内での瞬間pH転換に基づくN-カルボキシ無水物の高効率合成}, booktitle = {}, year = 2018, } @inproceedings{CTT100768273, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {マイクロフローリアクター内での瞬間pH転換に基づくN-カルボキシ無水物の高効率合成}, booktitle = {}, year = 2018, } @inproceedings{CTT100760761, author = {滝沢美織 and 布施新一郎 and 岡崎茂俊 and 中村浩之}, title = {光線力学療法用DπA色素の合成と作用機序解明}, booktitle = {}, year = 2018, } @inproceedings{CTT100822981, author = {K. C. S. Pradeepa and S. Fuse and H. Nakamura}, title = {AlCl3-meidated Dehydrogenative Cyclization of Diaryl-1,2-diones under Solvent-Free Conditions}, booktitle = {}, year = 2018, } @inproceedings{CTT100767978, author = {増井悠 and Santida Decharin and 布施新一郎 and 高橋孝志}, title = {α-ケトカルボン酸類縁体の簡便な合成法の開発とそのヘテロ環合成への応用}, booktitle = {}, year = 2018, } @inproceedings{CTT100767853, author = {植田大樹 and 佐藤伸一 and 布施新一郎 and 中村浩之}, title = {低酸素誘導因子(HIF-1)を標的としたα―ヘリックス模倣PPI阻害低分子の設計・合成・生物活性評価}, booktitle = {}, year = 2018, } @inproceedings{CTT100760767, author = {布施新一郎}, title = {マイクロフローアミド結合形成法を駆動力とするペプチド合成の革新}, booktitle = {}, year = 2018, } @inproceedings{CTT100760766, author = {Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor}, booktitle = {}, year = 2018, } @inproceedings{CTT100760765, author = {鈴木健介 and 布施新一郎 and 川村淳 and 佐藤伸一 and 中村浩之}, title = {低酸素誘導因子(HIF)阻害剤を志向した新規インデノピラゾロンの短段階合成と生物活性評価}, booktitle = {}, year = 2018, } @inproceedings{CTT100760764, author = {盛田大輝 and 佐藤伸一 and 布施新一郎 and 中村浩之}, title = {イソオキサゾールの光分解反応を利用したタンパク質の新規ラベル化法の開発}, booktitle = {}, year = 2018, } @inproceedings{CTT100760763, author = {福原信太郎 and 盛田大輝 and 布施新一郎 and 中村浩之}, title = {カチオン性金(I)触媒を用いたイソオキサゾール5位選択的環化反応}, booktitle = {}, year = 2018, } @inproceedings{CTT100760762, author = {小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフローリアクター内での瞬間pH転換に基づくN-カルボキシ無水物の高効率合成}, booktitle = {}, year = 2018, } @inproceedings{CTT100760760, author = {大石司 and 布施新一郎 and Xi Zeng and 中村健太郎 and 中村浩之}, title = {光音響イメージングを志向した新規DπA色素の合成と機能評価}, booktitle = {}, year = 2018, } @inproceedings{CTT100759567, author = {S. Fuse}, title = {Highly Efficient Amide Bond Formation using Micro-flow Technology}, booktitle = {}, year = 2018, } @inproceedings{CTT100758633, author = {Shinichiro Fuse}, title = {Highly Efficient Amide Bond Formation Using Micro-flow Technology}, booktitle = {}, year = 2018, } @inproceedings{CTT100758919, author = {布施新一郎}, title = {マイクロフローアミド化法を駆使するN-メチルアミノ酸の連結}, booktitle = {}, year = 2018, } @inproceedings{CTT100758678, author = {Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor}, booktitle = {}, year = 2018, } @inproceedings{CTT100757830, author = {布施新一郎}, title = {マイクロフローアミド結合形成法を駆動力とするペプチド合成の革新}, booktitle = {}, year = 2017, } @inproceedings{CTT100757411, author = {滝沢美織 and 布施新一郎 and 松村圭介 and 岡崎茂俊 and 中村浩之}, title = {光線力学療法用光増感剤の開発を志向したチオフェン含有DπA色素の合成と機能評価}, booktitle = {}, year = 2017, } @inproceedings{CTT100756736, author = {布施新一郎}, title = {マイクロフロー法を駆使するペプチドの高効率合成}, booktitle = {}, year = 2017, } @inproceedings{CTT100822976, author = {J. Kawamura and Y. Otake and S. Fuse and H. Nakamura}, title = {Preparation of boron cluster encapsulating liposomes using microflow system}, booktitle = {}, year = 2017, } @inproceedings{CTT100755338, author = {Shinichiro Fuse}, title = {Highly Efficienty Amide Bond Formation Using Micro-flow Technology}, booktitle = {}, year = 2017, } @inproceedings{CTT100757123, author = {布施新一郎}, title = {マイクロフロー法を駆使する天然物の高効率合成法の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100755026, author = {布施新一郎 and 御舩悠人 and 小竹佑磨 and 高橋孝志 and 田中浩士 and 中村浩之}, title = {迅速かつ強力なカルボン酸の活性化を基盤とするマイクロフローペプチド合成法の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100822971, author = {福原信太郎 and 盛田大輝 and 布施新一郎 and 中村浩之}, title = {カチオン性金(I)触媒を用いたイソオキサゾールの芳香族求電子置換型分子内環化反応}, booktitle = {}, year = 2017, } @inproceedings{CTT100755027, author = {布施新一郎 and 御舩悠人 and 小竹佑磨 and 高橋孝志 and 田中浩士 and 中村浩之}, title = {迅速かつ強力なカルボン酸の活性化を基盤とするマイクロフローペプチド合成法の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100753762, author = {布施新一郎}, title = {マイクロフローアミド化法を駆使するペプチドの高効率合成}, booktitle = {}, year = 2017, } @inproceedings{CTT100751945, author = {福原信太郎 and 盛田大輝 and 布施新一郎 and 中村浩之}, title = {カチオン性金(I)触媒を用いた4-(プロパルギルアミノ)イソオキサゾールの5位選択的環化反応の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100751684, author = {布施新一郎}, title = {ペプチドの低コスト生産を志向したマイクロフローアミド結合形成法の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100753208, author = {布施新一郎 and 御舩悠人 and 高橋孝志 and 田中浩士 and 中村浩之}, title = {マイクロフローアミド結合形成法を駆使するフェグリマイシンの全合成}, booktitle = {}, year = 2017, } @inproceedings{CTT100751683, author = {布施新一郎}, title = {超高速マイクロフローアミド化反応の開発とペプチド合成の革新}, booktitle = {}, year = 2017, } @inproceedings{CTT100752995, author = {布施新一郎}, title = {迅速かつ強力なカルボン酸の活性化を基盤とするマイクロフローペプチド合成法の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100749785, author = {布施新一郎}, title = {マイクロフロー法を駆使する最強のアミド化法開発を目指して}, booktitle = {}, year = 2017, } @inproceedings{CTT100749182, author = {布施新一郎}, title = {微小流路中での高速アミド化反応(秒単位)を駆使するペプチド合成}, booktitle = {}, year = 2017, } @inproceedings{CTT100747843, author = {滝沢美織 and 松村圭介 and 布施新一郎 and 岡崎茂俊 and 中村浩之}, title = {光線力学療法用有機DπA色素の作用機序解明}, booktitle = {}, year = 2017, } @inproceedings{CTT100747846, author = {布施新一郎 and 松村圭介 and 滝沢美織 and 岡崎茂俊 and 中村浩之}, title = {ジチエノピロール含有DπA色素の迅速合成と機能評価}, booktitle = {}, year = 2017, } @inproceedings{CTT100748738, author = {布施新一郎}, title = {マイクロフローアミド化法を駆使するN-メチルアミノ酸の連結}, booktitle = {}, year = 2017, } @inproceedings{CTT100747847, author = {洪瑛淳 and 稲井瑞穂 and 本多典広 and 間久直 and 布施新一郎 and 中村浩之 and 金田安史 and 粟津邦男}, title = {複製能欠損ウイルス粒子とプロトポルフィリンIX脂質を用いたPDTにおける腫瘍選択性向上のための治療条件の検討}, booktitle = {}, year = 2017, } @inproceedings{CTT100748737, author = {布施新一郎}, title = {マイクロフローアミド化法を駆使するN-メチルアミノ酸の連結}, booktitle = {}, year = 2017, } @inproceedings{CTT100745663, author = {布施新一郎}, title = {マイクロフロー法を駆使するペプチドの高効率合成}, booktitle = {}, year = 2017, } @inproceedings{CTT100744213, author = {小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフロー法を駆使するN-メチル化ペプチドの効率的合成}, booktitle = {}, year = 2017, } @inproceedings{CTT100744212, author = {Shinichiro Fuse}, title = {Highly Efficient Amide Bond Formation Using Micro‐flow Technology}, booktitle = {}, year = 2017, } @inproceedings{CTT100745540, author = {布施新一郎}, title = {マイクロフロー合成を駆使するアミド化法の開発とペプチド合成の革新}, booktitle = {}, year = 2017, } @inproceedings{CTT100743486, author = {盛田大輝 and 布施新一郎 and 中村浩之}, title = {イソオキサゾリルアニオンを利用するイソオキサゾール合成法の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100737273, author = {福原 信太郎 and 盛田 大輝 and 布施 新一郎 and 中村 浩之}, title = {カチオン性金(I)触媒を用いた4-(プロパルギルアミノ)イソオキサゾールの分子内ヒドロアリール化反応の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100737279, author = {布施 新一郎}, title = {マイクロフローペプチド合成法の開発 -奥深いアミド化の世界-}, booktitle = {}, year = 2017, } @inproceedings{CTT100737278, author = {Shinichiro Fuse}, title = {An efficient amide bond formation through rapid and strong activation of carboxylic acids in a micro-flow reactor}, booktitle = {}, year = 2017, } @inproceedings{CTT100737277, author = {布施 新一郎 and 御舩 悠人 and 中村 浩之}, title = {マイクロフローアミド化・光環化反応を駆使する高効率環状ペプチドの合成法の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100737276, author = {小竹 佑磨 and 中村 浩之 and 布施 新一郎}, title = {マイクロフロー法を駆使するN-メチル化ペプチドの革新的合成}, booktitle = {}, year = 2017, } @inproceedings{CTT100737275, author = {Keisuke Matsumura and Miori Takizawa and Shinichiro Fuse and Hiroyuki Nakamura}, title = {Synthesis and Evaluation of Organic DπA Dye Containing Dithienopyrrole as the Photosensitizer for Photodynamic Therapy}, booktitle = {}, year = 2017, } @inproceedings{CTT100737274, author = {滝沢 美織 and 松村 圭介 and 布施 新一郎 and 中村 浩之}, title = {光線力学療法のための有機DπA型色素の作用機序解明}, booktitle = {}, year = 2017, } @inproceedings{CTT100737272, author = {Taiki Morita and Shinichiro Fuse and Hiroyuki Nakamura}, title = {Generation of 4-Isoxazolyl Anion Species and Its Application for Synthesis of Multifunctionalized Isoxazoles}, booktitle = {}, year = 2017, } @inproceedings{CTT100737271, author = {石井 秀一 and 布施 新一郎 and 佐藤 伸一 and 中野 洋文 and 中村 浩之}, title = {多環性オルトキノン化合物の短段階合成法を指向したPd触媒による脱水素型環化反応の開発}, booktitle = {}, year = 2017, } @inproceedings{CTT100737270, author = {鈴木 健介 and 布施 新一郎 and 佐藤 伸一 and 中村 浩之}, title = {創薬を指向した新規インデノピラゾロンの短段階合成法の開発と生物活性評価}, booktitle = {}, year = 2017, } @inproceedings{CTT100737269, author = {稲葉 恵 and 峯岸 秀充 and 布施 新一郎 and 佐藤 伸一 and 中村 浩之}, title = {HIF阻害剤の創出を指向したベンゾフロピラゾールおよびピラゾロフロピラジンの合成法開発と生物活性評価}, booktitle = {}, year = 2017, } @inproceedings{CTT100735758, author = {布施 新一郎}, title = {マイクロフローアミド結合形成法を駆使するフェグリマイシンの全合成}, booktitle = {}, year = 2017, } @inproceedings{CTT100823014, author = {古山祐 and 稲井瑞穂 and 本多典広 and 間久直 and 布施新一郎 and 中村浩之 and 金田安史 and 粟津邦男}, title = {複製能欠損ウイルス粒子をキャリアとした新規光感受性物質による光線力学治療の作用機序の検討}, booktitle = {}, year = 2017, } @inproceedings{CTT100734629, author = {石井秀一 and 布施新一郎 and 佐藤伸一 and 中野洋文 and 中村浩之}, title = {天然物タンシノンIIAを基盤とした新規HIF-1α阻害剤の開発}, booktitle = {}, year = 2016, } @inproceedings{CTT100734630, author = {布施新一郎}, title = {マイクロフローアミド結合形成法の開発-単純なようで奥深いアミド化の世界-}, booktitle = {}, year = 2016, } @inproceedings{CTT100734508, author = {布施新一郎}, title = {強力かつ迅速なカルボン酸の活性化を基盤とするマイクロフローペプチド合成法の開発}, booktitle = {}, year = 2016, } @inproceedings{CTT100734182, author = {石井秀一 and 布施新一郎 and 中村浩之}, title = {多環性オルトキノン化合物の短段階合成を志向したPd触媒による脱水素型環化反応の開発}, booktitle = {}, year = 2016, } @inproceedings{CTT100734181, author = {小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフロー合成法を駆使するN-メチル化ペプチドの合成法開発}, booktitle = {}, year = 2016, } @inproceedings{CTT100734180, author = {布施新一郎}, title = {わずか5秒以内でアミノ酸を連結する超高速マイクロフローペプチド合成法の開発}, booktitle = {}, year = 2016, } @inproceedings{CTT100733983, author = {石井秀一 and 布施新一郎 and 佐藤伸一 and 中野洋文 and 中村浩之}, title = {天然物タンシノンIIAを基盤とした新規HIF-1α阻害剤の開発研究}, booktitle = {}, year = 2016, } @inproceedings{CTT100734360, author = {S. Fuse and Y. Mifune and H. Nakamura and H. Tanaka}, title = {Total Synthesis of Feglymycin based on a Linear/Convergent Hybrid Approach using Micro-flow Amide Bond Formation}, booktitle = {}, year = 2016, } @inproceedings{CTT100727127, author = {稲井瑞穂 and 古山祐 and 洪暎淳 and 本多典広 and 間久直 and 布施新一郎 and 中村浩之 and 金田安史 and 粟津邦男}, title = {複製能欠損ウイルス粒子を用いた光感受性薬剤の細胞内局在と腫瘍選択性の検討}, booktitle = {}, year = 2016, } @inproceedings{CTT100715879, author = {盛田大輝 and 布施新一郎 and 中村浩之}, title = {4-イソオキサゾリルアニオンを利用したイソオキサゾール4位の官能基化}, booktitle = {}, year = 2016, } @inproceedings{CTT100714388, author = {布施新一郎}, title = {フロー反応でしか実現できない高効率合成法開発を目指して}, booktitle = {}, year = 2016, } @inproceedings{CTT100720291, author = {洪暎淳 and 稲井瑞穂 and 古山祐 and 本多典広 and 間久直 and 布施新一郎 and 中村浩之 and 金田安史 and 粟津邦男}, title = {抗がん剤耐性前立腺がん細胞への迅速な薬剤輸送に向けた複製能欠損ウイルス粒子への光感受性物質の封入}, booktitle = {電気学会 光・量子デバイス研究会}, year = 2016, } @inproceedings{CTT100714978, author = {松村圭介 and 布施新一郎 and 池邊彩子 and 大角和也 and 柄澤智哉 and 田中浩士 and 廣瀬友靖 and 砂塚敏明 and 大村智 and 高橋孝志}, title = {ent-ピリピロペンAおよび構造簡略化ピリピロペン類縁体の合成と殺虫活性評価}, booktitle = {}, year = 2016, } @inproceedings{CTT100712718, author = {Shinichiro Fuse}, title = {Elucidating the structure-property relationship of donor-π-acceptor dyes for DSSCs through rapid library synthesis}, booktitle = {}, year = 2016, } @inproceedings{CTT100712717, author = {Taiki Morita and Shinichiro Fuse and Hiroyuki Nakamura}, title = {Preparation of 4-isoxazolyl Grignard reagent and its application for divergent synthesis of 4-substituted isoxazoles}, booktitle = {}, year = 2016, } @inproceedings{CTT100709162, author = {滝沢美織 and 布施新一郎 and 中村浩之}, title = {有機D-π-A色素の構造-PDT活性相関の解明}, booktitle = {}, year = 2016, } @inproceedings{CTT100822993, author = {布施新一郎 and 滝沢美織 and 中村浩之}, title = {新規PDT用有機色素の開発を志向したD-π-A色素の迅速合成と機能評価}, booktitle = {}, year = 2016, } @inproceedings{CTT100709164, author = {洪暎淳 and 稲井瑞穂 and 本多典広 and 間久直 and 布施新一郎 and 中村浩之 and 金田安史 and 粟津邦男}, title = {迅速な薬剤輸送に向けた複製能欠損センダイウイルス粒子への光感受性物質の封入条件の検討}, booktitle = {}, year = 2016, } @inproceedings{CTT100709163, author = {古山祐 and 稲井瑞穂 and 本多典広 and 間久直 and 布施新一郎 and 中村浩之 and 金田安史 and 粟津邦男}, title = {複製能欠損ウィルス粒子とプロトポルフィリンIV脂質を利用したPDT過程のタイムラプス撮影による作用機序の検討}, booktitle = {}, year = 2016, } @inproceedings{CTT100709161, author = {布施新一郎 and 滝沢美織 and 中村浩之}, title = {新規PDT用有機色素の開発を志向したD-π-A色素の迅速合成と機能評価}, booktitle = {}, year = 2016, } @inproceedings{CTT100708115, author = {布施新一郎 and 〇杉山寛崇 and 小林大輔 and 田中浩士}, title = {ワンポット[3+2]環化付加反応を基盤とした三置換ピラゾールの位置選択的合成法の開発}, booktitle = {}, year = 2016, } @inproceedings{CTT100708114, author = {稲葉恵 and 峯岸秀充 and 佐藤伸一 and 布施新一郎 and 中村浩之}, title = {ベンゾフロピラゾール類縁体の設計、合成およびHIF-1阻害能評価}, booktitle = {}, year = 2016, } @inproceedings{CTT100708308, author = {松村圭介 and 吉崎聡一 and 米谷真人 and 和田雄二 and 尾込裕平 and 早瀬修二 and 海宝龍夫 and 布施新一郎 and 田中浩士 and 中村浩之 and 高橋孝志}, title = {化学選択的ワンポット連結反応を駆使した色素増感太陽電池用DπA色素の効率的合成法の開発とその機能評価}, booktitle = {}, year = 2016, } @inproceedings{CTT100703101, author = {御舩悠人 and 田中浩士 and 中村浩之 and 布施新一郎}, title = {マイクロフローアミド結合形成法を基盤とするフェグリマイシンの全合成}, booktitle = {}, year = 2016, } @inproceedings{CTT100703100, author = {唐崎貴史 and 佐瀬祥平 and 布施新一郎 and 田中浩士 and 後藤敬}, title = {「クレードルドセレノシステイン」を活用した抗酸化酵素反応過程のモデル研究}, booktitle = {}, year = 2016, } @inproceedings{CTT100703099, author = {布施新一郎 and 池邊彩子 and 大角和也 and 柄澤智哉 and 松村圭介 and 泉川美穂 and 上本紘平 and 植草秀裕 and 新家一男 and 土井隆行 and 高橋孝志}, title = {塩化チタノセン触媒によるタンデムラジカル環化反応を駆使するピリピロペンAの不斉全合成}, booktitle = {}, year = 2016, } @inproceedings{CTT100718508, author = {稲葉 恵 and 峯岸 秀充 and 布施 新一郎 and 中村 浩之}, title = {ベンゾフロピラゾール骨格をもつ 新規HIF-1阻害剤の開発研究}, booktitle = {}, year = 2016, } @inproceedings{CTT100700897, author = {中村浩之 and 佐藤伸一 and 立川将士 and 布施新一郎 and 間久直 and 粟津邦男 and 金田安史}, title = {光感受性ポルフィリン脂質の開発とナノ粒子化による光線力学的治療効果}, booktitle = {}, year = 2016, } @inproceedings{CTT100700106, author = {Taiki Morita and Shinichiro Fuse and Keisuke Matsumura and Hirotaka Sugiyama and Daisuke Kobayashi and Hiroshi Tanaka and Hiroyuki Nakamura and Takashi Takahashi}, title = {Rapid synthesis of tri/tetraaryl-substituted pyrazoles via [3+2] cycloadditon and C-H direct arylation approaches}, booktitle = {}, year = 2015, } @inproceedings{CTT100700114, author = {Taku Aoyagi and Syuichi Ohira and Shinichiro Fuse and Hiroshi Tanaka}, title = {Partially Unprotected N-Acetyl Sialyl Donors Undergoing α-Sialylation without the Nitrile Effect}, booktitle = {}, year = 2015, } @inproceedings{CTT100700113, author = {Nana Shiraishi and Motofumi Kumazoe and Shinichiro Fuse and Hirofumi Tachibana and Hiroshi Tanaka}, title = {Synthesis of Optically Active 3-O-Acylated Catechin Analogs by Oxidative Cyclization}, booktitle = {}, year = 2015, } @inproceedings{CTT100700112, author = {Hiroki Hamagami and Yukinori Hatasa and Yoshiki Yamaguchi and Shinichiro Fuse and Takahiro Shibata and Hirofumi Tachibana and Koji Uchida and Hiroshi Tanaka}, title = {Synthesis of Sugar-Modified EGCGs by Direct C-Glycosylation and Its Application to a Chemical Biology}, booktitle = {}, year = 2015, } @inproceedings{CTT100699950, author = {布施新一郎}, title = {生物活性天然物のマイクロフロー合成:「マイクロフロー法ならでは」の手法論開発を目指して}, booktitle = {}, year = 2015, } @inproceedings{CTT100700055, author = {Shinichiro Fuse and Yuto Mifune and Nobutake Tanabe and Hiroyuki Nakamura and Takashi Takahashi}, title = {Utilization of microflow technology for the site-selective modification of multifunctionalized molecules}, booktitle = {}, year = 2015, } @inproceedings{CTT100700111, author = {Ryota Suzuki and Kou Sato and Shinichiro Fuse and Hiroshi Tanaka}, title = {One-pot Sequential Palladium-Catalyzed Cross-Coupling Reaction of Cyclic Boron Compounds}, booktitle = {}, year = 2015, } @inproceedings{CTT100698800, author = {盛田大輝 and 田中浩士 and 中村浩之 and 布施新一郎}, title = {4連続の直接アリール化による4置換ピラゾールの合成とその発光特性}, booktitle = {}, year = 2015, } @inproceedings{CTT100699088, author = {布施新一郎 and 小竹佑磨 and 御舩悠人 and 中村浩之 and 田中浩士}, title = {マイクロフローリアクター内での四連続反応によるαアリールカルボニル化合物合成法の開発}, booktitle = {}, year = 2015, } @inproceedings{CTT100697500, author = {Shinichiro Fuse}, title = {An efficient amide bond formation through the rapid and strong activation of carboxylic acids in a micro-flow reactor}, booktitle = {}, year = 2015, } @inproceedings{CTT100696265, author = {盛田大輝 and 田中浩士 and 中村浩之 and 布施新一郎}, title = {連続的C-H結合直接アリール化による4置換ピラゾールの合成}, booktitle = {}, year = 2015, } @inproceedings{CTT100696657, author = {御舩悠人 and 布施新一郎 and 田中浩士 and 中村浩之 and 高橋孝志}, title = {カルボン酸の迅速かつ強力な活性化を基盤とするマイクロフローペプチド合成法の開発とフェグリマイシンの合成研究}, booktitle = {}, year = 2015, } @inproceedings{CTT100691670, author = {布施新一郎}, title = {サイト選択的反応を駆使する多官能基性生物活性分子の合成}, booktitle = {}, year = 2015, } @inproceedings{CTT100684807, author = {布施新一郎 and 吉崎聡一 and 田中浩士}, title = {C-H結合直接アリール化を駆使するD-π-A色素合成法の開発}, booktitle = {}, year = 2015, } @inproceedings{CTT100684806, author = {入江俊介 and 布施新一郎 and 米谷真人 and 和田雄二 and 尾込裕平 and 早瀬修 二 and 海宝龍夫 and 増井悠 and 田中浩士 and 高橋孝志}, title = {DA’πA型近赤外光吸収色素の設計・合成およびその機能評価}, booktitle = {}, year = 2015, } @inproceedings{CTT100684805, author = {松村圭介 and 布施新一郎 and 藤田有紀 and 杉本八郎 and 高橋孝志}, title = {4成分ワンポット連結反応を駆使した機能性色素の合成とアミ ロイドβおよびタウタンパクの凝集阻害活性評価}, booktitle = {}, year = 2015, } @inproceedings{CTT100684812, author = {増井悠 and 布施新一郎 and 米谷真 人 and 和田雄二 and 尾込裕平 and 早瀬修二 and 高橋孝志}, title = {新規アンカー基含有色素の合成とその機能評価}, booktitle = {}, year = 2015, } @inproceedings{CTT100684815, author = {白石奈々 and 布施新一郎 and 田中浩士}, title = {酸化的環化反応を用いた光学活性3-O-アシル化カテキン類縁体の合成研究}, booktitle = {}, year = 2015, } @inproceedings{CTT100684814, author = {青栁拓 and 大平脩一 and 布施新一 郎 and 田中浩士}, title = {遊離水酸基を有するN-アセチルシアル酸供与体を用いたα選択的シアリル化反応}, booktitle = {}, year = 2015, } @inproceedings{CTT100684813, author = {布施新一郎}, title = {マイクロフロー合成法を駆使する高 選択的反応を基軸とした天然物合成}, booktitle = {}, year = 2015, } @inproceedings{CTT100684811, author = {御舩悠人 and 布施新一郎 and 田中浩 士}, title = {マイクロフロー合成法を駆使したペプチド系天然物フェグリマイシンの合成研究}, booktitle = {}, year = 2015, } @inproceedings{CTT100684810, author = {布施新一郎}, title = {マイクロフローリアクター内での四連続反応によるαアリールカルボニル化合物合成法の開発}, booktitle = {}, year = 2015, } @inproceedings{CTT100684809, author = {布施新一郎 and 盛田大輝 and 田 中浩士}, title = {4 連続のN-H およびC-H 結合直接アリール化を駆使した4置換ピラゾールの合成研究}, booktitle = {}, year = 2015, } @inproceedings{CTT100684808, author = {布施新一郎 and 杉山寛崇 and 小林大輔 and 田中浩士}, title = {ワンポット[3+2]環化付加反応を基盤とした三置換ピラゾールの位置選択的合成法の開発}, booktitle = {}, year = 2015, } @inproceedings{CTT100681145, author = {Hirotsugu Koinuma and Shinichiro Fuse and Atsushi Kimbara and Miho Izumikawa and Yuto Mifune and Haiyin He and Kazuo Shin-ya and Takashi Takahashi and Takayuki Doi}, title = {Total synthesis and stereochemistry revision of mannopeptimycin aglycone}, booktitle = {}, year = 2014, } @inproceedings{CTT100681143, author = {Shinichiro Fuse}, title = {Utilization of micro-flow technology for the site-selective modification of multi-functionalized molecules}, booktitle = {}, year = 2014, } @inproceedings{CTT100677374, author = {布施新一郎 and 入江俊介 and 杉山 栄 and 米谷真人 and 和田雄二 and 尾込裕平 and 早瀬修二 and 海宝龍夫 and 高橋孝志}, title = {ワンポットパラジウムカップリング反応によるD-π-A色素ライブラリーの迅速合成と構造-機能相関解明}, booktitle = {}, year = 2014, } @inproceedings{CTT100677872, author = {鈴木涼太 and 布施新一郎 and 田中浩士}, title = {環状ホウ素化合物の合成とその連続的クロスカップリング反応への応用}, booktitle = {}, year = 2014, } @inproceedings{CTT100677871, author = {鈴木涼太 and 布施新一郎 and 田中浩士}, title = {環状ホウ素化合物の合成とその連続的クロスカップリング反応への応用}, booktitle = {}, year = 2014, } @inproceedings{CTT100677375, author = {布施新一郎 and 盛田大輝 and 田中浩士}, title = {C-H結合直接アリール化を駆使した4置換ピラゾールの合成研究}, booktitle = {}, year = 2014, } @inproceedings{CTT100675095, author = {布施新一郎}, title = {フローでおこなうペプチドの超高速合成}, booktitle = {}, year = 2014, } @inproceedings{CTT100675094, author = {濱上大基 and 布施新一郎 and 田中浩士}, title = {C - グリコシルポリフェノール類の合成を指向した水中 C - グリコシル化反応の開発研究}, booktitle = {}, year = 2014, } @inproceedings{CTT100675093, author = {青柳拓 and 大平脩一 and 布施新一郎 and 田中浩士}, title = {4 位遊離水酸基を有する N - アセチルシアル酸供与体を用いる α 選択的シアリル化反応}, booktitle = {}, year = 2014, } @inproceedings{CTT100672535, author = {松村圭介 and 布施新一郎 and 増井悠 and 若宮淳志 and 吉川暹 and 高橋孝志 and 田中浩士}, title = {有機薄膜太陽電池用p 型有機半導体を指向したオリゴヘテロ芳香環化合物の効率的合成法の開発とその機能評価}, booktitle = {}, year = 2014, } @inproceedings{CTT100668755, author = {布施 新一郎 and 松村 圭介 and 増井 悠 and 若宮 淳志 and 吉川 暹 and 高橋 孝志 and 田中 浩士}, title = {有機薄膜太陽電池用p 型有機半導体を指向したオリゴヘテロ芳香環化合物の効率的合成法の開発とその機能評価}, booktitle = {}, year = 2014, } @inproceedings{CTT100668761, author = {増井悠 and 高橋良太 and 布施新一郎 and 若宮淳志 and 吉川暹 and 高橋孝志}, title = {高分子有機半導体のライブラリー合成とその評価}, booktitle = {}, year = 2014, } @inproceedings{CTT100668760, author = {布施 新一郎 and デーシャリン サンティダー and 増井 悠 and 高橋 孝志 and 田中 浩士}, title = {α-シアノ酢酸エステルを基盤とするアザビシクロ化合物の効率合成法の開発}, booktitle = {}, year = 2014, } @inproceedings{CTT100668759, author = {布施 新一郎 and 中村 研太郎 and 御舩 悠人 and 中村 沙季 and 高橋 孝志 and 田中 浩士}, title = {ジオキシノンを分子集積プラットフォームとして活用する非ラメラ液晶ライブラリーの構築と評価}, booktitle = {}, year = 2014, } @inproceedings{CTT100668758, author = {鈴木 涼太 and 布施 新一郎 and 田中 浩士}, title = {環状ボラン化合物に対する 連続的鈴木・宮浦クロスカップリング 反応の開発}, booktitle = {}, year = 2014, } @inproceedings{CTT100668757, author = {米谷 真人 and 尾込 裕平 and 布 施 新一郎 and 野上 顕吾 and 望月 大 and 鈴木 榮一 and 早瀬 修二 and 加藤 隆二 and 高橋 孝 志 and 和田 雄二}, title = {アナターゼ型酸化チタン表面の D-pi-A 系有機色素吸着形態による色素増感太陽電池の電子移動特性への影響}, booktitle = {}, year = 2014, } @inproceedings{CTT100668756, author = {布施 新一郎 and 盛田 大輝 and 小林 大輔 and 松村 圭介 and 高橋 孝志 and 田中 浩士}, title = {C-H 結合直接アリール化を駆使した アリール4 置換ピラゾールの合成}, booktitle = {}, year = 2014, } @inproceedings{CTT100668754, author = {布施 新一郎 and 高橋 良多 and 増井 悠 and 若宮 淳志 and 吉川 暹 and 高橋 孝志 and 田中 浩士}, title = {多様な側鎖構造の有機薄膜太陽電池用高分子p型半導体創出を指向したモノマーの迅速合成法の開発}, booktitle = {}, year = 2014, } @inproceedings{CTT100668753, author = {MIFUNE Yuto and Shinichiro and TANAKA Hiroshi and TAKAHASHI Takashi}, title = {Efficient Amide Bond Formation through a Rapid and Strong Activation of Carboxylic Acid, and its Application for a Synthesis of Feglymycin}, booktitle = {}, year = 2014, } @inproceedings{CTT100663547, author = {Shinichiro Fuse and Yuto Mifune and Takashi Takahashi}, title = {An Efficient Amide Bond Formation through the Rapid and Strong Activation of Carboxylic Acids in a Micro-flow Reactor}, booktitle = {}, year = 2013, } @inproceedings{CTT100665093, author = {Yuto Mifune and Shinichiro Fuse and Hiroshi Tanaka and Takashi Takahashi}, title = {An Efficient Micro-flow Peptide Synthesis through Rapid and Strong Activation of Carboxylic Acid}, booktitle = {}, year = 2013, } @inproceedings{CTT100665092, author = {Shinichiro Fuse}, title = {Highly Efficient Amide Bond Formation via Flash Activation of Carboxylic Acids in Microreactors}, booktitle = {}, year = 2013, } @inproceedings{CTT100663546, author = {御舩悠人 and 布施新一郎 and 田中浩士 and 高橋孝志}, title = {トリホスゲンを用いたペプチドの効率的マイクロフロー合成法の開発}, booktitle = {}, year = 2013, } @inproceedings{CTT100663545, author = {御舩悠人 and 布施新一郎 and 田中浩士 and 高橋孝志}, title = {トリホスゲンを用いたペプチドの効率的マイクロフロー合成法の開発}, booktitle = {}, year = 2013, } @inproceedings{CTT100661559, author = {布施新一郎 and 松村圭介 and 若宮淳志 and 吉川暹 