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Publication List - Hiroyuki Nakamura 2022 (49 / 1220 entries)
Journal Paper
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Kohei Umedera,
Atsushi Yoshimori,
Hengwei Chen,
Hiroyuki Kouji,
Hiroyuki Nakamura,
Jurgen Bajorath.
DeepCubist: Molecular Generator for Designing Peptidomimetics based on Complex three-dimensional scaffolds,
Journal of Computer-Aided Molecular Design,
Vol. 37,
No. 2,
pp. 107-115,
Dec. 2022.
Official location
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Hiroyuki Nakamura.
Design of MMP-1 Inhibitors via SAR Transfer and Experimental Validation,
Dec. 2022.
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S. Ogawa,
Y. Asawa,
M. Iiyama,
A. Yoshimori,
H. Nakamura,
M. Oda.
Regulation of binding between CD28 cytoplasmic region and SH2 domains of Grb2 and PI3K by carborane compounds for T-cell activation,
BIOORG. MED. CHEM. LETT.,
Vol. 78,
129049,
Dec. 2022.
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K. Umedera,
T. Morita,
H. Nakamura.
Asymmetric construction of densely functionalized three-dimensional aza-tetracyclic scaffolds for drug discovery,
Chem. Commun,
Nov. 2022.
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Kazuki Miura,
Yijin Wen,
Michihiko Tsushima,
Hiroyuki Nakamura.
Photodynamic therapy by glucose transporter 1–selective light inactivation,
ACS Omega,
7,
38,
34685–34692,
Sept. 2022.
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K. Nishimura,
S. Harrison,
K. Kawai,
T. Morita,
K. Miura,
S. Okada,
H. Nakamura.
Iodophenyl-conjugated closo-dodecaborate as a promising small boron molecule that binds to serum albumin and accumulates in tumor,
BIOORG. MED. CHEM. LETT.,
Vol. 72,
128869,
Sept. 2022.
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Hiroyuki Nakamura.
ホウ素の拓く創薬ワールド,
細胞「特集 低分子モダリティの進化―元素・光・分子機能に注目して」,
54,
9,
Aug. 2022.
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H. Kitamura,
Y. Otake,
N. Sugisawa,
H. Sugisawa,
T. Ida,
H. Nakamura,
S. Fuse,
Hiroyuki Nakamura.
Sequential Selective Introduction of Alcohols against Phosphorus Trichloride in a Continuous-Flow Reactor and Consideration of a Mechanism for Reduced Overreaction via the Addition of Imidazole,
Chemistry,
28,
37,
e202200932,
July 2022.
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A. M.Hughes,
J. A. Goldfinger,
M. A. Palmieri,
P. Ramos,
I. S. Santa Cruz,
L. De Leo,
M. A. Garabalino,
S. I. Thorp,
P. Curotto,
E. C.C. Pozzi,
K. Kawai,
S. Sato,
M. E. Itoiz,
V.A. Trivillin,
J. S. Guidobono,
H. Nakamura,
A. E. Schwint.
Boron neutron capture therapy (BNCT) mediated by maleimide-functionalized closo-dodecaborate albumin conjugates (MID:BSA) for oral cancer: Biodistribution studies and in vivo BNCT in the hamster cheek pouch oral cancer model,
Life (Basel),
12,
7,
1082,
July 2022.
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A. R Jalilian,
A. Shahi,
I. P. Swainson,
H. Nakamura,
M. Venkatesh,
J. A. Osso Jr.
Potential theranostic BNCT agents as multimodal radiopharmaceuticals,
Cancer Biotherapy and Radiopharmaceuticals,
Vol. 37,
5,
June 2022.
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S. Koyama,
H. Sato,
H. Sugai,
M. Murakoshi,
T. Kobayashi,
S. Usami,
K. Ikeda,
Y. Haga,
K. Tsumoto,
H. Nakamura,
N. Hirasawa,
Kenji ISHIHARA,
H. Wada.
Effects of Salicylate Derivatives on Changes in Localization of H723R Pendrin Mutant Expressed in HEK293 Cells,
Auris Nasus Larynx,
Mar. 2022.
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T. Morita,
H. Murakami,
Y. Asawa,
H. Nakamura.
Enantioselective Synthesis of Oxazaborolidines by Palladium-Catalyzed N−H/B−H Double Activation of 1,2-Azaborines,
Angew. Chem. Int. Ed.,
Vol. 61,
Issue 7,
Feb. 2022.
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Tae-Hee Han,
M. K. Park,
H. Nakamura,
H. S. Ban.
Capsaicin inhibits HIF-1α accumulation through suppression of mitochondrial respiration in lung cancer cells,
Biomedicine & Pharmacotherapy,
Volume 146,
112500,
Feb. 2022.
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R. Y. Utomo,
S. Okada,
A. Sumiyoshi,
I. Aoki,
H. Nakamura.
Development of an MRI contrast agent for both detection and inhibition of the amyloid-β fibrillation process,
RSC Adv.,
Feb. 2022.
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Hiroyuki Nakamura.
