@article{CTT100822319, author = {上野学 and 潘鉉承 and Hiroyuki Nakamura}, title = {リポソームを用いる中性子捕捉治療}, journal = {Drug Delivery System}, year = 2010, } @article{CTT100822322, author = {Hiroyuki Nakamura}, title = {中性子捕捉治療のためのナノカプセル型ホウ素薬剤送達システム(BDS)の開発}, journal = {Pharm. Tech. Japan (invited)}, year = 2010, } @article{CTT100684412, author = {Hyun Seung Ban and Hidemitsu Minegishi and Kazuki Shimizu and Minako Maruyama and Yuka Yasui and Hiroyuki Nakamura}, title = {Discovery of Carboranes as Inducers of 20S Proteasome Activity}, journal = {Chemmedchem}, year = 2010, } @article{CTT100827148, author = {Hiroyuki Nakamura}, title = {ホウ素の中性子捕捉反応を利用した低侵襲細胞選択的放射線療法}, journal = {Yakugaku Zasshi}, year = 2010, } @article{CTT100684616, author = {Manabu Ueno and Hyun Seung Ban and Kei Nakai and Ryu Inomata and Yasufumi Kaneda and Akira Matsumura and Hiroyuki Nakamura}, title = {Dodecaborate lipid liposomes as new vehicles for boron delivery system of neutron capture therapy}, journal = {Bioorganic & Medicinal Chemistry}, year = 2010, } @article{CTT100684605, author = {Tsuyuka Sugiishi and Akifumi Kimura and Hiroyuki Nakamura}, title = {Copper(I)-Catalyzed Substitution Reactions of Propargylic Amines: Importance of C(sp)-C(sp(3)) Bond Cleavage in Generation of Iminium Intermediates}, journal = {Journal of the American Chemical Society}, year = 2010, } @article{CTT100684603, author = {Kazuki Shimizu and Minako Maruyama and Yuka Yasui and Hidemitsu Minegishi and Hyun Seung Ban and Hiroyuki Nakamura}, title = {Boron-containing phenoxyacetanilide derivatives as hypoxia-inducible factor (HIF)-1 alpha inhibitors}, journal = {Bioorganic & Medicinal Chemistry Letters}, year = 2010, } @article{CTT100684541, author = {Hiroyuki Nakamura and Ryoji Horikoshi and Taikou Usui and Hyun Seung Ban}, title = {Selective inhibition of EGFR and VEGFR2 tyrosine kinases controlled by a boronic acid substituent on 4-anilinoquinazolines}, journal = {Medchemcomm}, year = 2010, } @article{CTT100684515, author = {Kenji Ishihara and Shuhei Okuyama and Shun Kumano and Koji Iida and Hiroshi Hamana and Michio Murakoshi and Toshimitsu Kobayashi and Shinichi Usami and Katsuhisa Ikeda and Yoichi Haga and Kohei Tsumoto and Hiroyuki Nakamura and Noriyasu Hirasawa and Hiroshi Wada}, title = {Salicylate restores transport function and anion exchanger activity of missense pendrin mutations}, journal = {Hearing Research}, year = 2010, } @article{CTT100684510, author = {Afaf R. Genady and Hiroyuki Nakamura}, title = {Undecahydro-closo-dodecaborates as good leaving groups in organic synthesis: generation of substituted styrenes via elimination of arylethyl dodecaborates}, journal = {Organic & Biomolecular Chemistry}, year = 2010, } @article{CTT100684508, author = {Mohamed E. El-Zaria and Afaf R. Genady and Hiroyuki Nakamura}, title = {Synthesis of triazolyl methyl-substituted amino- and oxy-undecahydrododecaborates for potential application in boron neutron capture therapy}, journal = {New Journal of Chemistry}, year = 