|
Publication List - Hiroyuki Nakamura 2020 (64 / 1220 entries)
Journal Paper
-
Naoto Sugisawa,
Hiroyuki Nakamura,
Sinichiro Fuse.
Recent advances in the continuous-flow reactions using metal-free homogeneous catalysts,
Catalysts,
Vol. 10,
No. 11,
pp. 1321,
Nov. 2020.
-
Somaraju Yugandar,
Taiki Moritai,
Hiroyuki Nakamura.
Rhodium(III)-Catalyzed Direct C-H Functionalization of Isoxazoles with Alkynes, Alkenes and Sulfoxonium Ylides,
Org. Biomol. Chem,
No. 18,
pp. 8625–8628,
Oct. 2020.
-
Shinichi Sato,
Hiroyuki Nakamura.
Labeling of Peroxidase-Induced Oxidative Stress Hotspots by Hemin-Catalyzed Tyrosine Click,
Chem. Pharm. Bull.,
Vol. 68,
No. 9,
pp. 885-890,
Sept. 2020.
-
S. A. Anufriev,
I. B. Sivaev,
Hiroyuki Nakamura.
Two possible ways to combine boron and gadolinium for Gd-guided BNCT. A concept,
Phosphorus, Sulfur and Silicon,
Vol. 195,
No. 11,
pp. 910-917,
Sept. 2020.
-
Yasunobu. Asawa,
A. Yoshimori,
J. Bajorath,
Hiroyuki. Nakamura.
Prediction of an MMP-1 Inhibitor Activity Cliff Using the SAR Matrix Approach and Its Experimental Validation,
Sci. Rep,
No. 10,
pp. 14710,
Sept. 2020.
-
T. Masuzawa,
S. Sato,
T. Niwa,
H. Taguchi,
H. Nakamura,
T. Oyoshi.
G-Quadruplex-Proximity Protein Labeling Based on Peroxidase Activity,
Chem. Commun.,
No. 56,
pp. 11641-11644,
Aug. 2020.
-
Kazuki Kawai,
Kai Nishimura,
Satoshi Okada,
Shinichi Sato,
Minoru Suzuki,
T. Takata,
Hiroyuki Nakamura.
Cyclic RGD-Functionalized closo-Dodecaborate Albumin Conjugates as Integrin Targeting Boron Carriers for Neutron Capture Therapy,
Mol. Pharm.,
Vol. 17,
No. 10,
pp. 3740–3747,
Aug. 2020.
-
Sei-ichi Tanuma,
Takahiro Oyama,
Atsushi Yoshimori,
Kiyotaka Katsuragi,
Yuri Shibasaki,
Yasunobu Asawa,
Hiroaki Yamazaki,
Kosho Makino,
Miwa Okazawa,
Yoko Ogino,
Yoshimi Sakamoto,
Miyuki Nomura,
Akira Sato,
Hideaki Abe,
Hiroyuki Nakamura,
Hideyo Takahashi,
Nobuhiro Tanuma,
Fumiaki Uchiumi.
Structural insights into the tunnel-shaped cavity of human nicotinamide phosphoribosyltransferase using a close structural set of azacyclohexane-motif inhibitors,
Molecules,
Vol. 25,
No. 16,
pp. 3633,
Aug. 2020.
-
Fumiko Nakagawa,
H. Kawashima,
Taiki. Morita,
Hiroyuki. Nakamura.
Water-soluble closo-Docecaborate-conjugated Pteroyl Derivatives for Boron Neutron Capture Therapy: Evidence of Targeting to Folate Receptor-Mediated Cell Uptake,
Cells,
Vol. 9,
No. 7,
pp. 1615,
July 2020.
-
Shinichiro. Fuse,
Wataru Moriya,
Shinichi Sato,
Hiroyuki Nakamura.
Investigation into the influence of an acrylic acid acceptor in organic D-π-A sensitizers against phototoxicity,
Bioorg. Med. Chem.,
Vol. 28,
No. 13,
pp. 115558,
July 2020.
-
Jun. Kawamura,
Hiroshi. Kitamura,
Yuma. Otake,
Shinichiro. Fuse,
Hiroyuki. Nakamura.
Size-Controllable and Scalable Production of Liposomes Using a V-Shape Mixer Micro-Flow Reactor,
Org. Process Res. Dev.,
Vol. 24,
No. 10,
pp. 2122-2127,
June 2020.
-
Michihiko Tsushima,
Shinichi Sato,
Keita Nakane,
Hiroyuki Nakamura.