and 高橋孝志}, title = {3成分ワンポット連結反応を基盤としたオリゴヘテロ芳香環化合物の効率的合成法の開発}, booktitle = {}, year = 2013, } @inproceedings{CTT100666502, author = {高橋孝志 and 布施新一郎 and 杉山 栄 and 田中恵多 and 米谷真人 and 和田雄二 and 田作優美 and 尾込裕平 and 早瀬修二 and 海宝龍夫}, title = {ワンポットパラジウムカップリング反応を駆使する太陽電池用色素ライブラリーの迅速構築と機能評価}, booktitle = {}, year = 2013, } @inproceedings{CTT100660860, author = {Hirotsugu Koinuma and Shinichiro Fuse and Atsushi Kinbara and Hiroshi Tanaka and Takashi Takahashi and Takayuki Doi}, title = {Total Synthesis of Mannopeptimycin Aglycon}, booktitle = {}, year = 2013, } @inproceedings{CTT100657772, author = {布施新一郎}, title = {自動・マイクロフロー合成法を駆使する高効率天然物合成}, booktitle = {}, year = 2013, } @inproceedings{CTT100654661, author = {布施新一郎}, title = {反応系内発生ホスゲンを用いるペプチドのマイクロフロー合成}, booktitle = {}, year = 2013, } @inproceedings{CTT100652362, author = {布施新一郎 and 小林大輔 and 飯島悠介 and 高橋孝志}, title = {連続的多成分カップリング反応を基盤とする多置換ピラゾール類の合成法の開発}, booktitle = {}, year = 2013, } @inproceedings{CTT100652360, author = {布施新一郎 and 松村圭介 and 吉川暹 and 高橋孝志}, title = {三成分ワンポットクロスカップリング反応による、オリゴヘテロ芳香環化合物ライブラリーの構築}, booktitle = {}, year = 2013, } @inproceedings{CTT100652358, author = {布施新一郎 and 御舩悠人 and 高橋孝志}, title = {反応系内で発生するホスゲンを用いたペプチドの効率的マイクロフロー合成法の開発}, booktitle = {}, year = 2013, } @inproceedings{CTT100652359, author = {増井悠 and 布施新一郎 and 高橋孝志}, title = {炭素-炭素結合形成を基盤とする環状α-イミノカルボキサミド化合物の新規合成法の開発}, booktitle = {}, year = 2013, } @inproceedings{CTT100652475, author = {布施新一郎}, title = {マイクロフロー合成法を駆使する高効率天然物合成}, booktitle = {}, year = 2013, } @inproceedings{CTT100652361, author = {布施新一郎 and 高橋良多 and 高橋孝志}, title = {連続的パラジウムカップリングを駆使するビシクロ骨格含有有機色素の合成と機能評価}, booktitle = {}, year = 2013, } @inproceedings{CTT100648439, author = {布施新一郎}, title = {フローマイクロリアクターを用いたビタミンD3類、ペプチドの効率合成}, booktitle = {}, year = 2013, } @inproceedings{CTT100646360, author = {布施新一郎 and 高橋孝志}, title = {マイクロフロー合成法を駆使する天然物合成}, booktitle = {}, year = 2012, } @inproceedings{CTT100639217, author = {布施新一郎 and 杉山栄 and 田中恵多 and 米谷真人 and 和田雄二 and 田作優美 and 尾込裕平 and 早瀬修二 and 高橋孝志}, title = {ワンポットパラジウムカップリング反応を駆使する太陽電池用色素ライブラリーの迅速構築と機能評価}, booktitle = {}, year = 2012, } @inproceedings{CTT100639071, author = {布施新一郎 and 杉山栄 and 田中恵多 and 米谷真人 and 和田雄二 and 田作優美 and 尾込裕平 and 早瀬修二 and 高橋孝志}, title = {ワンポットパラジウムカップリング反応を駆使する太陽電池用色素ライブラリーの迅速構築と機能評価}, booktitle = {}, year = 2012, } @inproceedings{CTT100634921, author = {布施新一郎 and 田邊暢偉 and 高橋孝志}, title = {マイクロリアクターを用いたカルボン酸の酸塩化物化―アミド化連続反応の制御}, booktitle = {}, year = 2012, } @inproceedings{CTT100634919, author = {布施新一郎 and 田子浩明 and 田中恵多 and 米谷真人 and 和田雄二 and 上本紘平 and 植草秀裕 and 高橋孝志}, title = {連続的鈴木-宮浦反応による近赤外光吸収色素群の合成研究}, booktitle = {}, year = 2012, } @inproceedings{CTT100634915, author = {布施新一郎 and 池邊彩子 and 柄澤智哉 and 上本紘平 and 植草秀裕 and 高橋孝志}, title = {ラジカル環化反応を用いたピリピロペンAの全合成研究}, booktitle = {}, year = 2012, } @inproceedings{CTT100634914, author = {増井悠 and 布施新一郎 and 丹那晃央 and 清水史彦 and 高橋孝志}, title = {α-イミノカルボキサミドニッケル(II)触媒のコンビナトリアル合成および重合活性評価}, booktitle = {}, year = 2012, } @inproceedings{CTT100634912, author = {布施新一郎 and 浅井裕也 and 杉山栄 and 高橋孝志}, title = {多成分ワンポットカップリング反応を基盤とする機能性色素の効率合成法開発}, booktitle = {}, year = 2012, } @inproceedings{CTT100634911, author = {杉山栄 and 布施新一郎 and 田中恵多 and 米谷真人 and 和田雄二 and 田作優美 and 尾込裕平 and 早瀬修二 and 高橋孝志}, title = {ワンポットパラジウムカップリング反応を鍵とする色素増感太陽電池用色素ライブラリーの効率的合成法の開発}, booktitle = {}, year = 2012, } @inproceedings{CTT100634492, author = {布施 新一郎}, title = {光・熱反応の空間的集積化を基盤とするビタミンD3類の効率的マイクロフロー合成法の開発}, booktitle = {}, year = 2012, } @inproceedings{CTT100634910, author = {布施新一郎 and 御舩悠人 and 田邊暢偉 and 高橋孝志}, title = {多段階連続マイクロフロー合成装置によるビタミンD類縁体の合成}, booktitle = {}, year = 2012, } @inproceedings{CTT100634908, author = {布施新一郎 and 吉田隼人 and 高橋孝志}, title = {アシルケテンをプラットフォームとする連続的四成分連結反応を駆使した1,3-ジカルボニル化合物群合成法の開発}, booktitle = {}, year = 2012, } @inproceedings{CTT100635481, author = {米谷真人 and 田中恵多 and 野上顕悟 and 高村 徹 and 望月 大 and 杉山 栄 and 布施新一郎 and 高橋 孝 and 和田雄二}, title = {酸化チタン(001)面による色素増感型太陽電池での電荷移動特性への影響}, booktitle = {}, year = 2012, } @inproceedings{CTT100635472, author = {布施 新一郎 and 田子 浩明 and 田中 恵多 and 米谷 真人 and 和田 雄二 and 上本 紘平 and 植草 秀裕 and 高橋 孝志}, title = {連続的鈴木-宮浦反応による近赤外光吸収色素群の合成研究}, booktitle = {}, year = 2012, } @inproceedings{CTT100635469, author = {田中 恵多 and 米谷 真人 and 望月 大 and 杉山 栄 and 布施 新一郎 and 高橋 孝志 and 和田 雄二}, title = {アナターゼ型酸化チタン結晶面による光誘起電荷移動への影響と色素増感型太陽電池への応用}, booktitle = {}, year = 2012, } @inproceedings{CTT100635465, author = {野上 顕悟 and 米谷 真人 and 望月 大 and 尾込 裕平 and 早瀬 修二 and 杉山 栄 and 布施 新一郎 and 高橋 孝志 and 和田 雄二}, title = {色素増感型太陽電池におけるアナターゼ型酸化チタン表面上色素吸着状態の光電変換特性への影響}, booktitle = {}, year = 2012, } @inproceedings{CTT100635462, author = {米谷 真人 and 田中 恵多 and 望月 大 and 尾込 裕平 and 早瀬 修二 and 杉山 栄 and 布施 新一郎 and 高橋 孝志 and 和田 雄二}, title = {色素増感型太陽電池における酸化チタン-色素界面の制御による高効率化}, booktitle = {}, year = 2012, } @inproceedings{CTT100634925, author = {肥沼宏次 and 布施新一郎 and 金原篤 and 土井隆行 and 高橋孝志}, title = {マンノペプチマイシンアグリコン提唱構造の全合成}, booktitle = {}, year = 2012, } @inproceedings{CTT100631805, author = {布施 新一郎}, title = {毒性ガスを利用する効率的な気液二相系連続マイクロフロー反応の開発}, booktitle = {}, year = 2011, } @inproceedings{CTT100631219, author = {布施新一郎 and 池邊彩子 and 柄澤智哉 and 高橋孝志}, title = {3価チタン試薬による触媒的ラジカル環化反応を用いたトランスデカリン骨格の構築}, booktitle = {}, year = 2011, } @inproceedings{CTT100631589, author = {Shinichiro Fuse and Yuto Mifune and Nobutake Tanabe and Masahito Yoshida and Hayato Yoshida and Takayuki Doi and Takashi Takahashi}, title = {Continuous-flow Synthesis of Vitamin D3 and Its Analogues}, booktitle = {}, year = 2011, } @inproceedings{CTT100631587, author = {Hisashi Masui and Shinichiro Fuse and Takashi Takahashi}, title = {Combinatorial Synthesis and Evaluation of a-Iminocarboxamide-Nickel(II) Catalysts for the Copolymerization