@book{CTT100793624, author = {布施新一郎}, title = {マイクロフローアミド化法を基盤とする高効率ペプチド合成法の開発}, publisher = {一般社団法人触媒学会}, year = 2019, } @article{CTT100810170, author = {S. Fuse and K. Suzuki and T. Kuchimaru and T. Kadonosono and H. Ueda and S. Sato and S. Kizaka-Kondoh and H. Nakamura}, title = {Design, synthesis, and evaluation of indeno[2,1-c]pyrazolones for use as inhibitors against hypoxia-inducible factor (HIF)-1 transcriptional activity}, journal = {Bioorg. Med. Chem}, year = 2019, } @article{CTT100809276, author = {S. Fuse and K. Masuda and Y. Otake and H. Nakamura}, title = {Peptide chain elongation using unprotected amino acids in a micro-flow reactor}, journal = {Chem. Eur. J}, year = 2019, } @article{CTT100793622, author = {T. Nakamura and Y. Ishikura and N. Arakawa and M. Hori and M. Sato and M. Endo and H. Masui and S. Fuse and T. Takahashi and Y. Murata and R. Murdey and A. Wakamiya}, title = {Donor–acceptor polymers containing thiazole-fused benzothiadiazole acceptor units for organic solar cells}, journal = {RSC Advances}, year = 2019, } @article{CTT100786555, author = {布施新一郎}, title = {マイクロフロー法によるペプチド合成}, journal = {月刊ファインケミカル}, year = 2019, } @article{CTT100809286, author = {N. Sugisawa and Y. Otake and H. Nakamura and S. Fuse}, title = {Single-step, rapid, and mild synthesis of β-amino acid N-carboxy anhydrides using micro-flow technologies}, journal = {Chem. Asian J.}, year = 2019, } @inproceedings{CTT100804153, author = {小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之 and 布施新一郎}, title = {アシルイミダゾリウムカチオン中間体を利用するマイクロフローN-メチル化ペプチド合成法の開発とPterulamide I-IVの全合成}, booktitle = {}, year = 2019, } @inproceedings{CTT100804000, author = {布施新一郎}, title = {奥深いアミド化の世界へのご招待ーマイクロフロー合成法を道具としてー}, booktitle = {}, year = 2019, } @inproceedings{CTT100806154, author = {森谷渉 and 布施新一郎 and 中村浩之}, title = {光線力学療法を指向したDπA光増感剤の合成と作用機序の解明}, booktitle = {}, year = 2019, } @inproceedings{CTT100802417, author = {布施新一郎}, title = {Nーメチル化ペプチドの超高効率マイクロフロー合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100800122, author = {布施新一郎 and 小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之}, title = {N-メチル化ペプチドの超高効率マイクロフロー合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100800890, author = {Shinichiro Fuse}, title = {Investigation of amide bond formation based on micro-flow technologies}, booktitle = {}, year = 2019, } @inproceedings{CTT100798810, author = {柴田裕介 and 林慶浩 and 小竹佑磨 and 中村浩之 and 布施新一郎 and 川内進}, title = {イミダゾール誘導体を触媒とするN-メチルアミド化反応機構の理論的解明}, booktitle = {}, year = 2019, } @inproceedings{CTT100822791, author = {Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor}, booktitle = {}, year = 2019, } @inproceedings{CTT100798655, author = {杉澤直斗 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフロー合成法による瞬間混合を駆使したβ-アミノ酸-N-カルボキシ無水物の合成とその応用}, booktitle = {}, year = 2019, } @inproceedings{CTT100798357, author = {布施新一郎}, title = {マイクロフロー法を駆使するN-メチル化ペプチドの高効率合成}, booktitle = {}, year = 2019, } @inproceedings{CTT100795962, author = {小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之 and 布施新一郎}, title = {アシルイミダゾリウムカチオン中間体を利用するマイクロフローNーメチル化ペプチド合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100795963, author = {増田耕志郎 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {無保護アミノ酸連結を基盤とするマイクロフローペプチド鎖伸長法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100793958, author = {布施新一郎}, title = {高速マイクロフローアミド結合形成法の開発とペプチド合成の革新}, booktitle = {}, year = 2019, } @inproceedings{CTT100793957, author = {Shinichiro Fuse}, title = {Innovation of Peptide Synthesisbased on Micro-Flow Technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100792102, author = {Taiki Morita and Shinichiro Fuse and Hiroyuki Nakamura}, title = {Photochemical conversion of isoxazoles to 5-hydroxyimidazolines and its application for protein labeling}, booktitle = {}, year = 2019, } @inproceedings{CTT100792099, author = {福原信太郎 and Somaraju Yugandar and 布施新一郎 and 中村浩之}, title = {イソキサゾロピリジン形成と窒素ー酸素結合開裂を経由するプロパルギルイソオキサゾールからの3ーヒドロキシー4ー置換ピコリノニトリルの一気合成}, booktitle = {}, year = 2019, } @inproceedings{CTT100792096, author = {増田 耕志郎 and 小竹 佑磨 and 中村 浩之 and 布施 新一郎}, title = {マイクロフロー法を駆使する無保護アミノ酸を用いたペプチド鎖伸長法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100792094, author = {Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {An efficient synthesis of N-methylated peptides using micro-flow technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100792085, author = {Shinichiro Fuse and Yuma Otake and Hiroyuki Nakamura}, title = {Development of Amide Bond Formation of N-Methyl Amino Acids Using Micro-Flow Technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100792418, author = {布施新一郎}, title = {高速混合技術を基盤とする効率的有機合成手法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100789460, author = {Shinichiro Fuse}, title = {Highly Efficient Amide Bond Formation using Micro-Flow Technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100787105, author = {布施新一郎}, title = {マイクロフロー技術を駆使する高収率・省スペースかつ低コストの革新的ペプチド合成法の開発}, booktitle = {}, year = 2019, } @misc{CTT100866375, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-563042(2019/12/11), 再表2020/137545(2021/11/04)} } @misc{CTT100826091, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {フローリアクターを用いるN-カルボキシ無水物の合成方法}, howpublished = {登録特許}, year = 2023, month = {}, note = {特願2019-094952(2019/05/21), 特開2020-011948(2020/01/23), 特許第7362055号(2023/10/06)} } @misc{CTT100845903, author = {布施新一郎 and 中村浩之 and 小竹佑磨 and 宮崎 俊一 and 伊東 篤志 and 小川 潤一}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-525410(2019/05/28), 再表2019/239879(2021/02/12)} } @misc{CTT100845916, author = {布施新一郎 and 中村浩之 and 小竹佑磨 and 宮崎 俊一 and 伊東 篤志 and 小川 潤一}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-525411(2019/05/28), 再表2019/239880(2021/02/12)} } @misc{CTT100746386, author = {布施新一郎 and 和田雄二 and 米谷真人 and 高橋 孝志 and 増井 悠  and 海宝 龍夫  and 早瀬 修二  and 尾込 裕平}, title = {色素増感型光電変換素子用のヘテロ環リンカー基を有する完全有機色素化合物、およびそれを用いた光電変換素子}, howpublished = {登録特許}, year = 2019, month = {}, note = {特願2015-201952(2015/10/13), 特開2017-076648(2017/04/20), 特許第6534331号(2019/06/07)} }