Target protein identification on the photocatalyst-functionalized magnetic affinity beads,
Current Protocol.,
Vol. 101,
Issue 1,
June 2020.
-
Guangzhe Li,,
Chengdong Wang,
Yueqing Li,,
Kun Shao,
Guo Yu,
Shisheng Wang,,
Xiuhan Guo,,
Weijie Zhao,
H. Nakamura.
Zinc (II)-Catalyzed Intramolecular Hydroarylation-Redox Cross-Dehydrogenative Coupling of N-Propargylamines with sp and sp3 Carbon Pronucleophiles: Facile Access to Multifunctionalized Tetrahydroquinolines,
Chem. Commun.,
Issue 56,
pp. Chem. Commun.,
May 2020.
-
S. Sato,
K. Nakane,
H. Nakamura.
Laccase-Catalysed Tyrosine Click Reaction,
Org. Biomol. Chem,
Vol. 2020,
No. 18,
pp. 3664-3668,
May 2020.
-
Wanaporn Yimchuen,
Tetsuya Kadonosono,
Yumi Ota,
Shinichi Sato,
Maika Kitazawa,
Tadashi Shiozawa,
Takahiro Kuchimaru,
Masumi Taki,
Yuji Ito,
Hiroyuki Nakamura,
Shinae Kizaka-Kondoh.
Strategic design to create HER2-targeting proteins with target-binding peptides immobilized on a fibronectin type III domain scaffold,
RSC Advances,
Vol. 10,
pp. 15154-15162,
Apr. 2020.
Official location
-
T. Morita,
S. Fuse,
H. Nakamura.
Novel Photochemical Conversion of Isoxazoles to 5-Hydroxyimidazolines: Possible Protein Labeling at Lysine Residues,
Org. Lett,
Apr. 2020.
-
Y. Otake,
Y. Shibata,
Y. Hayashi,
S. Kawauchi,
H. Nakamura,
S. Fuse.
N-Methylated Peptide Synthesis through Acyl N-Methylimidazolium Cation Generation Accelerated by a Brønsted Acid,
Angew. Chem. Int. Ed.,
Vol. 59,
No. 31,
pp. 12925-12930,
Apr. 2020.
-
Shinichi Sato,
Masaki Matsumura,
Tetsuya Kadonosono,
Satoshi Abe,
Takafumi Ueno,
Hiroshi Ueda,
Hiroyuki Nakamura.
Site-selective protein chemical modification of exposed tyrosine residues using tyrosine click reaction,
Bioconjugate Chemistry,
Mar. 2020.
Official location
-
Hiroyuki Nakamura.
ホウ素中性子捕捉療法:がん細胞内でα線を発生させる次世代放射線治療,
DDS学会誌,
Vol. 35,
No. 2,
pp. 129-136,
Mar. 2020.
-
Hiroyuki Nakamura.
Carrier proteins-based boron delivery to tumor,
Applied Radiation and Isotopes,
Mar. 2020.
Official location
-
Hiroyuki Nakamura.
Suppression of HIF-1α accumulation by betulinic acid through proteasome activation in hypoxic cervical cancer,
Biochemical and Biophysical Research Communications,
Mar. 2020.
Official location
-
Hiroyuki Nakamura.
Boron Neutron Capture Therapy Study of 10B Enriched Nanostructured Boron Carbide Against Cervical Cancer and Glioblastoma Cell Line,
Journal of Cluster Science,
Mar. 2020.
Official location
-
Hiroyuki Nakamura.
中性子捕捉療法のためホウ素薬剤研究開発の進展-ホウ素薬剤が今後適応疾患拡大の鍵を握る!,
日本原子力学会誌,
Jan. 2020.
-
Naoto Sugisawa,
Yuma Otake,
Hiroyuki Nakamura,
Shinichiro Fuse.
Single‐Step, Rapid, and Mild Synthesis of β‐Amino Acid N ‐Carboxy Anhydrides Using Micro‐Flow Technology,
Chemistry – An Asian Journal,
Vol. 15,
No. 1,
pp. 79-84,
Jan. 2020.
Official location
-
A. Kumar; M. Kaur; P. Singh; K. Singh; U. S. Gaharwar; R. Meena; M. Kumar; K. Nakagawa; S. Wu; M. Suzuki; H. Nakamura,
Hiroyuki Nakamura.
Boron Nitride (10BN) a prospective material for treatment of cancer by Boron Neutron Capture Therapy (BNCT),
Materials Letters,
Jan. 2020.
