@article{CTT100883765, author = {K. Umedera and T. Morita and H. Nakamura}, title = {Asymmetric construction of densely functionalized three-dimensional aza-tetracyclic scaffolds for drug discovery}, journal = {Chem. Commun}, year = 2022, } @article{CTT100877628, author = {K. Nishimura and S. Harrison and K. Kawai and T. Morita and K. Miura and S. Okada and H. Nakamura}, title = {Iodophenyl-conjugated closo-dodecaborate as a promising small boron molecule that binds to serum albumin and accumulates in tumor}, journal = {BIOORG. MED. CHEM. LETT.}, year = 2022, } @article{CTT100866095, author = {T. Morita and H. Murakami and Y. Asawa and H. Nakamura}, title = {Enantioselective Synthesis of Oxazaborolidines by Palladium-Catalyzed N−H/B−H Double Activation of 1,2-Azaborines}, journal = {Angew. Chem. Int. Ed.}, year = 2022, } @article{CTT100866101, author = {M. Tsuda and T. Morita and H. Nakamura}, title = {Synthesis of isoxazoloazaborines via gold(i)-catalyzed propargyl aza-Claisen rearrangement/borylative cyclization cascade}, journal = {Chem. Commun.}, year = 2022, } @article{CTT100864848, author = {G. Li and G. Yu and C. Wang and T. Morita and X. Zhang and H. Nakamura}, title = {Copper(I)-catalysed intramolecular hydroarylation-redox cross-dehydrogenative coupling of N-propargylanilines with phosphites}, journal = {Org. biomol. chem.}, year = 2022, } @inproceedings{CTT100884130, author = {H. Nakamura and T. Morita and H. Murakami}, title = {Development of 1,2-Azaborine-fused Heterocycles and Their Novel Functionalization}, booktitle = {}, year = 2022, } @inproceedings{CTT100881419, author = {Taiki Morita and Hiroki Murakami and Hiroyuki Nakamura}, title = {Asymmetric Synthesis of Oxazaborolidines via Palladium-Catalyzed N-H/B-H Double Functionalization of 1,2-Azaborines}, booktitle = {}, year = 2022, } @inproceedings{CTT100877625, author = {中村浩之 and 西村開 and 盛田大輝 and 岡田智 and 三浦一輝 and 柏木秀基 and 福尾祐介 and 松本孔貴 and 鈴木実 and 中井啓 and 川端信司}, title = {中性子捕捉療法のための血清アルブミンを利用したホウ素キャリアの開発}, booktitle = {}, year = 2022, } @inproceedings{CTT100875468, author = {西村開 and 盛田大輝 and 岡田智 and 三浦一輝 and 柏木秀基 and 福尾祐介 and 松本孔貴 and 高田卓志 and 鈴木実 and 中井啓 and 川端信司 and 中村浩之}, title = {中性子捕捉療法のための、アルブミンリガンドを基軸としたホウ素キャリアの開発}, booktitle = {}, year = 2022, } @inproceedings{CTT100875461, author = {津田正仁 and 盛田大輝 and 中村浩之}, title = {金(I)触媒によるプロパルギルアザClaisen転位反応を用いたイソオキサゾロアザボリンの合成と亜鉛カルベノイドによるN−O結合へのメチレン挿入反応の開発}, booktitle = {}, year = 2022, } @inproceedings{CTT100875462, author = {村上弘樹 and 盛田大輝 and 中村浩之}, title = {パラジウム触媒を用いた1,2-アザボリン類の不斉N-H/B-H二官能基化法の開発}, booktitle = {}, year = 2022, } @inproceedings{CTT100875464, author = {盛田大輝 and 中村浩之}, title = {ピペラジン酸およびN-ヒドロキシアミノ酸の直接縮合を基盤としたDentigerumycin Aの合成研究}, booktitle = {}, year = 2022, } @inproceedings{CTT100875466, author = {植原彩奈 and 盛田大輝 and 佐々木雄彦 and 中村浩之}, title = {リゾホスファチジルイノシトール(4,5)ビスリン酸の合成研究}, booktitle = {}, year = 2022, } @misc{CTT100884602, author = {中村浩之 and 盛田大輝 and 岡田智 and 西村開 and 川端 信司 and 鰐渕 昌彦 and 福尾 祐介 and 柏木 秀基}, title = {新規ホウ素薬剤}, howpublished = {公開特許}, year = 2022, month = {}, note = {PCT/JP2022/010452(2022/03/10), WO 2022/191262(2022/09/15)} } @misc{CTT100882394, author = {中村浩之 and 梅寺倖平 and 盛田大輝 and 小路 弘行 and 吉森 篤史}, title = {新規含窒素三環性骨格化合物およびその使用}, howpublished = {公開特許}, year = 2022, month = {}, note = {特願2020-204328(2020/12/09), 特開2022-091476(2022/06/21)} }