@article{CTT100921038, author = {Taiki Morita and Kentaro Makino and Masato Tsuda and Hiroyuki Nakamura}, title = {Chemoselective α-Trifluoroacetylation of Amides Using Highly Electrophilic Trifluoroacetic Anhydrides and 2,4,6-Collidine}, journal = {Organic Letters}, year = 2023, } @article{CTT100921039, author = {Satoshi Okada and Kai Nishimura and Qarri Ainaya and Kouichi Shiraishi and Sergey A. Anufriev and Igor B. Sivaev and Yoshinori Sakurai and Minoru Suzuki and Masayuki Yokoyama and Hiroyuki Nakamura}, title = {Development of a Gadolinium–Boron-Conjugated Albumin for MRI-Guided Neutron Capture Therapy}, journal = {Molecular Pharmaceutics}, year = 2023, } @article{CTT100921475, author = {Y. Hattori and T. Andoh and S. Kawabata and N. Hu and H. Michiue and H. Nakamura and T. Nomoto and M. Suzuki and T. Takata and H. Tanaka and T. Watanabe and K. Ono}, title = {Proposal of recommended experimental protocols for in vitro and in vivo evaluation methods of boron agents for neutron capture therapy}, journal = {Journal of Radiation Research}, year = 2023, } @article{CTT100921040, author = {Kazuki Miura and Manjusha Joshi and Taiki Morita and Hiroyuki Nakamura}, title = {Discovery of three-dimensional bicyclo[3.3.1]nonanols as novel heat shock protein 90 inhibitors}, journal = {Bioorganic & Medicinal Chemistry}, year = 2023, } @article{CTT100921041, author = {Yoshiki Fujikawa and Yusuke Fukuo and Kai Nishimura and Kohei Tsujino and Hideki Kashiwagi and Ryo Hiramatsu and Naosuke Nonoguchi and Motomasa Furuse and Toshihiro Takami and Naonori Hu and Shin-Ichi Miyatake and Takushi Takata and Hiroki Tanaka and Tsubasa Watanabe and Minoru Suzuki and Shinji Kawabata and Hiroyuki Nakamura and Masahiko Wanibuchi}, title = {Evaluation of the Effectiveness of Boron Neutron Capture Therapy with Iodophenyl-Conjugated closo-Dodecaborate on a Rat Brain Tumor Model}, journal = {Biology}, year = 2023, } @article{CTT100917054, author = {Hung Wei Lai and Yukitaka Tani and Udomlak Sukatta and Prapassorn Rugthaworn and Asada Thepyos and Shinkuro Yamamoto and Hideo Fukuhara and Keiji Inoue and Hideya Yuasa and Hiroyuki Nakamura and Shun-ichiro Ogura}, title = {Mangostin enhances efficacy of aminolevulinic acid-photodynamic therapy against cancer through inhibition of ABCG2 activity}, journal = {Photodiagnosis and Photodynamic Therapy}, year = 2023, } @article{CTT100921042, author = {Taiki Morita and Non Ito and Hiroyuki Nakamura}, title = {Asymmetric Synthesis of Bicyclic Isoxazolines via Dearomative Cycloaddition of 4-Nitroisoxazoles with Zwitterionic π-Allyl Palladium Species}, journal = {Organic Letters}, year = 2023, } @article{CTT100921477, author = {Kai Nishimura and Hideki Kashiwagi and Taiki Morita and Yusuke Fukuo and Satoshi Okada and Kazuki Miura and Yoshitaka Matsumoto and Yu Sugawara and Takayuki Enomoto and Minoru Suzuki and Kei Nakai and Shinji Kawabata and Hiroyuki Nakamura}, title = {Efficient neutron capture therapy of glioblastoma with pteroyl-closo-dodecaborate-conjugated 4-(p-iodophenyl)butyric acid (PBC-IP)}, journal = {Journal of Controlled Release}, year = 2023, } @article{CTT100921043, author = {Domenico Loreto and Basudev Maity and Taiki Morita and Hiroyuki Nakamura and Antonello Merlino and Takafumi Ueno}, title = {Cross-Linked Crystals of Dirhodium Tetraacetate/RNase A Adduct Can Be Used as Heterogeneous Catalysts}, journal = {Inorganic Chemistry}, year = 2023, } @article{CTT100921479, author = {Otoka Shamoto and Keiji Komuro and Naoto Sugisawa and Ting-Ho Chen and Hiroyuki Nakamura