-
Shinichiro Fuse,
Tsukasa Oishi,
Keisuke Matsumura,
Yoshihiro Hayashi,
Susumu Kawauchi,
Hiroyuki Nakamura.
Design, synthesis, and evaluation of azo D–π-A dyes as photothermal agents,
Organic & Biomolecular Chemistry,
2020.
Official location
-
Naoto Sugisawa,
Hiroyuki Nakamura,
Shinichiro Fuse.
Micro-flow synthesis of β-amino acid derivatives via a rapid dual activation approach,
Chemical Communications,
2020.
Official location
-
Hiroyuki Nakamura.
Suppression of HIF-1α accumulation by betulinic acid through proteasome activation in hypoxic cervical cancer,
Biochemical and Biophysical Research Communications,
Vol. 523,
No. 3,
pp. 726 - 732,
2020.
Official location
International Conference (Not reviewed / Unknown)
-
Hiroyuki Nakamura.
Development of Protein Chemical Labeling: From Target Identification to Cancer Therapy,
The 21st RIES-Hokudai International Symposium, Invited Lecture (online, Sapporo),
Dec. 2020.
-
Hiroyuki Nakamura.
Albumin-Dodecaborate Conjugates as Efficient Boron Carriers for Neutron Capture Therapy,
A3-Five star symposium, Invited Lecture (online, Osaka),
Dec. 2020.
-
Hiroyuki Nakamura.
Development of Boron Agents for BNCT,
The 11th Annual Indonesian Society for Cancer Chemoprevention Conference and Congress (ISCC-11),
Nov. 2020.
-
Hiroyuki Nakamura,
Kazuki Kawai,
Kai Nishimura,
Satoshi Okada,
Takushi Takata,
Minoru Suzuki.
Albumin-Based Boron Delivery for Active Targeting to Tumor,
22nd Taiwan-Japan Neutron Capture Therapy Academic Conference of Elite, oral (online, Taiwan),
Oct. 2020.
-
Hiroyuki Nakamura,
Eva Hey-Hawkins.
Boron Compounds,
IAEA Virtual Technical Meeting on Advances in Boron Neutron Capture Therapy (EVT1905174) Session Speaker (online, Austria),
July 2020.
-
Hiroyuki Nakamura.
Boron Delivery Agents for BNCT: Current Status and Future Prospects,
IAEA Virtual Technical Meeting on Advances in Boron Neutron Capture Therapy (EVT1905174) oral (online, Austria),
July 2020.
Domestic Conference (Not reviewed / Unknown)
-
Hiroyuki Nakamura,
Taiki Morita,
福原 信太郎,
Hiroyuki Nakamura.
金(I)触媒を用いたプロパルギルアザClaisen転位反応による5-アレニルイソオキサゾールの合成,
第10回CSJ化学フェスタ2020(オンライン),
Oct. 2020.
-
Hiroyuki Nakamura.
がんの低侵襲治療法(中性子捕捉療法):承認までの軌跡と今後の展望,
第15 回四大学連合文化講演会、招待講演(東京),
Oct. 2020.
-
Hiroyuki Nakamura,
Yuma Otake,
Hiroyuki Nakamura,
Shinichiro Fuse.
マイクロフローリアクター内でのpH瞬間転換と両基質同時活性化を駆使したβ-アミノ酸-N-カルボン酸無水物の合成と誘導体化,
第117回有機合成シンポジウム(オンライン),
Oct. 2020.
-
Hiroyuki Nakamura,
高門輝,
岩本真幸,
老木成稔,
Hiroyuki Nakamura,
岩田耕一.
ピコ秒時間分解けい光分光法を用いて評価した局所麻酔薬の脂質二重膜への影響,
日本分光学会分光学会年次講演会,
Oct. 2020.
-
YU Guo,
ZHANG Xuhai,
LI Guangzhe,
Hiroyuki Nakamura.
Synthesis of 2-Phosphonotetrahydroquinoline with Site-Selective C-H Bond Functionalization through Intramolecular Hydroarylation-Redox CDC Reaction,
第10回CSJ化学フェスタ2020(オンライン),
Oct. 2020.
-
Hiroyuki Nakamura,
Yuma Otake,
Hiroyuki Nakamura,
布施 新一郎.
マイクロフローリアクター内でのトリホスゲンを用いた環状ペプチド合成法の開発,
第10回CSJ化学フェスタ2020(オンライン),
Oct. 2020.
-
Yasunobu Asawa,
吉森 篤史,
BAJORATH J?rgen,
Hiroyuki Nakamura.