of Ethylene and a Polar Monomer}, booktitle = {}, year = 2011, } @inproceedings{CTT100631521, author = {Shinichiro Fuse}, title = {Efficient Organic Synthesis Using a Continuous-flow System}, booktitle = {}, year = 2011, } @inproceedings{CTT100631591, author = {Hirotsugu Koinuma and Shinichiro Fuse and Atsushi Kinbara and Takayuki Doi and Takashi Takahashi}, title = {Synthetic Study of Mannopeptimycin Aglycon}, booktitle = {}, year = 2011, } @inproceedings{CTT100630469, author = {布施 新一郎}, title = {自動合成・フロー合成技術を活用した天然物合成}, booktitle = {}, year = 2011, } @inproceedings{CTT100630121, author = {布施新一郎 and 肥沼宏次 and 金原篤 and 土井隆行 and 高橋孝志}, title = {マンノペプチマイシンアグリコンの全合成}, booktitle = {}, year = 2011, } @inproceedings{CTT100628384, author = {布施新一郎 and 吉田隼人 and 高橋孝志}, title = {パラジウム触媒による有機ケイ 素カップリングを基盤とするπ共役オリ ゴ複素環の効率的合成法開発}, booktitle = {}, year = 2011, } @inproceedings{CTT100624956, author = {増井悠 and 布施新一郎 and 高橋孝志}, title = {連続分子内[3+2]環化付加反応を用いた高酸化スピロ骨格の構築}, booktitle = {}, year = 2011, } @inproceedings{CTT100624955, author = {田邊暢偉 and 布施新一郎 and 吉田将人 and 御舩悠人 and 吉田隼人 and 土井隆行 and 高橋孝志}, title = {マイクロリアクターを活用した光熱異性化反応によるビタミンD3及び活性型ビタミンD3の効率合成}, booktitle = {}, year = 2011, } @inproceedings{CTT100619444, author = {布施新一郎 and 吉田隼人 and 高橋孝志}, title = {パラジウム触媒による有機ケイ素カップリングを基盤とするπ共役オリゴヘテロ環の効率合成法の開発}, booktitle = {}, year = 2011, } @inproceedings{CTT100635494, author = {米谷真人 and 田中恵多 and 野上顕吾 and 高村 徹 and 望月大 and 杉山 栄 and 布施新一郎 and 高橋孝 and 和田雄二}, title = {色素増感型太陽電池における酸化チタン(001)面の光電変換特性への影響}, booktitle = {}, year = 2011, } @inproceedings{CTT100619445, author = {田邊暢偉 and 布施新一郎 and 高橋孝志}, title = {マイクロリアクターを用いた酸塩化物を経由する高効率アミド形成反応の開発}, booktitle = {}, year = 2011, } @inproceedings{CTT100619443, author = {杉山栄 and 布施新一郎 and 高橋孝志}, title = {連続的パラジウムカップリング反応を鍵とするレゾルシン酸ラクトン類の迅速合成法の開発}, booktitle = {}, year = 2011, } @inproceedings{CTT100619442, author = {増井悠 and 布施新一郎 and 高橋孝志}, title = {分子内[3+2]環化付加反応を用いたスピロ[4,4]ノナン骨格の効率的合成法の開発}, booktitle = {}, year = 2011, } @inproceedings{CTT100619441, author = {布施新一郎 and 芹沢貴之 and 宮本滋 and 土井隆行 and 高橋孝志}, title = {立体選択的ワンポット三成分連結反応を基盤とするタキサン骨格の構築}, booktitle = {}, year = 2011, } @inproceedings{CTT100619440, author = {布施新一郎 and 大角和也 and 柄澤智哉 and 高橋孝志}, title = {ピリピロペンAの合成研究}, booktitle = {}, year = 2011, } @inproceedings{CTT100619439, author = {布施新一郎 and 池邊彩子 and 柄澤智哉 and 高橋孝志}, title = {ラジカル環化反応を用いるピリピロペンAのAB環部の合成研究}, booktitle = {}, year = 2011, } @inproceedings{CTT100619438, author = {肥沼宏次 and 金原篤 and 布施新一郎 and 高橋孝志 and 土井隆行}, title = {マンノペプチマイシンアグリコンの合成研究}, booktitle = {}, year = 2011, } @inproceedings{CTT100618152, author = {布施 新一郎}, title = {一酸化炭素ナノバブルを活用するフロー系超高効率連続的カルボニル化反応の開発}, booktitle = {}, year = 2011, } @inproceedings{CTT100616662, author = {Hisashi Masui and Shinichiro Fuse and Takashi Takahashi}, title = {Combinatorial Synthesis of alpha-Iminocarboxamide Library}, booktitle = {}, year = 2010, } @inproceedings{CTT100616661, author = {Takashi Takahashi and Yoshikazu Tanaka and Shinichiro Fuse}, title = {Efficient Syntheses of 9-Membered Masked Enediyne and Taxol Aided by an Automated Synthesizer}, booktitle = {}, year = 2010, } @inproceedings{CTT100616660, author = {Shinichiro Fuse and Nobutake Tanabe and Masahito Yoshida and Hayato Yoshida and Takayuki Doi and Takashi Takahashi}, title = {Continuous-Flow Synthesis of Vitamin D3}, booktitle = {}, year = 2010, } @inproceedings{CTT100616659, author = {Shinichiro Fuse and Sakae Sugiyama and Takashi Takahashi}, title = {Rapid Assembly of Resorcylic Acid Lactone Frameworks through Sequential Palladium-Catalyzed Coupling Reactions}, booktitle = {}, year = 2010, } @inproceedings{CTT100611976, author = {土井隆行 and 吉田将人 and 布施新一郎 and 田中正洋 and 稲葉健一 and Le Anh Tuan and 飯島悠介 and 田中浩士 and 高橋孝志 and 高木基樹 and 新家一男 and 広川貴次}, title = {インシリコ連携による天然物合成を基盤とする生体制御化合物の開発}, booktitle = {}, year = 2010, } @inproceedings{CTT100611972, author = {Sakae Sugiyama and Shinichiro Fuse and Takashi TAKAHASHI}, title = {An Efficient Synthesis of Resorcylic Acid Lactones via Sequential Palladium-Catalyzed Cross-Coupling and Ring-Closing Metathesis}, booktitle = {}, year = 2010, } @inproceedings{CTT100611971, author = {増井悠 and 布施新一郎 and 高橋孝志}, title = {高機能性分子の創製を指向したα-イミノカルボキサミド類縁体群の迅速合成法の確立}, booktitle = {}, year = 2010, } @inproceedings{CTT100611975, author = {Shinichiro Fuse and Yoshikazu Tanaka and Takashi Takahashi}, title = {Efficient Syntheses of Taxol and 9-Membered Masked Enediyne Using Automated Synthesizers}, booktitle = {}, year = 2010, } @inproceedings{CTT100611974, author = {Shinichiro Fuse}, title = {Efficient Syntheses of Taxol and 9-Membered Masked Enediyne Using Automated Synthesizers}, booktitle = {}, year = 2010, } @inproceedings{CTT100611973, author = {Nobutake Tanabe and Shinichiro Fuse and Hayato Yoshida and Takahashi Takashi}, title = {Flow Synthesis of Vitamin D3 Using a Microreactor}, booktitle = {}, year = 2010, } @inproceedings{CTT100608209, author = {増井悠 and 布施新一郎 and 高橋孝志}, title = {ライブラリー構築を指向したα-イミノカルボキサミドの効率的合成}, booktitle = {}, year = 2010, } @inproceedings{CTT100607729, author = {杉山栄 and 布施新一郎 and 高橋孝志}, title = {連続的パラジウムカップリング反応-閉環メタセシス反応を鍵とするレゾルシン酸ラクトンライブラリーの構築}, booktitle = {}, year = 2010, } @inproceedings{CTT100605278, author = {布施新一郎 and 田邊暢偉 and 土井隆行 and 吉田将人 and 高橋孝志}, title = {マイクロリアクターを活用した光熱異性化反応による高効率的なビタミンD3の合成}, booktitle = {}, year = 2010, } @inproceedings{CTT100605277, author = {布施新一郎 and 大角和也 and 柄澤智哉 and 高橋孝志}, title = {ラジカル環化反応を利用したピリピロペンAの合成研究}, booktitle = {}, year = 2010, } @inproceedings{CTT100603595, author = {布施新一郎 and 増井悠 and 高橋孝志}, title = {炭素-炭素結合形成反応を用いたα-イミノカルボキサミド類縁体群の合成}, booktitle = {}, year = 2010, } @inproceedings{CTT100603596, author = {田中義一 