2010, } @article{CTT100684507, author = {Mohamed E. El-Zaria and Hyun Seung Ban and Hiroyuki Nakamura}, title = {Boron-Containing Protoporphyrin IX Derivatives and Their Modification for Boron Neutron Capture Therapy: Synthesis, Characterization, and Comparative In Vitro Toxicity Evaluation}, journal = {Chemistry-a European Journal}, year = 2010, } @article{CTT100684497, author = {Hyun Seung Ban and Masaharu Uno and Hiroyuki Nakamura}, title = {Suppression of hypoxia-induced HIF-1 alpha accumulation by VEGFR inhibitors: Different profiles of AAL993 versus SU5416 and KRN633}, journal = {Cancer Letters}, year = 2010, } @article{CTT100684495, author = {Hyun Seung Ban and Yuko Tanaka and Wataru Nabeyama and Masako Hatori and Hiroyuki Nakamura}, title = {Enhancement of EGFR tyrosine kinase inhibition by C-C multiple bonds-containing anilinoquinazolines}, journal = {Bioorganic & Medicinal Chemistry}, year = 2010, } @article{CTT100684492, author = {Hyun Seung Ban and Kazuki Shimizu and Hidemitsu Minegishi and Hiroyuki Nakamura}, title = {Identification of HSP60 as a Primary Target of o-Carboranylphenoxyacetanilide, an HIF-1 alpha Inhibitor}, journal = {Journal of the American Chemical Society}, year = 2010, } @inproceedings{CTT100845724, author = {H. Nakamura and M. Ueno and N. Ueda and R. Inomata and H. Ban}, title = {Development of boron lipid liposomes for neutron capture therapy}, booktitle = {}, year = 2010, } @inproceedings{CTT100845732, author = {H. Minegishi and M. Maruyama and Y. Yasui and K. Shimizu and H. Ban and H. Nakamura}, title = {Discovery of carboranes as 20S proteasome activators}, booktitle = {}, year = 2010, } @inproceedings{CTT100845730, author = {Y. Koma and M. Uno and H. Ban and H. Nakamura}, title = {Structure-activity relationship of 1-[4-(N-benzylamino)phenyl]-3-phenylurea derivatives as HIF-1α inhibitors}, booktitle = {}, year = 2010, } @inproceedings{CTT100845729, author = {S. Tachikawa and H. Nakamura}, title = {Development of closo-dodecaborates for liposomal boron delivery of neutron capture therapy}, booktitle = {}, year = 2010, } @inproceedings{CTT100845728, author = {A. Takeuchi and A. Shoji and H. Ban and T. Yamori and H. Nakamura}, title = {Discovery of carborane-conjugated triazines as topoisomerase inhibitors}, booktitle = {}, year = 2010, } @inproceedings{CTT100845727, author = {H. Ban and K. Shimizu and H. Minegishi and H. Nakamura}, title = {Action mechanism of HIF-1α inhibitor GN26361: Identification of target protein with multifunctional molecular probe}, booktitle = {}, year = 2010, } @inproceedings{CTT100845726, author = {H. Nakamura and M. E. El-Zaria and H. Ban and A. R. Genady}, title = {Synthesis of triazolyl methyl-substituted thio-, amino-, and oxy-undecahydrododecaborates for potential application to boron neutron capture therapy}, booktitle = {}, year = 2010, } @inproceedings{CTT100845725, author = {H. Nakamura and M. Ueno and N. Ueda and R. Inomata and H. Ban}, title = {Development of boron lipid liposomes for