@article{CTT100935224, author = {Y. Honda and Haruna Haraguchi and T. Tsuda and Rui Ko and K. Muguruma and H. Guo and T. Nomoto and Y. Miura and N. Nishiyama}, title = {Metal-phenolic network-based polymeric nanocarriers facilitating antibody cytoplasmic delivery and anti-tumor effects to orthotopic breast tumors}, journal = {J. Control. Release}, year = 2025, } @article{CTT100917900, author = {Imai Kyosuke and Kyohei Muguruma and Ambara R. Pradipta and Katsunori Tanaka}, title = {In vivo synthetic anticancer approach by resourcing mouse blood albumin as a biocompatible artificial metalloenzyme}, journal = {Angewandte Chemie International Edition}, year = 2024, } @article{CTT100911561, author = {Minagi Mukaiyama and Chihiro Uchiyama and Akane Fukuda and Yoshiki Nakazawa and Yuka Kuramochi and Yudai Shibata and Sho Konno and Kyohei Muguruma and Naohiro Matsugaki and Tomo Asari and Kazuyoshi Ogawa and Akihiro Taguchi and Kentaro Takayama and Atsuhiko Taniguchi and Yoko Nagumo and Toshiya Senda and Yoshio Hayashi and Takeo Usui}, title = {X-Ray Conformation and Structure–Activity Relationships of MA026, a Reversible Tight Junction Opener}, journal = {Journal of Medicinal Chemistry}, year = 2023, } @article{CTT100911562, author = {Yudai Ode and Ambara R. Pradipta and Peni Ahmadi and Akihiro Ishiwata and Akiko Nakamura and Yasuko Egawa and Yuriko Kusakari and Kyohei Muguruma and Yang Wang and Xiaojie Yin and Nozomi Sato and Hiromitsu Haba and Katsunori Tanaka}, title = {Therapeutic efficacy of 211At-radiolabeled 2,6-diisopropylphenyl azide in mouse models of human lung cancer}, journal = {Chemical Science}, year = 2023, } @article{CTT100911563, author = {Tsung-Che Chang and Igor Nasibullin and Kyohei Muguruma and Yuriko Kusakari and Taiji Shimoda and Katsunori Tanaka}, title = {Evaluation of acute toxicity of cancer-targeting albumin-based artificial metalloenzymes}, journal = {Bioorganic & Medicinal Chemistry}, year = 2022, } @article{CTT100911564, author = {Ahmadi P and Muguruma K and Chang TC and Tamura S and Tsubokura K and Egawa Y and Suzuki T and Dohmae N and Nakao Y and Tanaka K}, title = {In vivo metal-catalyzed SeCT therapy by a proapoptotic peptide.}, journal = {Chemical science}, year = 2021, } @article{CTT100911565, author = {Pradipta AR and Ahmadi P and Terashima K and Muguruma K and Fujii M and Ichino T and Maeda S and Tanaka K}, title = {Targeted 1,3-dipolar cycloaddition with acrolein for cancer prodrug activation.}, journal = {Chemical science}, year = 2021, } @article{CTT100911566, author = {Muguruma K and Osawa R and Fukuda A and Ishikawa N and Fujita K and Taguchi A and Takayama K and Taniguchi A and Ito Y and Hayashi Y}, title = {Development of a High-Affinity Antibody-Binding Peptide for Site-Specific Modification.}, journal = {ChemMedChem}, year = 2021, } @article{CTT100911567, author = {Sasaki K and Muguruma K and Osawa R and Fukuda A and Taniguchi A and Kishimura A and Hayashi Y and Mori T and Katayama Y}, title = {Synthesis and biological evaluation of a monocyclic Fc-binding antibody-recruiting molecule for cancer immunotherapy.}, journal = {RSC medicinal chemistry}, year = 2021, } @article{CTT100911568, author = {Muguruma K and Pradipta AR and Ode Y and Terashima K and Michiba H and Fujii M and Tanaka K}, title = {Disease-associated acrolein: A possible diagnostic and therapeutic substrate for in vivo synthetic chemistry.}, journal = {Bioorganic & medicinal chemistry}, year = 2020, } @article{CTT100911569, author = {Muguruma K and Fujita K and Fukuda A and Kishimoto S and Sakamoto S and Arima R and Ito M and Kawasaki M and Nakano S and Ito S and Shimizu K and Taguchi A and Takayama K and Taniguchi A and Hayashi Y}, title = {Kinetics-Based Structural Requirements of Human Immunoglobulin G Binding Peptides.}, journal = {ACS omega}, year = 2019, } @article{CTT100911570, author = {Muguruma K and Ito M and Fukuda A and Kishimoto S and Taguchi A and Takayama K and Taniguchi A and Ito Y and Hayashi Y}, title = {Synthesis and structure-activity relationship studies of IgG-binding peptides focused on the C-terminal histidine residue.}, journal = {MedChemComm}, year = 2019, } @article{CTT100911571, author = {Muguruma K and Shirasaka T and Akiyama D and Fukumoto K and Taguchi A and Takayama K and Taniguchi A and Hayashi Y}, title = {An Efficient Method for the Conjugation of Hydrophilic and Hydrophobic Components by Solid-Phase-Assisted Disulfide Ligation.