and 布施新一郎 and 川内進 and 田中浩士 and 土井隆行 and 高橋孝志}, title = {光照射によりビラジカル発生が誘起される環状エンジイン化合物の合成}, booktitle = {}, year = 2010, } @inproceedings{CTT100603594, author = {布施新一郎 and 岡田久美子 and 高橋孝志}, title = {固相合成法を利用したヒメグルシン類の合成研究}, booktitle = {}, year = 2010, } @inproceedings{CTT100592412, author = {Shinichiro Fuse and Nobutake Tanabe and Masahito Yoshida and Takayuki Doi and Takashi Takahashi}, title = {Synthesis of VitaminD3 by Photo and Thermal Isomerization Using Microreactor}, booktitle = {}, year = 2009, } @inproceedings{CTT100611977, author = {土井隆行 and 吉田将人 and 布施新一郎 and 飯島悠介 and 田中浩士 and 高橋孝志 and 広川貴次}, title = {インシリコ連携による天然物合成を基盤とする生体制御化合物の開発}, booktitle = {}, year = 2009, } @inproceedings{CTT100590218, author = {Nobutake Tanabe and Shinichiro Fuse and Masahito Yoshida and Takayuki Doi and Takashi Takahashi}, title = {Microflow Synthesis of Vitamin D3 by Photo and Thermal Isomerization}, booktitle = {}, year = 2009, } @inproceedings{CTT100590219, author = {Sakae Sugiyama and Shinichiro Fuse and Takashi Takahashi}, title = {An Efficient Synthesis of Resorcylic Acid Lactones via Sequential Palladium-Catalyzed Cross-Coupling and Ring-Closing Metathesis}, booktitle = {}, year = 2009, } @inproceedings{CTT100590061, author = {杉山栄 and 布施新一郎 and 高橋孝志}, title = {連続的パラジウムカップリング反応‐閉環メタセシス反応を鍵とするレゾルシン酸ラクト}, booktitle = {}, year = 2009, } @inproceedings{CTT100608208, author = {布施新一郎 and 柄澤智哉 and 大角和也 and 土井隆行 and 高橋孝志}, title = {N置換型BeauveriolideIII類縁体群の固相合成法の開発}, booktitle = {}, year = 2009, } @inproceedings{CTT100577094, author = {布施新一郎 and 杉山 栄 and 高橋孝志}, title = {3成分連結法を基盤とするレゾルシン酸ラクトン類の効率的合成法の開発}, booktitle = {}, year = 2009, } @inproceedings{CTT100577110, author = {布施新一郎 and 岡田久美子 and 宗像麻未 and 飯島悠介 and 土井隆行 and 高橋孝志}, title = {ラボオートメーション技術を利用したスピルコスタチンB の全合成}, booktitle = {}, year = 2009, } @inproceedings{CTT100577106, author = {布施新一郎 and 増井悠 and 高橋孝志}, title = {ライブラリーの構築を指向したα‐イミノカルボキサミドの合成}, booktitle = {}, year = 2009, } @inproceedings{CTT100577107, author = {布施新一郎 and 田邊暢偉 and 高橋孝志}, title = {マイクロリアクターを用いたカルボン酸の酸塩化物化―アミド化連続反応の制御}, booktitle = {}, year = 2009, } @inproceedings{CTT100577109, author = {田中義一 and 布施新一郎 and 田中浩士 and 土井隆行 and 高橋孝志}, title = {DNA 塩基配列認識部位を有する9 員環エンジイン化合物の合成研究}, booktitle = {}, year = 2009, } @inproceedings{CTT100577108, author = {布施新一郎 and 柄澤智哉 and 土井隆行 and 高橋孝志}, title = {ラジカル環化反応を利用したピリピロペンA の合成研究}, booktitle = {}, year = 2009, } @inproceedings{CTT100577111, author = {布施新一郎 and 肥沼宏次 and 金原篤 and 高橋孝志 and 土井隆行}, title = {マンノペプチマイシンアグリコンの合成研究}, booktitle = {}, year = 2009, } @inproceedings{CTT100577095, author = {Takayuki Doi and Masahito Yoshida and Nobutake Tanabe and Shinichiro Fuse and Takashi Takahashi}, title = {Synthesis of Vitamin D3 by Photo and Thermal Isomerization Using a Microreactor}, booktitle = {}, year = 2008, } @inproceedings{CTT100611978, author = {高橋孝志 and 田中浩士 and 布施新一郎 and 土井隆行 and 吉田将人}, title = {天然物を基盤とするコンビナトリアル合成とラボラトリーオートメーションの活用}, booktitle = {}, year = 2008, } @inproceedings{CTT100584140, author = {田中義一 and 布施新一郎 and 田中浩士 and 土井 隆行 and 高橋 孝志}, title = {ラボオートメーション技術を利用する9員環エンジイン分子の合成研究}, booktitle = {}, year = 2008, } @inproceedings{CTT100608207, author = {土井 隆行 and 肥沼 宏次 and 金原 篤 and 布施 新一郎 and 高橋 孝志}, title = {Mannopeptimycin aglyconの全合成研究}, booktitle = {}, year = 2008, } @inproceedings{CTT100577078, author = {布施新一郎 and 土井隆行 and 飯島悠介 and 宗像麻未 and 高橋孝志 and Ganesan A and 新家一男 and 千々和修平 and 家村俊一郎 and 夏目徹}, title = {スピルコスタチンAの全合成と結合タンパク質ネットワーク解析}, booktitle = {}, year = 2008, } @inproceedings{CTT100577100, author = {Shinichiro Fuse}, title = {Synthesis and Evaluation of Moenomycin Analogs}, booktitle = {}, year = 2007, } @inproceedings{CTT100577103, author = {布施新一郎}, title = {減生、再構築法を基盤とする抗生物質Moenomycin Aの構造活性相関研究}, booktitle = {}, year = 2007, } @inproceedings{CTT100577097, author = {Shinichiro Fuse and Yi Zhang and Masaatsu Adachi and Daniel Kahne}, title = {Dissecting the structural requirements for moenomycin A activity using semi-synthetic analogues with modified phosphoglycerate lipids}, booktitle = {}, year = 2007, } @inproceedings{CTT100577092, author = {Takashi Takahashi and Shinichiro Fuse and Takayuki Doi.}, title = {Total synthesis of taxol utilizing an automated synthesizer, ChemKonzert}, booktitle = {}, year = 2005, } @inproceedings{CTT100577091, author = {Shinichiro Fuse and 宮本滋 and 中井一宙 and 廣瀬洋一郎 and 流石大輔 and Takashi TAKAHASHI}, title = {A Total Synthesis of (±)-Baccatin III utilizing Automated Synthesizers}, booktitle = {}, year = 2005, } @inproceedings{CTT100577105, author = {布施新一郎}, title = {ラボオートメーションの導入による有機合成の効率化を指向したタキソールの全合成研究}, booktitle = {}, year = 2005, } @inproceedings{CTT100577090, author = {布施新一郎 and 宮本滋 and 中井一宙 and 土井隆行 and 高橋孝志}, title = {LA(ラボオートメーション)導入による有機合成の効率化を指向したタキソールの全合成研究}, booktitle = {}, year = 2005, } @inproceedings{CTT100577089, author = {布施 新一郎 and 土井 隆行 and 高橋 孝志}, title = {自動合成ロボットを活用したタキソールの効率的な全合成研究}, booktitle = {}, year = 2005, } @inproceedings{CTT100577098, author = {布施新一郎 and 宮本滋 and 中井一宙 and 土井隆行 and 高橋孝志}, title = {LA(ラボオートメーション)導入による有機合成の効率化を指向したタキソールの全合成研究}, booktitle = {}, year = 2004, } @inproceedings{CTT100577088, author = {布施新一郎 and 宮本滋 and 中井一宙 and 土井隆行 and 高橋孝志}, title = {LA(ラボオートメーション)導入による有機合成の効率化を指向したタキソールの全合成研究}, booktitle = {}, year = 2004, } @inproceedings{CTT100577096, author = {Shinichiro Fuse and Shigeru Miyamoto and Kazuoki Nakai and Takayuki Doi and Takashi Takahashi}, title = {Utilization of an Automated Synthesizer Toward an Efficient Synthesis of Natural Product The Application for the Total Synthesis of Taxol}, booktitle = {}, year = 2004, } @inproceedings{CTT100577099, author = {Shinichiro Fuse and Shigeru Miyamoto and Kazuoki