and Shinichiro Fuse}, title = {Peptide Cyclization by the Use of Acylammonium Species}, journal = {Angewandte Chemie International Edition}, year = 2023, } @article{CTT100921490, author = {Annette G. Beck-Sickinger and Daniel P. Becker and Oksana Chepurna and Bhaskar Das and Sebastian Flieger and Evamarie Hey-Hawkins and Narayan Hosmane and Satish S. Jalisatgi and Hiroyuki Nakamura and Rameshwar Patil and Maria da Graテァa H. Vicente and Clara Viテアas}, title = {New Boron Delivery Agents}, journal = {Cancer Biotherapy and Radiopharmaceuticals}, year = 2023, } @article{CTT100903969, author = {Satoshi Okada and Yuka Muto and Bo Zhu and Hiroshi Ueda and Hiroyuki Nakamura}, title = {Development of a Peptide Sensor Derived from Human ACE2 for Fluorescence Polarization Assays of the SARS-CoV-2 Receptor Binding Domain}, journal = {Analytical Chemistry}, year = 2023, } @article{CTT100885782, author = {Yasuhiko Orita and Susumu Shimanuki and Satoshi Okada and Kentaro Nakamura and Hiroyuki Nakamura and Yoshitaka Kitamoto and Yusuke Shimoyama and Yuta Kurashina*}, title = {Acoustic-responsive carbon dioxide-loaded liposomes for efficient drug release}, journal = {Ultrasonics Sonochemistry}, year = 2023, } @article{CTT100887613, author = {Hiroyuki Nakamura}, title = {イソオキサゾールの新規官能基化法の開発}, journal = {有機合成化学協会誌}, year = 2023, } @article{CTT100921045, author = {Kohei Tsujino and Hideki Kashiwagi and Kai Nishimura and Ryo Kayama and Kohei Yoshimura and Yusuke Fukuo and Hiroyuki Shiba and Ryo Hiramatsu and Naosuke Nonoguchi and Motomasa Furuse and Toshihiro Takami and Shin-Ichi Miyatake and Naonori Hu and Takushi Takata and Hiroki Tanaka and Minoru Suzuki and Shinji Kawabata and Hiroyuki Nakamura and Masahiko Wanibuchi}, title = {Improved Boron Neutron Capture Therapy Using Integrin αvβ3-Targeted Long-Retention-Type Boron Carrier in a F98 Rat Glioma Model}, journal = {Biology}, year = 2023, } @article{CTT100887612, author = {Hiroyuki Nakamura}, title = {中性子捕捉療法の鍵を握る10B薬剤開発}, journal = {Precision Medicine}, year = 2023, } @article{CTT100921046, author = {Tomoya Doi and Kohei Umedera and Kazuki Miura and Taiki Morita and Hiroyuki Nakamura}, title = {Synthesis of the diazatricycloundecane scaffold via gold(i)-catalysed Conia-ene-type 5-exo-dig cyclization and stepwise substituent assembly for the construction of an sp3-rich compound library}, journal = {Organic & Biomolecular Chemistry}, year = 2023, } @article{CTT100921476, author = {Manjot Kaur and Ramovatar Meena and Kai Nishimura and Kazuki Miura and Hiroyuki Nakamura and Minoru Suzuki and Ram K. Sharma and Akshay Kumar}, title = {Boron neutron capture therapy anti-tumor effect of nanostructured boron carbon nitride: A new potential candidate}, journal = {Inorganic Chemistry Communications}, year = 2023, } @inproceedings{CTT100921529, author = {Hiroyuki Nakamura}, title = {Photocatalytic Target Protein Knockdown and Its Application to Intracellular Molecular Targeted Photodynamic Therapy}, booktitle = {}, year = 2023, } @inproceedings{CTT100921528, author = {Hiroyuki Nakamura}, title = {Photocatalytic Target Protein Knockdown and Its Application to Intracellular Molecular Targeted Photodynamic Therapy}, booktitle = {}, year = 2023, } @inproceedings{CTT100921523, author = {Hiroyuki Nakamura}, title = {Photocatalytic Target Protein Knockdown and Its Application to Molecular Targeted Photodynamic Therapy}, booktitle = {}, year = 2023, } @inproceedings{CTT100921543, author = {Hiroyuki Nakamura and Kazuki Miura and Michihiko Tsushima and Yijin Wen}, title = {がん特異的分子の光不活性化を作用機序とする分子標的型光線力学療法}, booktitle = {}, year = 2023, } @inproceedings{CTT100921544, author = {Tomoya Doi and Kazuki Miura and Kohei Umedera and Taiki Morita and Hiroyuki Nakamura}, title = {新規ジアザトリシクロウンデカン骨格を基盤とする化合物ライブラリーの構築と生物活性分子の創出}, booktitle = {}, year = 2023, } @inproceedings{CTT100921545, author = {Kentaro Makino and Masato Tsuda and Taiki Morita and Hiroyuki Nakamura}, title = {アミド選択的α-アシル化反応の開発}, booktitle = {}, year = 2023, } @inproceedings{CTT100921548, author = {Taiki Morita and Non Ito and Hiroyuki Nakamura}, title = {パラジウム触媒を用いた1,2-アザボリン類のB -アレニル化反応の開発}, booktitle = {}, year = 2023, } @inproceedings{CTT100921547, author = {Masato Tsuda and Taiki Morita and Hiroyuki Nakamura}, title = {亜鉛カルベノイドによる1,2-アゾール類へのメチレン挿入反応の開発}, booktitle = {}, year = 2023, } @inproceedings{CTT100921546, author = {Non Ito and Taiki Morita and Hiroyuki Nakamura}, title = {パラジウム触媒によるイソオキサゾールの脱芳香族化を伴う不斉環化付加反応の開発}, booktitle = {}, year = 2023, } @inproceedings{CTT100921522, author = {Hiroyuki Nakamura}, title = {Efficient therapeutic approach for glioblastoma with a novel boron agent PBC-IP on neutron capture therapy}, booktitle = {}, year = 2023, } @inproceedings{CTT100921551, author = {辻野晃平 and 川端信司 and 柏木秀基 and 福尾祐介 and 宮武伸一 and Hiroki Tanaka and Minori Suzuki and Kai Nishimura and Hiroyuki Nakamura and 鰐渕昌彦}, title = {葉酸受容体標的ホウ素キャリアを局所投与で使用するホウ素中性子捕捉療法の可能性}, booktitle = {}, year = 2023, } @inproceedings{CTT100921550, author = {第19回日本中性子捕捉療法学会学術大会 and Hiroyuki Nakamura}, title = {MRIガイド下での中性子捕捉療法を指向したガドリニウム-ホウ素-アルブミン複合体の開発、○西村開、岡田智、Qarri Ainaya、白石貢一、鈴木実、横山昌幸、中村浩之}, booktitle = {}, year = 2023, } @inproceedings{CTT100921519, author = {Hiroyuki Nakamura}, title = {Prospects for Boron Compounds Beyond BPA}, booktitle = {}, year = 2023, } @inproceedings{CTT100921552, author = {Kazuki Miura and Tomoyuki Araki and Kai Nishimura and Taiki Morita and Tomoyasu Okada and Hiroyuki Nakamura}, title = {アミノ酸トランスポーターASCT2を標的とした新規低分子ホウ素薬剤の開発}, booktitle = {}, year = 2023, } @inproceedings{CTT100921515, author = {Hiroyuki Nakamura}, title = {Intramolecular Molecular-targeted Photodynamic Therapy}, booktitle = {}, year = 2023, } @inproceedings{CTT100921517, author = {Hiroyuki Nakamura}, title = {Intracellular Molecular-Targeted Photodynamic Therapy,}, booktitle = {}, year = 2023, } @inproceedings{CTT100921554, author = {Kazuki Miura and Michihiko Tsushima and Hiroyuki Nakamura}, title = {新規光線力学療法戦略としてのがん分子標的型光線力学療法の開発}, booktitle = {}, year = 2023, } @inproceedings{CTT100921555, author = {Tomoyasu Okada and Kai Nishimura and Qarri Ainaya and 白石貢一 and Minori Suzuki and 横山昌幸 and Hiroyuki Nakamura}, title = {MRI誘導型ホウ素中性子捕捉療法を指向したアルブミン薬剤の開発}, booktitle = {}, year = 2023, } @inproceedings{CTT100921553, author = {Dhina Fitriastuti and Kazuki Miura and Tomoyasu Okada and 平野弘之 and 長田裕之 and Hiroyuki Nakamura}, title = {HIF-1α/p300タンパク質間相互作用評価系の構築と新規阻害剤探索への展開}, booktitle = {}, year = 2023, } @inproceedings{CTT100887758, author = {Hiroyuki Nakamura}, title = {ペプチド模倣分子への応用を指向した籠型骨格の構造生成器”DeepCubist”の開発}, booktitle = {}, year = 2023, } @misc{CTT100909669, author = {Hiroyuki Nakamura and Satoshi Okada}, title = {新規蛍光検出薬}, howpublished = {PublishedPatent}, year = 2023, month = {}, note = {特願2022-079168(2022/05/13), 特開2023-167748(2023/11/24)} } @misc{CTT100826091, author = {Shinichiro Fuse and Yuma Otake and Hiroyuki Nakamura}, title = {フローリアクターを用いるN-カルボキシ無水物の合成方法}, howpublished = {RegisteredPatent}, year = 2023, month = {}, note = {特願2019-094952(2019/05/21), 特開2020-011948(2020/01/23), 特許第7362055号(2023/10/06)} }