neutron capture therapy}, booktitle = {}, year = 2010, } @inproceedings{CTT100845721, author = {峯岸秀充 and 潘鉉承 and 丸山美菜子 and 安井友香 and 清水一希 and 中村浩之 and Hiroyuki Nakamura}, title = {カルボラン含有低分子20S プロテアソーム活性化剤の開発}, booktitle = {}, year = 2010, } @inproceedings{CTT100845723, author = {Hiroyuki Nakamura}, title = {低酸素誘導因子シグナルを標的とした創薬研究の現状}, booktitle = {}, year = 2010, } @inproceedings{CTT100845722, author = {三好達郎 and Mohamed E. El-Zaria and 潘鉉承 and Hiroyuki Nakamura}, title = {カルボラニルトリアジン誘導体の選択的トポイソメラーゼ阻害活性}, booktitle = {}, year = 2010, } @inproceedings{CTT100845720, author = {竹内彩乃 and 東海林篤 and 潘鉉承 and 矢守隆夫 and Hiroyuki Nakamura}, title = {ホウ素含有コレステロールの開発:クリック反応によるイメージングとリポソーム化}, booktitle = {}, year = 2010, } @inproceedings{CTT100845712, author = {Hiroyuki Nakamura}, title = {ホウ素の力でがんに挑む}, booktitle = {}, year = 2010, } @inproceedings{CTT100845715, author = {R. Inomata and M. E. El-Zaria and H. S. Ban and H. Nakamura}, title = {Development of Boron-Containing Protoporphyrin IX Derivatives for Boron Neutron Capture Therapy and Photodynamic Therapy}, booktitle = {}, year = 2010, } @inproceedings{CTT100845713, author = {東海林篤 and 竹内彩乃 and 潘鉉承 and Kang Sang Ook and 矢守隆夫 and Hiroyuki Nakamura}, title = {カルボラン含有トリアジン誘導体のトポイソメラーゼ阻害活性}, booktitle = {}, year = 2010, } @inproceedings{CTT100845718, author = {F. Yoshida and K. Nakai and T. Isobe and R. Inomata and A. Zaboronok and Y. Yamamoto and M. Shirakawa and T. Yamamoto and A. Matsumura and H. Nakamura}, title = {Biodistribution of BSH-encapsulated boron liposome in mouse glioma}, booktitle = {}, year = 2010, } @inproceedings{CTT100845717, author = {H. Nakamura and N. Ueda and H. S. Ban and K. Maruyama and M. E. El-Zaria}, title = {Boron Lipid Liposomes: EPR Effect and Fluorescence Imaging}, booktitle = {}, year = 2010, } @inproceedings{CTT100845716, author = {R. Inomata and M. E. El-Zaria and H. S. Ban and H. Nakamura}, title = {Development of Boron-Containing Protoporphyrin IX Derivatives for Boron Neutron Capture Therapy and Photodynamic Therapy}, booktitle = {}, year = 2010, } @inproceedings{CTT100845711, author = {杉石露佳 and Hiroyuki Nakamura}, title = {1価の銅触媒存在下におけるプロパルギルアミン類のアルキン置換反応}, booktitle = {}, year = 2010, } @inproceedings{CTT100845708, author = {猪俣竜 and 上野学 and 立川将士 and 三好達郎 and Mohamed E. El-Zaria and 潘鉉承 and 小田雄介 and 鈴木亮 and 丸山一雄 and Hiroyuki Nakamura}, title = {トランスフェリン修飾ホウ素リポソームによるBNCT効果}, booktitle = {}, year = 2010, } @inproceedings{CTT100845710, author = {Hiroyuki Nakamura}, title = {がんの低酸素環境応答に着目した創薬アプローチ}, booktitle = {}, year = 2010, } @inproceedings{CTT100845709, author = {M. E. El- Zaria and A. R. Genady and 中村浩之}, title = {New Strategy for Synthesis of Mercaptoundecahydrododecaborate Derivatives via Click Chemistry: Possible Boron Carriers and Visualization in Cells for Neutron Capture Therapy}, booktitle = {}, year = 2010, } @inproceedings{CTT100845707, author = {潘鉉承 and 清水一希 and 峯岸秀充 and Hiroyuki Nakamura}, title = {カルボラン含有小分子化合物GN26361による低酸素誘導因子(HIF)阻害と作用機序}, booktitle = {}, year = 