Nakai and Takayuki Doi and Takashi Takahashi}, title = {Utilization of an Automated Synthesizer Toward an Efficient Synthesis of Natural Product The Application for the Total Synthesis of Taxol}, booktitle = {}, year = 2004, } @inproceedings{CTT100577087, author = {布施 新一郎 and 宮本 茂 and 土井 隆行 and 高橋 孝志}, title = {LA(ラボオートメーション)導入による天然物合成の効率化を指向したタキソール合成研究 (東工大院理工)}, booktitle = {}, year = 2004, } @inproceedings{CTT100577086, author = {布施新一郎 and 中井一宙 and 宮本滋 and 土井隆行 and 高橋孝志}, title = {LA(ラボオートメーション)導入による天然物合成の効率化を指向したタキソール合成研究}, booktitle = {}, year = 2003, } @inproceedings{CTT100577085, author = {土井隆行 and 羽後丸訓 and 布施新一郎 and 中井一宙 and 高橋孝志}, title = {触媒量のチタノセンクロリド(III)によるエポキシアルケンのラジカル環化反応に関する研究}, booktitle = {}, year = 2003, } @inproceedings{CTT100577084, author = {Takashi Takahashi and Shinichiro Fuse and Kazuoki Nakai and Takayuki Doi}, title = {Utilization of an Automated Synthesizer Toward an Efficient Synthesis of the C-ring of Taxol}, booktitle = {}, year = 2002, } @inproceedings{CTT100577083, author = {高橋孝志 and 布施新一郎 and 中井一宙 and 土井隆行}, title = {ラボラトリーオートメーションの導入によるタキソールC環部合成の効率化}, booktitle = {}, year = 2001, } @inproceedings{CTT100577080, author = {宮本滋 and 中井一宙 and 布施新一郎 and 土井隆行 and 高橋孝志}, title = {分子内アルキル化を用いるタキソールABC環骨格の合成研究}, booktitle = {}, year = 2001, } @inproceedings{CTT100577082, author = {高橋孝志 and 布施新一郎 and 中井一宙 and 土井隆行}, title = {自動合成ロボットを活用する天然物合成の効率化 -タキソールC環の自動合成研究-}, booktitle = {}, year = 2001, } @misc{CTT100785003, author = {Shinichiro Fuse and Yuma Otake and Hiroyuki Nakamura}, title = {Peptide Synthesis Utilizing Micro‐flow Technology}, year = 2018, } @misc{CTT100755068, author = {Shinichiro Fuse and Yuma Otake and Hiroyuki Nakamura}, title = {Integrated Micro-Flow Synthesis Based on Photochemical Wolff Rearrangement}, year = 2017, } @misc{CTT100673491, author = {布施新一郎 and 高橋孝志}, title = {マイクロフローリアクターを駆使したペプチドの迅速合成}, year = 2014, } @misc{CTT100633627, author = {布施 新一郎}, title = {マイクロフロー合成法を駆使する有機合成}, year = 2012, } @misc{CTT100617869, author = {布施 新一郎 and 高橋孝志}, title = {天然物を基盤としたケミカルバイオロジー研究を加速させる合成工学的新技術}, year = 2011, } @misc{CTT100561141, author = {高橋孝志 and 布施新一郎}, title = {合成ロボットを使った天然物合成}, year = 2004, } @misc{CTT100572424, author = {布施 新一郎}, title = {ラボオートメーションの導入による有機合成の効率化を指向したタキソールの合成研究}, year = 2005, } @misc{CTT100595000, author = {Shinichiro Fuse}, title = {ラボオートメーションの導入による有機合成の効率化を指向したタキソールの合成研究}, year = 2005, } @misc{CTT100601945, author = {布施新一郎}, title = {ラボオートメーションの導入による有機合成の効率化を指向したタキソールの合成研究}, year = 2005, } @misc{CTT100596313, author = {Shinichiro Fuse}, title = {ラボオートメーション(LA)導入による有機合成の効率化を指向したタキソール合成研究}, year = 2002, } @misc{CTT100884601, author = {布施新一郎 and 北村宙士 and 小竹佑磨 and 中村浩之}, title = {非対称型リン酸トリエステルの製造方法、対称型リン酸トリエステルの製造方法、リン酸エステルの製造方法、及び、有機リン化合物の製造方法}, howpublished = {公開特許}, year = 2022, month = {}, note = {PCT/JP2022/004557(2022/02/04), WO 2022/185843(2022/09/09)} } @misc{CTT100868492, author = {布施新一郎 and 増田耕志郎 and 小竹佑磨 and 中村浩之}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2021-501811(2020/02/03), 再表2020/175023(2021/12/16)} } @misc{CTT100866375, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-563042(2019/12/11), 再表2020/137545(2021/11/04)} } @misc{CTT100845916, author = {布施新一郎 and 中村浩之 and 小竹佑磨 and 宮崎 俊一 and 伊東 篤志 and 小川 潤一}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-525411(2019/05/28), 再表2019/239880(2021/02/12)} } @misc{CTT100845903, author = {布施新一郎 and 中村浩之 and 小竹佑磨 and 宮崎 俊一 and 伊東 篤志 and 小川 潤一}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-525410(2019/05/28), 再表2019/239879(2021/02/12)} } @misc{CTT100826091, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {フローリアクターを用いるN-カルボキシ無水物の合成方法}, howpublished = {登録特許}, year = 2023, month = {}, note = {特願2019-094952(2019/05/21), 特開2020-011948(2020/01/23), 特許第7362055号(2023/10/06)} } @misc{CTT100746386, author = {布施新一郎 and 和田雄二 and 米谷真人 and 高橋 孝志 and 増井 悠  and 海宝 龍夫  and 早瀬 修二  and 尾込 裕平}, title = {色素増感型光電変換素子用のヘテロ環リンカー基を有する完全有機色素化合物、およびそれを用いた光電変換素子}, howpublished = {登録特許}, year = 2019, month = {}, note = {特願2015-201952(2015/10/13), 特開2017-076648(2017/04/20), 特許第6534331号(2019/06/07)} } @misc{CTT100734427, author = {布施新一郎 and 和田雄二 and 米谷真人 and 高橋 孝志 and 増井 悠 and 海宝 龍夫 and 早瀬 修二 and 尾込 裕平}, title = {光電変換用増感色素、その製造方法および該色素を用いた光電変換素子}, howpublished = {公開特許}, year = 2016, month = {}, note = {特願2015-035123(2015/02/25), 特開2016-157837(2016/09/01)} } @misc{CTT100698843, author = {高橋孝志 and 布施新一郎 and 和田雄二 and 米谷真人 and 海会 龍夫 and 早瀬 修二  and 伊牟田 聡}, title = {色素増感型光電変換素子用の非平面型構造を有する完全有機色素化合物、およびそれを用いた光電変換素子}, howpublished = {公開特許}, year = 2015, month = {}, note = {特願2014-502382(2013/02/28), 特開(再表)2013/129605(2015/07/30)} } @misc{CTT100666214, author = {高橋孝志 and 布施新一郎 and 和田雄二 and 米谷真人 and 海宝 龍夫 and 早瀬 修二 and 伊牟田 聡}, title = {色素増感型光電変換素子用の高活性完全有機色素化合物、およびそれを用いた光電変換素子}, howpublished = {公開特許}, year = 2013, month = {}, note = {特願2012-045914(2012/03/01), 特開2013-181108(2013/09/12)} } @misc{CTT100660973, author = {高橋孝志 and 土井隆行 and 布施新一郎 and 新家 一男 and 高木 基樹 and 広川 貴次 and 稲葉 健一 and 田中 正洋}, title = {TDP1阻害活性を有する環状エノン化合物}, howpublished = {公開特許}, year = 2013, month = {}, note = {特願2011-270875(2011/12/12), 特開2013-121930(2013/06/20)} } @phdthesis{CTT100572424, author = {布施 新一郎}, title = {ラボオートメーションの導入による有機合成の効率化を指向したタキソールの合成研究}, school = {}, year = 2005, } @phdthesis{CTT100595000, author = {Shinichiro Fuse}, title = {ラボオートメーションの導入による有機合成の効率化を指向したタキソールの合成研究}, school = {東京工業大学}, year = 2005, } @phdthesis{CTT100601945, author = {布施新一郎}, title = {ラボオートメーションの導入による有機合成の効率化を指向したタキソールの合成研究}, school = {東京工業大学}, year = 2005, } @mastersthesis{CTT100596313, author = {Shinichiro Fuse}, title = {ラボオートメーション(LA)導入による有機合成の効率化を指向したタキソール合成研究}, school = {東京工業大学}, year = 2002, }