SAR空間の可視化によるActivity cliffの予測とその実験的検証,
第10回CSJ化学フェスタ2020(オンライン),
Oct. 2020.
-
Michihiko Tsushima,
Yijin Wen,
津賀雄輝,
金森功吏,
湯浅英哉,
Hiroyuki Nakamura.
リガンド連結型有機光触媒を用いた標的タンパク質の酸化的不活性化と抗腫瘍活性,
LASER WEEK IN KOCHI(オンライン),
Oct. 2020.
-
岡田夏実,
岩本真幸,
高門輝,
Hiroyuki Nakamura,
老木成稔,
岩田耕一.
ピコ秒時間分解けい光分光法で評価した脂質二重膜の粘度に対する局所麻酔薬の影響―脂質分子の極性基による違い,
分子科学オンライン討論会,
Sept. 2020.
-
塩野晴菜,
高門輝,
髙屋智久,
Hiroyuki Nakamura,
岩田耕一.
時間分解けい光分光法による脂質二重膜ナノディスクの粘度評価,
分子科学オンライン討論会,
Sept. 2020.
-
Hiroyuki Nakamura,
Kawai Kazuki,
Shinichi Sato,
Minoru Suzuki,
.
Albumin-Based Boron Delivery to Tumor by Active Targeting via αvβ3 Integrin,
the 59th ANNUAL CONFERENCE OF THE PARTICLE THERAPY CO-OPERATIVE GROUP (PTCOG-59)(online, Taiwan),
Sept. 2020.
-
Shinichi Sato,
増澤樹,
大吉崇文,
丹羽達也,
田口英樹,
Hiroyuki Nakamura.
ペルオキシダーゼ活性の変化と近接標識を利用したグアニン四重鎖結合タンパク質の選択的化学修飾,
第14回バイオ関連化学シンポジウム2020(オンライン),
Sept. 2020.
-
Michihiko Tsushima,
Shinichi Sato,
Hiroyuki Nakamura.
タンパク質-タンパク質相互作用の解析を志向した細胞内触媒近接ラベル化の開発,
第64回日本薬学会関東支部大会(オンライン),
Sept. 2020.
-
Rohmad Yudi Utomo,
Yasunobu Asawa,
Atsushi Yoshimori,
Hiroyuki Nakamura.
Novel Curcumin Derivatives Generated from SAR Matrix Possess as Amyloid β Inhibitors for Alzheimer?s Disease,
第64回日本薬学会関東支部大会(オンライン),
Sept. 2020.
-
Hiroyuki Nakamura.
BNCT 用ホウ素薬剤:現在の状況と将来の展望、,
第2回生体量子捕獲反応研究会 特別講演(オンライン),
Aug. 2020.
-
Hiroyuki Nakamura.
細胞内タンパク質-タンパク質相互作用解析を可能とする光ラベル化技術の開発,
分子夾雑の生命化学 第3回オンラインセミナー,
Aug. 2020.
-
Yasunobu Asawa,
吉森篤史,
山田健太郎,
邵玉潔,
李廣晢,
加藤明良,
小路弘行,
Hiroyuki Nakamura.
タンパク質の2次構造を模倣した新規カルボランPPI制御分子の設計・合成とその機能評価,
日本薬学会第140年会,
Mar. 2020.
-
増澤樹,
Shinichi Sato,
Hiroyuki Nakamura,
大吉崇文.
ヘミンによって活性化したルミノール誘導体によるグアニン四重鎖結合タンパク質の選択的修飾,
日本化学会第100春季年会,
Mar. 2020.
-
Takahiro Shimizu,
Huber Vincent,
Atsushi Yoshimori,
Hiroki Ueda,
Hiroyuki Nakamura,
Hiroyuki Koji,
Hiroki Oguri.
Design, synthesis and biological evaluation of α-helix mimetics composed of skeletally diverse macrocyclic mid-sized scaffolds,,
日本化学会第100春季年会,
Mar. 2020.
-
Guo Yu,
Xuhai Zhang,
Guangzhe Li,
Hiroyuki Nakamura.
Synthesis of tetrahydroquinoline with site-selective C-H bond functionalization through IH-Redox CDC reaction,
日本化学会第100春季年会,
Mar. 2020.
-
Masato Tsuda,
Taiki Morita,
Shintaro Fukuhara,
Hiroyuki Nakamura.
金(I)触媒を用いたアザプロパルギルClaisen転位反応による5-アレニルイソオキサゾールの合成,
日本化学会第100春季年会,
Mar. 2020.