2010, } @inproceedings{CTT100845704, author = {東海林篤 and 潘鉉承 and 矢守隆夫 and Hiroyuki Nakamura}, title = {カルボラン含有トリアジン類のトポイソメラーゼ阻害活性}, booktitle = {}, year = 2010, } @inproceedings{CTT100845706, author = {潘鉉承 and 清水一希 and 峯岸秀充 and Hiroyuki Nakamura}, title = {低酸素誘導因子(HIF) 阻害剤GN26361 の作用機序の解明}, booktitle = {}, year = 2010, } @inproceedings{CTT100845705, author = {峯岸秀充 and 清水一希 and 潘鉉承 and Hiroyuki Nakamura}, title = {カルボラン含有低分子20S プロテアソーム活性化剤の開発}, booktitle = {}, year = 2010, } @inproceedings{CTT100845703, author = {Hiroyuki Nakamura and 宇野正治 and 潘鉉承}, title = {脱SUMO 化酵素SENP-1 阻害剤の発見}, booktitle = {}, year = 2010, } @inproceedings{CTT100845701, author = {Hiroyuki Nakamura}, title = {Boron-Containing Phenoxyacetanilide DHypoxia-Inducible Factor (HIF)-1α Inhibitors}, booktitle = {}, year = 2010, } @inproceedings{CTT100845702, author = {Hiroyuki Nakamura}, title = {Liposomal Boron Delivery System for Neutron Capture Therapy of Cancers}, booktitle = {}, year = 2010, } @inproceedings{CTT100845700, author = {高麗洋佑 and 宇野正治 and 潘鉉承 and Hiroyuki Nakamura}, title = {低酸素誘導因子(HIF)-1α阻害剤の開発}, booktitle = {}, year = 2010, } @inproceedings{CTT100845699, author = {峯岸秀充 and 潘鉉承 and 丸山美菜子 and 安井友香 and 清水一希 and Hiroyuki Nakamura}, title = {カルボラン含有低分子20Sプロテアソーム活性化剤の開発}, booktitle = {}, year = 2010, } @inproceedings{CTT100845698, author = {竹内彩乃 and 東海林篤 and 潘鉉承 and 矢守隆夫 and Hiroyuki Nakamura}, title = {カルボラン含有トリアジン類のトポイソメラーゼ阻害活性}, booktitle = {}, year = 2010, } @inproceedings{CTT100845697, author = {Hiroyuki Nakamura and 宇野正治 and 潘鉉承}, title = {脱SUMO化酵素SENP-1阻害剤の発見と低酸素誘導因子抑制作用}, booktitle = {}, year = 2010, } @inproceedings{CTT100845696, author = {M. E. El-Zaria and A. R. Genady and 潘鉉承 and Hiroyuki Nakamura}, title = {イオン性ホウ素クラスターのクリック型環化反応の開発と細胞内イメージング}, booktitle = {}, year = 2010, } @inproceedings{CTT100845695, author = {Hiroyuki Nakamura}, title = {ホウ素の中性子捕捉反応を利用した低侵襲細胞選択的放射線療法}, booktitle = {}, year = 2010, } @inproceedings{CTT100845694, author = {上田記子 and 潘鉉承 and Hiroyuki Nakamura}, title = {蛍光標識ホウ素ナノカプセルの開発と細胞内イメージング}, booktitle = {}, year = 2010, } @inproceedings{CTT100845693, author = {潘鉉承 and 宇野正治 and Hiroyuki Nakamura}, title = {VEGFR阻害剤によるHIF活性化抑制とその作用機序}, booktitle = {}, year = 2010, } @inproceedings{CTT100845692, author = {田中優子 and 臼井大晃 and 潘鉉承 and 浅井章良 and Hiroyuki Nakamura}, title = {インデノピラゾール骨格を有する新規HIF-1α 阻害剤の開発}, booktitle = {}, year = 2010, } @inproceedings{CTT100845690, author = {清水一希 and Hiroyuki Nakamura}, title = {アリルトリフルオロボレートを用いた触媒的ビス-π- アリルパラジウム反応}, booktitle = {}, year = 2010, } @inproceedings{CTT100845689, author = {峯岸秀充 and 丸山美菜子 and 安井友香 and 清水一希 and 潘鉉承 and Hiroyuki Nakamura}, title = {カルボラン含有低分子プロテアソーム活性化剤の開発}, booktitle = {}, year = 2010, } @inproceedings{CTT100845688, author = {宇野正治 and 潘鉉承 and Hiroyuki Nakamura}, title = {新規SUMO 特異的プロテアーゼ(SENP)阻害剤の開発}, booktitle = {}, year = 2010, } @inproceedings{CTT100845687, author = {高麗洋佑 and 潘鉉承 and Shinae Kizaka-Kondoh and 平岡眞寛 and Hiroyuki Nakamura}, title = {HIF-1α 抑制剤GN6767誘導体の創薬研究 宇野正治}, booktitle = {}, year = 2010, }