BODIPY Catalyzes Proximity‐Dependent Histidine Labellin,
Feb. 2022.
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G. Li,
G. Yu,
C. Wang,
T. Morita,
X. Zhang,
H. Nakamura.
Copper(I)-catalysed intramolecular hydroarylation-redox cross-dehydrogenative coupling of N-propargylanilines with phosphites,
Org. biomol. chem.,
20,
113-116,
Jan. 2022.
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H. Ueda,
P.Wipf,
H. Nakamura.
Synthesis of sp3-rich chiral bicyclo[3.3.1]nonanes for chemical space expansion and study of biological activities,
Bioorganic & Medicinal Chemistry,
Volume 54,
116561,
Jan. 2022.
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R. Y. Utomo,
A. Sugie,
S. Okada,
K. Miura,
H. Nakamura.
Detoxification of amyloid β fibrils by curcumin derivatives and their verification in a Drosophila Alzheimer's model,
Chem. Commun.,
58,
2576-2579,
Jan. 2022.
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M. Tsuda,
T. Morita,
H. Nakamura.
Synthesis of isoxazoloazaborines via gold(i)-catalyzed propargyl aza-Claisen rearrangement/borylative cyclization cascade,
Chem. Commun.,
58,
1942-1945,
Jan. 2022.
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M. Tsushima,
S. Sato,
K. Miura,
T. Niwa,
HIDEKI TAGUCHI,
H. Nakamura.
Intracellular photocatalytic-proximity labeling for profiling protein–protein interactions in microenvironments,
Chem. Commun.,
58,
1926-1929,
Jan. 2022.
International Conference (Reviewed)
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Hiroyuki Nakamura.
Chemical Manipulation of Target Proteins Using Ruthenium bis(Bipyridine) Complexes,
The 27th International SPACC Symposium,
Dec. 2022.
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Hiroyuki Nakamura.
Development of Intracellular Photocatalytic Proximity Protein Labeling (iPPL) for Profiling Protein–Protein Interactions,
International Congress of Pure and Applied Chemistry (ICPACK)2022,
Nov. 2022.
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H. Nakamura,
T. Morita,
H. Murakami.
Development of 1,2-Azaborine-fused Heterocycles and Their Novel Functionalization,
The VIth International Conference,
Sept. 2022.
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Taiki Morita,
Hiroki Murakami,
Hiroyuki Nakamura.
Asymmetric Synthesis of Oxazaborolidines via Palladium-Catalyzed N-H/B-H Double Functionalization of 1,2-Azaborines,
The 9th European Conference on Boron Chemistry,
July 2022.
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Hiroyuki Nakamura,
Yasunobu Asawa.
Comprehensive Exploration of Chemical Space Using Trisubstituted Carboranes,
The 9th European Conference on Boron Chemistry,
July 2022.
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Hiroyuki Nakamura.
Boron Delivery using Serum Albumin,
NCI Workshop on Neutron Capture Therapy for Cancer,
Apr. 2022.
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Hiroyuki Nakamura.
Development of Intracellular Photocatalytic Proximity Protein Labeling (iPPL),
9th International Conference on Chemical and Biological Sciences (ICCBS 2022),
Mar. 2022.
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Michihiko Tsushima,
Kazuki Miura,
Shinichi Sato,
Hiroyuki Nakamura.
Intrecellular photocatalytic proximity labeling for profiling protein-protein interactins in multimolecular crowding,
The 2nd International Symposium on Chemistry for Multimolecular Vrouding Biosystems,
Jan. 2022.
Domestic Conference (Reviewed)
Domestic Conference (Not reviewed / Unknown)
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Hiroshi Kitamura,
Yuma Otake,
Naoto Sugisawa,
杉澤宏樹,
井田朋智,
Hiroyuki Nakamura,
Shinichiro Fuse.
非対称リン酸トリエステルのマイクロフロー合成および反応機構解明,
第120回有機合成シンポジウム,
June 2022.
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Hiroshi Kitamura,
Yuma Otake,
Naoto Sugisawa,
杉澤宏樹,
井田朋智,
Hiroyuki Nakamura,
Shinichiro Fuse.
非対称リン酸トリエステルのマイクロフロー合成および反応機構解明,
創薬懇話会2022,
June 2022.
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Hiroyuki Nakamura,
Kai Nishimura,
Taiki Morita,
Satoshi Okada,
Kazuki Miura,
柏木秀基,
福尾祐介,
松本孔貴,
Minoru Suzuki,
中井啓,
川端信司.
中性子捕捉療法のための血清アルブミンを利用したホウ素キャリアの開発,
第27 回癌治療増感研究会,
Apr. 2022.
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Kazuki Miura,
Yijin Wen,
Michihiko Tsushima,
Hiroyuki Nakamura.
細胞透過型有機光触媒による標的タンパク質選択的不活性化と抗腫瘍活性プローブへの応用,
日本薬学会142春季年会,
Mar. 2022.
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Kai Nishimura,
Taiki Morita,
Satoshi Okada,
Kazuki Miura,
柏木秀基,
福尾祐介,
松本孔貴,
高田卓志,
Minoru Suzuki,
中井啓,
川端信司,
Hiroyuki Nakamura.