}, journal = {Angewandte Chemie (International ed. in English)}, year = 2018, } @article{CTT100911572, author = {Takayama K and Rentier C and Asari T and Nakamura A and Saga Y and Shimada T and Nirasawa K and Sasaki E and Muguruma K and Taguchi A and Taniguchi A and Negishi Y and Hayashi Y}, title = {Development of Potent Myostatin Inhibitory Peptides through Hydrophobic Residue-Directed Structural Modification.}, journal = {ACS medicinal chemistry letters}, year = 2017, } @article{CTT100911573, author = {Taguchi A and Kobayashi K and Kotani A and Muguruma K and Kobayashi M and Fukumoto K and Takayama K and Hakamata H and Hayashi Y}, title = {3-Nitro-2-pyridinesulfenates as Efficient Solution- and Solid-Phase Disulfide Bond Forming Agents.}, journal = {Chemistry (Weinheim an der Bergstrasse, Germany)}, year = 2017, } @article{CTT100911574, author = {Yakushiji F and Muguruma K and Hayashi Y and Shirasaka T and Kawamata R and Tanaka H and Yoshiwaka Y and Taguchi A and Takayama K and Hayashi Y}, title = {Click strategy using disodium salts of amino acids improves the water solubility of plinabulin and KPU-300.}, journal = {Bioorganic & medicinal chemistry}, year = 2017, } @article{CTT100911575, author = {Muguruma K and Yakushiji F and Kawamata R and Akiyama D and Arima R and Shirasaka T and Kikkawa Y and Taguchi A and Takayama K and Fukuhara T and Watabe T and Ito Y and Hayashi Y}, title = {Novel Hybrid Compound of a Plinabulin Prodrug with an IgG Binding Peptide for Generating a Tumor Selective Noncovalent-Type Antibody-Drug Conjugate.}, journal = {Bioconjugate chemistry}, year = 2016, } @article{CTT100911576, author = {Hayashi Y and Takeno H and Chinen T and Muguruma K and Okuyama K and Taguchi A and Takayama K and Yakushiji F and Miura M and Usui T and Hayashi Y}, title = {Development of a new benzophenone-diketopiperazine-type potent antimicrotubule agent possessing a 2-pyridine structure.}, journal = {ACS medicinal chemistry letters}, year = 2014, } @article{CTT100911577, author = {Yakushiji F and Tanaka H and Muguruma K and Iwahashi T and Yamazaki Y and Hayashi Y}, title = {Water-soluble prodrug of antimicrotubule agent plinabulin: effective strategy with click chemistry.}, journal = {Chemistry (Weinheim an der Bergstrasse, Germany)}, year = 2011, } @inproceedings{CTT100935250, author = {飯田啓介 and 松井 誠 and 六車 共平 and 本田雄士 and 三浦 裕 and 西山 伸宏}, title = {一型糖尿病の治療を目指した抗体フラグメント-高分子結合型医薬品の創製}, booktitle = {}, year = 2025, } @inproceedings{CTT100935249, author = {柳田浩毅 and 小林基晃 and Chintrakulchai Wanphiwat and 高田 郁人 and 尾木 公一 and 道西 准也 and 大嶽 知之 and 六車 共平 and 本田 雄士 and 武元 宏泰 and 三浦 裕 and 西山 伸宏}, title = {PEGジレンマを解決する新規脂質ナノ粒子の開発とがん治療への展開}, booktitle = {}, year = 2025, } @inproceedings{CTT100935237, author = {千野利純 and 松尾 拓海 and 本田 雄士 and 刑部 祐里子 and Guo Haochen and 六車 共平 and 三浦裕 and 西山 伸宏}, title = {CRISPR/Cas9-sgRNA RNP搭載三元系複合体による臓器選択的in vivoゲノム編集}, booktitle = {}, year = 2025, } @inproceedings{CTT100935236, author = {Nozomi Matsudaira and Yuto Honda and Kyohei Muguruma and Haochen Guo and Yutaka Miura and Nobuhiro Nishiyama}, title = {Self-Assembly Ternary Complex Comprising Cyclic RGD-installed Polymer and Tannic Acid for Selective and Effective Protein Delivery to Tumor}, booktitle = {}, year = 2024, } @inproceedings{CTT100935244, author = {千野利純 and 松尾拓海 and 本田雄士 and 刑部 祐里子 and Guo Haochen and 六車共平 and 三浦裕 and 西山伸宏}, title = {Cas9 RNP三元系複合体の高分子側鎖アミン構造調整によるゲノム編集制御}, booktitle = {}, year = 2024, } @inproceedings{CTT100935247, author = {津田雄流 and 本田雄士 and リチャードソンJ.ジョセフ and 六車共平 and Guo Haochen and 三浦裕 and 西山伸宏}, title = {金属イオン‐ポリフェノール錯体を基盤としたPEG被覆技術の構築及び物性評価}, booktitle = {}, year = 2024, } @inproceedings{CTT100935246, author = {松平 望 and 本田 雄士 and 六車 共平 and GUO Haochen and 三浦 裕 and 西山 伸宏}, title = {環状RGDペプチド導入高分子とタンニン酸からなる腫瘍細胞標的型三元系複合体の開発}, booktitle = {}, year = 2024, } @inproceedings{CTT100935245, author = {金子彩海 and 本田雄士 and 松平望 and Guo Haochen and 喜納宏昭 and 六車共平 and 三浦裕 and 西山伸宏}, title = {肝実質細胞を標的可能にするGalNAc搭載アデノ随伴ウイルス三元系複合体の開発}, booktitle = {}, year = 2024, } @inproceedings{CTT100935243, author = {黄 若言 and 津田 雄流 and 本田 雄士 and Haochen Guo and 六車 共平 and 三浦 裕 and 西山伸宏}, title = {CRISPR-Cas9/sgRNA RNPのゲノム編集効率を向上させる高分子ナノキャリアの開発}, booktitle = {}, year = 2024, } @inproceedings{CTT100935235, author = {津田雄流 and 本田雄士 and リチャードソンJ.ジョセフ and 六車共平 and 三浦裕 and 西山伸宏}, title = {金属イオン‐ポリフェノール錯体を基盤としたPEG被覆中空マイクロカプセルの 構築及び物性評価}, booktitle = {}, year = 2024, }