-
Naoto Sugisawa,
Yuma Otake,
Hiroyuki Nakamura,
Shinichiro Fuse.
β-アミノ酸-N-カルボン酸無水物の迅速かつ温和なワンフロー合成,
日本化学会第100春季年会,
Mar. 2020.
-
Kohei Umedera,
Taiki Morita,
Hiroyuki Nakamura.
飽和炭素に富むアザトリシクロドデセン骨格の合成,
日本化学会第100春季年会,
Mar. 2020.
-
Wataru Moriya,
Shinichiro Fuse,
Hiroyuki Nakamura.
光線力学療法を志向したDπA光増感剤の構造光毒性相関の解明,
日本化学会第100春季年会,
Mar. 2020.
-
Keita Nakane,
Shinichi Sato,
Michihiko Tsushima,
丹羽達也,
田口英樹,
Hiroyuki Nakamura.
アフィニティー担体上でのチロシン残基修飾による抗体の部位選択的修飾,
日本化学会第100春季年会,
Mar. 2020.
-
Shinichi Sato,
Hiroyuki Nakamura.
チロシン残基ラベル化における触媒的手法と電気化学的手法の比較,
日本化学会第100春季年会,
Mar. 2020.
-
Takahiro Shimizu,
Huber Vincent,
Atsushi Yoshimori,
Hiroki Ueda,
Hiroyuki Nakamura,
Hiroyuki Koji,
Hiroki Oguri.
Design, synthesis and biological evaluation of α-helix mimetics composed of skeletally diverse macrocyclic mid-sized scaffolds,
The Fourth A3 Young Scientist Meeting,
Mar. 2020.
-
Rohmad Yudi Utomo,
Yasunobu Asawa,
Shinichi Sato,
Atsushi Yoshimori,
Hiroyuki Nakamura.
Novel Curcumin Derivatives Generated from SAR Matrix Possess as Amyloid β Inhibitors,
日本薬学会第140年会,
Mar. 2020.
Patent
-
Hiroyuki Nakamura,
Kohei Umedera,
Taiki Morita.
新規含窒素三環性骨格化合物およびその使用.
Patent.
Published.
国立大学法人東京工業大学, 株式会社大分大学先端医学研究所.
2020/12/09.
特願2020-204328.
2022/06/21.
特開2022-091476.
2022.
-
Shinichiro Fuse,
Koshiro Masuda,
Yuma Otake,
Hiroyuki Nakamura.
アミドの製造方法.
Patent.
Published.
国立大学法人東京工業大学, 横河電機株式会社.
2020/02/03.
特願2021-501811.
2021/12/16.
再表2020/175023.
2021.
-
Shinichiro Fuse,
Yuma Otake,
Hiroyuki Nakamura.
フローリアクターを用いるN-カルボキシ無水物の合成方法.
Patent.
Registered.
国立大学法人東京工業大学, 保土谷化学工業株式会社.
2019/05/21.
特願2019-094952.
2020/01/23.
特開2020-011948.
特許第7362055号.
2023/10/06
2023.
-
Hiroyuki Nakamura,
Shinichi Sato.
電気化学的手法を用いたハロゲン化物の製造方法.
Patent.
Registered.
国立大学法人東京工業大学, 国立大学法人大阪大学.
2018/12/21.
特願2018-239130.
2020/07/02.
特開2020-100865.
特許第7166531号.
2022/10/28
2022.
-
Shinichi Sato,
Hiroyuki Nakamura.
電気化学的手法による修飾タンパク質の製造方法.
Patent.
Published.
国立大学法人東京工業大学.
2018/06/29.
特願2018-124834.
2020/01/09.
特開2020-002095.
2020.
-
Shinichi Sato,
Hiroyuki Nakamura.
チロシンホスファターゼ及びチロシンキナーゼ活性の測定方法.
Patent.
Registered.
国立大学法人東京工業大学.
2016/09/26.
特願2017-544450.
2018/09/06.
特開(再表)2017/061288.
特許第6770750号.
2020/09/30
2020.
-
Hiroyuki Nakamura.
ホウ素含有化合物とタンパク質とのコンジュゲートを含む医薬組成物.
Patent.
Registered.
国立大学法人東京工業大学.
2016/07/26.
特願2017-534171.
2018/05/24.
再表2017/026276.
特許第6788278号.
2020/11/04
2020.
[ Save as BibTeX ]
[ Paper, Presentations, Books, Others, Degrees: Save as CSV
]
[ Patents: Save as CSV
]
|