中性子捕捉療法のための、アルブミンリガンドを基軸としたホウ素キャリアの開発,
日本薬学会142春季年会,
Mar. 2022.
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社本乙華,
Keiji Komuro,
Naoto Sugisawa,
Hiroyuki Nakamura,
Shinichiro Fuse.
マイクロフローリアクター内での環状ペプチド合成法の開発,
日本化学会第102春季年会,
Mar. 2022.
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Ayana Uehara,
Taiki Morita,
佐々木雄彦,
Hiroyuki Nakamura.
リゾホスファチジルイノシトール(4,5)ビスリン酸の合成研究,
日本化学会第102春季年会,
Mar. 2022.
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Taiki Morita,
Hiroyuki Nakamura.
ピペラジン酸およびN-ヒドロキシアミノ酸の直接縮合を基盤としたDentigerumycin Aの合成研究,
日本化学会第102春季年会,
Mar. 2022.
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Hiroyuki Nakamura,
Rohmad.Yudi Utomo,
Satoshi Okada,
住吉晃,
Ichio Aoki.
アミロイドβ繊維化を検出・阻害するMRIプローブの開発,
日本化学会第102春季年会,
Mar. 2022.
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Hiroki Murakami,
Taiki Morita,
Hiroyuki Nakamura.
パラジウム触媒を用いた1,2-アザボリン類の不斉N-H/B-H二官能基化法の開発,
日本化学会第102春季年会,
Mar. 2022.
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Masato Tsuda,
Taiki Morita,
Hiroyuki Nakamura.
金(I)触媒によるプロパルギルアザClaisen転位反応を用いたイソオキサゾロアザボリンの合成と亜鉛カルベノイドによるN−O結合へのメチレン挿入反応の開発,
日本化学会第102春季年会,
Mar. 2022.
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Hiroyuki Nakamura.
中性子捕捉療法:承認までの軌跡と今後の展望,
第19回同位体科学研究会,
Mar. 2022.
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Rohmad.Yudi Utomo,
Atsushi Sugie,
Satoshi Okada,
Kazuki Miura,
Hiroyuki Nakamura.
Curcumin誘導体のアミロイドβ繊維の解離を介した解毒作用とショウジョウバエのアルツハイマー病モデルにおける検証,
日本薬学会142春季年会,
Mar. 2022.
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Hiroyuki Nakamura.
タンパク質夾雑空間解析のための細胞内光触媒近接場標識法(iPPL法)の開発,
新学術領域研究「分子夾雑の生命化学」第6回班会議,
Jan. 2022.
Patent
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Hiroyuki Nakamura,
Satoshi Okada.
新規蛍光検出薬.
Patent.
Published.
国立大学法人東京工業大学.
2022/05/13.
特願2022-079168.
2023/11/24.
特開2023-167748.
2023.
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Hiroyuki Nakamura,
Taiki Morita,
Satoshi Okada,
Kai Nishimura.
新規ホウ素薬剤.
Patent.
Published.
国立大学法人東京工業大学, 学校法人大阪医科薬科大学.
2022/03/10.
PCT/JP2022/010452.
2022/09/15.
WO 2022/191262.
2022.
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Shinichiro Fuse,
Hiroshi Kitamura,
Yuma Otake,
Hiroyuki Nakamura.
非対称型リン酸トリエステルの製造方法、対称型リン酸トリエステルの製造方法、リン酸エステルの製造方法、及び、有機リン化合物の製造方法.
Patent.
Published.
国立大学法人東京工業大学, 横河電機株式会社.
2022/02/04.
PCT/JP2022/004557.
2022/09/09.
WO 2022/185843.
2022.
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Hiroyuki Nakamura,
Yasunobu Asawa.
カルボラン化合物若しくはその塩又はこれらの溶媒和物.
Patent.
Published.
国立大学法人東京工業大学, 京都府公立大学法人.
2021/10/26.
PCT/JP2021/039442.
2022/05/05.
WO 2022/092068.
2022.
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Hiroyuki Nakamura,
Kohei Umedera,
Taiki Morita.
新規含窒素三環性骨格化合物およびその使用.
Patent.
Published.
国立大学法人東京工業大学, 株式会社大分大学先端医学研究所.
2020/12/09.
特願2020-204328.
2022/06/21.
特開2022-091476.
2022.
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Hiroyuki Nakamura,
Shinichi Sato.
電気化学的手法を用いたハロゲン化物の製造方法.
Patent.
Registered.
国立大学法人東京工業大学, 国立大学法人大阪大学.
2018/12/21.
特願2018-239130.
2020/07/02.
特開2020-100865.
特許第7166531号.
2022/10/28
2022.
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Hiroyuki Nakamura.
ホウ素含有葉酸誘導体.
Patent.
Registered.
国立大学法人東京工業大学, ステラファーマ株式会社.
2017/08/25.
特願2017-162387.
2019/03/14.
特開2019-038778.
特許第7154528号.
2022/10/07
2022.
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