@book{CTT100685021, author = {中村浩之}, title = {機能性DDSキャリアの製剤設計}, publisher = {シーエムシー出版}, year = 2008, } @book{CTT100822150, author = {Hiroyuki Nakamura}, title = {Nanoparticle Synthesis in Microreactors}, publisher = {}, year = 2008, } @article{CTT100822323, author = {中村浩之}, title = {がん中性子捕捉療法と次世代ホウ素デリバリーシステム}, journal = {臨床血液}, year = 2008, } @article{CTT100828173, author = {Hiroyuki Nakamura}, title = {Minimally Invasive Cytoselective Radiation Therapy Using Boron Neutron Capture Reaction}, journal = {Yakugaku Zasshi}, year = 2008, } @article{CTT100828171, author = {Hiroyuki Nakamura}, title = {Development of Boron Delivery System for Neutron Capture Therapy of Cancer}, journal = {Progress in Drug Delivery System XVII}, year = 2008, } @article{CTT100768326, author = {Hiroyuki Nakamura}, title = {Triazinyl Architecture on Bifunctional Carboranyl Templates for the Production of Potential Neutron Capture Therapy Agents: Synthesis and Characterization of 1, 3, 5-Triazinylcarborane Derivatives}, journal = {Synthesis}, year = 2008, } @article{CTT100684954, author = {Hiroyuki Nakamura and Hiroyuki Saito and Masato Nanjo}, title = {Synthesis of 1,2-dihydroisoquinolines via palladium(0)-catalyzed addition-cyclization of chloroform to ortho-alkynylaldimines}, journal = {Tetrahedron Letters}, year = 2008, } @article{CTT100684621, author = {Taikou Usui and Hyun Seung Ban and Junpei Kawada and Takatsugu Hirokawa and Hiroyuki Nakamura}, title = {Discovery of indenopyrazoles as EGFR and VEGFR-2 tyrosine kinase inhibitors by in silico high-throughput screening}, journal = {Bioorganic & Medicinal Chemistry Letters}, year = 2008, } @article{CTT100684618, author = {Masaharu Uno and Hyun Seung Ban and Wataru Nabeyama and Hiroyuki Nakamura}, title = {de novo Design and synthesis of N-benzylanilines as new candidates for VEGFR tyrosinekinase inhibitors}, journal = {Organic & Biomolecular Chemistry}, year = 2008, } @article{CTT100684604, author = {Natsuko Sogabe and Kimimitsu Oda and Hiroyuki Nakamura and Hideo Orimo and Hisashi Watanabe and Takayuki Hosoi and Masae Goseki-Sone}, title = {Molecular effects of the tissue-nonspecific alkaline phosphatase gene polymorphism (787T > C) associated with bone mineral density}, journal = {Biomedical Research-Tokyo}, year = 2008, } @article{CTT100684597, author = {Ilhyong Ryu and Hiroshi Matsubara and Hiroyuki Nakamura and Dennis P. Curran}, title = {Phase-Vanishing Methods Based on Fluorous Phase Screen: A Simple Way for Efficient Execution of Organic Synthesis}, journal = {Chemical Record}, year = 2008, } @article{CTT100684554, author = {Hiroyuki Nakamura and Tsuyuka Sugiishi and Yuko Tanaka}, title = {Synthesis of allenes via CuBr-catalyzed homologation of alk-1-ynes accelerated by microwave}, journal = {Tetrahedron Letters}, year = 2008, } @article{CTT100684542, author = {Hiroyuki Nakamura and Makoto Ishikura and Tsuyuka Sugiishi and Takaya Kamakura and Jean-Francois Biellmann}, title = {Synthesis of mono- and 1,3-disubstituted allenes from propargylic amines via palladium-catalysed hydride-transfer reaction}, journal = {Organic & Biomolecular Chemistry}, year = 2008, } @article{CTT100684537, author = {Hiroyuki Nakamura}, title = {Liposomal boron delivery system for neutron capture therapy}, journal = {Yakugaku Zasshi-Journal of the Pharmaceutical Society of Japan}, year = 2008, } @article{CTT100684524, author = {Chai-Ho Lee and Guo Fan Jin and Ji Ho Yoon and Young Ju Jung and Jong-Dae Lee and Sungdong Cho and Hiroyuki Nakamura