@article{CTT100864841, author = {Y. Asawa and S. Hatsuzawa and A. Yoshimori and K. Yamada and A. Katoh and H. Kouji and H. Nakamura}, title = {Comprehensive Exploration of Chemical Space Using Trisubstituted Carboranes}, journal = {Sci. Rep.}, year = 2021, } @article{CTT100863388, author = {Yasunobu Asawa and Kei Nishida and Kazuki Kawai and Kiyotaka Domae and Hyun Seung Ban and Akihiro Kitazaki and Hiroya Asami and Jun-Ya Kohno and Satoshi Okada and Hiraku Tokuma and Daisuke Sakano and Shoen Kume and Masaru Tanaka and Hiroyuki Nakamura}, title = {Carborane as an Alternative Efficient Hydrophobic Tag for Protein Degradation}, journal = {Bioconjugate Chemistry}, year = 2021, } @article{CTT100845898, author = {Y. Asawa and A. V. Arsent’eva and S. A. Anufriev and A. A. Anisimov and K. Yu. Suponitsky and O. A. Filippov and H. Nakamura and I. B. Sivaev}, title = {Synthesis of Bis(Carboranyl)amides 1,1’-μ-(CH2NH(O)C(CH2)n- 1,2-C2B10H11)2 (n = 0, 1) and Attempt of Synthesis of Gadolinium Bis(Dicarbollide}, journal = {Molecules}, year = 2021, } @article{CTT100853226, author = {R. Yudi Utomo and Y. Asawa and S. Okada and A. Yoshimori and J. Bajorath and H. Nakamura}, title = {Development of curcumin-based amyloid β aggregation inhibitors for Alzheimer's disease using the SAR matrix-approach}, journal = {Bioorg. Med. Chem.}, year = 2021, } @article{CTT100842476, author = {Takahiro Shimizu and NorihitoTakahashi and Vincent J.Huber and Yasunobu Asawa and Hiroki Ueda and Atsushi Yoshimori and Yukiko Muramatsu and Hiroyuki Seimiya and Hiroyuki Kouji and Hiroyuki Nakamura and Hiroki Oguri}, title = {Design and synthesis of 14 and 15-membered macrocyclic scaffolds exhibiting inhibitory activities of hypoxia-inducible factor 1α}, journal = {Bioorg. Med. Chem.}, year = 2021, } @inproceedings{CTT100858346, author = {浅輪 泰允 and 中村 浩之}, title = {カルボランを基盤とした立体的分子による3次元ケミカルスペースの探索と新規PPI制御分子の創成}, booktitle = {}, year = 2021, } @inproceedings{CTT100864816, author = {Yasunobu Asawa and Saki Hatsuzawa and Atsushi Yoshimori and Kentaro Yamada and Akira Katoh and Hiroyuki Kouji and Hiroyuki Nakamura}, title = {Comprehensive exploration of three-dimensional chemical space by trisubstituted carboranes for discovery of bioactive molecule}, booktitle = {}, year = 2021, } @inproceedings{CTT100864739, author = {浅輪泰允 and 中村浩之}, title = {疎水性ホウ素クラスターによる新規タンパク質分解誘導剤の開発とその機構解明}, booktitle = {}, year = 2021, } @inproceedings{CTT100853239, author = {浅輪泰允 and 吉森篤史 and 山田健太郎 and 小路弘行 and 中村浩之}, title = {カルボランを基盤とした立体的分子による3次元ケミカルスペースの探索とそのPPI制御機能評価}, booktitle = {}, year = 2021, } @inproceedings{CTT100853233, author = {村上弘樹 and 盛田大輝 and 浅輪泰允 and 中村浩之}, title = {パラジウム触媒を用いた1,2-アザボリン類のN-H/B-H二官能基化法の開発}, booktitle = {}, year = 2021, } @inproceedings{CTT100853240, author = {初澤早貴 and 浅輪泰允 and 吉森篤史 and 山田健太郎 and 小路弘行 and 真崎康博 and 中村浩之}, title = {PPI阻害剤を志向した三置換メタカルボランライブラリー化合物の合成とその生物活性評価}, booktitle = {}, year = 2021, } @misc{CTT100881786, author = {中村浩之 and 浅輪泰允 and 織田 昌幸}, title = {カルボラン化合物若しくはその塩又はこれらの溶媒和物}, howpublished = {公開特許}, year = 2022, month = {}, note = {PCT/JP2021/039442(2021/10/26), WO 2022/092068(2022/05/05)} }