@article{CTT100809276, author = {S. Fuse and K. Masuda and Y. Otake and H. Nakamura}, title = {Peptide chain elongation using unprotected amino acids in a micro-flow reactor}, journal = {Chem. Eur. J}, year = 2019, } @article{CTT100809286, author = {N. Sugisawa and Y. Otake and H. Nakamura and S. Fuse}, title = {Single-step, rapid, and mild synthesis of β-amino acid N-carboxy anhydrides using micro-flow technologies}, journal = {Chem. Asian J.}, year = 2019, } @inproceedings{CTT100822811, author = {増田耕志郎 and 小竹佑磨 and 中村浩之}, title = {マイクロフロー法を駆使する無保護アミノ酸直接連結によるペプチド鎖伸長法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100804153, author = {小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之 and 布施新一郎}, title = {アシルイミダゾリウムカチオン中間体を利用するマイクロフローN-メチル化ペプチド合成法の開発とPterulamide I-IVの全合成}, booktitle = {}, year = 2019, } @inproceedings{CTT100800122, author = {布施新一郎 and 小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之}, title = {N-メチル化ペプチドの超高効率マイクロフロー合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100798810, author = {柴田裕介 and 林慶浩 and 小竹佑磨 and 中村浩之 and 布施新一郎 and 川内進}, title = {イミダゾール誘導体を触媒とするN-メチルアミド化反応機構の理論的解明}, booktitle = {}, year = 2019, } @inproceedings{CTT100822791, author = {Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {Rapid and Mild Synthesis of Amino Acid N-Carboxy Anhydrides Using Basic-to-Acidic Flash Switching in a Micro-flow Reactor}, booktitle = {}, year = 2019, } @inproceedings{CTT100798655, author = {杉澤直斗 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {マイクロフロー合成法による瞬間混合を駆使したβ-アミノ酸-N-カルボキシ無水物の合成とその応用}, booktitle = {}, year = 2019, } @inproceedings{CTT100795963, author = {増田耕志郎 and 小竹佑磨 and 中村浩之 and 布施新一郎}, title = {無保護アミノ酸連結を基盤とするマイクロフローペプチド鎖伸長法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100795962, author = {小竹佑磨 and 柴田裕介 and 林慶浩 and 川内進 and 中村浩之 and 布施新一郎}, title = {アシルイミダゾリウムカチオン中間体を利用するマイクロフローNーメチル化ペプチド合成法の開発}, booktitle = {}, year = 2019, } @inproceedings{CTT100792094, author = {Yuma Otake and Hiroyuki Nakamura and Shinichiro Fuse}, title = {An efficient synthesis of N-methylated peptides using micro-flow technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100792085, author = {Shinichiro Fuse and Yuma Otake and Hiroyuki Nakamura}, title = {Development of Amide Bond Formation of N-Methyl Amino Acids Using Micro-Flow Technology}, booktitle = {}, year = 2019, } @inproceedings{CTT100792096, author = {増田 耕志郎 and 小竹 佑磨 and 中村 浩之 and 布施 新一郎}, title = {マイクロフロー法を駆使する無保護アミノ酸を用いたペプチド鎖伸長法の開発}, booktitle = {}, year = 2019, } @misc{CTT100866375, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-563042(2019/12/11), 再表2020/137545(2021/11/04)} } @misc{CTT100845903, author = {布施新一郎 and 中村浩之 and 小竹佑磨 and 宮崎 俊一 and 伊東 篤志 and 小川 潤一}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-525410(2019/05/28), 再表2019/239879(2021/02/12)} } @misc{CTT100845916, author = {布施新一郎 and 中村浩之 and 小竹佑磨 and 宮崎 俊一 and 伊東 篤志 and 小川 潤一}, title = {アミドの製造方法}, howpublished = {公開特許}, year = 2021, month = {}, note = {特願2020-525411(2019/05/28), 再表2019/239880(2021/02/12)} } @misc{CTT100826091, author = {布施新一郎 and 小竹佑磨 and 中村浩之}, title = {フローリアクターを用いるN-カルボキシ無水物の合成方法}, howpublished = {登録特許}, year = 2023, month = {}, note = {特願2019-094952(2019/05/21), 特開2020-011948(2020/01/23), 特許第7362055号(2023/10/06)} }