and Sang Ook Kang}, title = {Synthesis and characterization of polar functional group substituted mono- and bis-(o-carboranyl)-1,3,5-triazine derivatives}, journal = {Tetrahedron Letters}, year = 2008, } @article{CTT100684522, author = {Chai-Ho Lee and Guo Fan Jin and Hyo-Suk Kim and Hiroyuki Nakamura and Jong-Dae Lee}, title = {Synthesis and characterization of o-carboranylthiolate substituted 1,3,5-triazines}, journal = {Bulletin of the Korean Chemical Society}, year = 2008, } @article{CTT100684490, author = {Hyun Seung Ban and Shinya Onagi and Masaharu Uno and Wataru Nabeyama and Hiroyuki Nakamura}, title = {Allene as an alternative functional group for drug design: Effect of C - C multiple bonds conjugated with on the inhibition of EGFR tyrosine kinase}, journal = {Chemmedchem}, year = 2008, } @article{CTT100684521, author = {Chai-Ho Lee and Guo Fan Jin and Hyo-Suk Kim and Hiroyuki Nakamura and Yongseog Chung and Jong-Dae Lee}, title = {Preparation of boronated heterocyclic compounds using intramolecular cyclization reaction}, journal = {Bulletin of the Korean Chemical Society}, year = 2008, } @inproceedings{CTT100839275, author = {潘鉉承 and 宇野正治 and 中村浩之}, title = {VEGFR 阻害剤 AAL993 による HIF 活性化抑制作用}, booktitle = {}, year = 2008, } @inproceedings{CTT100839273, author = {田中優子 and 羽鳥雅子 and 潘鉉承 and 中村浩之}, title = {EGFRチロシンキナーゼへの非可逆的阻害作用を指向したアレニルキナゾリンの開発と生物活性評価}, booktitle = {}, year = 2008, } @inproceedings{CTT100839272, author = {中村 浩之}, title = {BNCTにおける薬剤開発の現状と展望}, booktitle = {}, year = 2008, } @inproceedings{CTT100839271, author = {Hiroyuki Nakamura and M. Ueno and H. S. Ban and K. Nakai and K. Tsuruta and Y. Kaneda and A. Matsumura}, title = {Development of Boron Nano Capsules for Neutron Capture Therapy}, booktitle = {}, year = 2008, } @inproceedings{CTT100839270, author = {T. Tsurubuchi and T. Yamamoto and K. Nakai and F. Yoshida and M. Miyakawa and M. Shirakawa and M. Ueno and M. Matsuda and Y. Nakae and R. Asano and A. Matsumura and Hiroyuki Nakamura}, title = {Intracellular uptake of a new boronated porphyrin EC032}, booktitle = {}, year = 2008, } @inproceedings{CTT100839279, author = {潘鉉承 and 宇野正治 and 中村浩之}, title = {VEGFR 阻害剤AAL993によるHIF活性化抑制作用}, booktitle = {}, year = 2008, } @inproceedings{CTT100839278, author = {宇野正治 and 潘鉉承 and 中村浩之}, title = {酸素誘導因子(HIF)-1alpha活性化阻害剤:1-[4-(N-Benzylamino)]phenyl-3-phenylurea誘導体の合成及び生物活性評価}, booktitle = {}, year = 2008, } @inproceedings{CTT100839277, author = {丸山美菜子 and 清水一希 and 潘鉉承 and 中村浩之}, title = {カルボランの立体電子的効果を利用した HIF-1α阻害剤の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100839276, author = {清水一希 and 丸山美菜子 and 潘鉉承 and 中村浩之}, title = {Hypoxia-Inducible Factor (HIF)活性化阻害能を有するホウ素化合物の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100839274, author = {宇野正治 and 潘鉉承 and 中村浩之}, title = {低酸素誘導因子(HIF)-1alpha活性化阻害剤:1-[4-(N-Benzylamino)phenyI]-3-phenylurea誘導体の合成及び生物活性評価}, booktitle = {}, year = 2008, } @inproceedings{CTT100839267, author = {潘鉉承 and 宇野正治 and Hiroyuki Nakamura}, title = {Development of HIF-1a inhibitor: Inhibition by VEGFR inhibitor AAL993 ofHIF-1a activation}, booktitle = {}, year = 2008, } @inproceedings{CTT100839268, author = {中村 浩之}, title = {中性子捕捉がん治療のための次世代ホウ素デリバリーシステム}, booktitle = {}, year = 2008, } @inproceedings{CTT100839269, author = {Hiroyuki Nakamura}, title = {Design and Synthesis of closo-Dodecaborate Lipids: Application to LiposomalBoron Delivery System for Neutron Capture Therapy}, booktitle = {}, year = 2008, } @inproceedings{CTT100839265, author = {中村浩之}, title = {DDS型ホウ素デリバリーシステムの現在地}, booktitle = {}, year = 2008, } @inproceedings{CTT100839264, author = {上野学 and 野村直裕 and 潘鉉承 and 中村浩之}, title = {ホウ素リポソームの血中安定性向上を目指した新規ホウ素脂質の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100839263, author = {Hiroyuki Nakamura and M. Ueno and H. S. Ban and K. Nakai and K. Tsuruta and Y. Kaneda and A. Matsumura}, title = {Boronated Liposomes for Neutron Capture Therapy of Cancer}, booktitle = {}, year = 2008, } @inproceedings{CTT100839262, author = {Hiroyuki Nakamura and M. Ueno and H. S. Ban and K. Nakai and K. Tsuruta and Y. Kaneda and A. Matsumura}, title = {Boron Nano Capsules for neutron Capture Therapy of Cancer}, booktitle = {}, year = 2008, } @inproceedings{CTT100839266, author = {中村浩之 and 上野学 and 潘鉉承 and J.-D. Lee and 中井啓 and 鶴田和太郎 and 松村明 and 金田安史}, title = {ホウ素ナノカプセルを用いた中性子捕捉治療}, booktitle = {}, year = 2008, } @inproceedings{CTT100839261, author = {中村浩之 and 上野学 and 潘鉉承 and 中井啓 and 金田安史 and 松村明}, title = {ホウ素ナノカプセルの開発と中性子捕捉治療効果}, booktitle = {}, year = 2008, } @inproceedings{CTT100839258, author = {上田記子 and 潘鉉承 and 中村浩之}, title = {ホウ酸基を導入したBelactosin誘導体によるプロテアソーム阻害作用}, booktitle = {}, year = 2008, } @inproceedings{CTT100839257, author = {清水一希 and 潘鉉承 and Hiroyuki Nakamura}, title = {Hypoxia-Inducible Factor-1 (HIF-1)活性化阻害能を有するホウ素化合物の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100839259, author = {田中優子 and 潘鉉承 and 中村浩之}, title = {アレンの特異的な反応性を利用した非可逆的EGFRチロシンキナーゼ阻害剤の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100839260, author = {中村 浩之}, title = {ホウ素を基軸とした創薬アプローチ}, booktitle = {}, year = 2008, } @inproceedings{CTT100839236, author = {宇野正治 and 潘鉉承 and 中村浩之}, title = {de novo 分子設計法を用いた血管内皮増殖因子受容体チロシンキナーゼ阻害剤の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100839243, author = {K. Nakai and Hiroyuki Nakamura and Lee. Chunman and Y. Kaneda and A. Matsumura}, title = {Develop ment of Boron Nano-Capsules for Neturon CaptureTherapy}, booktitle = {}, year = 2008, } @inproceedings{CTT100839237, author = {Hiroyuki Nakamura}, title = {Boronic Acid as an Alternative Functional Group for Drug Design}, booktitle = {}, year = 2008, } @inproceedings{CTT100836858, author = {上野学 and 丸山美菜子 and 野村直裕 and 潘鉉承 and 中井啓 and 鶴田和太郎 and 松村明 and 金田安史 and 中村浩之}, title = {中性子捕捉療法のためのホウ素リポソームの開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100836851, author = {田中優子 and 杉石露佳 and 中村浩之}, title = {マイクロウェーブによるCrabb?型アレン合成反応の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100836852, author = {杉石露佳 and 木村聡文 and 小名木信耶 and 中村浩之}, title = {1価の銅触媒を用いたプロパルギルアミンのアミン交換反応}, booktitle = {}, year = 2008, } @inproceedings{CTT100836853, author = {上田 記子・渡邉 自由・谷中 佳代子・潘 鉉承・中村 浩之}, title = {プロテアソーム阻害剤を指向した新規ペプチドホウ酸の合成と生物活性評価}, booktitle = {}, year = 2008, } @inproceedings{CTT100836854, author = {丸山美菜子 and 潘 鉉承 and 丸山美菜子 and 潘 鉉承 and 中村浩之}, title = {De novo分子設計法を用いた上皮細胞増殖因子受容体の細胞外ドメイン標的阻害剤の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100836855, author = {上野学 and 丸山美菜子 and 野村直裕 and 潘鉉承 and 中井啓 and 鶴田和太郎 and 松村明 and 金田安史 and 中村浩之}, title = {ホウ素と中性子でがんを治す! 、講演ハイライト(ポスター展 示:医薬化学}, booktitle = {}, year = 2008, } @inproceedings{CTT100836856, author = {渡邉自由 and 谷中佳代子 and 上田記子 and 潘鉉承 and 中村浩之}, title = {プロテアソーム阻害剤を指向した新規ペプチドホウ酸の合成と生物活性評価}, booktitle = {}, year = 2008, } @inproceedings{CTT100836857, author = {宇野正治 and 潘鉉承 and 鍋山航 and 中村浩之}, title = {de novo分子設計法を用いた血管内皮増殖因子受容体チロシンキナーゼ阻害剤の開発}, booktitle = {}, year = 2008, } @inproceedings{CTT100836850, author = {中村 浩之}, title = {ホウ素デリバリーシステムを用いた中性子捕捉がん治療}, booktitle = {}, year = 2008, }