@article{CTT100917900, author = {Imai Kyosuke and Kyohei Muguruma and Ambara R. Pradipta and Katsunori Tanaka}, title = {In vivo synthetic anticancer approach by resourcing mouse blood albumin as a biocompatible artificial metalloenzyme}, journal = {Angewandte Chemie International Edition}, year = 2024, } @article{CTT100911561, author = {Minagi Mukaiyama and Chihiro Uchiyama and Akane Fukuda and Yoshiki Nakazawa and Yuka Kuramochi and Yudai Shibata and Sho Konno and Kyohei Muguruma and Naohiro Matsugaki and Tomo Asari and Kazuyoshi Ogawa and Akihiro Taguchi and Kentaro Takayama and Atsuhiko Taniguchi and Yoko Nagumo and Toshiya Senda and Yoshio Hayashi and Takeo Usui}, title = {X-Ray Conformation and Structure–Activity Relationships of MA026, a Reversible Tight Junction Opener}, journal = {Journal of Medicinal Chemistry}, year = 2023, } @article{CTT100911562, author = {Yudai Ode and Ambara R. Pradipta and Peni Ahmadi and Akihiro Ishiwata and Akiko Nakamura and Yasuko Egawa and Yuriko Kusakari and Kyohei Muguruma and Yang Wang and Xiaojie Yin and Nozomi Sato and Hiromitsu Haba and Katsunori Tanaka}, title = {Therapeutic efficacy of 211At-radiolabeled 2,6-diisopropylphenyl azide in mouse models of human lung cancer}, journal = {Chemical Science}, year = 2023, } @article{CTT100911563, author = {Tsung-Che Chang and Igor Nasibullin and Kyohei Muguruma and Yuriko Kusakari and Taiji Shimoda and Katsunori Tanaka}, title = {Evaluation of acute toxicity of cancer-targeting albumin-based artificial metalloenzymes}, journal = {Bioorganic & Medicinal Chemistry}, year = 2022, } @article{CTT100911564, author = {Ahmadi P and Muguruma K and Chang TC and Tamura S and Tsubokura K and Egawa Y and Suzuki T and Dohmae N and Nakao Y and Tanaka K}, title = {In vivo metal-catalyzed SeCT therapy by a proapoptotic peptide.}, journal = {Chemical science}, year = 2021, } @article{CTT100911565, author = {Pradipta AR and Ahmadi P and Terashima K and Muguruma K and Fujii M and Ichino T and Maeda S and Tanaka K}, title = {Targeted 1,3-dipolar cycloaddition with acrolein for cancer prodrug activation.}, journal = {Chemical science}, year = 2021, } @article{CTT100911566, author = {Muguruma K and Osawa R and Fukuda A and Ishikawa N and Fujita K and Taguchi A and Takayama K and Taniguchi A and Ito Y and Hayashi Y}, title = {Development of a High-Affinity Antibody-Binding Peptide for Site-Specific Modification.}, journal = {ChemMedChem}, year = 2021, } @article{CTT100911567, author = {Sasaki K and Muguruma K and Osawa R and Fukuda A and Taniguchi A and Kishimura A and Hayashi Y and Mori T and Katayama Y}, title = {Synthesis and biological evaluation of a monocyclic Fc-binding antibody-recruiting molecule for cancer immunotherapy.}, journal = {RSC medicinal chemistry}, year = 2021, } @article{CTT100911568, author = {Muguruma K and Pradipta AR and Ode Y and Terashima K and Michiba H and Fujii M and Tanaka K}, title = {Disease-associated acrolein: A possible diagnostic and therapeutic substrate for in vivo synthetic chemistry.}, journal = {Bioorganic & medicinal chemistry}, year = 2020, } @article{CTT100911570, author = {Muguruma K and Ito M and Fukuda A and Kishimoto S and Taguchi A and Takayama K and Taniguchi A and Ito Y and Hayashi Y}, title = {Synthesis and structure-activity relationship studies of IgG-binding peptides focused on the C-terminal histidine residue.}, journal = {MedChemComm}, year = 2019, } @article{CTT100911569, author = {Muguruma K and Fujita K and Fukuda A and Kishimoto S and Sakamoto S and Arima R and Ito M and Kawasaki M and Nakano S and Ito S and Shimizu K and Taguchi A and Takayama K and Taniguchi A and Hayashi Y}, title = {Kinetics-Based Structural Requirements of Human Immunoglobulin G Binding Peptides.}, journal = {ACS omega}, year = 2019, } @article{CTT100911571, author = {Muguruma K and Shirasaka T and Akiyama D and Fukumoto K and Taguchi A and Takayama K and Taniguchi A and Hayashi Y}, title = {An Efficient Method for the Conjugation of Hydrophilic and Hydrophobic Components by Solid-Phase-Assisted Disulfide Ligation.}, journal = {Angewandte Chemie (International ed. in English)}, year = 2018, } @article{CTT100911572, author = {Takayama K and Rentier C and Asari T and Nakamura A and Saga Y and Shimada T and Nirasawa K and Sasaki E and Muguruma K and Taguchi A and Taniguchi A and Negishi Y and Hayashi Y}, title = {Development of Potent Myostatin Inhibitory Peptides through Hydrophobic Residue-Directed Structural Modification.}, journal = {ACS medicinal chemistry letters}, year = 2017, } @article{CTT100911573, author = {Taguchi A and Kobayashi K and Kotani A and Muguruma K and Kobayashi M and Fukumoto K and Takayama K and Hakamata H and Hayashi Y}, title = {3-Nitro-2-pyridinesulfenates as Efficient Solution- and Solid-Phase Disulfide Bond Forming Agents.}, journal = {Chemistry (Weinheim an der Bergstrasse, Germany)}, year = 2017, } @article{CTT100911574, author = {Yakushiji F and Muguruma K and Hayashi Y and Shirasaka T and Kawamata R and Tanaka H and Yoshiwaka Y and Taguchi A and Takayama K and Hayashi Y}, title = {Click strategy using disodium salts of amino acids improves the water solubility of plinabulin and KPU-300.}, journal = {Bioorganic & medicinal chemistry}, year = 2017, } @article{CTT100911575, author = {Muguruma K and Yakushiji F and Kawamata R and Akiyama D and Arima R and Shirasaka T and Kikkawa Y and Taguchi A and Takayama K and Fukuhara T and Watabe T and Ito Y and Hayashi Y}, title = {Novel Hybrid Compound of a Plinabulin Prodrug with an IgG Binding Peptide for Generating a Tumor Selective Noncovalent-Type Antibody-Drug Conjugate.}, journal = {Bioconjugate chemistry}, year = 2016, } @article{CTT100911576, author = {Hayashi Y and Takeno H and Chinen T and Muguruma K and Okuyama K and Taguchi A and Takayama K and Yakushiji F and Miura M and Usui T and Hayashi Y}, title = {Development of a new benzophenone-diketopiperazine-type potent antimicrotubule agent possessing a 2-pyridine structure.}, journal = {ACS medicinal chemistry letters}, year = 2014, } @article{CTT100911577, author = {Yakushiji F and Tanaka H and Muguruma K and Iwahashi T and Yamazaki Y and Hayashi Y}, title = {Water-soluble prodrug of antimicrotubule agent plinabulin: effective strategy with click chemistry.}, journal = {Chemistry (Weinheim an der Bergstrasse, Germany)}, year = 2011, }